CRIS Current Research Information System

ROBERTI, MARINELLA
 Distribuzione geografica
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Continente #
NA - Nord America 3.931
EU - Europa 3.088
AS - Asia 1.159
AF - Africa 227
SA - Sud America 17
OC - Oceania 5
Totale 8.427
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Nazione #
US - Stati Uniti d'America 3.914
IT - Italia 817
GB - Regno Unito 679
DE - Germania 409
CN - Cina 346
SE - Svezia 342
SG - Singapore 288
VN - Vietnam 215
IN - India 189
UA - Ucraina 167
IE - Irlanda 151
FR - Francia 115
TG - Togo 84
RU - Federazione Russa 74
CH - Svizzera 64
EE - Estonia 57
BG - Bulgaria 53
ZA - Sudafrica 46
NG - Nigeria 42
JO - Giordania 40
CI - Costa d'Avorio 38
FI - Finlandia 24
ES - Italia 22
TW - Taiwan 21
BE - Belgio 19
HR - Croazia 18
NL - Olanda 16
BR - Brasile 13
CA - Canada 13
JP - Giappone 13
PL - Polonia 11
SC - Seychelles 11
GR - Grecia 10
HK - Hong Kong 10
MT - Malta 10
AT - Austria 7
CZ - Repubblica Ceca 7
IR - Iran 7
KR - Corea 7
TR - Turchia 7
PH - Filippine 6
PT - Portogallo 6
AU - Australia 5
RO - Romania 5
CL - Cile 4
EG - Egitto 4
MX - Messico 4
BD - Bangladesh 3
AE - Emirati Arabi Uniti 2
LB - Libano 2
DK - Danimarca 1
IL - Israele 1
IQ - Iraq 1
LI - Liechtenstein 1
MU - Mauritius 1
NO - Norvegia 1
RS - Serbia 1
SM - San Marino 1
SN - Senegal 1
UZ - Uzbekistan 1
Totale 8.427
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Città #
Southend 589
Fairfield 532
Chandler 416
Ashburn 365
Bologna 275
Woodbridge 272
Seattle 252
Singapore 245
Houston 222
Wilmington 209
Cambridge 197
Ann Arbor 172
Princeton 152
Dublin 149
Dong Ket 138
Jacksonville 99
Lomé 84
Nanjing 62
Westminster 60
Berlin 59
Padova 59
Santa Clara 52
Sofia 50
Abeokuta 41
Amman 40
Milan 40
Abidjan 38
Redmond 37
Bern 36
Shenyang 33
Jinan 32
New York 32
Turin 31
Dearborn 28
Hebei 27
Beijing 25
Changsha 21
Genoa 21
Helsinki 21
Mülheim 20
Bremen 19
Rome 18
Saint Petersburg 18
San Diego 18
Hyderabad 17
Nanchang 17
Brussels 16
Leawood 16
Tianjin 16
Boardman 13
Shanghai 13
Redwood City 12
Stockholm 12
Chicago 11
Des Moines 11
Haikou 11
Nürnberg 11
Bengaluru 10
Hangzhou 10
Mahé 10
Medford 10
Nerviano 10
Palermo 10
Amsterdam 9
Guangzhou 9
Olalla 9
Taipei 9
Zurich 9
Ahmedabad 8
Exeter 7
Lausanne 7
Norwalk 7
San Venanzo 7
Tokyo 7
Carlsbad 6
Cento 6
Florence 6
Forlì 6
Modena 6
Mountain View 6
Ningbo 6
Paris 6
Porto Alegre 6
Taizhou 6
Valletta 6
Vienna 6
Wanchai 6
Zhengzhou 6
Ancona 5
Cebu City 5
Falls Church 5
Frankfurt am Main 5
Genova 5
Gothenburg 5
Hefei 5
Istanbul 5
Jiaxing 5
Los Angeles 5
New Taipei City 5
Taiyuan 5
Totale 5.774
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Nome #
A Focused Library of Psychotropic Analogues with Neuroprotective and Neuroregenerative Potential 230
A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation 200
Antioxidant Activity of Hydroxystilbene Derivatives in Homogeneous Solution 197
Rad51/Brca2 Disruptors Inhibit Homologous Recombination and Synergize with Olaparib in Pancreatic Cancer Cells 174
Synthetic Lethality in Pancreatic Cancer: Discovery of a New RAD51-BRCA2 Small Molecule Disruptor That Inhibits Homologous Recombination and Synergizes with Olaparib 174
A RAD51/BRCA2 small molecule inhibitor enhances the antineoplastic effect of the PARPi talazoparib in pancreatic cancer 171
Computational design and discovery of "minimally structured" hERG blockers. 165
Characterisation of bioactive compounds in wine by-products: toward the valorisation of sustainable resources 153
Arylsulphones: A Promising Class on Non-Nucleoside Antiviral Agents 152
SINTESI PARALLELA DI UNA COLLEZIONE DI PICCOLE MOLECOLE SIMIL-NATURALI MEDIANTE REAZIONE DOMINO KNOEVENAGEL/ DIELS-ALDER 147
Antiproliferative agents that interfere with the cell cycle at the G(1)-->S transition: further development and characterization of a small library of stilbene-derived compounds 146
Berberine and its metabolites: Relationship between physicochemical properties and plasma levels after administration to human subjects 146
Capitolo 2. Proprietà chimico-fisiche e attività biologica 142
Domino Knovenaegel/Diels-Alder Sequence Coupled to Suzuki Reaction: a Powerful Synthetic Platform for Chemical Biology 134
Parallel Synthesis, Evaluation, and Preliminary Structure-Activity Relationship of 2,5-Diamino-1,4-benzoquinones as a Novel Class of Bivalent Anti-Prion Compound. 134
Benzimidazole derivatives as kinase inhibitors 134
LDH inhibition impacts on heat shock response and induces senescence of hepatocellular carcinoma cells 134
Galloflavin, a new lactate dehydrogenase inhibitor, induces the death of human breast cancer cells with different glycolytic attitude by affecting distinct signaling pathways. 133
Multitarget Drug Design Strategy: Quinone–Tacrine Hybrids Designed To Block Amyloid-β Aggregation and To Exert Anticholinesterase and Antioxidant Effects 133
Lactate dehydrogenase inhibitors can reverse inflammation induced changes in colon cancer cells 132
Enriching Proteolysis Targeting Chimeras with a Second Modality: When Two Are Better Than One 131
Galloflavin (CAS 568-80-9), a novel inhibitor of lactate dehydrogenase. 129
A natural-like synthetic small molecule impairs bcr-abl signaling cascades and induces megakaryocyte differentiation in erythroleukemia cells 127
Differential antiproliferative activity of new benzimidazole- 4,7-diones. 126
Diaryl Urea: A Privileged Structure in Anticancer Agents 123
Lactate dehydrogenase inhibitors sensitize lymphoma cells to cisplatin without enhancing the drug effects on immortalized normal lymphocytes. 122
Hybrid Lipoic Acid Derivatives to Attack Prion Disease on Multiple Fronts 121
Synthetic Lethality Triggered by Combining Olaparib with BRCA2-Rad51 Disruptors 120
Domino Knoevenagel/Diels–Alder sequence coupled to Suzuki reaction: a valuable synthetic platform for chemical biology 119
Effects of trans-stilbene and terphenyl compounds on different strains of Leishmania and on cytokines production from infected macrophages 119
Inhibition of Urease, a Ni-Enzyme: The Reactivity of a Key Thiol With Mono- and Di-Substituted Catechols Elucidated by Kinetic, Structural, and Theoretical Studies 118
Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A 113
Pterostilbene and 3'-hydroxypterostilbene are effective apoptosis-inducing agents in MDR and BCR-ABL-expressing leukemia cells 113
Docking ligands on protein surfaces: the case study of prion protein. 110
Novel antiproliferative chimeric compounds with marked histone deacetylase inhibitory activity. 109
Non-ATP competitive protein kinase inhibitors 107
Identification of a terphenyl derivative that blocks the cell cycle in the G0-G1 phase and induces differentiation in leukemia cells. 107
Suppression of human monocyte tissue factor induction by red wine phenolics and synthetic derivatives of resveratrol 105
Lactate dehydrogenase inhibition affects homologous recombination repair independently of cell metabolic asset; implications for anticancer treatment 103
Polo-like kinases inhibitors 102
TTAS a New Stilbene Derivative that Induces Apoptosis in Leishmania Infantum 102
Synthesis and Pharmacology of 6-Substituted Benztropines: Discovery of Novel Dopamine Uptake Inhibitors Possessing Low Binding Affinity to the Dopamine Transporter 102
null 101
null 101
Nitrogen-containing heterocyclic quinones: a class of potential selective antitumor agents 101
null 98
Stilbene-based anticancer agents: Resveratrol analogues active toward HL60 leukemic cells with a non-specific phase mechanism. 96
Probing the binding sites and mechanisms of action of two human ether-a-go-go-related gene channel activators, 1,3-bis-(2-hydroxy-5-trifluoromethyl-phenyl)-urea (NS1643) and 2-[2-(3,4-dichloro-phenyl)-2,3-dihydro-1H-isoindol-5-ylamino]-nicotinic acid (PD307243) 96
Thermal and catalytic reactions of ethyl diazopiruvate with [60]fullerene 93
Heterocyclic and Phenyl Double-Bond-Locked Combretastatin Analogues Possessing Potent Apoptosis-Inducing Activity in HL60 and in MDR Cell Lines 92
Identification of biphenyl-based hybrid molecules able to decrease the intracellular level of Bcl-2 protein in Bcl-2 overexpressing leukemia cells 91
Small molecule aurora kinases inhibitors 91
A journey through targeting BRCA2-RAD51 protein-protein interaction to establish synthetic lethality as paradigm for anticancer drug discovery 90
Identification of a Terphenyl-Based Small Molecule That Induces Differentiation in Leukemia Cells 88
null 87
Sequential Virtual Screening Approach to the Identification of Small Organic Molecules as Potential BACE-1 Inhibitors 87
Synthesis and Biological Evaluation of Novel 1'-Branched and Spiro-Nucleoside Analogues 86
Studies on the Apoptotic Activity of Natural and Synthetic Retinoids: Discovery of a New Class of Synthetic Terphenyls That Potently Support Cell Growth and Inhibit Apoptosis in Neuronal and HL-60 Cells 85
null 81
Identification and characterization of a terphenyl derivative blocking the G1-S transition in neoplastic cells 74
null 74
Insights into the activity of ARN24089, a new RAD51-BRCA2 disruptor that inhibits homologous recombination and achieves synthetic lethality in pancreatic cancer 72
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign 72
null 68
Proteostasis Regulators in Cystic Fibrosis: Current Development and Future Perspectives 66
DESIGN OF LIGANDS WITH A HIGH AFFINITY TO PrPC 65
Combined analytical approaches to define biodistribution and biological activity of semi-synthetic berberrubine, the active metabolite of natural berberine 60
null 56
Identification and subsequent development of RAD51-BRCA2 disruptors through a fragment-based approach 55
Multiple Ligand Strategy in anticancer drug discovery 55
Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors 54
Antiparasitic effect of stilbene and terphenyl compounds against trypanosoma cruzi parasites 54
null 53
Free-radical-mediated formation of trans-cardiolipin isomers, analytical approaches for lipidomics and consequences of the structural organization of membranes 51
null 51
Identification of RAD51-BRCA2 Inhibitors Using N-Acylhydrazone-Based Dynamic Combinatorial Chemistry 49
The Mechanistic Understanding of RAD51 Defibrillation: A Critical Step in BRCA2-Mediated DNA Repair by Homologous Recombination 44
Multi-kinase inhibitors 42
Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease 40
In vitro antileishmanial activity of trans-stilbene and terphenyl compounds 38
Synthetic small molecule Cdc25 phosphatases inhibitors 36
An 19F NMR fragment-based approach for the discovery and development of BRCA2-RAD51 inhibitors to pursuit synthetic lethality in combination with PARP inhibition in pancreatic cancer 35
The use of stilbene scaffold in medicinal chemistry and multi-target drug design 32
A ligand-based virtual screening approach to identify small molecules as hERG channel activators 25
Innovative Strategy toward Mutant CFTR Rescue in Cystic Fibrosis: Design and Synthesis of Thiadiazole Inhibitors of the E3 Ligase RNF5 22
Irreversible protein kinase inhibitors 18
New Horizons of Synthetic Lethality in Cancer: Current Development and Future Perspectives 16
RAD51 nuclear recruitment and inhibition towards innovative strategies against pancreatic cancer 15
Preomic profile of BxPC-3 cells after treatment with BRC4 11
Application of an “inhalation by design” approach to the identification and in-vitro evaluation of novel purine based PI3Kδ inhibitors 11
Proteomic profile of BxPC-3 cells after treatment with BRC4 6
Totale 8.643
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Categoria #
all - tutte 21.447
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 21.447
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/20201.765 0 0 27 112 217 217 285 301 284 142 68 112
2020/20211.240 203 97 31 62 76 118 31 76 113 79 62 292
2021/20221.254 107 31 113 82 112 72 45 117 62 82 224 207
2022/20231.887 148 301 130 218 159 139 62 122 294 76 108 130
2023/2024973 98 102 49 94 64 126 68 68 29 79 100 96
2024/2025524 137 338 49 0 0 0 0 0 0 0 0 0
Totale 8.643