CAVALLI, ANDREA
CAVALLI, ANDREA
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di Ia fascia
Cavalli, ANDREA
A chemical biology probe identified through 19F NMR screening stimulates RAD51 oligomerization and disrupts BRC4 binding
2026 Rinaldi, F.; Veronesi, M.; Masi, M.; Andonaia, A.; Bosio, S.; Varignani, G.; Catalano, F.; Marotta, R.; Falchi, F.; Girotto, S.; Cavalli, A.
A Metabolites' Interplay Can Modulate DNA Repair by Homologous Recombination
2026 Rossi, Valentina; Masi, Mirco; Govoni, Marzia; Veronesi, Marina; Duca, Martina; Girotto, Stefania; Cavalli, Andrea; Di Stefano, Giuseppina
An integrated biophysical and structural biology approach to investigate the BRCA2-RAD51 interaction
2026 Rinaldi, F.; Franco, P.; Langer, G.; Girotto, S.; Cavalli, A.
Critical Assessment of a Structure-Based Pipeline for Targeting the Long Noncoding RNA MALAT1
2026 Aguti, Riccardo; Bernetti, Mattia; Elisi, Gian Marco; Cavalli, Andrea; Masetti, Matteo
Decoding the RAD51–BRC repeats interplay in Homologous Recombination
2026 Rinaldi, F.; Franco, P.; Langer, J. D.; Girotto, S.; Cavalli, A.
Molecular determinants of the BRC Repeats - RAD51 recognition
2026 Rinaldi, F.; Franco, P.; Langer, J. D.; Girotto, S.; Cavalli, A.
Targeting RAD51-BRCA2 Interaction to Enhance Synthetic Lethality with Olaparib in Pancreatic Cancer: Development of a Novel Phenyl Furan-Quinoline-Carboxylic Acid Series
2026 Ferrandi, G; Bagnolini, G; Poppi, L; Masi, M; Previtali, V; Andonaia, A; Varignani, G; Veronesi, M; De Franco, F; Falchi, F; Di Stefano, G; Girotto, S; Roberti, M; Cavalli, A
An integrative structural study of RAD52, an emerging target in anticancer drug discovery
2025 Rinaldi, F.; Balboni, B.; Girotto, S.; Cavalli, A.
Dissecting the RAD51-BRC4 Interaction Landscape through Integrative Molecular Simulations and Experimental Biophysics
2025 Bresciani, V.; Rinaldi, F.; Franco, P.; Girotto, S.; Cavalli, A.; Langer, J. D.; Masetti, M.; Bernetti, M.
Elucidating RAD52 architecture through an integrated structural biology approach
2025 Rinaldi, F.; Balboni, B.; Marotta, R.; Girotto, S.; Cavalli, A.
Elucidating the BRCA2-RAD51 interaction through an integrated biophysical and structural biology approach
2025 Rinaldi, F.; Bresciani, V.; Franco, P.; Bernetti, M.; Langer, J.; Cavalli, A.; Girotto, S.
Exploration of the Neuromodulatory Properties of Fyn and GSK-3β Kinases Exploiting 7-Azaindole-Based Inhibitors
2025 Marotta, Giambattista; Massenzio, Francesca; Ortega, Jose; Russo, Debora; Penna, Ilaria; Falchi, Federico; Babini, Giorgia; Petralla, Sabrina; Scarpelli, Rita; Roggiolani, Elena; Fricker, Gert; Rosini, Michela; Cavalli, Andrea; Monti, Barbara; Minarini, Anna; Basagni, Filippo
IN SEARCH OF SMALL MOLECULES TARGETING RAD52 FOR SYNTHETIC LETHALITY
2025 Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Varignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli, Rita; Girotto, Stefania; Cavalli, Andrea
Investigating synthetic lethality and PARP inhibitor resistance in pancreatic cancer through enantiomer differential activity
2025 Masi, Mirco; Poppi, Laura; Previtali, Viola; Nelson, Shannon R; Wynne, Kieran; Varignani, Giulia; Falchi, Federico; Veronesi, Marina; Albanesi, Ennio; Tedesco, Daniele; De Franco, Francesca; Ciamarone, Andrea; Myers, Samuel H; Ortega, Jose Antonio; Bagnolini, Greta; Ferrandi, Giovanni; Farabegoli, Fulvia; Tirelli, Nicola; Di Stefano, Giuseppina; Oliviero, Giorgio; Walsh, Naomi; Roberti, Marinella; Girotto, Stefania; Cavalli, Andrea
IsoBayes: a Bayesian approach for single-isoform proteomics inference
2025 Bollon, Jordy; R Shortreed, Michael; Jeffery, Erin; T Jordan, Ben; Miller, Rachel; Cavalli, Andrea; M Smith, Lloyd; N Dewey, Colin; M Sheynkman, Gloria; Tiberi, Simone
Probing the BRC repeats RAD51 interaction by integrating computational and experimental biophysics
2025 Rinaldi, F.; Bresciani, V.; Franco, P.; Veronesi, M.; Bernetti, M.; Masetti, M.; Langer, J.; Cavalli, A.; Girotto, S.
Rational optimization of D3R/GSK-3β dual target-directed ligands as potential treatment for bipolar disorder: Design, synthesis, X-ray crystallography, molecular dynamics simulations, in vitro ADME, and in vivo pharmacokinetic studies
2025 Di Martino, R. M. C.; Russo, D.; Penna, I.; Demuro, S.; Dalle Vedove, A.; Spagnuolo, R.; Ottonello, G.; Bertozzi, S. M.; Summa, M.; Desantis, J.; Valeri, A.; Pruccoli, L.; Tripathi, S. K.; Tarozzi, A.; Storici, P.; Girotto, S.; Bertorelli, R.; Armirotti, A.; Cruciani, G.; Bandiera, T.; Cavalli, A.; Bottegoni, G.
TARGETING RAD52 FOR SYNTHETIC LETHALITY: DISCOVERY OF A NOVEL SMALL MOLECULE AS A PROMISING INHIBITOR FOR CANCER THERAPY
2025 Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Varignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli Stefania Girotto, Rita; Cavalli, Andrea
The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study
2025 Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A.
The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study
2025 Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A.
| Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
|---|---|---|---|---|---|---|
| A chemical biology probe identified through 19F NMR screening stimulates RAD51 oligomerization and disrupts BRC4 binding | Rinaldi, F.; Veronesi, M.; Masi, M.; Andonaia, A.; Bosio, S.; Varignani, G.; Catalano, F.; Marott...a, R.; Falchi, F.; Girotto, S.; Cavalli, A. | 2026-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| A Metabolites' Interplay Can Modulate DNA Repair by Homologous Recombination | Rossi, Valentina; Masi, Mirco; Govoni, Marzia; Veronesi, Marina; Duca, Martina; Girotto, Stefania...; Cavalli, Andrea; Di Stefano, Giuseppina | 2026-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | IJMS 2026.pdf |
| An integrated biophysical and structural biology approach to investigate the BRCA2-RAD51 interaction | Rinaldi, F.; Franco, P.; Langer, G.; Girotto, S.; Cavalli, A. | 2026-01-01 | - | - | 4.03 Poster | - |
| Critical Assessment of a Structure-Based Pipeline for Targeting the Long Noncoding RNA MALAT1 | Aguti, Riccardo; Bernetti, Mattia; Elisi, Gian Marco; Cavalli, Andrea; Masetti, Matteo | 2026-01-01 | JOURNAL OF CHEMICAL INFORMATION AND MODELING | - | 1.01 Articolo in rivista | 2026_Aguti_critical-assessment-of-a-structure-based-pipeline-for-targeting-the-long-noncoding-rna-malat1.pdf; 2026_Aguti_SI_critical-assessment-of-a-structure-based-pipeline-for-targeting-the-long-noncoding-rna-malat1.pdf |
| Decoding the RAD51–BRC repeats interplay in Homologous Recombination | Rinaldi, F.; Franco, P.; Langer, J. D.; Girotto, S.; Cavalli, A. | 2026-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Molecular determinants of the BRC Repeats - RAD51 recognition | Rinaldi, F.; Franco, P.; Langer, J. D.; Girotto, S.; Cavalli, A. | 2026-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Targeting RAD51-BRCA2 Interaction to Enhance Synthetic Lethality with Olaparib in Pancreatic Cancer: Development of a Novel Phenyl Furan-Quinoline-Carboxylic Acid Series | Ferrandi, G; Bagnolini, G; Poppi, L; Masi, M; Previtali, V; Andonaia, A; Varignani, G; Veronesi, ...M; De Franco, F; Falchi, F; Di Stefano, G; Girotto, S; Roberti, M; Cavalli, A | 2026-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | targeting-rad51-brca2-interaction-to-enhance-synthetic-lethality-with-olaparib-in-pancreatic-cancer-development-of-a.pdf |
| An integrative structural study of RAD52, an emerging target in anticancer drug discovery | Rinaldi, F.; Balboni, B.; Girotto, S.; Cavalli, A. | 2025-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Dissecting the RAD51-BRC4 Interaction Landscape through Integrative Molecular Simulations and Experimental Biophysics | Bresciani, V.; Rinaldi, F.; Franco, P.; Girotto, S.; Cavalli, A.; Langer, J. D.; Masetti, M.; Ber...netti, M. | 2025-01-01 | JOURNAL OF CHEMICAL INFORMATION AND MODELING | - | 1.01 Articolo in rivista | dissecting-the-rad51-brc4-interaction-landscape-through-integrative-molecular-simulations-and-experimental-biophysics.pdf |
| Elucidating RAD52 architecture through an integrated structural biology approach | Rinaldi, F.; Balboni, B.; Marotta, R.; Girotto, S.; Cavalli, A. | 2025-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Elucidating the BRCA2-RAD51 interaction through an integrated biophysical and structural biology approach | Rinaldi, F.; Bresciani, V.; Franco, P.; Bernetti, M.; Langer, J.; Cavalli, A.; Girotto, S. | 2025-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Exploration of the Neuromodulatory Properties of Fyn and GSK-3β Kinases Exploiting 7-Azaindole-Based Inhibitors | Marotta, Giambattista; Massenzio, Francesca; Ortega, Jose; Russo, Debora; Penna, Ilaria; Falchi, ...Federico; Babini, Giorgia; Petralla, Sabrina; Scarpelli, Rita; Roggiolani, Elena; Fricker, Gert; Rosini, Michela; Cavalli, Andrea; Monti, Barbara; Minarini, Anna; Basagni, Filippo | 2025-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Exploration of the neuromodulatory properties of fyn and gsk-3β kinases exploiting 7-azaindole-based inhibitors_compressed.pdf; Supporting Information.pdf |
| IN SEARCH OF SMALL MOLECULES TARGETING RAD52 FOR SYNTHETIC LETHALITY | Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Va...rignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli, Rita; Girotto, Stefania; Cavalli, Andrea | 2025-01-01 | - | - | 4.03 Poster | - |
| Investigating synthetic lethality and PARP inhibitor resistance in pancreatic cancer through enantiomer differential activity | Masi, Mirco; Poppi, Laura; Previtali, Viola; Nelson, Shannon R; Wynne, Kieran; Varignani, Giulia;... Falchi, Federico; Veronesi, Marina; Albanesi, Ennio; Tedesco, Daniele; De Franco, Francesca; Ciamarone, Andrea; Myers, Samuel H; Ortega, Jose Antonio; Bagnolini, Greta; Ferrandi, Giovanni; Farabegoli, Fulvia; Tirelli, Nicola; Di Stefano, Giuseppina; Oliviero, Giorgio; Walsh, Naomi; Roberti, Marinella; Girotto, Stefania; Cavalli, Andrea | 2025-01-01 | CELL DEATH DISCOVERY | - | 1.01 Articolo in rivista | Masi_et_al-2025-Cell_Death_Discovery.pdf; 41420_2025_2382_MOESM3_ESM.xlsx; 41420_2025_2382_MOESM2_ESM.pdf; 41420_2025_2382_MOESM1_ESM.docx |
| IsoBayes: a Bayesian approach for single-isoform proteomics inference | Bollon, Jordy; R Shortreed, Michael; Jeffery, Erin; T Jordan, Ben; Miller, Rachel; Cavalli, Andre...a; M Smith, Lloyd; N Dewey, Colin; M Sheynkman, Gloria; Tiberi, Simone | 2025-01-01 | BIOINFORMATICS | - | 1.01 Articolo in rivista | btaf450.pdf |
| Probing the BRC repeats RAD51 interaction by integrating computational and experimental biophysics | Rinaldi, F.; Bresciani, V.; Franco, P.; Veronesi, M.; Bernetti, M.; Masetti, M.; Langer, J.; Cava...lli, A.; Girotto, S. | 2025-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
| Rational optimization of D3R/GSK-3β dual target-directed ligands as potential treatment for bipolar disorder: Design, synthesis, X-ray crystallography, molecular dynamics simulations, in vitro ADME, and in vivo pharmacokinetic studies | Di Martino, R. M. C.; Russo, D.; Penna, I.; Demuro, S.; Dalle Vedove, A.; Spagnuolo, R.; Ottonell...o, G.; Bertozzi, S. M.; Summa, M.; Desantis, J.; Valeri, A.; Pruccoli, L.; Tripathi, S. K.; Tarozzi, A.; Storici, P.; Girotto, S.; Bertorelli, R.; Armirotti, A.; Cruciani, G.; Bandiera, T.; Cavalli, A.; Bottegoni, G. | 2025-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | h_11585_1026573.pdf; ScienceDirect_files_05Nov2025_12-04-15.802.zip |
| TARGETING RAD52 FOR SYNTHETIC LETHALITY: DISCOVERY OF A NOVEL SMALL MOLECULE AS A PROMISING INHIBITOR FOR CANCER THERAPY | Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Va...rignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli Stefania Girotto, Rita; Cavalli, Andrea | 2025-01-01 | - | - | 4.03 Poster | - |
| The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study | Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A. | 2025-01-01 | - | - | 4.03 Poster | - |
| The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study | Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A. | 2025-01-01 | - | - | 4.03 Poster | - |