CAVALLI, ANDREA
CAVALLI, ANDREA
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di Ia fascia
Cavalli, ANDREA
An integrative structural study of RAD52, an emerging target in anticancer drug discovery
2025 Rinaldi, F.; Balboni, B.; Girotto, S.; Cavalli, A.
Dissecting the RAD51-BRC4 Interaction Landscape through Integrative Molecular Simulations and Experimental Biophysics
2025 Bresciani, V.; Rinaldi, F.; Franco, P.; Girotto, S.; Cavalli, A.; Langer, J. D.; Masetti, M.; Bernetti, M.
Elucidating RAD52 architecture through an integrated structural biology approach
2025 Rinaldi, F.; Balboni, B.; Marotta, R.; Girotto, S.; Cavalli, A.
Elucidating the BRCA2-RAD51 interaction through an integrated biophysical and structural biology approach
2025 Rinaldi, F.; Bresciani, V.; Franco, P.; Bernetti, M.; Langer, J.; Cavalli, A.; Girotto, S.
Exploration of the Neuromodulatory Properties of Fyn and GSK-3β Kinases Exploiting 7-Azaindole-Based Inhibitors
2025 Marotta, Giambattista; Massenzio, Francesca; Ortega, Jose; Russo, Debora; Penna, Ilaria; Falchi, Federico; Babini, Giorgia; Petralla, Sabrina; Scarpelli, Rita; Roggiolani, Elena; Fricker, Gert; Rosini, Michela; Cavalli, Andrea; Monti, Barbara; Minarini, Anna; Basagni, Filippo
IN SEARCH OF SMALL MOLECULES TARGETING RAD52 FOR SYNTHETIC LETHALITY
2025 Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Varignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli, Rita; Girotto, Stefania; Cavalli, Andrea
Investigating synthetic lethality and PARP inhibitor resistance in pancreatic cancer through enantiomer differential activity
2025 Masi, Mirco; Poppi, Laura; Previtali, Viola; Nelson, Shannon R; Wynne, Kieran; Varignani, Giulia; Falchi, Federico; Veronesi, Marina; Albanesi, Ennio; Tedesco, Daniele; De Franco, Francesca; Ciamarone, Andrea; Myers, Samuel H; Ortega, Jose Antonio; Bagnolini, Greta; Ferrandi, Giovanni; Farabegoli, Fulvia; Tirelli, Nicola; Di Stefano, Giuseppina; Oliviero, Giorgio; Walsh, Naomi; Roberti, Marinella; Girotto, Stefania; Cavalli, Andrea
IsoBayes: a Bayesian approach for single-isoform proteomics inference
2025 Bollon, Jordy; R Shortreed, Michael; Jeffery, Erin; T Jordan, Ben; Miller, Rachel; Cavalli, Andrea; M Smith, Lloyd; N Dewey, Colin; M Sheynkman, Gloria; Tiberi, Simone
Probing the BRC repeats RAD51 interaction by integrating computational and experimental biophysics
2025 Rinaldi, F.; Bresciani, V.; Franco, P.; Veronesi, M.; Bernetti, M.; Masetti, M.; Langer, J.; Cavalli, A.; Girotto, S.
Rational optimization of D3R/GSK-3β dual target-directed ligands as potential treatment for bipolar disorder: Design, synthesis, X-ray crystallography, molecular dynamics simulations, in vitro ADME, and in vivo pharmacokinetic studies
2025 Di Martino, R. M. C.; Russo, D.; Penna, I.; Demuro, S.; Dalle Vedove, A.; Spagnuolo, R.; Ottonello, G.; Bertozzi, S. M.; Summa, M.; Desantis, J.; Valeri, A.; Pruccoli, L.; Tripathi, S. K.; Tarozzi, A.; Storici, P.; Girotto, S.; Bertorelli, R.; Armirotti, A.; Cruciani, G.; Bandiera, T.; Cavalli, A.; Bottegoni, G.
TARGETING RAD52 FOR SYNTHETIC LETHALITY: DISCOVERY OF A NOVEL SMALL MOLECULE AS A PROMISING INHIBITOR FOR CANCER THERAPY
2025 Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Varignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli Stefania Girotto, Rita; Cavalli, Andrea
The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study
2025 Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A.
The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study
2025 Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A.
A journey through targeting BRCA2-RAD51 protein-protein interaction to establish synthetic lethality as paradigm for anticancer drug discovery
2024 Bagnolini G., Poppi L., Previtali V., Ferrandi G., Rinaldi F., Girotto S., Hirsch A.K.H., Roberti M., Cavalli A.
AMCG: a graph dual atomic-molecular conditional molecular generator
2024 Abate, Carlo; Decherchi, Sergio; Cavalli, Andrea
An integrative structural study of the human full-length RAD52 at 2.2 Å resolution
2024 Balboni, Beatrice; Marotta, Roberto; Rinaldi, Francesco; Milordini, Giulia; Varignani, Giulia; Girotto, Stefania; Cavalli, Andrea
Bidirectional path-based non-equilibrium simulations for binding free energy
2024 Ghidini, Alessia; Serra, Eleonora; Decherchi, Sergio; Cavalli, Andrea
Design and synthesis of RAD51-BRCA2 disruptors to inhibit homologous recombination and achieve synthetic lethality in pancreatic cancer cells
2024 Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Previtali, Viola; Roberti, Marinella; Cavalli, Andrea
Design and synthesis of RAD51-BRCA2 protein-protein interaction disruptors to trigger synthetic lethality with Olaparib in pancreatic cancer cells
2024 Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Falchi, Federico; Previtali, Viola; Girotto, Stefania; Roberti, Marinella; Cavalli, Andrea
Differential enantiomers activity of ARN24089 to achieve synthetic lethality in pancreatic cancer
2024 Previtali, Viola; Masi, Mirco; Poppi, Laura; Varignani, Giulia; Falchi, Federico; Tedesco, Daniele; Wynne, Kieran; Oliviero, Giorgio; Bagnolini, Greta; Farabegoli, Fulvia; DI STEFANO, Giuseppina; Girotto, Stefania; Roberti, Marinella; Cavalli, Andrea
| Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
|---|---|---|---|---|---|---|
| An integrative structural study of RAD52, an emerging target in anticancer drug discovery | Rinaldi, F.; Balboni, B.; Girotto, S.; Cavalli, A. | 2025-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Dissecting the RAD51-BRC4 Interaction Landscape through Integrative Molecular Simulations and Experimental Biophysics | Bresciani, V.; Rinaldi, F.; Franco, P.; Girotto, S.; Cavalli, A.; Langer, J. D.; Masetti, M.; Ber...netti, M. | 2025-01-01 | JOURNAL OF CHEMICAL INFORMATION AND MODELING | - | 1.01 Articolo in rivista | - |
| Elucidating RAD52 architecture through an integrated structural biology approach | Rinaldi, F.; Balboni, B.; Marotta, R.; Girotto, S.; Cavalli, A. | 2025-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Elucidating the BRCA2-RAD51 interaction through an integrated biophysical and structural biology approach | Rinaldi, F.; Bresciani, V.; Franco, P.; Bernetti, M.; Langer, J.; Cavalli, A.; Girotto, S. | 2025-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Exploration of the Neuromodulatory Properties of Fyn and GSK-3β Kinases Exploiting 7-Azaindole-Based Inhibitors | Marotta, Giambattista; Massenzio, Francesca; Ortega, Jose; Russo, Debora; Penna, Ilaria; Falchi, ...Federico; Babini, Giorgia; Petralla, Sabrina; Scarpelli, Rita; Roggiolani, Elena; Fricker, Gert; Rosini, Michela; Cavalli, Andrea; Monti, Barbara; Minarini, Anna; Basagni, Filippo | 2025-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Exploration of the neuromodulatory properties of fyn and gsk-3β kinases exploiting 7-azaindole-based inhibitors_compressed.pdf; Supporting Information.pdf |
| IN SEARCH OF SMALL MOLECULES TARGETING RAD52 FOR SYNTHETIC LETHALITY | Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Va...rignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli, Rita; Girotto, Stefania; Cavalli, Andrea | 2025-01-01 | - | - | 4.03 Poster | - |
| Investigating synthetic lethality and PARP inhibitor resistance in pancreatic cancer through enantiomer differential activity | Masi, Mirco; Poppi, Laura; Previtali, Viola; Nelson, Shannon R; Wynne, Kieran; Varignani, Giulia;... Falchi, Federico; Veronesi, Marina; Albanesi, Ennio; Tedesco, Daniele; De Franco, Francesca; Ciamarone, Andrea; Myers, Samuel H; Ortega, Jose Antonio; Bagnolini, Greta; Ferrandi, Giovanni; Farabegoli, Fulvia; Tirelli, Nicola; Di Stefano, Giuseppina; Oliviero, Giorgio; Walsh, Naomi; Roberti, Marinella; Girotto, Stefania; Cavalli, Andrea | 2025-01-01 | CELL DEATH DISCOVERY | - | 1.01 Articolo in rivista | Masi_et_al-2025-Cell_Death_Discovery.pdf; 41420_2025_2382_MOESM3_ESM.xlsx; 41420_2025_2382_MOESM2_ESM.pdf; 41420_2025_2382_MOESM1_ESM.docx |
| IsoBayes: a Bayesian approach for single-isoform proteomics inference | Bollon, Jordy; R Shortreed, Michael; Jeffery, Erin; T Jordan, Ben; Miller, Rachel; Cavalli, Andre...a; M Smith, Lloyd; N Dewey, Colin; M Sheynkman, Gloria; Tiberi, Simone | 2025-01-01 | BIOINFORMATICS | - | 1.01 Articolo in rivista | btaf450.pdf |
| Probing the BRC repeats RAD51 interaction by integrating computational and experimental biophysics | Rinaldi, F.; Bresciani, V.; Franco, P.; Veronesi, M.; Bernetti, M.; Masetti, M.; Langer, J.; Cava...lli, A.; Girotto, S. | 2025-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
| Rational optimization of D3R/GSK-3β dual target-directed ligands as potential treatment for bipolar disorder: Design, synthesis, X-ray crystallography, molecular dynamics simulations, in vitro ADME, and in vivo pharmacokinetic studies | Di Martino, R. M. C.; Russo, D.; Penna, I.; Demuro, S.; Dalle Vedove, A.; Spagnuolo, R.; Ottonell...o, G.; Bertozzi, S. M.; Summa, M.; Desantis, J.; Valeri, A.; Pruccoli, L.; Tripathi, S. K.; Tarozzi, A.; Storici, P.; Girotto, S.; Bertorelli, R.; Armirotti, A.; Cruciani, G.; Bandiera, T.; Cavalli, A.; Bottegoni, G. | 2025-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | h_11585_1026573.pdf; ScienceDirect_files_05Nov2025_12-04-15.802.zip |
| TARGETING RAD52 FOR SYNTHETIC LETHALITY: DISCOVERY OF A NOVEL SMALL MOLECULE AS A PROMISING INHIBITOR FOR CANCER THERAPY | Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Va...rignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli Stefania Girotto, Rita; Cavalli, Andrea | 2025-01-01 | - | - | 4.03 Poster | - |
| The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study | Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A. | 2025-01-01 | - | - | 4.03 Poster | - |
| The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study | Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A. | 2025-01-01 | - | - | 4.03 Poster | - |
| A journey through targeting BRCA2-RAD51 protein-protein interaction to establish synthetic lethality as paradigm for anticancer drug discovery | Bagnolini G., Poppi L., Previtali V., Ferrandi G., Rinaldi F., Girotto S., Hirsch A.K.H., Roberti... M., Cavalli A. | 2024-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
| AMCG: a graph dual atomic-molecular conditional molecular generator | Abate, Carlo; Decherchi, Sergio; Cavalli, Andrea | 2024-01-01 | MACHINE LEARNING: SCIENCE AND TECHNOLOGY | - | 1.01 Articolo in rivista | - |
| An integrative structural study of the human full-length RAD52 at 2.2 Å resolution | Balboni, Beatrice; Marotta, Roberto; Rinaldi, Francesco; Milordini, Giulia; Varignani, Giulia; Gi...rotto, Stefania; Cavalli, Andrea | 2024-01-01 | COMMUNICATIONS BIOLOGY | - | 1.01 Articolo in rivista | s42003-024-06644-1.pdf |
| Bidirectional path-based non-equilibrium simulations for binding free energy | Ghidini, Alessia; Serra, Eleonora; Decherchi, Sergio; Cavalli, Andrea | 2024-01-01 | MOLECULAR PHYSICS | - | 1.01 Articolo in rivista | - |
| Design and synthesis of RAD51-BRCA2 disruptors to inhibit homologous recombination and achieve synthetic lethality in pancreatic cancer cells | Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Previtali, Viola; Roberti, Marinella; Cavalli..., Andrea | 2024-01-01 | - | - | 4.03 Poster | - |
| Design and synthesis of RAD51-BRCA2 protein-protein interaction disruptors to trigger synthetic lethality with Olaparib in pancreatic cancer cells | Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Falchi, Federico; Previtali, Viola; Girotto, ...Stefania; Roberti, Marinella; Cavalli, Andrea | 2024-01-01 | - | - | 4.03 Poster | - |
| Differential enantiomers activity of ARN24089 to achieve synthetic lethality in pancreatic cancer | Previtali, Viola; Masi, Mirco; Poppi, Laura; Varignani, Giulia; Falchi, Federico; Tedesco, Daniel...e; Wynne, Kieran; Oliviero, Giorgio; Bagnolini, Greta; Farabegoli, Fulvia; DI STEFANO, Giuseppina; Girotto, Stefania; Roberti, Marinella; Cavalli, Andrea | 2024-01-01 | - | - | 4.03 Poster | - |