CAVALLI, ANDREA
CAVALLI, ANDREA
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di Ia fascia
Cavalli, ANDREA
The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study
2025 Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A.
The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study
2025 Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A.
A journey through targeting BRCA2-RAD51 protein-protein interaction to establish synthetic lethality as paradigm for anticancer drug discovery
2024 Bagnolini G., Poppi L., Previtali V., Ferrandi G., Rinaldi F., Girotto S., Hirsch A.K.H., Roberti M., Cavalli A.
AMCG: a graph dual atomic-molecular conditional molecular generator
2024 Abate, Carlo; Decherchi, Sergio; Cavalli, Andrea
An integrative structural study of the human full-length RAD52 at 2.2 Å resolution
2024 Balboni, Beatrice; Marotta, Roberto; Rinaldi, Francesco; Milordini, Giulia; Varignani, Giulia; Girotto, Stefania; Cavalli, Andrea
Bidirectional path-based non-equilibrium simulations for binding free energy
2024 Ghidini, Alessia; Serra, Eleonora; Decherchi, Sergio; Cavalli, Andrea
Design and synthesis of RAD51-BRCA2 disruptors to inhibit homologous recombination and achieve synthetic lethality in pancreatic cancer cells
2024 Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Previtali, Viola; Roberti, Marinella; Cavalli, Andrea
Design and synthesis of RAD51-BRCA2 protein-protein interaction disruptors to trigger synthetic lethality with Olaparib in pancreatic cancer cells
2024 Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Falchi, Federico; Previtali, Viola; Girotto, Stefania; Roberti, Marinella; Cavalli, Andrea
Faster ISNet for Background Bias Mitigation on Deep Neural Networks
2024 Bassi, Pedro R. A. S.; Decherchi, Sergio; Cavalli, Andrea
Improving deep neural network generalization and robustness to background bias via layer-wise relevance propagation optimization
2024 Bassi P.R.A.S.; Dertkigil S.S.J.; Cavalli A.
Machine learning for precision diagnostics of autoimmunity
2024 Kruta, J.; Carapito, R.; Trendelenburg, M.; Martin, T.; Rizzi, M.; Voll, R. E.; Cavalli, A.; Natali, E.; Meier, P.; Stawiski, M.; Mosbacher, J.; Mollet, A.; Santoro, A.; Capri, M.; Giampieri, E.; Schkommodau, E.; Miho, E.
New Horizons of Synthetic Lethality in Cancer: Current Development and Future Perspectives
2024 Previtali, Viola; Bagnolini, Greta; Ciamarone, Andrea; Ferrandi, Giovanni; Rinaldi, Francesco; Myers, Samuel Harry; Roberti, Marinella; Cavalli, Andrea
OBIWAN: An Element-Wise Scalable Feed-Forward Neural Network Potential
2024 Martire, Stefano; Decherchi, Sergio; Cavalli, Andrea
A RAD51/BRCA2 small molecule inhibitor enhances the antineoplastic effect of the PARPi talazoparib in pancreatic cancer
2023 Laura Poppi, Samuel H Myers, Viola Previtali, Francesco Rinaldi, Fulvia Farabegoli, Giuseppina Di Stefano, Naomi Walsh, Marinella Roberti, Andrea Cavalli
An 19F NMR fragment-based approach for the discovery and development of BRCA2-RAD51 inhibitors to pursuit synthetic lethality in combination with PARP inhibition in pancreatic cancer
2023 Myers, S. H.; Poppi, L.; Rinaldi, F.; Veronesi, M.; Ciamarone, A.; Previtali, V.; Bagnolini, G.; Schipani, F.; Ortega Martínez, J. A.; Girotto, S.; Di Stefano, G.; Farabegoli, F.; Walsh, N.; De Franco, F.; Roberti, M.; Cavalli, A.
Design and synthesis of RAD51-BRCA disruptors to inhibit homologous recombination and achieve synthetic lethality in cancer cells
2023 Ferrandi, Giovanni; Bagnolini, Greta; Roberti, Marinella; Cavalli, Andrea
Dissecting the BRCA2 - RAD51 interaction by integrating computational and experimental biophysics
2023 Rinaldi F., Bernetti M., Bresciani V., Girotto S., Cavalli A.
Elucidating the BRCA2 - RAD51 interaction by integrating computational and experimental biophysics
2023 Rinaldi F., Bernetti M., Bresciani V., Girotto S., Cavalli A.
Elucidating the BRCA2-RAD51 interaction through an integrated structural biophysics approach
2023 Rinaldi Francesco, Girotto Stefania, Cavalli Andrea
Galantamine-memantine hybrids for Alzheimer's disease: The influence of linker rigidity in biological activity and pharmacokinetic properties
2023 Basagni, Filippo; Ortega, Jose A; Bertozzi, Sine M; Armirotti, Andrea; Summa, Maria; Bertorelli, Rosalia; Bartolini, Manuela; Mellor, Ian R; Bedeschi, Martina; Bottegoni, Giovanni; Lembo, Vittorio; Minarini, Anna; Cavalli, Andrea; Rosini, Michela
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study | Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A. | 2025-01-01 | - | - | 4.03 Poster | - |
The mechanistic understanding of the BRCA2-RAD51 interaction: an integrated structural biophysics study | Rinaldi, F.; Bernetti, M.; Bresciani, V.; Veronesi, M.; Masetti, M.; Girotto, S.; Cavalli, A. | 2025-01-01 | - | - | 4.03 Poster | - |
A journey through targeting BRCA2-RAD51 protein-protein interaction to establish synthetic lethality as paradigm for anticancer drug discovery | Bagnolini G., Poppi L., Previtali V., Ferrandi G., Rinaldi F., Girotto S., Hirsch A.K.H., Roberti... M., Cavalli A. | 2024-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
AMCG: a graph dual atomic-molecular conditional molecular generator | Abate, Carlo; Decherchi, Sergio; Cavalli, Andrea | 2024-01-01 | MACHINE LEARNING: SCIENCE AND TECHNOLOGY | - | 1.01 Articolo in rivista | - |
An integrative structural study of the human full-length RAD52 at 2.2 Å resolution | Balboni, Beatrice; Marotta, Roberto; Rinaldi, Francesco; Milordini, Giulia; Varignani, Giulia; Gi...rotto, Stefania; Cavalli, Andrea | 2024-01-01 | COMMUNICATIONS BIOLOGY | - | 1.01 Articolo in rivista | - |
Bidirectional path-based non-equilibrium simulations for binding free energy | Ghidini, Alessia; Serra, Eleonora; Decherchi, Sergio; Cavalli, Andrea | 2024-01-01 | MOLECULAR PHYSICS | - | 1.01 Articolo in rivista | - |
Design and synthesis of RAD51-BRCA2 disruptors to inhibit homologous recombination and achieve synthetic lethality in pancreatic cancer cells | Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Previtali, Viola; Roberti, Marinella; Cavalli..., Andrea | 2024-01-01 | - | - | 4.03 Poster | - |
Design and synthesis of RAD51-BRCA2 protein-protein interaction disruptors to trigger synthetic lethality with Olaparib in pancreatic cancer cells | Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Falchi, Federico; Previtali, Viola; Girotto, ...Stefania; Roberti, Marinella; Cavalli, Andrea | 2024-01-01 | - | - | 4.03 Poster | - |
Faster ISNet for Background Bias Mitigation on Deep Neural Networks | Bassi, Pedro R. A. S.; Decherchi, Sergio; Cavalli, Andrea | 2024-01-01 | IEEE ACCESS | - | 1.01 Articolo in rivista | - |
Improving deep neural network generalization and robustness to background bias via layer-wise relevance propagation optimization | Bassi P.R.A.S.; Dertkigil S.S.J.; Cavalli A. | 2024-01-01 | NATURE COMMUNICATIONS | - | 1.01 Articolo in rivista | Nat_Commun.pdf |
Machine learning for precision diagnostics of autoimmunity | Kruta, J.; Carapito, R.; Trendelenburg, M.; Martin, T.; Rizzi, M.; Voll, R. E.; Cavalli, A.; Nata...li, E.; Meier, P.; Stawiski, M.; Mosbacher, J.; Mollet, A.; Santoro, A.; Capri, M.; Giampieri, E.; Schkommodau, E.; Miho, E. | 2024-01-01 | SCIENTIFIC REPORTS | - | 1.01 Articolo in rivista | Kruta et al_2024_Scient_rep_Machine_Learning.pdf; 41598_2024_76093_MOESM1_ESM.pdf |
New Horizons of Synthetic Lethality in Cancer: Current Development and Future Perspectives | Previtali, Viola; Bagnolini, Greta; Ciamarone, Andrea; Ferrandi, Giovanni; Rinaldi, Francesco; My...ers, Samuel Harry; Roberti, Marinella; Cavalli, Andrea | 2024-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
OBIWAN: An Element-Wise Scalable Feed-Forward Neural Network Potential | Martire, Stefano; Decherchi, Sergio; Cavalli, Andrea | 2024-01-01 | JOURNAL OF CHEMICAL THEORY AND COMPUTATION | - | 1.01 Articolo in rivista | - |
A RAD51/BRCA2 small molecule inhibitor enhances the antineoplastic effect of the PARPi talazoparib in pancreatic cancer | Laura Poppi, Samuel H Myers, Viola Previtali, Francesco Rinaldi, Fulvia Farabegoli, Giuseppina Di... Stefano, Naomi Walsh, Marinella Roberti, Andrea Cavalli | 2023-01-01 | - | FEBS PRESS | 4.03 Poster | - |
An 19F NMR fragment-based approach for the discovery and development of BRCA2-RAD51 inhibitors to pursuit synthetic lethality in combination with PARP inhibition in pancreatic cancer | Myers, S. H.; Poppi, L.; Rinaldi, F.; Veronesi, M.; Ciamarone, A.; Previtali, V.; Bagnolini, G.; ...Schipani, F.; Ortega Martínez, J. A.; Girotto, S.; Di Stefano, G.; Farabegoli, F.; Walsh, N.; De Franco, F.; Roberti, M.; Cavalli, A. | 2023-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | 1-s2.0-S0223523423010814-mmc1.docx; 1-s2.0-S0223523423010814-main.pdf |
Design and synthesis of RAD51-BRCA disruptors to inhibit homologous recombination and achieve synthetic lethality in cancer cells | Ferrandi, Giovanni; Bagnolini, Greta; Roberti, Marinella; Cavalli, Andrea | 2023-01-01 | - | - | 4.03 Poster | - |
Dissecting the BRCA2 - RAD51 interaction by integrating computational and experimental biophysics | Rinaldi F., Bernetti M., Bresciani V., Girotto S., Cavalli A. | 2023-01-01 | - | - | 4.03 Poster | - |
Elucidating the BRCA2 - RAD51 interaction by integrating computational and experimental biophysics | Rinaldi F., Bernetti M., Bresciani V., Girotto S., Cavalli A. | 2023-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
Elucidating the BRCA2-RAD51 interaction through an integrated structural biophysics approach | Rinaldi Francesco, Girotto Stefania, Cavalli Andrea | 2023-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
Galantamine-memantine hybrids for Alzheimer's disease: The influence of linker rigidity in biological activity and pharmacokinetic properties | Basagni, Filippo; Ortega, Jose A; Bertozzi, Sine M; Armirotti, Andrea; Summa, Maria; Bertorelli, ...Rosalia; Bartolini, Manuela; Mellor, Ian R; Bedeschi, Martina; Bottegoni, Giovanni; Lembo, Vittorio; Minarini, Anna; Cavalli, Andrea; Rosini, Michela | 2023-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Eur. J. Med.Chem. 2023.pdf; 1-s2.0-S0223523423007705-mmc1.docx |