FALCHI, FEDERICO

FALCHI, FEDERICO  

DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE  

Ricercatori a tempo determinato  

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Risultati 1 - 20 di 45 (tempo di esecuzione: 0.061 secondi).
Titolo Autore(i) Anno Periodico Editore Tipo File
Probing allosteric communication with combined molecular dynamics simulations and network analysis Bernetti, Mattia; Bosio, Stefano; Bresciani, Veronica; Falchi, Federico; Masetti, Matteo 2024-01-01 CURRENT OPINION IN STRUCTURAL BIOLOGY - 1.01 Articolo in rivista -
Innovative Strategy toward Mutant CFTR Rescue in Cystic Fibrosis: Design and Synthesis of Thiadiazole Inhibitors of the E3 Ligase RNF5 Brusa, Irene; Sondo, Elvira; Pesce, Emanuela; Tomati, Valeria; Gioia, Dario; Falchi, Federico; Ba...lboni, Beatrice; Ortega Martínez, Jose Antonio; Veronesi, Marina; Romeo, Elisa; Margaroli, Natasha; Recanatini, Maurizio; Girotto, Stefania; Pedemonte, Nicoletta; Roberti, Marinella; Cavalli, Andrea 2023-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista brusa-et-al-2023-innovative-strategy-toward-mutant-cftr-rescue-in-cystic-fibrosis-design-and-synthesis-of-thiadiazole.pdf
Proteostasis Regulators in Cystic Fibrosis: Current Development and Future Perspectives Brusa I.; Sondo E.; Falchi F.; Pedemonte N.; Roberti M.; Cavalli A. 2022-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista acs.jmedchem.1c01897.pdf
Divide et impera: An in silico screening targeting hcmv ppul44 processivity factor homodimerization identifies small molecules inhibiting viral replication Ghassabian H.; Falchi F.; Timmoneri M.; Mercorelli B.; Loregian A.; Palu G.; Alvisi G. 2021-01-01 VIRUSES - 1.01 Articolo in rivista Divide et impera_ An In Silico Screening Targeting HCMV ppUL44 Processivity Factor Homodimerization Identifies Small Molecules Inhibiting Viral Replication.pdf
Searching for New Microbiome-Targeted Therapeutics through a Drug Repurposing Approach Barone M.; Rampelli S.; Biagi E.; Bertozzi S.M.; Falchi F.; Cavalli A.; Armirotti A.; Brigidi P.;... Turroni S.; Candela M. 2021-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista acs.jmedchem.1c01333.pdf
Synthetic Lethality in Pancreatic Cancer: Discovery of a New RAD51-BRCA2 Small Molecule Disruptor That Inhibits Homologous Recombination and Synergizes with Olaparib Bagnolini G.; Milano D.; Manerba M.; Schipani F.; Ortega J.A.; Gioia D.; Falchi F.; Balboni A.; F...arabegoli F.; De Franco F.; Robertson J.; Pellicciari R.; Pallavicini I.; Peri S.; Minucci S.; Girotto S.; Di Stefano G.; Roberti M.; Cavalli A. 2020-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista ASAP_acs.jmedchem.9b01526.pdf
Targeting the Protein Tunnels of the Urease Accessory Complex: A Theoretical Investigation Masetti, Matteo; Falchi, Federico; Gioia, Dario; Recanatini, Maurizio; Ciurli, Stefano; Musiani, ...Francesco 2020-01-01 MOLECULES - 1.01 Articolo in rivista 63_2020_Masetti_Molecules.pdf
Rad51/Brca2 Disruptors Inhibit Homologous Recombination and Synergize with Olaparib in Pancreatic Cancer Cells Marinella Roberti, Fabrizio Schipani, Greta Bagnolini, Domenico Milano, Elisa Giacomini, Federico... Falchi, Andrea Balboni, Marcella Manerba, Fulvia Farabegoli, Francesca De Franco, Janet Robertson, Saverio Minucci, Isabella Pallavicini, Giuseppina Di Stefano, Stefania Girotto, Roberto Pellicciari, and Andrea Cavalli 2019-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Structure-based virtual screening allows the identification of efficient modulators of E-cadherin-mediated cell-cell adhesion Vedove A.D.; Falchi F.; Donini S.; Dobric A.; Germain S.; Martino G.P.D.; Prosdocimi T.; Vettrain...o C.; Torretta A.; Cavalli A.; Rigot V.; Andre F.; Parisini E. 2019-01-01 INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES - 1.01 Articolo in rivista -
Pharmacological Inhibition of the Ubiquitin Ligase RNF5 Rescues F508del-CFTR in Cystic Fibrosis Airway Epithelia Sondo, Elvira; Falchi, Federico; Caci, Emanuela; Ferrera, Loretta; Giacomini, Elisa; Pesce, Emanu...ela; Tomati, Valeria; Mandrup Bertozzi, Sine; Goldoni, Luca; Armirotti, Andrea; Ravazzolo, Roberto; Cavalli, Andrea; Pedemonte, Nicoletta 2018-01-01 CELL CHEMICAL BIOLOGY - 1.01 Articolo in rivista -
Chalcone-based carbamates for Alzheimer's disease treatment Rampa, Angela; Montanari, Serena; Pruccoli, Letizia; Bartolini, Manuela; Falchi, Federico; Feoli,... Alessandra; Cavalli, Andrea; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra 2017-01-01 FUTURE MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Crassiflorone derivatives that inhibit Trypanosoma brucei glyceraldehyde-3-phosphate dehydrogenase (TbGAPDH) and Trypanosoma cruzi trypanothione reductase (TcTR) and display trypanocidal activity Uliassi, Elisa; Fiorani, Giulia; Krauth-Siegel, R. Luise; Bergamini, Christian; Fato, Romana; Bia...nchini, Giulia; Carlos Menéndez, J.; Molina, Maria Teresa; López-Montero, Eulogio; Falchi, Federico; Cavalli, Andrea; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Witt, Gesa; Moraes, Carolina B.; Freitas-Junior, Lucio H.; Borsari, Chiara; Costi, Maria Paola; Bolognesi, Maria Laura* 2017-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Development of a multisite model for Ni(II) ion in solution from thermodynamic and kinetic data Masetti, Matteo; Musiani, Francesco; Bernetti, Mattia; Falchi, Federico; Cavalli, Andrea; Ciurli,... Stefano; Recanatini, Maurizio 2017-01-01 JOURNAL OF COMPUTATIONAL CHEMISTRY - 1.01 Articolo in rivista -
Discovery of Multitarget Agents Active as Broad-Spectrum Antivirals and Correctors of Cystic Fibrosis Transmembrane Conductance Regulator for Associated Pulmonary Diseases Tassini, Sabrina; Sun, Liang; Lanko, Kristina; Crespan, Emmanuele; Langron, Emily; Falchi, Federi...co; Kissova, Miroslava; Armijos-Rivera, Jorge I.; Delang, Leen; Mirabelli, Carmen; Neyts, Johan; Pieroni, Marco; Cavalli, Andrea; Costantino, Gabriele; Maga, Giovanni; Vergani, Paola; Leyssen, Pieter; Radi, Marco 2017-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Protein Tunnels: The Case of Urease Accessory Proteins Musiani, Francesco; Gioia, Dario; Masetti, Matteo; Falchi, Federico; Cavalli, Andrea; Recanatini,... Maurizio; Ciurli, Stefano 2017-01-01 JOURNAL OF CHEMICAL THEORY AND COMPUTATION - 1.01 Articolo in rivista Musiani_2017_JCTC(1).pdf
Synthetic Lethality Triggered by Combining Olaparib with BRCA2-Rad51 Disruptors Falchi, Federico; Giacomini, Elisa; Masini, Tiziana; Boutard, Nicolas; Di Ianni, Lorenza; Manerba..., Marcella; Farabegoli, Fulvia; Rossini, Lara; Robertson, Janet; Minucci, Saverio; Pallavicini, Isabella; Di Stefano, Giuseppina; Roberti, Marinella; Pellicciari, Roberto; Cavalli, Andrea 2017-01-01 ACS CHEMICAL BIOLOGY - 1.01 Articolo in rivista -
Kernel-Based, Partial Least Squares Quantitative Structure-Retention Relationship Model for UPLC Retention Time Prediction: A Useful Tool for Metabolite Identification Falchi, Federico; Bertozzi, Sine Mandrup; Ottonello, Giuliana; Ruda, Gian Filippo; Colombano, Gia...mpiero; Fiorelli, Claudio; Martucci, Cataldo; Bertorelli, Rosalia; Scarpelli, Rita; Cavalli, Andrea; Bandiera, Tiziano; Armirotti, Andrea 2016-01-01 ANALYTICAL CHEMISTRY - 1.01 Articolo in rivista -
Multitarget Strategy to Address Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and Computational Studies of Coumarin-Based Derivatives Montanari, Serena; Bartolini, Manuela; Neviani, Paolo; Belluti, Federica; Gobbi, Silvia; Pruccoli..., Letizia; Tarozzi, Andrea; Falchi, Federico; Andrisano, Vincenza; Miszta, Przemysław; Cavalli, Andrea; Filipek, Sławomir; Bisi, Alessandra; Rampa, Angela 2016-01-01 CHEMMEDCHEM - 1.01 Articolo in rivista ChemMedChem VQR.pdf
Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A Rupiani, Sebastiano; Guidotti, Laura; Manerba, Marcella; Di Ianni, Lorenza; Giacomini, Elisa; Fal...chi, Federico; Di Stefano, Giuseppina; Roberti, Marinella; Recanatini, Maurizio 2016-01-01 ORGANIC & BIOMOLECULAR CHEMISTRY - 1.01 Articolo in rivista -
2-Phenoxy-1,4-naphthoquinones: From a Multitarget Antitrypanosomal to a Potential Antitumor Profile Prati, Federica; Bergamini, Christian; Molina, Maria Teresa; Falchi, Federico; Cavalli, Andrea; K...aiser, Marcel; Brun, Reto; Fato, Romana; Bolognesi, Maria Laura 2015-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -