FALCHI, FEDERICO
FALCHI, FEDERICO
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di IIa fascia
Design and synthesis of small molecules targeting pre-miRNA21 toward the development of ribonuclease targeting chimeras (RIBOTACs) to regulate the oncogenic miRNA21
2025 Sdei, F.; Bagnolini, G.; Falchi, F.; Sosic, A.; Fabbian, S.; Duca, M.; Bolognesi, M. L.
Exploration of the Neuromodulatory Properties of Fyn and GSK-3β Kinases Exploiting 7-Azaindole-Based Inhibitors
2025 Marotta, Giambattista; Massenzio, Francesca; Ortega, Jose; Russo, Debora; Penna, Ilaria; Falchi, Federico; Babini, Giorgia; Petralla, Sabrina; Scarpelli, Rita; Roggiolani, Elena; Fricker, Gert; Rosini, Michela; Cavalli, Andrea; Monti, Barbara; Minarini, Anna; Basagni, Filippo
IN SEARCH OF SMALL MOLECULES TARGETING RAD52 FOR SYNTHETIC LETHALITY
2025 Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Varignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli, Rita; Girotto, Stefania; Cavalli, Andrea
Investigating synthetic lethality and PARP inhibitor resistance in pancreatic cancer through enantiomer differential activity
2025 Masi, Mirco; Poppi, Laura; Previtali, Viola; Nelson, Shannon R; Wynne, Kieran; Varignani, Giulia; Falchi, Federico; Veronesi, Marina; Albanesi, Ennio; Tedesco, Daniele; De Franco, Francesca; Ciamarone, Andrea; Myers, Samuel H; Ortega, Jose Antonio; Bagnolini, Greta; Ferrandi, Giovanni; Farabegoli, Fulvia; Tirelli, Nicola; Di Stefano, Giuseppina; Oliviero, Giorgio; Walsh, Naomi; Roberti, Marinella; Girotto, Stefania; Cavalli, Andrea
Morphological inhibitors of aggregation-prone amyloid-β conformers: A computational exploration
2025 Bosio, S.; Falchi, F.; Rauzi, C.; Bellucci, L.
Target Identification with Live-Cell Photoaffinity Labeling and Mechanism of Action Elucidation of ARN23765, a Highly Potent CFTR Corrector
2025 Romeo, E.; Saccoliti, F.; Ocello, R.; Andonaia, A.; Allegretta, C.; Pastorino, C.; Pedemonte, N.; Falchi, F.; Laselva, O.; Bandiera, T.; Bertozzi, F.
TARGETING RAD52 FOR SYNTHETIC LETHALITY: DISCOVERY OF A NOVEL SMALL MOLECULE AS A PROMISING INHIBITOR FOR CANCER THERAPY
2025 Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Varignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli Stefania Girotto, Rita; Cavalli, Andrea
Design and synthesis of RAD51-BRCA2 protein-protein interaction disruptors to trigger synthetic lethality with Olaparib in pancreatic cancer cells
2024 Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Falchi, Federico; Previtali, Viola; Girotto, Stefania; Roberti, Marinella; Cavalli, Andrea
DESIGN AND SYNTHESIS OF SMALL MOLECULES TARGETING PRE-MIRNA21 TOWARD THE DEVELOPMENT OF RIBONUCLEASE TARGETING CHIMERAS (RIBOTACS) TO REGULATE THE ONCOGENIC MIRNA21
2024 Sdei, F.; Bagnolini, G.; Falchi, F.; Sosic, A.; Bolognesi, M. L.
Differential enantiomers activity of ARN24089 to achieve synthetic lethality in pancreatic cancer
2024 Previtali, Viola; Masi, Mirco; Poppi, Laura; Varignani, Giulia; Falchi, Federico; Tedesco, Daniele; Wynne, Kieran; Oliviero, Giorgio; Bagnolini, Greta; Farabegoli, Fulvia; DI STEFANO, Giuseppina; Girotto, Stefania; Roberti, Marinella; Cavalli, Andrea
Probing allosteric communication with combined molecular dynamics simulations and network analysis
2024 Bernetti, Mattia; Bosio, Stefano; Bresciani, Veronica; Falchi, Federico; Masetti, Matteo
Structure-based targeting of the lipid A-modifying enzyme PmrC to contrast colistin resistance in Acinetobacter baumannii
2024 Romano, M.; Falchi, F.; De Gregorio, E.; Stabile, M.; Migliaccio, A.; Ruggiero, A.; Napolitano, V.; Autiero, I.; Squeglia, F.; Berisio, R.
Targeting RNA degradation with small molecules: design and synthesis of selective RNA binders and development of ribonuclease targeting chimeras (RIBOTACs)
2024 Sdei, Federico; Bagnolini, Greta; Falchi, Federico; Ghezzo, M.; Sosic, Alice; Sissi, Claudia; Roberti, Marinella; Bolognesi, MARIA LAURA
Innovative Strategy toward Mutant CFTR Rescue in Cystic Fibrosis: Design and Synthesis of Thiadiazole Inhibitors of the E3 Ligase RNF5
2023 Brusa, Irene; Sondo, Elvira; Pesce, Emanuela; Tomati, Valeria; Gioia, Dario; Falchi, Federico; Balboni, Beatrice; Ortega Martínez, Jose Antonio; Veronesi, Marina; Romeo, Elisa; Margaroli, Natasha; Recanatini, Maurizio; Girotto, Stefania; Pedemonte, Nicoletta; Roberti, Marinella; Cavalli, Andrea
Triggering RNA degradation with small molecules: development of RIBOnuclease TArgeting Chimeras (RIBOTACs)
2023 Bagnolini, G.; Falchi, F.; Sdei, F.; Roberti, M.; Sosic, A.; Sissi, C.; Bolognesi, M. L.
Proteostasis Regulators in Cystic Fibrosis: Current Development and Future Perspectives
2022 Brusa I.; Sondo E.; Falchi F.; Pedemonte N.; Roberti M.; Cavalli A.
Divide et impera: An in silico screening targeting hcmv ppul44 processivity factor homodimerization identifies small molecules inhibiting viral replication
2021 Ghassabian H.; Falchi F.; Timmoneri M.; Mercorelli B.; Loregian A.; Palu G.; Alvisi G.
Searching for New Microbiome-Targeted Therapeutics through a Drug Repurposing Approach
2021 Barone M.; Rampelli S.; Biagi E.; Bertozzi S.M.; Falchi F.; Cavalli A.; Armirotti A.; Brigidi P.; Turroni S.; Candela M.
Synthetic Lethality in Pancreatic Cancer: Discovery of a New RAD51-BRCA2 Small Molecule Disruptor That Inhibits Homologous Recombination and Synergizes with Olaparib
2020 Bagnolini G.; Milano D.; Manerba M.; Schipani F.; Ortega J.A.; Gioia D.; Falchi F.; Balboni A.; Farabegoli F.; De Franco F.; Robertson J.; Pellicciari R.; Pallavicini I.; Peri S.; Minucci S.; Girotto S.; Di Stefano G.; Roberti M.; Cavalli A.
Targeting the Protein Tunnels of the Urease Accessory Complex: A Theoretical Investigation
2020 Masetti, Matteo; Falchi, Federico; Gioia, Dario; Recanatini, Maurizio; Ciurli, Stefano; Musiani, Francesco
| Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
|---|---|---|---|---|---|---|
| Design and synthesis of small molecules targeting pre-miRNA21 toward the development of ribonuclease targeting chimeras (RIBOTACs) to regulate the oncogenic miRNA21 | Sdei, F.; Bagnolini, G.; Falchi, F.; Sosic, A.; Fabbian, S.; Duca, M.; Bolognesi, M. L. | 2025-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
| Exploration of the Neuromodulatory Properties of Fyn and GSK-3β Kinases Exploiting 7-Azaindole-Based Inhibitors | Marotta, Giambattista; Massenzio, Francesca; Ortega, Jose; Russo, Debora; Penna, Ilaria; Falchi, ...Federico; Babini, Giorgia; Petralla, Sabrina; Scarpelli, Rita; Roggiolani, Elena; Fricker, Gert; Rosini, Michela; Cavalli, Andrea; Monti, Barbara; Minarini, Anna; Basagni, Filippo | 2025-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Exploration of the neuromodulatory properties of fyn and gsk-3β kinases exploiting 7-azaindole-based inhibitors_compressed.pdf; Supporting Information.pdf |
| IN SEARCH OF SMALL MOLECULES TARGETING RAD52 FOR SYNTHETIC LETHALITY | Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Va...rignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli, Rita; Girotto, Stefania; Cavalli, Andrea | 2025-01-01 | - | - | 4.03 Poster | - |
| Investigating synthetic lethality and PARP inhibitor resistance in pancreatic cancer through enantiomer differential activity | Masi, Mirco; Poppi, Laura; Previtali, Viola; Nelson, Shannon R; Wynne, Kieran; Varignani, Giulia;... Falchi, Federico; Veronesi, Marina; Albanesi, Ennio; Tedesco, Daniele; De Franco, Francesca; Ciamarone, Andrea; Myers, Samuel H; Ortega, Jose Antonio; Bagnolini, Greta; Ferrandi, Giovanni; Farabegoli, Fulvia; Tirelli, Nicola; Di Stefano, Giuseppina; Oliviero, Giorgio; Walsh, Naomi; Roberti, Marinella; Girotto, Stefania; Cavalli, Andrea | 2025-01-01 | CELL DEATH DISCOVERY | - | 1.01 Articolo in rivista | Masi_et_al-2025-Cell_Death_Discovery.pdf; 41420_2025_2382_MOESM3_ESM.xlsx; 41420_2025_2382_MOESM2_ESM.pdf; 41420_2025_2382_MOESM1_ESM.docx |
| Morphological inhibitors of aggregation-prone amyloid-β conformers: A computational exploration | Bosio, S.; Falchi, F.; Rauzi, C.; Bellucci, L. | 2025-01-01 | COMPUTERS IN BIOLOGY AND MEDICINE | - | 1.01 Articolo in rivista | - |
| Target Identification with Live-Cell Photoaffinity Labeling and Mechanism of Action Elucidation of ARN23765, a Highly Potent CFTR Corrector | Romeo, E.; Saccoliti, F.; Ocello, R.; Andonaia, A.; Allegretta, C.; Pastorino, C.; Pedemonte, N.;... Falchi, F.; Laselva, O.; Bandiera, T.; Bertozzi, F. | 2025-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
| TARGETING RAD52 FOR SYNTHETIC LETHALITY: DISCOVERY OF A NOVEL SMALL MOLECULE AS A PROMISING INHIBITOR FOR CANCER THERAPY | Quatraccioni, Martina; Ocello, Riccardo; Falchi, Federico; Previtali, Viola; Veronesi, Marina; Va...rignani, Giulia; Margaroli, Natasha; Andonaia, Angela; Masi, Mirco; Scarpelli Stefania Girotto, Rita; Cavalli, Andrea | 2025-01-01 | - | - | 4.03 Poster | - |
| Design and synthesis of RAD51-BRCA2 protein-protein interaction disruptors to trigger synthetic lethality with Olaparib in pancreatic cancer cells | Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Falchi, Federico; Previtali, Viola; Girotto, ...Stefania; Roberti, Marinella; Cavalli, Andrea | 2024-01-01 | - | - | 4.03 Poster | - |
| DESIGN AND SYNTHESIS OF SMALL MOLECULES TARGETING PRE-MIRNA21 TOWARD THE DEVELOPMENT OF RIBONUCLEASE TARGETING CHIMERAS (RIBOTACS) TO REGULATE THE ONCOGENIC MIRNA21 | Sdei, F.; Bagnolini, G.; Falchi, F.; Sosic, A.; Bolognesi, M. L. | 2024-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
| Differential enantiomers activity of ARN24089 to achieve synthetic lethality in pancreatic cancer | Previtali, Viola; Masi, Mirco; Poppi, Laura; Varignani, Giulia; Falchi, Federico; Tedesco, Daniel...e; Wynne, Kieran; Oliviero, Giorgio; Bagnolini, Greta; Farabegoli, Fulvia; DI STEFANO, Giuseppina; Girotto, Stefania; Roberti, Marinella; Cavalli, Andrea | 2024-01-01 | - | - | 4.03 Poster | - |
| Probing allosteric communication with combined molecular dynamics simulations and network analysis | Bernetti, Mattia; Bosio, Stefano; Bresciani, Veronica; Falchi, Federico; Masetti, Matteo | 2024-01-01 | CURRENT OPINION IN STRUCTURAL BIOLOGY | - | 1.01 Articolo in rivista | 2024_Bernetti_OPEN_ACCESS.pdf |
| Structure-based targeting of the lipid A-modifying enzyme PmrC to contrast colistin resistance in Acinetobacter baumannii | Romano, M.; Falchi, F.; De Gregorio, E.; Stabile, M.; Migliaccio, A.; Ruggiero, A.; Napolitano, V....; Autiero, I.; Squeglia, F.; Berisio, R. | 2024-01-01 | FRONTIERS IN MICROBIOLOGY | - | 1.01 Articolo in rivista | fmicb-1-1501051.pdf |
| Targeting RNA degradation with small molecules: design and synthesis of selective RNA binders and development of ribonuclease targeting chimeras (RIBOTACs) | Sdei, Federico; Bagnolini, Greta; Falchi, Federico; Ghezzo, M.; Sosic, Alice; Sissi, Claudia; Rob...erti, Marinella; Bolognesi, MARIA LAURA | 2024-01-01 | - | - | 4.03 Poster | - |
| Innovative Strategy toward Mutant CFTR Rescue in Cystic Fibrosis: Design and Synthesis of Thiadiazole Inhibitors of the E3 Ligase RNF5 | Brusa, Irene; Sondo, Elvira; Pesce, Emanuela; Tomati, Valeria; Gioia, Dario; Falchi, Federico; Ba...lboni, Beatrice; Ortega Martínez, Jose Antonio; Veronesi, Marina; Romeo, Elisa; Margaroli, Natasha; Recanatini, Maurizio; Girotto, Stefania; Pedemonte, Nicoletta; Roberti, Marinella; Cavalli, Andrea | 2023-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | brusa-et-al-2023-innovative-strategy-toward-mutant-cftr-rescue-in-cystic-fibrosis-design-and-synthesis-of-thiadiazole.pdf |
| Triggering RNA degradation with small molecules: development of RIBOnuclease TArgeting Chimeras (RIBOTACs) | Bagnolini, G.; Falchi, F.; Sdei, F.; Roberti, M.; Sosic, A.; Sissi, C.; Bolognesi, M. L. | 2023-01-01 | - | - | 4.03 Poster | - |
| Proteostasis Regulators in Cystic Fibrosis: Current Development and Future Perspectives | Brusa I.; Sondo E.; Falchi F.; Pedemonte N.; Roberti M.; Cavalli A. | 2022-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | acs.jmedchem.1c01897.pdf |
| Divide et impera: An in silico screening targeting hcmv ppul44 processivity factor homodimerization identifies small molecules inhibiting viral replication | Ghassabian H.; Falchi F.; Timmoneri M.; Mercorelli B.; Loregian A.; Palu G.; Alvisi G. | 2021-01-01 | VIRUSES | - | 1.01 Articolo in rivista | Divide et impera_ An In Silico Screening Targeting HCMV ppUL44 Processivity Factor Homodimerization Identifies Small Molecules Inhibiting Viral Replication.pdf |
| Searching for New Microbiome-Targeted Therapeutics through a Drug Repurposing Approach | Barone M.; Rampelli S.; Biagi E.; Bertozzi S.M.; Falchi F.; Cavalli A.; Armirotti A.; Brigidi P.;... Turroni S.; Candela M. | 2021-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | acs.jmedchem.1c01333.pdf |
| Synthetic Lethality in Pancreatic Cancer: Discovery of a New RAD51-BRCA2 Small Molecule Disruptor That Inhibits Homologous Recombination and Synergizes with Olaparib | Bagnolini G.; Milano D.; Manerba M.; Schipani F.; Ortega J.A.; Gioia D.; Falchi F.; Balboni A.; F...arabegoli F.; De Franco F.; Robertson J.; Pellicciari R.; Pallavicini I.; Peri S.; Minucci S.; Girotto S.; Di Stefano G.; Roberti M.; Cavalli A. | 2020-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | ASAP_acs.jmedchem.9b01526.pdf |
| Targeting the Protein Tunnels of the Urease Accessory Complex: A Theoretical Investigation | Masetti, Matteo; Falchi, Federico; Gioia, Dario; Recanatini, Maurizio; Ciurli, Stefano; Musiani, ...Francesco | 2020-01-01 | MOLECULES | - | 1.01 Articolo in rivista | 63_2020_Masetti_Molecules.pdf |