TAROZZI, ANDREA
TAROZZI, ANDREA
QUVI - DIPARTIMENTO DI SCIENZE PER LA QUALITA' DELLA VITA
Docenti di ruolo di Ia fascia
Antioxidant and neuroprotective effects of ubiquinol diacetate: Insights from SH-SY5Y cell line and Caenorhabditis elegans models of Parkinson's disease
2026 Micucci, Matteo; Battistelli, Michela; Burattini, Sabrina; Osman, Riham; Onesimo, Francesco; Mari, Michele; Retini, Michele; Versari, Ilaria; Pagliarani, Barbara; Tarozzi, Andrea; Zappia, Giovanni; Gianfanti, Federico; Pruccoli, Letizia
Exploring the anti-inflammatory activity of sulforaphane metabolites
2026 Pagliarani, B.; Pruccoli, L.; Chemello, C.; Zusso, M.; Fonseca Moreira, J. C.; Tarozzi, A.; Gomes, H. M.
AR-A014418-based dual Glycogen Synthase Kinase 3β/Histone Deacetylase inhibitors as potential therapeutics for Alzheimer's disease
2025 Santini, Alan; Tassinari, Elisa; Altomare, Alessandra; Loi, Manuela; Ciani, Elisabetta; Trazzi, Stefania; Piccarducci, Rebecca; Daniele, Simona; Martini, Claudia; Pagliarani, Barbara; Tarozzi, Andrea; Bersani, Matteo; Spyrakis, Francesca; Danková, Daniela; Poeta, Eleonora; Raimondi, Simone; Davani, Lara; Aldini, Giancarlo; Andrisano, Vincenza; De Simone, Angela; Milelli, Andrea
Effetti Antiossidanti e Antinfiammatori del Nutraceutico Sulforafano e dei suoi Metaboliti: uno Studio Comparativo in Modelli in vitro
2025 Pagliarani, B.; Mautone Gomes, H.; Pruccoli, L.; Tarozzi, A.
Glycosylation of chrysin with β-d-glucose tetraacetate (LQFM280) enhances its in vitro and in vivo neuroprotective effects against the toxicity induced by 3-nitropropionic acid
2025 Pereira, R. M.; Campos, H. M.; De Oliveira Ferreira, P. Y.; Uchenna, N.; Silva, Y. S.; Okoh, V. I.; Pruccoli, L.; Arruda, E. L.; Liao, L. M.; Mota, P. A. A.; Leite, J. A.; De Castro Georg, R.; Damatta, D.; Dos Santos, F. C. A.; Costa, E. A.; Tarozzi, A.; Menegatti, R.; Ghedini, P. C.
Rational optimization of D3R/GSK-3β dual target-directed ligands as potential treatment for bipolar disorder: Design, synthesis, X-ray crystallography, molecular dynamics simulations, in vitro ADME, and in vivo pharmacokinetic studies
2025 Di Martino, R. M. C.; Russo, D.; Penna, I.; Demuro, S.; Dalle Vedove, A.; Spagnuolo, R.; Ottonello, G.; Bertozzi, S. M.; Summa, M.; Desantis, J.; Valeri, A.; Pruccoli, L.; Tripathi, S. K.; Tarozzi, A.; Storici, P.; Girotto, S.; Bertorelli, R.; Armirotti, A.; Cruciani, G.; Bandiera, T.; Cavalli, A.; Bottegoni, G.
Targeting Alzheimer’s disease neurotoxicity by functionalization of the chalcone scaffold
2025 Da Fermo, A.; Tarozzi, A.; Pruccoli, L.; Zusso, M.; Orioli, R.; Bisi, A.; Gobbi, S.; Belluti, F.
A novel arylpiperazine derivative (LQFM181) protects against neurotoxicity induced by 3- nitropropionic acid in in vitro and in vivo models
2024 Mesquita Campos, Hericles; Mota Pereira, Robbert; Yasmin de Oliveira Ferreira, Pamela; Uchenna, Nkaa; Rio Branco da Silva, Cínthia; Pruccoli, Letizia; Sanz, German; Ferreira Rodrigues, Marcella; Gontijo Vaz, Boniek; Gonçalves Rivello, Barbara; Luís Batista da Rocha, Andre; Silva de Carvalho, Flavio; de Almeida Ribeiro Oliveira, Gerlon; Morais Liao, Luciano; de Castro Georg, Raphaela; Alves Leite, Jacqueline; Cristina Alcantara dos Santos, Fernanda; Alves Costa, Elson; Menegatti, Ricardo; Tarozzi, Andrea; Cesar Ghedini, Paulo
Antioxidant and Anti-Melanogenesis Effects of Teucrium chamaedrys L. Cell Suspension Extract and Its Main Phenylethanoid Glycoside in B16-F10 Cells
2024 Pruccoli, Letizia; Nicolini, Benedetta; Lianza, Mariacaterina; Teti, Gabriella; Falconi, Mirella; Tarozzi, Andrea; Antognoni, Fabiana
Antioxidant and Neuroprotective Effects of Fucoxanthin and Its Metabolite Fucoxanthinol: A Comparative In Vitro Study
2024 Pruccoli, Letizia; Balducci, Martina; Pagliarani, Barbara; Tarozzi, Andrea
Chrysin bonded to β-d-glucose tetraacetate enhances its protective effects against the neurotoxicity induced by aluminum in Swiss mice
2024 Ifeanyi Okoh, Victor; Mesquita Campos, Hericles; Yasmin de Oliveira Ferreira, Pâmela; Mota Pereira, Robbert; Souza Silva, Yohanny; Lima Arruda, Evilanna; Pagliarani, Barbara; de Almeida Ribeiro Oliveira, Gerlon; Morais Lião, Luciano; Franco Dos Santos, Gabriel; Gontijo Vaz, Boniek; Ricardo Sabino, José; Cristina Alcantara Dos Santos, Fernanda; Alves Costa, Elson; Tarozzi, Andrea; Menegatti, Ricardo; César Ghedini, Paulo
Erucin, a Natural Isothiocyanate, Prevents Polyglutamine-Induced Toxicity in Caenorhabditis elegans via aak-2/AMPK and daf-16/FOXO Signaling
2024 Balducci, M.; Perez, J. T.; del Rio, C. T.; Perez, M. C.; Carranza, A. D. V.; Gomez Escribano, A. P.; Vazquez-Manrique, R. P.; Tarozzi, A.
First in Class Dual Non-ATP-Competitive Glycogen Synthase Kinase 3β/Histone Deacetylase Inhibitors as a Potential Therapeutic to Treat Alzheimer’s Disease
2024 Santini, A.; Tassinari, E.; Poeta, E.; Loi, M.; Ciani, E.; Trazzi, S.; Piccarducci, R.; Daniele, S.; Martini, C.; Pagliarani, B.; Tarozzi, A.; Bersani, M.; Spyrakis, F.; Danková, D.; Olsen, C. A.; Soldati, R.; Tumiatti, V.; Montanari, S.; De Simone, A.; Milelli, A.
Synthesis and pharmacological evaluation of novel N-aryl-cinnamoyl-hydrazone hybrids designed as neuroprotective agents for the treatment of Parkinson’s disease
2024 De Freitas Silva, Matheus; Juliet Cristancho Ortiz, Cindy; Ferreira Coelho, Letícia; Pruccoli, Letizia; Pagliarani, Barbara; Pisani, Leonardo; Catto, Marco; Poli, Giulio; Tuccinardi, Tiziano; Cardoso Vilela, Fabiana; Giusti-Paiva, Alexandre; Amaral Alves, Marina; Ribeiro De Souza, Hygor M.; Tarozzi, Andrea; Silva Gontijo, Vanessa; Jr., Claudio Viegas
Heat stress as a potential risk factor for vitamin D deficiency
2023 Balducci M.; Pruccoli L.; Tarozzi A.
Neuroprotection by Drugs, Nutraceuticals and Physical Activity
2023 Tarozzi A.; Angeloni C.
PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease
2023 Guardigni M.; Pruccoli L.; Santini A.; Simone A.D.; Bersani M.; Spyrakis F.; Frabetti F.; Uliassi E.; Andrisano V.; Pagliarani B.; Fernández-Gómez P.; Palomo V.; Bolognesi M.L.; Tarozzi A.; Milelli A.
Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold
2023 De Lorenzi, Ersilia; Seghetti, Francesca; Tarozzi, Andrea; Pruccoli, Letizia; Contardi, Cecilia; Serra, Massimo; Bisi, Alessandra; Gobbi, Silvia; Vistoli, Giulio; Gervasoni, Silvia; Argentini, Carla; Ghirardo, Giulia; Guarato, Giulia; Orso, Genny; Belluti, Federica; Di Martino, Rita Maria Concetta; Zusso, Morena
Addressing a Trapped High-Energy Water: Design and Synthesis of Highly Potent Pyrimidoindole-Based Glycogen Synthase Kinase-3β Inhibitors
2022 Andreev S.; Pantsar T.; Tesch R.; Kahlke N.; El-Gokha A.; Ansideri F.; Gratz L.; Romasco J.; Sita G.; Geibel C.; Lammerhofer M.; Tarozzi A.; Knapp S.; Laufer S.A.; Koch P.
Design, synthesis, and biological evaluation of new thalidomide–donepezil hybrids as neuroprotective agents targeting cholinesterases and neuroinflammation
2022 Cindy Juliet Cristancho Ortiz, Matheus de Freitas Silva, Letizia Pruccoli, Nathália Fonseca Nadur, Luciana Luíza de Azevedo, Arthur Eugen Kümmerle, Isabella Alvim Guedes, Laurent Emmanuel Dardenne, Luiz Felipe Leomil Coelho, Marcos J. Guimarães, Fernanda M. R. da Silva, Newton Castro, Vanessa Silva Gontijo, Viviana C. T. Rojas, Merelym Ketterym de Oliveira, Fabiana Cardoso Vilela, Alexandre Giusti-Paiva, Gisele Barbosa, Lídia Moreira Lima, Gabriela Beserra Pinheiro, Letícia Germino Veras, Márcia Renata Mortari, Andrea Tarozzi, Claudio Viegas Jr
| Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
|---|---|---|---|---|---|---|
| Antioxidant and neuroprotective effects of ubiquinol diacetate: Insights from SH-SY5Y cell line and Caenorhabditis elegans models of Parkinson's disease | Micucci, Matteo; Battistelli, Michela; Burattini, Sabrina; Osman, Riham; Onesimo, Francesco; Mari..., Michele; Retini, Michele; Versari, Ilaria; Pagliarani, Barbara; Tarozzi, Andrea; Zappia, Giovanni; Gianfanti, Federico; Pruccoli, Letizia | 2026-01-01 | EXPERIMENTAL AND MOLECULAR PATHOLOGY | - | 1.01 Articolo in rivista | Antioxidant-and-neuroprotective-effects-of-ubiquinol-diac_2026_Experimental-.pdf; 1-s2.0-S001448002600002X-mmc1.pdf |
| Exploring the anti-inflammatory activity of sulforaphane metabolites | Pagliarani, B.; Pruccoli, L.; Chemello, C.; Zusso, M.; Fonseca Moreira, J. C.; Tarozzi, A.; Gomes..., H. M. | 2026-01-01 | PHARMACOLOGICAL REPORTS | - | 1.01 Articolo in rivista | Revised Article POSTPRINT Embargo.pdf; 43440_2026_823_MOESM1_ESM.pdf |
| AR-A014418-based dual Glycogen Synthase Kinase 3β/Histone Deacetylase inhibitors as potential therapeutics for Alzheimer's disease | Santini, Alan; Tassinari, Elisa; Altomare, Alessandra; Loi, Manuela; Ciani, Elisabetta; Trazzi, S...tefania; Piccarducci, Rebecca; Daniele, Simona; Martini, Claudia; Pagliarani, Barbara; Tarozzi, Andrea; Bersani, Matteo; Spyrakis, Francesca; Danková, Daniela; Poeta, Eleonora; Raimondi, Simone; Davani, Lara; Aldini, Giancarlo; Andrisano, Vincenza; De Simone, Angela; Milelli, Andrea | 2025-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | AR-A014418-based dual Glycogen Synthase Kinase 3β_Histone Deacetylase inhibitors as potential therapeutics for Alzheimer_s disease.pdf; 1-s2.0-S0223523425006038-mmc1.docx |
| Effetti Antiossidanti e Antinfiammatori del Nutraceutico Sulforafano e dei suoi Metaboliti: uno Studio Comparativo in Modelli in vitro | Pagliarani, B.; Mautone Gomes, H.; Pruccoli, L.; Tarozzi, A. | 2025-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Glycosylation of chrysin with β-d-glucose tetraacetate (LQFM280) enhances its in vitro and in vivo neuroprotective effects against the toxicity induced by 3-nitropropionic acid | Pereira, R. M.; Campos, H. M.; De Oliveira Ferreira, P. Y.; Uchenna, N.; Silva, Y. S.; Okoh, V. I....; Pruccoli, L.; Arruda, E. L.; Liao, L. M.; Mota, P. A. A.; Leite, J. A.; De Castro Georg, R.; Damatta, D.; Dos Santos, F. C. A.; Costa, E. A.; Tarozzi, A.; Menegatti, R.; Ghedini, P. C. | 2025-01-01 | NAUNYN-SCHMIEDEBERG'S ARCHIVES OF PHARMACOLOGY | - | 1.01 Articolo in rivista | ARTICL~1.PDF |
| Rational optimization of D3R/GSK-3β dual target-directed ligands as potential treatment for bipolar disorder: Design, synthesis, X-ray crystallography, molecular dynamics simulations, in vitro ADME, and in vivo pharmacokinetic studies | Di Martino, R. M. C.; Russo, D.; Penna, I.; Demuro, S.; Dalle Vedove, A.; Spagnuolo, R.; Ottonell...o, G.; Bertozzi, S. M.; Summa, M.; Desantis, J.; Valeri, A.; Pruccoli, L.; Tripathi, S. K.; Tarozzi, A.; Storici, P.; Girotto, S.; Bertorelli, R.; Armirotti, A.; Cruciani, G.; Bandiera, T.; Cavalli, A.; Bottegoni, G. | 2025-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | h_11585_1026573.pdf; ScienceDirect_files_05Nov2025_12-04-15.802.zip |
| Targeting Alzheimer’s disease neurotoxicity by functionalization of the chalcone scaffold | Da Fermo, A.; Tarozzi, A.; Pruccoli, L.; Zusso, M.; Orioli, R.; Bisi, A.; Gobbi, S.; Belluti, F. | 2025-01-01 | - | - | 4.03 Poster | - |
| A novel arylpiperazine derivative (LQFM181) protects against neurotoxicity induced by 3- nitropropionic acid in in vitro and in vivo models | Mesquita Campos, Hericles; Mota Pereira, Robbert; Yasmin de Oliveira Ferreira, Pamela; Uchenna, N...kaa; Rio Branco da Silva, Cínthia; Pruccoli, Letizia; Sanz, German; Ferreira Rodrigues, Marcella; Gontijo Vaz, Boniek; Gonçalves Rivello, Barbara; Luís Batista da Rocha, Andre; Silva de Carvalho, Flavio; de Almeida Ribeiro Oliveira, Gerlon; Morais Liao, Luciano; de Castro Georg, Raphaela; Alves Leite, Jacqueline; Cristina Alcantara dos Santos, Fernanda; Alves Costa, Elson; Menegatti, Ricardo; Tarozzi, Andrea; Cesar Ghedini, Paulo | 2024-01-01 | CHEMICO-BIOLOGICAL INTERACTIONS | - | 1.01 Articolo in rivista | Final Article not marked POSTPRINT.pdf |
| Antioxidant and Anti-Melanogenesis Effects of Teucrium chamaedrys L. Cell Suspension Extract and Its Main Phenylethanoid Glycoside in B16-F10 Cells | Pruccoli, Letizia; Nicolini, Benedetta; Lianza, Mariacaterina; Teti, Gabriella; Falconi, Mirella;... Tarozzi, Andrea; Antognoni, Fabiana | 2024-01-01 | PLANTS | - | 1.01 Articolo in rivista | plants-13-00808 (1).pdf; plants-2894275-supplementary.pdf |
| Antioxidant and Neuroprotective Effects of Fucoxanthin and Its Metabolite Fucoxanthinol: A Comparative In Vitro Study | Pruccoli, Letizia; Balducci, Martina; Pagliarani, Barbara; Tarozzi, Andrea | 2024-01-01 | CURRENT ISSUES IN MOLECULAR BIOLOGY | - | 1.01 Articolo in rivista | cimb-46-00357 (2).pdf; cimb-46-00357-s001.zip |
| Chrysin bonded to β-d-glucose tetraacetate enhances its protective effects against the neurotoxicity induced by aluminum in Swiss mice | Ifeanyi Okoh, Victor; Mesquita Campos, Hericles; Yasmin de Oliveira Ferreira, Pâmela; Mota Pereir...a, Robbert; Souza Silva, Yohanny; Lima Arruda, Evilanna; Pagliarani, Barbara; de Almeida Ribeiro Oliveira, Gerlon; Morais Lião, Luciano; Franco Dos Santos, Gabriel; Gontijo Vaz, Boniek; Ricardo Sabino, José; Cristina Alcantara Dos Santos, Fernanda; Alves Costa, Elson; Tarozzi, Andrea; Menegatti, Ricardo; César Ghedini, Paulo | 2024-01-01 | JOURNAL OF PHARMACY AND PHARMACOLOGY | - | 1.01 Articolo in rivista | Postprint.pdf |
| Erucin, a Natural Isothiocyanate, Prevents Polyglutamine-Induced Toxicity in Caenorhabditis elegans via aak-2/AMPK and daf-16/FOXO Signaling | Balducci, M.; Perez, J. T.; del Rio, C. T.; Perez, M. C.; Carranza, A. D. V.; Gomez Escribano, A.... P.; Vazquez-Manrique, R. P.; Tarozzi, A. | 2024-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | ijms-25-12220.pdf; ijms-25-12220-s001.zip |
| First in Class Dual Non-ATP-Competitive Glycogen Synthase Kinase 3β/Histone Deacetylase Inhibitors as a Potential Therapeutic to Treat Alzheimer’s Disease | Santini, A.; Tassinari, E.; Poeta, E.; Loi, M.; Ciani, E.; Trazzi, S.; Piccarducci, R.; Daniele, ...S.; Martini, C.; Pagliarani, B.; Tarozzi, A.; Bersani, M.; Spyrakis, F.; Danková, D.; Olsen, C. A.; Soldati, R.; Tumiatti, V.; Montanari, S.; De Simone, A.; Milelli, A. | 2024-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | acs-cn.pdf |
| Synthesis and pharmacological evaluation of novel N-aryl-cinnamoyl-hydrazone hybrids designed as neuroprotective agents for the treatment of Parkinson’s disease | De Freitas Silva, Matheus; Juliet Cristancho Ortiz, Cindy; Ferreira Coelho, Letícia; Pruccoli, Le...tizia; Pagliarani, Barbara; Pisani, Leonardo; Catto, Marco; Poli, Giulio; Tuccinardi, Tiziano; Cardoso Vilela, Fabiana; Giusti-Paiva, Alexandre; Amaral Alves, Marina; Ribeiro De Souza, Hygor M.; Tarozzi, Andrea; Silva Gontijo, Vanessa; Jr., Claudio Viegas | 2024-01-01 | BIOORGANIC CHEMISTRY | - | 1.01 Articolo in rivista | Manuscript ridotto.pdf |
| Heat stress as a potential risk factor for vitamin D deficiency | Balducci M.; Pruccoli L.; Tarozzi A. | 2023-01-01 | MEDICAL HYPOTHESES | - | 1.01 Articolo in rivista | Revised manuscript.pdf |
| Neuroprotection by Drugs, Nutraceuticals and Physical Activity | Tarozzi A.; Angeloni C. | 2023-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | ijms-24-03176.pdf |
| PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease | Guardigni M.; Pruccoli L.; Santini A.; Simone A.D.; Bersani M.; Spyrakis F.; Frabetti F.; Uliassi... E.; Andrisano V.; Pagliarani B.; Fernández-Gómez P.; Palomo V.; Bolognesi M.L.; Tarozzi A.; Milelli A. | 2023-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | acschemneuro.3c00096.pdf |
| Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold | De Lorenzi, Ersilia; Seghetti, Francesca; Tarozzi, Andrea; Pruccoli, Letizia; Contardi, Cecilia; ...Serra, Massimo; Bisi, Alessandra; Gobbi, Silvia; Vistoli, Giulio; Gervasoni, Silvia; Argentini, Carla; Ghirardo, Giulia; Guarato, Giulia; Orso, Genny; Belluti, Federica; Di Martino, Rita Maria Concetta; Zusso, Morena | 2023-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold.pdf; 1-s2.0-S0223523423002635-mmc1.pdf |
| Addressing a Trapped High-Energy Water: Design and Synthesis of Highly Potent Pyrimidoindole-Based Glycogen Synthase Kinase-3β Inhibitors | Andreev S.; Pantsar T.; Tesch R.; Kahlke N.; El-Gokha A.; Ansideri F.; Gratz L.; Romasco J.; Sita... G.; Geibel C.; Lammerhofer M.; Tarozzi A.; Knapp S.; Laufer S.A.; Koch P. | 2022-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | J Med Chem 2022.pdf |
| Design, synthesis, and biological evaluation of new thalidomide–donepezil hybrids as neuroprotective agents targeting cholinesterases and neuroinflammation | Cindy Juliet Cristancho Ortiz, Matheus de Freitas Silva, Letizia Pruccoli, Nathália Fonseca Nadur..., Luciana Luíza de Azevedo, Arthur Eugen Kümmerle, Isabella Alvim Guedes, Laurent Emmanuel Dardenne, Luiz Felipe Leomil Coelho, Marcos J. Guimarães, Fernanda M. R. da Silva, Newton Castro, Vanessa Silva Gontijo, Viviana C. T. Rojas, Merelym Ketterym de Oliveira, Fabiana Cardoso Vilela, Alexandre Giusti-Paiva, Gisele Barbosa, Lídia Moreira Lima, Gabriela Beserra Pinheiro, Letícia Germino Veras, Márcia Renata Mortari, Andrea Tarozzi, Claudio Viegas Jr | 2022-01-01 | RSC MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Manuscript RSC TAROZZI Andrea.pdf |