TAROZZI, ANDREA
TAROZZI, ANDREA
QUVI - DIPARTIMENTO DI SCIENZE PER LA QUALITA' DELLA VITA
Docenti di ruolo di Ia fascia
Antioxidant and neuroprotective effects of ubiquinol diacetate: Insights from SH-SY5Y cell line and Caenorhabditis elegans models of Parkinson's disease
2026 Micucci, Matteo; Battistelli, Michela; Burattini, Sabrina; Osman, Riham; Onesimo, Francesco; Mari, Michele; Retini, Michele; Versari, Ilaria; Pagliarani, Barbara; Tarozzi, Andrea; Zappia, Giovanni; Gianfanti, Federico; Pruccoli, Letizia
Exploring the anti-inflammatory activity of sulforaphane metabolites
2026 Pagliarani, B.; Pruccoli, L.; Chemello, C.; Zusso, M.; Fonseca Moreira, J. C.; Tarozzi, A.; Gomes, H. M.
AR-A014418-based dual Glycogen Synthase Kinase 3β/Histone Deacetylase inhibitors as potential therapeutics for Alzheimer's disease
2025 Santini, Alan; Tassinari, Elisa; Altomare, Alessandra; Loi, Manuela; Ciani, Elisabetta; Trazzi, Stefania; Piccarducci, Rebecca; Daniele, Simona; Martini, Claudia; Pagliarani, Barbara; Tarozzi, Andrea; Bersani, Matteo; Spyrakis, Francesca; Danková, Daniela; Poeta, Eleonora; Raimondi, Simone; Davani, Lara; Aldini, Giancarlo; Andrisano, Vincenza; De Simone, Angela; Milelli, Andrea
Effetti Antiossidanti e Antinfiammatori del Nutraceutico Sulforafano e dei suoi Metaboliti: uno Studio Comparativo in Modelli in vitro
2025 Pagliarani, B.; Mautone Gomes, H.; Pruccoli, L.; Tarozzi, A.
Glycosylation of chrysin with β-d-glucose tetraacetate (LQFM280) enhances its in vitro and in vivo neuroprotective effects against the toxicity induced by 3-nitropropionic acid
2025 Pereira, R. M.; Campos, H. M.; De Oliveira Ferreira, P. Y.; Uchenna, N.; Silva, Y. S.; Okoh, V. I.; Pruccoli, L.; Arruda, E. L.; Liao, L. M.; Mota, P. A. A.; Leite, J. A.; De Castro Georg, R.; Damatta, D.; Dos Santos, F. C. A.; Costa, E. A.; Tarozzi, A.; Menegatti, R.; Ghedini, P. C.
Rational optimization of D3R/GSK-3β dual target-directed ligands as potential treatment for bipolar disorder: Design, synthesis, X-ray crystallography, molecular dynamics simulations, in vitro ADME, and in vivo pharmacokinetic studies
2025 Di Martino, R. M. C.; Russo, D.; Penna, I.; Demuro, S.; Dalle Vedove, A.; Spagnuolo, R.; Ottonello, G.; Bertozzi, S. M.; Summa, M.; Desantis, J.; Valeri, A.; Pruccoli, L.; Tripathi, S. K.; Tarozzi, A.; Storici, P.; Girotto, S.; Bertorelli, R.; Armirotti, A.; Cruciani, G.; Bandiera, T.; Cavalli, A.; Bottegoni, G.
Targeting Alzheimer’s disease neurotoxicity by functionalization of the chalcone scaffold
2025 Da Fermo, A.; Tarozzi, A.; Pruccoli, L.; Zusso, M.; Orioli, R.; Bisi, A.; Gobbi, S.; Belluti, F.
A novel arylpiperazine derivative (LQFM181) protects against neurotoxicity induced by 3- nitropropionic acid in in vitro and in vivo models
2024 Mesquita Campos, Hericles; Mota Pereira, Robbert; Yasmin de Oliveira Ferreira, Pamela; Uchenna, Nkaa; Rio Branco da Silva, Cínthia; Pruccoli, Letizia; Sanz, German; Ferreira Rodrigues, Marcella; Gontijo Vaz, Boniek; Gonçalves Rivello, Barbara; Luís Batista da Rocha, Andre; Silva de Carvalho, Flavio; de Almeida Ribeiro Oliveira, Gerlon; Morais Liao, Luciano; de Castro Georg, Raphaela; Alves Leite, Jacqueline; Cristina Alcantara dos Santos, Fernanda; Alves Costa, Elson; Menegatti, Ricardo; Tarozzi, Andrea; Cesar Ghedini, Paulo
Antioxidant and Anti-Melanogenesis Effects of Teucrium chamaedrys L. Cell Suspension Extract and Its Main Phenylethanoid Glycoside in B16-F10 Cells
2024 Pruccoli, Letizia; Nicolini, Benedetta; Lianza, Mariacaterina; Teti, Gabriella; Falconi, Mirella; Tarozzi, Andrea; Antognoni, Fabiana
Antioxidant and Neuroprotective Effects of Fucoxanthin and Its Metabolite Fucoxanthinol: A Comparative In Vitro Study
2024 Pruccoli, Letizia; Balducci, Martina; Pagliarani, Barbara; Tarozzi, Andrea
Chrysin bonded to β-d-glucose tetraacetate enhances its protective effects against the neurotoxicity induced by aluminum in Swiss mice
2024 Ifeanyi Okoh, Victor; Mesquita Campos, Hericles; Yasmin de Oliveira Ferreira, Pâmela; Mota Pereira, Robbert; Souza Silva, Yohanny; Lima Arruda, Evilanna; Pagliarani, Barbara; de Almeida Ribeiro Oliveira, Gerlon; Morais Lião, Luciano; Franco Dos Santos, Gabriel; Gontijo Vaz, Boniek; Ricardo Sabino, José; Cristina Alcantara Dos Santos, Fernanda; Alves Costa, Elson; Tarozzi, Andrea; Menegatti, Ricardo; César Ghedini, Paulo
Erucin, a Natural Isothiocyanate, Prevents Polyglutamine-Induced Toxicity in Caenorhabditis elegans via aak-2/AMPK and daf-16/FOXO Signaling
2024 Balducci, M.; Perez, J. T.; del Rio, C. T.; Perez, M. C.; Carranza, A. D. V.; Gomez Escribano, A. P.; Vazquez-Manrique, R. P.; Tarozzi, A.
First in Class Dual Non-ATP-Competitive Glycogen Synthase Kinase 3β/Histone Deacetylase Inhibitors as a Potential Therapeutic to Treat Alzheimer’s Disease
2024 Santini, A.; Tassinari, E.; Poeta, E.; Loi, M.; Ciani, E.; Trazzi, S.; Piccarducci, R.; Daniele, S.; Martini, C.; Pagliarani, B.; Tarozzi, A.; Bersani, M.; Spyrakis, F.; Danková, D.; Olsen, C. A.; Soldati, R.; Tumiatti, V.; Montanari, S.; De Simone, A.; Milelli, A.
Synthesis and pharmacological evaluation of novel N-aryl-cinnamoyl-hydrazone hybrids designed as neuroprotective agents for the treatment of Parkinson’s disease
2024 De Freitas Silva, Matheus; Juliet Cristancho Ortiz, Cindy; Ferreira Coelho, Letícia; Pruccoli, Letizia; Pagliarani, Barbara; Pisani, Leonardo; Catto, Marco; Poli, Giulio; Tuccinardi, Tiziano; Cardoso Vilela, Fabiana; Giusti-Paiva, Alexandre; Amaral Alves, Marina; Ribeiro De Souza, Hygor M.; Tarozzi, Andrea; Silva Gontijo, Vanessa; Jr., Claudio Viegas
Heat stress as a potential risk factor for vitamin D deficiency
2023 Balducci M.; Pruccoli L.; Tarozzi A.
Neuroprotection by Drugs, Nutraceuticals and Physical Activity
2023 Tarozzi A.; Angeloni C.
PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease
2023 Guardigni M.; Pruccoli L.; Santini A.; Simone A.D.; Bersani M.; Spyrakis F.; Frabetti F.; Uliassi E.; Andrisano V.; Pagliarani B.; Fernández-Gómez P.; Palomo V.; Bolognesi M.L.; Tarozzi A.; Milelli A.
Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold
2023 De Lorenzi, Ersilia; Seghetti, Francesca; Tarozzi, Andrea; Pruccoli, Letizia; Contardi, Cecilia; Serra, Massimo; Bisi, Alessandra; Gobbi, Silvia; Vistoli, Giulio; Gervasoni, Silvia; Argentini, Carla; Ghirardo, Giulia; Guarato, Giulia; Orso, Genny; Belluti, Federica; Di Martino, Rita Maria Concetta; Zusso, Morena
Addressing a Trapped High-Energy Water: Design and Synthesis of Highly Potent Pyrimidoindole-Based Glycogen Synthase Kinase-3β Inhibitors
2022 Andreev S.; Pantsar T.; Tesch R.; Kahlke N.; El-Gokha A.; Ansideri F.; Gratz L.; Romasco J.; Sita G.; Geibel C.; Lammerhofer M.; Tarozzi A.; Knapp S.; Laufer S.A.; Koch P.
Design, synthesis, and biological evaluation of new thalidomide–donepezil hybrids as neuroprotective agents targeting cholinesterases and neuroinflammation
2022 Juliet Cristancho Ortiz, Cindy; De Freitas Silva, Matheus; Pruccoli, Letizia; Fonseca Nadur, Nathália; Luíza De Azevedo, Luciana; Eugen Kümmerle, Arthur; Alvim Guedes, Isabella; Emmanuel Dardenne, Laurent; Felipe Leomil Coelho, Luiz; Guimarães, Marcos J.; Da Silva, Fernanda M. R.; Castro, Newton; Silva Gontijo, Vanessa; Rojas, Viviana C. T.; Ketterym De Oliveira, Merelym; Cardoso Vilela, Fabiana; Giusti-Paiva, Alexandre; Barbosa, Gisele; Moreira Lima, Lídia; Beserra Pinheiro, Gabriela; Germino Veras, Letícia; Renata Mortari, Márcia; Tarozzi, Andrea; Viegas Jr, Claudio
| Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
|---|---|---|---|---|---|---|
| Antioxidant and neuroprotective effects of ubiquinol diacetate: Insights from SH-SY5Y cell line and Caenorhabditis elegans models of Parkinson's disease | Micucci, Matteo; Battistelli, Michela; Burattini, Sabrina; Osman, Riham; Onesimo, Francesco; Mari..., Michele; Retini, Michele; Versari, Ilaria; Pagliarani, Barbara; Tarozzi, Andrea; Zappia, Giovanni; Gianfanti, Federico; Pruccoli, Letizia | 2026-01-01 | EXPERIMENTAL AND MOLECULAR PATHOLOGY | - | 1.01 Articolo in rivista | Antioxidant-and-neuroprotective-effects-of-ubiquinol-diac_2026_Experimental-.pdf; 1-s2.0-S001448002600002X-mmc1.pdf |
| Exploring the anti-inflammatory activity of sulforaphane metabolites | Pagliarani, B.; Pruccoli, L.; Chemello, C.; Zusso, M.; Fonseca Moreira, J. C.; Tarozzi, A.; Gomes..., H. M. | 2026-01-01 | PHARMACOLOGICAL REPORTS | - | 1.01 Articolo in rivista | Revised Article POSTPRINT Embargo.pdf; 43440_2026_823_MOESM1_ESM.pdf |
| AR-A014418-based dual Glycogen Synthase Kinase 3β/Histone Deacetylase inhibitors as potential therapeutics for Alzheimer's disease | Santini, Alan; Tassinari, Elisa; Altomare, Alessandra; Loi, Manuela; Ciani, Elisabetta; Trazzi, S...tefania; Piccarducci, Rebecca; Daniele, Simona; Martini, Claudia; Pagliarani, Barbara; Tarozzi, Andrea; Bersani, Matteo; Spyrakis, Francesca; Danková, Daniela; Poeta, Eleonora; Raimondi, Simone; Davani, Lara; Aldini, Giancarlo; Andrisano, Vincenza; De Simone, Angela; Milelli, Andrea | 2025-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | AR-A014418-based dual Glycogen Synthase Kinase 3β_Histone Deacetylase inhibitors as potential therapeutics for Alzheimer_s disease.pdf; 1-s2.0-S0223523425006038-mmc1.docx |
| Effetti Antiossidanti e Antinfiammatori del Nutraceutico Sulforafano e dei suoi Metaboliti: uno Studio Comparativo in Modelli in vitro | Pagliarani, B.; Mautone Gomes, H.; Pruccoli, L.; Tarozzi, A. | 2025-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Glycosylation of chrysin with β-d-glucose tetraacetate (LQFM280) enhances its in vitro and in vivo neuroprotective effects against the toxicity induced by 3-nitropropionic acid | Pereira, R. M.; Campos, H. M.; De Oliveira Ferreira, P. Y.; Uchenna, N.; Silva, Y. S.; Okoh, V. I....; Pruccoli, L.; Arruda, E. L.; Liao, L. M.; Mota, P. A. A.; Leite, J. A.; De Castro Georg, R.; Damatta, D.; Dos Santos, F. C. A.; Costa, E. A.; Tarozzi, A.; Menegatti, R.; Ghedini, P. C. | 2025-01-01 | NAUNYN-SCHMIEDEBERG'S ARCHIVES OF PHARMACOLOGY | - | 1.01 Articolo in rivista | ARTICL~1.PDF |
| Rational optimization of D3R/GSK-3β dual target-directed ligands as potential treatment for bipolar disorder: Design, synthesis, X-ray crystallography, molecular dynamics simulations, in vitro ADME, and in vivo pharmacokinetic studies | Di Martino, R. M. C.; Russo, D.; Penna, I.; Demuro, S.; Dalle Vedove, A.; Spagnuolo, R.; Ottonell...o, G.; Bertozzi, S. M.; Summa, M.; Desantis, J.; Valeri, A.; Pruccoli, L.; Tripathi, S. K.; Tarozzi, A.; Storici, P.; Girotto, S.; Bertorelli, R.; Armirotti, A.; Cruciani, G.; Bandiera, T.; Cavalli, A.; Bottegoni, G. | 2025-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | h_11585_1026573.pdf; ScienceDirect_files_05Nov2025_12-04-15.802.zip |
| Targeting Alzheimer’s disease neurotoxicity by functionalization of the chalcone scaffold | Da Fermo, A.; Tarozzi, A.; Pruccoli, L.; Zusso, M.; Orioli, R.; Bisi, A.; Gobbi, S.; Belluti, F. | 2025-01-01 | - | - | 4.03 Poster | - |
| A novel arylpiperazine derivative (LQFM181) protects against neurotoxicity induced by 3- nitropropionic acid in in vitro and in vivo models | Mesquita Campos, Hericles; Mota Pereira, Robbert; Yasmin de Oliveira Ferreira, Pamela; Uchenna, N...kaa; Rio Branco da Silva, Cínthia; Pruccoli, Letizia; Sanz, German; Ferreira Rodrigues, Marcella; Gontijo Vaz, Boniek; Gonçalves Rivello, Barbara; Luís Batista da Rocha, Andre; Silva de Carvalho, Flavio; de Almeida Ribeiro Oliveira, Gerlon; Morais Liao, Luciano; de Castro Georg, Raphaela; Alves Leite, Jacqueline; Cristina Alcantara dos Santos, Fernanda; Alves Costa, Elson; Menegatti, Ricardo; Tarozzi, Andrea; Cesar Ghedini, Paulo | 2024-01-01 | CHEMICO-BIOLOGICAL INTERACTIONS | - | 1.01 Articolo in rivista | Final Article not marked POSTPRINT.pdf |
| Antioxidant and Anti-Melanogenesis Effects of Teucrium chamaedrys L. Cell Suspension Extract and Its Main Phenylethanoid Glycoside in B16-F10 Cells | Pruccoli, Letizia; Nicolini, Benedetta; Lianza, Mariacaterina; Teti, Gabriella; Falconi, Mirella;... Tarozzi, Andrea; Antognoni, Fabiana | 2024-01-01 | PLANTS | - | 1.01 Articolo in rivista | plants-13-00808 (1).pdf; plants-2894275-supplementary.pdf |
| Antioxidant and Neuroprotective Effects of Fucoxanthin and Its Metabolite Fucoxanthinol: A Comparative In Vitro Study | Pruccoli, Letizia; Balducci, Martina; Pagliarani, Barbara; Tarozzi, Andrea | 2024-01-01 | CURRENT ISSUES IN MOLECULAR BIOLOGY | - | 1.01 Articolo in rivista | cimb-46-00357 (2).pdf; cimb-46-00357-s001.zip |
| Chrysin bonded to β-d-glucose tetraacetate enhances its protective effects against the neurotoxicity induced by aluminum in Swiss mice | Ifeanyi Okoh, Victor; Mesquita Campos, Hericles; Yasmin de Oliveira Ferreira, Pâmela; Mota Pereir...a, Robbert; Souza Silva, Yohanny; Lima Arruda, Evilanna; Pagliarani, Barbara; de Almeida Ribeiro Oliveira, Gerlon; Morais Lião, Luciano; Franco Dos Santos, Gabriel; Gontijo Vaz, Boniek; Ricardo Sabino, José; Cristina Alcantara Dos Santos, Fernanda; Alves Costa, Elson; Tarozzi, Andrea; Menegatti, Ricardo; César Ghedini, Paulo | 2024-01-01 | JOURNAL OF PHARMACY AND PHARMACOLOGY | - | 1.01 Articolo in rivista | Postprint.pdf |
| Erucin, a Natural Isothiocyanate, Prevents Polyglutamine-Induced Toxicity in Caenorhabditis elegans via aak-2/AMPK and daf-16/FOXO Signaling | Balducci, M.; Perez, J. T.; del Rio, C. T.; Perez, M. C.; Carranza, A. D. V.; Gomez Escribano, A.... P.; Vazquez-Manrique, R. P.; Tarozzi, A. | 2024-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | ijms-25-12220.pdf; ijms-25-12220-s001.zip |
| First in Class Dual Non-ATP-Competitive Glycogen Synthase Kinase 3β/Histone Deacetylase Inhibitors as a Potential Therapeutic to Treat Alzheimer’s Disease | Santini, A.; Tassinari, E.; Poeta, E.; Loi, M.; Ciani, E.; Trazzi, S.; Piccarducci, R.; Daniele, ...S.; Martini, C.; Pagliarani, B.; Tarozzi, A.; Bersani, M.; Spyrakis, F.; Danková, D.; Olsen, C. A.; Soldati, R.; Tumiatti, V.; Montanari, S.; De Simone, A.; Milelli, A. | 2024-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | acs-cn.pdf |
| Synthesis and pharmacological evaluation of novel N-aryl-cinnamoyl-hydrazone hybrids designed as neuroprotective agents for the treatment of Parkinson’s disease | De Freitas Silva, Matheus; Juliet Cristancho Ortiz, Cindy; Ferreira Coelho, Letícia; Pruccoli, Le...tizia; Pagliarani, Barbara; Pisani, Leonardo; Catto, Marco; Poli, Giulio; Tuccinardi, Tiziano; Cardoso Vilela, Fabiana; Giusti-Paiva, Alexandre; Amaral Alves, Marina; Ribeiro De Souza, Hygor M.; Tarozzi, Andrea; Silva Gontijo, Vanessa; Jr., Claudio Viegas | 2024-01-01 | BIOORGANIC CHEMISTRY | - | 1.01 Articolo in rivista | Manuscript ridotto.pdf |
| Heat stress as a potential risk factor for vitamin D deficiency | Balducci M.; Pruccoli L.; Tarozzi A. | 2023-01-01 | MEDICAL HYPOTHESES | - | 1.01 Articolo in rivista | Revised manuscript.pdf |
| Neuroprotection by Drugs, Nutraceuticals and Physical Activity | Tarozzi A.; Angeloni C. | 2023-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | ijms-24-03176.pdf |
| PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease | Guardigni M.; Pruccoli L.; Santini A.; Simone A.D.; Bersani M.; Spyrakis F.; Frabetti F.; Uliassi... E.; Andrisano V.; Pagliarani B.; Fernández-Gómez P.; Palomo V.; Bolognesi M.L.; Tarozzi A.; Milelli A. | 2023-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | acschemneuro.3c00096.pdf |
| Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold | De Lorenzi, Ersilia; Seghetti, Francesca; Tarozzi, Andrea; Pruccoli, Letizia; Contardi, Cecilia; ...Serra, Massimo; Bisi, Alessandra; Gobbi, Silvia; Vistoli, Giulio; Gervasoni, Silvia; Argentini, Carla; Ghirardo, Giulia; Guarato, Giulia; Orso, Genny; Belluti, Federica; Di Martino, Rita Maria Concetta; Zusso, Morena | 2023-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold.pdf; 1-s2.0-S0223523423002635-mmc1.pdf |
| Addressing a Trapped High-Energy Water: Design and Synthesis of Highly Potent Pyrimidoindole-Based Glycogen Synthase Kinase-3β Inhibitors | Andreev S.; Pantsar T.; Tesch R.; Kahlke N.; El-Gokha A.; Ansideri F.; Gratz L.; Romasco J.; Sita... G.; Geibel C.; Lammerhofer M.; Tarozzi A.; Knapp S.; Laufer S.A.; Koch P. | 2022-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | J Med Chem 2022.pdf |
| Design, synthesis, and biological evaluation of new thalidomide–donepezil hybrids as neuroprotective agents targeting cholinesterases and neuroinflammation | Juliet Cristancho Ortiz, Cindy; De Freitas Silva, Matheus; Pruccoli, Letizia; Fonseca Nadur, Nath...ália; Luíza De Azevedo, Luciana; Eugen Kümmerle, Arthur; Alvim Guedes, Isabella; Emmanuel Dardenne, Laurent; Felipe Leomil Coelho, Luiz; Guimarães, Marcos J.; Da Silva, Fernanda M. R.; Castro, Newton; Silva Gontijo, Vanessa; Rojas, Viviana C. T.; Ketterym De Oliveira, Merelym; Cardoso Vilela, Fabiana; Giusti-Paiva, Alexandre; Barbosa, Gisele; Moreira Lima, Lídia; Beserra Pinheiro, Gabriela; Germino Veras, Letícia; Renata Mortari, Márcia; Tarozzi, Andrea; Viegas Jr, Claudio | 2022-01-01 | RSC MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Manuscript RSC TAROZZI Andrea.pdf; d1md00374g1_suppl.pdf |