DE SIMONE, ANGELA
Dettaglio
DE SIMONE, ANGELA
DIPARTIMENTO DI SCIENZE PER LA QUALITA' DELLA VITA
Assegnisti
Pubblicazioni
Risultati 1 - 20 di 73 (tempo di esecuzione: 0.0 secondi).
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File | |
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1 | 3,4-Dihydro-1,3,5-triazin-2(1H)-ones as the First Dual BACE-1/GSK-3β Fragment Hits against Alzheimer's Disease | Prati, Federica; De Simone, Angela; Armirotti, Andrea; Summa, Maria; Pizzirani, Daniela; Scarpell...i, Rita; Bertozzi, Sine Mandrup; Perez, Daniel I.; Andrisano, Vincenza; Perez-Castillo, Ana; Monti, Barbara; Massenzio, Francesca; Polito, Letizia; Racchi, Marco; Sabatino, Piera; Bottegoni, Giovanni; Martinez, Ana; Cavalli, Andrea; Bolognesi, Maria L. | 2015 | ACS CHEMICAL NEUROSCIENCE | 1.01 Articolo in rivista | ||
2 | A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation | G. P. Chiriano; A. De Simone; F. Mancini; D. I. Perez; A. Cavalli; M. L. Bolognesi; G. Legname; A.... Martinez; V. Andrisano; P. Carloni; M. Roberti | 2012 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 1.01 Articolo in rivista | - | |
3 | Advanced analytical methodologies in Alzheimer's disease drug discovery | De Simone A.; Naldi M.; Tedesco D.; Bartolini M.; Davani L.; Andrisano V. | 2020 | JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS | 1.01 Articolo in rivista | - | |
4 | An Advanced Multiple Receptor Conformations Virtual Ligand Screening Protocol for the Identification of Novel BACE-1 Inhibitors | Kacker, Puneet; Masetti, Matteo; De Simone, Angela; Bottegoni, Giovanni; Cavalli, Andrea | 2011 | 4.03 Poster | - | ||
5 | Amaryllidaceae alkaloids from Narcissus pseudonarcissus L. cv. Dutch Master as potential drugs in treatment of Alzheimer's disease | Hulcova D.; Marikova J.; Korabecny J.; Hostalkova A.; Jun D.; Kunes J.; Chlebek J.; Opletal L.; D...e Simone A.; Novakova L.; Andrisano V.; Ruzicka A.; Cahlikova L. | 2019 | PHYTOCHEMISTRY | 1.01 Articolo in rivista | - | |
6 | Amyloid beta-Peptide 25-35 Self Assembly and Its Inhibition: A Model Undecapeptide System to Gain Atomistic and Secondary Structure Details of the Alzheimer's Disease Process and Treatment | Naldi M.; Fiori J.; Pistolozzi M.; Drake A.F.; Bertucci C.; Wu R.; Mlynarczyk K.; Filipek S.; De ...Simone A.; Andrisano V. | 2012 | ACS CHEMICAL NEUROSCIENCE | 1.01 Articolo in rivista | - | |
7 | Analytical approaches in Alzheimer’s disease Drug Discovery | De Simone, Angela; Bartolini, Manuela; Fiori, Jessica; D’Urzo, Annalisa; Naldi, Marina.; Andrisan...o, Vincenza | 2015 | 4.01 Contributo in Atti di convegno | - | ||
8 | Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors. | De Simone, A; Milelli, A; Naldi, M; Andrisano, V. | 2016 | 4.03 Poster | - | ||
9 | - Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors. | Angela, De Simone; Andrea, Milelli; Marina, Naldi; Vincenza, Andrisano | 2016 | 4.03 Poster | - | ||
10 | Application of an ESI-QTOF method for the detailed characterization of GSK-3β inhibitors | DE SIMONE, Angela; Fiori, Jessica; Naldi, Marina; D'Urzo, Annalisa; Tumiatti, Vincenzo; Milelli, ...Andrea; Andrisano, Vincenza | 2017 | JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS | 1.01 Articolo in rivista | - | |
11 | Application of BACE1 immobilized enzyme reactor for the characterization of multifunctional alkaloids from Corydalis cava (Fumariaceae) as Alzheimer's disease targets | Chlebek, Jakub; De Simone, Angela; Hoš͗álková, Anna; Opletal, Lubomír; Pérez, Concepción; Pérez, ...Daniel I.; Havlíková, Lucie; Cahlíková, Lucie; Andrisano, Vincenza | 2016 | FITOTERAPIA | 1.01 Articolo in rivista | - | |
12 | Application of ESI-MS method for detailed characterization of GSK-3β inhibitors by monitoring GSM peptide phosphorylation.Angelini Farmaceutici. | De Simone, A; Naldi, M; Milelli, A; Andrisano, V | 2016 | 4.01 Contributo in Atti di convegno | - | ||
13 | Beta-secretase as a target for Alzheimer's disease drug discovery: an overview of in vitro methods for characterization of inhibitors. | F. Mancini; A. De Simone; V. Andrisano | 2011 | ANALYTICAL AND BIOANALYTICAL CHEMISTRY | 1.01 Articolo in rivista | - | |
14 | (±)- BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3β Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease | Ismaili L.; Monnin J.; Etievant A.; Arribas R.L.; Viejo L.; Refouvelet B.; Soukup O.; Janockova J....; Hepnarova V.; Korabecny J.; Kucera T.; Jun D.; Andrys R.; Musilek K.; Baguet A.; Garcia-Frutos E.M.; De Simone A.; Andrisano V.; Bartolini M.; De Los Rios C.; Marco-Contelles J.; Haffen E. | 2021 | ACS CHEMICAL NEUROSCIENCE | 1.01 Articolo in rivista | - | |
15 | Characterization of essential oil components in cosmetic products by GC-MS. | De Simone, A.; Andrisano, V. | 2015 | 4.03 Poster | - | ||
16 | Circular dichroism in drug discovery and development: an abridged review. | Bertucci C; Pistolozzi M; De Simone A. | 2010 | ANALYTICAL AND BIOANALYTICAL CHEMISTRY | 1.01 Articolo in rivista | - | |
17 | Circular Dichroism: a Study of Reversible Binding HSA Binding of Lipocrine. | A. De Simone; M. Pistolozzi; M. Rosini; C. Melchiorre; C. Bertucci | 2009 | 4.01 Contributo in Atti di convegno | - | ||
18 | Combined Methodologies for Determining In Vitro Bioavailability of Drugs and Prediction of In Vivo Bioequivalence From Pharmaceutical Oral Formulations | De Simone A.; Davani L.; Montanari S.; Tumiatti V.; Avanessian S.; Testi F.; Andrisano V. | 2021 | FRONTIERS IN CHEMISTRY | 1.01 Articolo in rivista | - | |
19 | Correction: Discovery of the First-in-Class GSK-3β/HDAC Dual Inhibitor as Disease-Modifying Agent to Combat Alzheimer's Disease (ACS Medicinal Chemistry Letters (2019) 10: 4 (469−474) DOI: 10.1021/acsmedchemlett.8b00507) | De Simone A.; La Pietra V.; Betari N.; Petragnani N.; Conte M.; Daniele S.; Pietrobono D.; Martin...i C.; Petralla S.; Casadei R.; Davani L.; Frabetti F.; Russomanno P.; Novellino E.; Montanari S.; Tumiatti V.; Ballerini P.; Sarno F.; Nebbioso A.; Altucci L.; Monti B.; Andrisano V.; Milelli A. | 2019 | ACS MEDICINAL CHEMISTRY LETTERS | 1.01 Articolo in rivista | - | |
20 | Curcumin derivatives as beta-secretase (BACE1) inhibitors. | De Simone, A; Mancini, F; Belluti, F; Bartolini, M; Bottegoni, G.; Rampa, A.; Cavalli, A.; Andris...ano, V. | 2012 | 4.03 Poster | - |