DE SIMONE, ANGELA

DE SIMONE, ANGELA  

DIPARTIMENTO DI SCIENZE PER LA QUALITA' DELLA VITA  

Assegnisti  

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Risultati 1 - 20 di 77 (tempo di esecuzione: 0.023 secondi).
Titolo Autore(i) Anno Periodico Editore Tipo File
(±)- BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3β Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease Ismaili L.; Monnin J.; Etievant A.; Arribas R.L.; Viejo L.; Refouvelet B.; Soukup O.; Janockova J....; Hepnarova V.; Korabecny J.; Kucera T.; Jun D.; Andrys R.; Musilek K.; Baguet A.; Garcia-Frutos E.M.; De Simone A.; Andrisano V.; Bartolini M.; De Los Rios C.; Marco-Contelles J.; Haffen E. 2021-01-01 ACS CHEMICAL NEUROSCIENCE - 1.01 Articolo in rivista -
- Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors. Angela, De Simone; Andrea, Milelli; Marina, Naldi; Vincenza, Andrisano 2016-01-01 - - 4.03 Poster -
3,4-Dihydro-1,3,5-triazin-2(1H)-ones as the First Dual BACE-1/GSK-3β Fragment Hits against Alzheimer's Disease Prati, Federica; De Simone, Angela; Armirotti, Andrea; Summa, Maria; Pizzirani, Daniela; Scarpell...i, Rita; Bertozzi, Sine Mandrup; Perez, Daniel I.; Andrisano, Vincenza; Perez-Castillo, Ana; Monti, Barbara; Massenzio, Francesca; Polito, Letizia; Racchi, Marco; Sabatino, Piera; Bottegoni, Giovanni; Martinez, Ana; Cavalli, Andrea; Bolognesi, Maria L. 2015-01-01 ACS CHEMICAL NEUROSCIENCE - 1.01 Articolo in rivista accepted11585-546374.pdf
A multi-approach study for BACE-1 inhibitors characterization. Angela De Simone; F. Mancini; C. Bertucci; V. Andrisano 2010-01-01 - - 4.01 Contributo in Atti di convegno -
A multi-methodological approach for the investigation of β-Amyloid-CORMs interaction: an LC-ESI/MS and Circular Dichroism study. de simone a, naldi m, tedesco d, bartolini m, andrisano v 2018-01-01 - - 4.01 Contributo in Atti di convegno -
A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors Perez-Areales F.J.; Turcu A.L.; Barniol-Xicota M.; Pont C.; Pivetta D.; Espargaro A.; Bartolini M....; De Simone A.; Andrisano V.; Perez B.; Sabate R.; Sureda F.X.; Vazquez S.; Munoz-Torrero D. 2019-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
A patent review of butyrylcholinesterase inhibitors and reactivators 2010–2017 Andrisano, Vincenza*; Naldi, Marina; De Simone, Angela; Bartolini, Manuela 2018-01-01 EXPERT OPINION ON THERAPEUTIC PATENTS - 1.01 Articolo in rivista -
A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation G. P. Chiriano; A. De Simone; F. Mancini; D. I. Perez; A. Cavalli; M. L. Bolognesi; G. Legname; A.... Martinez; V. Andrisano; P. Carloni; M. Roberti 2012-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Advanced analytical methodologies in Alzheimer's disease drug discovery De Simone A.; Naldi M.; Tedesco D.; Bartolini M.; Davani L.; Andrisano V. 2020-01-01 JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS - 1.01 Articolo in rivista -
Amaryllidaceae alkaloids from Narcissus pseudonarcissus L. cv. Dutch Master as potential drugs in treatment of Alzheimer's disease Hulcova D.; Marikova J.; Korabecny J.; Hostalkova A.; Jun D.; Kunes J.; Chlebek J.; Opletal L.; D...e Simone A.; Novakova L.; Andrisano V.; Ruzicka A.; Cahlikova L. 2019-01-01 PHYTOCHEMISTRY - 1.01 Articolo in rivista -
Amyloid beta-Peptide 25-35 Self Assembly and Its Inhibition: A Model Undecapeptide System to Gain Atomistic and Secondary Structure Details of the Alzheimer's Disease Process and Treatment Naldi M.; Fiori J.; Pistolozzi M.; Drake A.F.; Bertucci C.; Wu R.; Mlynarczyk K.; Filipek S.; De ...Simone A.; Andrisano V. 2012-01-01 ACS CHEMICAL NEUROSCIENCE - 1.01 Articolo in rivista -
An Advanced Multiple Receptor Conformations Virtual Ligand Screening Protocol for the Identification of Novel BACE-1 Inhibitors Kacker, Puneet; Masetti, Matteo; De Simone, Angela; Bottegoni, Giovanni; Cavalli, Andrea 2011-01-01 - - 4.03 Poster -
An immobilized enzyme reactor based on human recombinant betasecretase (hrBACE-1-IMER) for the fast processing of substrates and screening of inhibitors Chlebek, Jakub; De Simone, Angela; Mancini, Francesca; Andrisano, Vincenza 2012-01-01 - - 4.03 Poster -
Analytical approaches in Alzheimer’s disease Drug Discovery De Simone, Angela; Bartolini, Manuela; Fiori, Jessica; D’Urzo, Annalisa; Naldi, Marina.; Andrisan...o, Vincenza 2015-01-01 - - 4.01 Contributo in Atti di convegno -
Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors. De Simone, A; Milelli, A; Naldi, M; Andrisano, V. 2016-01-01 - - 4.03 Poster -
Application of an ESI-QTOF method for the detailed characterization of GSK-3β inhibitors De Simone, Angela; Fiori, Jessica; Naldi, Marina; D'Urzo, Annalisa; Tumiatti, Vincenzo; Milelli, ...Andrea; Andrisano, Vincenza 2017-01-01 JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS - 1.01 Articolo in rivista -
Application of BACE1 immobilized enzyme reactor for the characterization of multifunctional alkaloids from Corydalis cava (Fumariaceae) as Alzheimer's disease targets Chlebek, Jakub; De Simone, Angela; Hoš͗álková, Anna; Opletal, Lubomír; Pérez, Concepción; Pérez, ...Daniel I.; Havlíková, Lucie; Cahlíková, Lucie; Andrisano, Vincenza 2016-01-01 FITOTERAPIA - 1.01 Articolo in rivista -
Application of ESI-MS method for detailed characterization of GSK-3β inhibitors by monitoring GSM peptide phosphorylation.Angelini Farmaceutici. De Simone, A; Naldi, M; Milelli, A; Andrisano, V 2016-01-01 - - 4.01 Contributo in Atti di convegno -
Aß42 peptide toxicity on neuronal cells: a lipidomic study in view of Alzheimer’s Disease drug discovery Lara Davani, Xiaoqing Fu, Angela De Simone, Peng Li, Serena Montanari, Michael Lämmerhofer, Vince...nza Andrisano 2021-01-01 - - 4.03 Poster -
Beta-secretase as a target for Alzheimer's disease drug discovery: an overview of in vitro methods for characterization of inhibitors. F. Mancini; A. De Simone; V. Andrisano 2011-01-01 ANALYTICAL AND BIOANALYTICAL CHEMISTRY - 1.01 Articolo in rivista -