GENTILUCCI, LUCA
GENTILUCCI, LUCA
DIPARTIMENTO DI CHIMICA "GIACOMO CIAMICIAN"
Docenti di ruolo di IIa fascia
Conjecturing about Small-Molecule Agonists and Antagonists of α4β1 Integrin: From Mechanistic Insight to Potential Therapeutic Applications
2024 He, Tingting; Giacomini, Daria; Tolomelli, Alessandra; Baiula, Monica; Gentilucci, Luca
Expedient recycling of peptide organocatalysts using a nanocrystalline hydroxyapatite catching system
2024 He, T.; Valagussa, B.; Boanini, E.; Gentilucci, L.
Identification of c[D-Trp-Phe-β-Ala-β-Ala], the First κ-Opioid Receptor-Specific Negative Allosteric Modulator
2024 Zhao, Junwei; Baiula, Monica; Cuna, Elisabetta; Francescato, Marco; Matalińska, Joanna; Lipiński, Piotr F.J.; Bedini, Andrea; Gentilucci, Luca
Peptide direct growth on poly(acrylic acid)/poly(vinyl alcohol) electrospun fibers coated with branched poly(ethylenimine): A solid-phase approach for scaffolds biofunctionalization
2024 Liguori, Anna; Zhao, Junwei; Di Gesù, Roberto; De Marco, Rossella; Gualandi, Chiara; Calonghi, Natalia; Pollicino, Antonino; Gentilucci, Luca; Focarete, Maria Letizia
Peptides inhibiting the assembly of monomeric human l‐lactate dehydrogenase into catalytically active homotetramer decrease the synthesis of lactate in cultured cells
2024 Stefan, Alessandra; Gentilucci, Luca; Ruffolo, Francesca; Rossi, Valentina; Sordi, Sofia; He, Tingting; di Stefano, Giuseppina; Santino, Federica; Brigotti, Maurizio; Scotti, Claudia; Iamele, Luisa; de Jonge, Hugo; Piaz, Fabrizio Dal; Santarcangelo, Danilo Rocco; Hochkoeppler, Alejandro
Design and Pharmacological Characterization of α4β1 Integrin Cyclopeptide Agonists: Computational Investigation of Ligand Determinants for Agonism versus Antagonism
2023 Anselmi, Michele; Baiula, Monica; Spampinato, Santi; Artali, Roberto; He, Tingting; Gentilucci, Luca
Design of κ-Opioid Receptor Agonists for the Development of Potential Treatments of Pain with Reduced Side Effects
2023 Santino, Federica; Gentilucci, Luca
Design, Pharmacological Characterization, and Molecular Docking of Minimalist Peptidomimetic Antagonists of α4β1 Integrin
2023 Baiula, Monica; Anselmi, Michele; Musiani, Francesco; Ghidini, Alessia; Carbone, Jacopo; Caligiana, Alberto; Maurizio, Andrea; Spampinato, Santi; Gentilucci, Luca
Synthesis and Antiproliferative Activity against Cancer Cells of Indole-Aryl-Amide Derivatives
2023 Zhao, Junwei; Carbone, Jacopo; Farruggia, Giovanna; Janecka, Anna; Gentilucci, Luca; Calonghi, Natalia
PacDOCK: A Web Server for Positional Distance-Based and Interaction-Based Analysis of Docking Results
2022 Carbone, Jacopo; Ghidini, Alessia; Romano, Antonio; Gentilucci, Luca; Musiani, Francesco
Preparation of Non-Toxic Fluorescent Peptide-Coated Silica/PEG Nanoparticles from Peptide-Block Copolymer Conjugates
2022 Federica Santino; Pasquale Stavole; Tingting He; Silvia Pieraccini; Mayra Paolillo; Luca Prodi; Enrico Rampazzo; Luca Gentilucci
Synthesis, Biological Activity and Molecular Docking of Chimeric Peptides Targeting Opioid and NOP Receptors
2022 Wtorek, Karol; Ghidini, Alessia; Gentilucci, Luca; Adamska-Bartłomiejczyk, Anna; Piekielna-Ciesielska, Justyna; Ruzza, Chiara; Sturaro, Chiara; Calò, Girolamo; Pieretti, Stefano; Kluczyk, Alicja; McDonald, John; Lambert, David G; Janecka, Anna
Design of α/β-hybrid peptide ligands of α4β1 integrin equipped with a linkable side chain for chemoselective biofunctionalization of microstructured materials
2021 Anselmi M.; Baiula M.; Santino F.; Zhao J.; Spampinato S.; Calonghi N.; Gentilucci L.
Leukocyte Integrin Antagonists as a Novel Option to Treat Dry Age-Related Macular Degeneration
2021 Baiula, Monica; Caligiana, Alberto; Bedini, Andrea; Zhao, Junwei; Santino, Federica; Cirillo, Martina; Gentilucci, Luca; Giacomini, Daria; Spampinato, Santi
Linker Hydrophilicity Modulates the Anticancer Activity of RGD–Cryptophycin Conjugates
2021 Anselmi M.; Borbely A.; Figueras E.; Michalek C.; Kemker I.; Gentilucci L.; Sewald N.
Peptide bond formation using unprotected N-carboxyanhydrides under green chemistry conditions
2021 Santino F.; Petruzzelli R.; Zhao J.; Boanini E.; Gentilucci L.
Pharmacological Characterization of µ-Opioid Receptor Agonists with Biased G Protein or β-Arrestin Signaling, and Computational Study of Conformational Changes during Receptor Activation
2021 Piekielna-Ciesielska, Justyna; Artali, Roberto; Azzam, Ammar A H; Lambert, David G; Kluczyk, Alicja; Gentilucci, Luca; Janecka, Anna
Functional Selectivity and Antinociceptive Effects of a Novel KOPr Agonist
2020 Bedini A.; Di Cesare Mannelli L.; Micheli L.; Baiula M.; Vaca G.; De Marco R.; Gentilucci L.; Ghelardini C.; Spampinato S.
Green synthesis of bioactive oligopeptides promoted by recyclable nanocrystalline hydroxyapatite
2020 Anselmi M.; Stavole P.; Boanini E.; Bigi A.; Juaristi E.; Gentilucci L.
Integrin-targeting dye-doped peg-shell/silica-core nanoparticles mimicking the proapoptotic Smac/DIABLO protein
2020 De Marco R.; Rampazzo E.; Zhao J.; Prodi L.; Paolillo M.; Picchetti P.; Gallo F.; Calonghi N.; Gentilucci L.