MINARINI, ANNA
MINARINI, ANNA
DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di Ia fascia
"Non-canonical” structures of Braf promoter as novel target in anticancer therapy
2015 Maria Laura Greco; Marco Folini; Andrea Milelli; Anna Minarini; Claudia Sissi
4-AMINO-2-PYRIDO-BICYCLIC PYRIMIDINES AND USE THEREOF AS MEDICAMENTS - 4 AMINO-2-PIRIDO-BICICLO PIRIMIDINE E LORO USO COME MEDICAMENTI
2016 Marco, DE VIVO; Antonio, ORTEGA MARTINEZ JOSE; Manuel, ARENCIBIA JIMENEZ JOSE; Minarini, Anna; Claudia, Sissi
A kinetic study of new polyamine analogs oxidized by bovine serum amine oxidase .
2011 S Saccoccio; Minarini A; A Milelli; V Tumiatti; G Tempera; N Viceconte; R Stevanato; E Agostinelli
Affinity and selectivity at M2 and M3 muscarinic receptor subtypes of cyclic and open oxygenated analogues of 4-DAMP
1992 Tumiatti V.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R.; Bolognesi M.L.
Alzheimer's disease: new approaches to drug discovery.
2009 Bolognesi M.L.; Matera R.; Minarini A.; Rosini M.; Melchiorre C.
An optimized polyamine moiety boosts the potency of human type II topoisomerase poisons as quantified by comparative analysis centered on the clinical candidate F14512
2015 Palermo, G.; Minniti, E.; Greco, M.L.; Riccardi, L.; Simoni, E.; Convertino, M.; Marchetti, C.; Rosini, M.; Sissi, C.; Minarini, A.; De Vivo, M.
Analogues of prazosin that bear a benextramine-related polyamine backbone exhibit different antagonism toward α1-adrenoreceptor subtypes
2001 Bolognesi M.L.; Marucci G.; Angeli P.; Buccioni M.; Minarini A.; Rosini M.; Tumiatti V.; Melchiorre C.
Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines
2001 Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Spampinato S.; Tumiatti V.; Melchiorre C.
Antagonist binding profile of the split chimeric muscarinic m2-trunc/m3-tail receptor
1998 Barbier P.; Colelli A.; Bolognesi M.L.; Minarini A.; Tumiatti V.; Corsini G.U.; Melchiorre C.; Maggio R.
Antidepressivi e antipsicotici
2015 Minarini, Anna; Melchiorre, Carlo
Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach
2019 Di Paolo, Maria Luisa; Cozza, Giorgio; Milelli, Andrea; Zonta, Francesca; Sarno, Stefania; Minniti, Elirosa; Ursini, Fulvio; Rosini, Michela; Minarini, Anna
Benextramine derivatives as probes to target human monoamine oxidases
2015 Maria Luisa Di Paolo; Andrea Milelli; Giorgio Cozza; Monica Rossetto; Michela Rosini; Anna Minarini
Beta-secretase monolithic micro-IMER (immobilized enzyme reactor) for on-line HPLC screening of quinone-bearing polyamine inhibitors.
2007 Mancini F.; Bolognesi ML.; Minarini A.; Melchiorre C.; Andrisano V.
Binding profile of the selective muscarinic receptor antagonist tripitramine
1994 Maggio R.; Barbier P.; Bolognesi M.L.; Minarini A.; Tedeschi D.; Melchiorre C.
Bovine Serum Amine Oxidase and Polyamine Analogues: Chemical Synthesis and Biological Evaluation Integrated with Molecular Docking and 3-D QSAR Studies
2022 Ragno, Rino; Minarini, Anna; Proia, Eleonora; Lorenzo, Antonini; Milelli, Andrea; Tumiatti, Vincenzo; Fiore, Marco; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Di Paolo, Maria Luisa; Agostinelli, Enzo
Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate.
2016 Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E; Lodola, A; Mor, M; Milelli, A; Minarini, A.
Cystamine-tacrine dimer: A new multi-target-directed ligand as potential therapeutic agent for Alzheimer's disease treatment.
2012 Minarini A.; Milelli A.; Tumiatti V.; Rosini M.; Simoni E.; Bolognesi M.L.; Andrisano V.; Bartolini M.; Motori E.; Angeloni C.; Hrelia S.
Cystamine-tacrine dimer: a new multi-target-directed ligand as potential therapeutic agent for Alzheimer’s disease treatment
2011 A. Minarini; A. Milelli; V. Tumiatti; E. Simoni; M. L. Bolognesi; V. Andrisano; M. Bartolini; E. Motori; C. Angeloni ; S. Hrelia; C.Melchiorre
Cytotoxicity of methoctramine and methoctramine-related polyamines.
2009 Zini M.; Passariello C.L.; Gottardi D.; Cetrullo S.; Flamigni F.; Pignatti C.; Minarini A.; Tumiatti V.; Milelli A.; Melchiorre C.; Stefanelli C.
Cytotoxicity of Methoctramine and related Spermine analogues
2007 A. Minarini; V. Tumiatti; F. Flamigni; M. Zini; C. Stefanelli
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
"Non-canonical” structures of Braf promoter as novel target in anticancer therapy | Maria Laura Greco; Marco Folini; Andrea Milelli; Anna Minarini; Claudia Sissi | 2015-01-01 | - | - | 4.03 Poster | - |
4-AMINO-2-PYRIDO-BICYCLIC PYRIMIDINES AND USE THEREOF AS MEDICAMENTS - 4 AMINO-2-PIRIDO-BICICLO PIRIMIDINE E LORO USO COME MEDICAMENTI | Marco, DE VIVO; Antonio, ORTEGA MARTINEZ JOSE; Manuel, ARENCIBIA JIMENEZ JOSE; Minarini, Anna; Cl...audia, Sissi | 2016-01-01 | - | - | 6.01 Brevetto | - |
A kinetic study of new polyamine analogs oxidized by bovine serum amine oxidase . | S Saccoccio; Minarini A; A Milelli; V Tumiatti; G Tempera; N Viceconte; R Stevanato; E Agostinelli | 2011-01-01 | - | (sine nomine) | 4.02 Riassunto (Abstract) | - |
Affinity and selectivity at M2 and M3 muscarinic receptor subtypes of cyclic and open oxygenated analogues of 4-DAMP | Tumiatti V.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R.; Bolognesi M.L. | 1992-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |
Alzheimer's disease: new approaches to drug discovery. | Bolognesi M.L.; Matera R.; Minarini A.; Rosini M.; Melchiorre C. | 2009-01-01 | CURRENT OPINION IN CHEMICAL BIOLOGY | - | 1.01 Articolo in rivista | - |
An optimized polyamine moiety boosts the potency of human type II topoisomerase poisons as quantified by comparative analysis centered on the clinical candidate F14512 | Palermo, G.; Minniti, E.; Greco, M.L.; Riccardi, L.; Simoni, E.; Convertino, M.; Marchetti, C.; R...osini, M.; Sissi, C.; Minarini, A.; De Vivo, M. | 2015-01-01 | CHEMICAL COMMUNICATIONS | - | 1.01 Articolo in rivista | 84. Chem. Comm. 2015.pdf |
Analogues of prazosin that bear a benextramine-related polyamine backbone exhibit different antagonism toward α1-adrenoreceptor subtypes | Bolognesi M.L.; Marucci G.; Angeli P.; Buccioni M.; Minarini A.; Rosini M.; Tumiatti V.; Melchior...re C. | 2001-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines | Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Sp...ampinato S.; Tumiatti V.; Melchiorre C. | 2001-01-01 | BRITISH JOURNAL OF PHARMACOLOGY | - | 1.01 Articolo in rivista | British J Pharmacology - 2009 - Budriesi - Analysis of the muscarinic receptor subtype mediating inhibition of the.pdf |
Antagonist binding profile of the split chimeric muscarinic m2-trunc/m3-tail receptor | Barbier P.; Colelli A.; Bolognesi M.L.; Minarini A.; Tumiatti V.; Corsini G.U.; Melchiorre C.; Ma...ggio R. | 1998-01-01 | EUROPEAN JOURNAL OF PHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Antidepressivi e antipsicotici | Minarini, Anna; Melchiorre, Carlo | 2015-01-01 | - | CEA- Casa Editrice Ambrosiana | 2.01 Capitolo / saggio in libro | - |
Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach | Di Paolo, Maria Luisa; Cozza, Giorgio; Milelli, Andrea; Zonta, Francesca; Sarno, Stefania; Minnit...i, Elirosa; Ursini, Fulvio; Rosini, Michela; Minarini, Anna | 2019-01-01 | THE FEBS JOURNAL | - | 1.01 Articolo in rivista | - |
Benextramine derivatives as probes to target human monoamine oxidases | Maria Luisa Di Paolo; Andrea Milelli; Giorgio Cozza; Monica Rossetto; Michela Rosini; Anna Minarini | 2015-01-01 | AMINO ACIDS | - | 1.06 Abstract in rivista | - |
Beta-secretase monolithic micro-IMER (immobilized enzyme reactor) for on-line HPLC screening of quinone-bearing polyamine inhibitors. | Mancini F.; Bolognesi ML.; Minarini A.; Melchiorre C.; Andrisano V. | 2007-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Binding profile of the selective muscarinic receptor antagonist tripitramine | Maggio R.; Barbier P.; Bolognesi M.L.; Minarini A.; Tedeschi D.; Melchiorre C. | 1994-01-01 | EUROPEAN JOURNAL OF PHARMACOLOGY-MOLECULAR PHARMACOLOGY SECTION | - | 1.01 Articolo in rivista | - |
Bovine Serum Amine Oxidase and Polyamine Analogues: Chemical Synthesis and Biological Evaluation Integrated with Molecular Docking and 3-D QSAR Studies | Ragno, Rino; Minarini, Anna; Proia, Eleonora; Lorenzo, Antonini; Milelli, Andrea; Tumiatti, Vince...nzo; Fiore, Marco; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Di Paolo, Maria Luisa; Agostinelli, Enzo | 2022-01-01 | JOURNAL OF CHEMICAL INFORMATION AND MODELING | - | 1.01 Articolo in rivista | Accepted.20220504_con link.pdf; SI JCIM 2022.pdf |
Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate. | Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E...; Lodola, A; Mor, M; Milelli, A; Minarini, A. | 2016-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Cystamine-tacrine dimer: A new multi-target-directed ligand as potential therapeutic agent for Alzheimer's disease treatment. | Minarini A.; Milelli A.; Tumiatti V.; Rosini M.; Simoni E.; Bolognesi M.L.; Andrisano V.; Bartoli...ni M.; Motori E.; Angeloni C.; Hrelia S. | 2012-01-01 | NEUROPHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Cystamine-tacrine dimer: a new multi-target-directed ligand as potential therapeutic agent for Alzheimer’s disease treatment | A. Minarini; A. Milelli; V. Tumiatti; E. Simoni; M. L. Bolognesi; V. Andrisano; M. Bartolini; E. ...Motori; C. Angeloni ; S. Hrelia; C.Melchiorre | 2011-01-01 | - | 2011 Università del Salento – Coordinamento SIBA- | 4.02 Riassunto (Abstract) | - |
Cytotoxicity of methoctramine and methoctramine-related polyamines. | Zini M.; Passariello C.L.; Gottardi D.; Cetrullo S.; Flamigni F.; Pignatti C.; Minarini A.; Tumia...tti V.; Milelli A.; Melchiorre C.; Stefanelli C. | 2009-01-01 | CHEMICO-BIOLOGICAL INTERACTIONS | - | 1.01 Articolo in rivista | - |
Cytotoxicity of Methoctramine and related Spermine analogues | A. Minarini; V. Tumiatti; F. Flamigni; M. Zini; C. Stefanelli | 2007-01-01 | - | CSU Università degli Studi di Roma La Sapienza | 4.02 Riassunto (Abstract) | - |