MINARINI, ANNA
MINARINI, ANNA
DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di Ia fascia
"Non-canonical” structures of Braf promoter as novel target in anticancer therapy
2015 Maria Laura Greco; Marco Folini; Andrea Milelli; Anna Minarini; Claudia Sissi
4-AMINO-2-PYRIDO-BICYCLIC PYRIMIDINES AND USE THEREOF AS MEDICAMENTS - 4 AMINO-2-PIRIDO-BICICLO PIRIMIDINE E LORO USO COME MEDICAMENTI
2016 Marco, DE VIVO; Antonio, ORTEGA MARTINEZ JOSE; Manuel, ARENCIBIA JIMENEZ JOSE; Minarini, Anna; Claudia, Sissi
A kinetic study of new polyamine analogs oxidized by bovine serum amine oxidase .
2011 S Saccoccio; Minarini A; A Milelli; V Tumiatti; G Tempera; N Viceconte; R Stevanato; E Agostinelli
Affinity and selectivity at M2 and M3 muscarinic receptor subtypes of cyclic and open oxygenated analogues of 4-DAMP
1992 Tumiatti V.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R.; Bolognesi M.L.
Alzheimer's disease: new approaches to drug discovery.
2009 Bolognesi M.L.; Matera R.; Minarini A.; Rosini M.; Melchiorre C.
An optimized polyamine moiety boosts the potency of human type II topoisomerase poisons as quantified by comparative analysis centered on the clinical candidate F14512
2015 Palermo, G.; Minniti, E.; Greco, M.L.; Riccardi, L.; Simoni, E.; Convertino, M.; Marchetti, C.; Rosini, M.; Sissi, C.; Minarini, A.; De Vivo, M.
Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines
2001 Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Spampinato S.; Tumiatti V.; Melchiorre C.
Antidepressivi e antipsicotici
2015 Minarini, Anna; Melchiorre, Carlo
Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach
2019 Di Paolo, Maria Luisa; Cozza, Giorgio; Milelli, Andrea; Zonta, Francesca; Sarno, Stefania; Minniti, Elirosa; Ursini, Fulvio; Rosini, Michela; Minarini, Anna
Benextramine derivatives as probes to target human monoamine oxidases
2015 Maria Luisa Di Paolo; Andrea Milelli; Giorgio Cozza; Monica Rossetto; Michela Rosini; Anna Minarini
Beta-secretase monolithic micro-IMER (immobilized enzyme reactor) for on-line HPLC screening of quinone-bearing polyamine inhibitors.
2007 Mancini F.; Bolognesi ML.; Minarini A.; Melchiorre C.; Andrisano V.
Bovine Serum Amine Oxidase and Polyamine Analogues: Chemical Synthesis and Biological Evaluation Integrated with Molecular Docking and 3-D QSAR Studies
2022 Ragno, Rino; Minarini, Anna; Proia, Eleonora; Lorenzo, Antonini; Milelli, Andrea; Tumiatti, Vincenzo; Fiore, Marco; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Di Paolo, Maria Luisa; Agostinelli, Enzo
Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate.
2016 Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E; Lodola, A; Mor, M; Milelli, A; Minarini, A.
Cystamine-tacrine dimer: A new multi-target-directed ligand as potential therapeutic agent for Alzheimer's disease treatment.
2012 Minarini A.; Milelli A.; Tumiatti V.; Rosini M.; Simoni E.; Bolognesi M.L.; Andrisano V.; Bartolini M.; Motori E.; Angeloni C.; Hrelia S.
Cystamine-tacrine dimer: a new multi-target-directed ligand as potential therapeutic agent for Alzheimer’s disease treatment
2011 A. Minarini; A. Milelli; V. Tumiatti; E. Simoni; M. L. Bolognesi; V. Andrisano; M. Bartolini; E. Motori; C. Angeloni ; S. Hrelia; C.Melchiorre
Cytotoxicity of methoctramine and methoctramine-related polyamines.
2009 Zini M.; Passariello C.L.; Gottardi D.; Cetrullo S.; Flamigni F.; Pignatti C.; Minarini A.; Tumiatti V.; Milelli A.; Melchiorre C.; Stefanelli C.
Cytotoxicity of Methoctramine and related Spermine analogues
2007 A. Minarini; V. Tumiatti; F. Flamigni; M. Zini; C. Stefanelli
Cytotoxicity of methoctramine-related polyamines
2011 V. Tumiatti; A. Minarini; A. Milelli; C. Cappadone; M. Zini; C. Stefanelli
Design and synthesis of new multitarget agents for the study of neuroinflammation in Alzheimer's disease
2021 Giambattista Marotta, Rita Maria Concetta Di Martino, Debora Russo, Ilaria Penna, Michela Rosini, Jose Antonio Ortega, Anna Minarini
Design, synthesis and biological activity of some 4-DAMP- related compounds
1995 Tumiatti V.; Santi S.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R.
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
"Non-canonical” structures of Braf promoter as novel target in anticancer therapy | Maria Laura Greco; Marco Folini; Andrea Milelli; Anna Minarini; Claudia Sissi | 2015-01-01 | - | - | 4.03 Poster | - |
4-AMINO-2-PYRIDO-BICYCLIC PYRIMIDINES AND USE THEREOF AS MEDICAMENTS - 4 AMINO-2-PIRIDO-BICICLO PIRIMIDINE E LORO USO COME MEDICAMENTI | Marco, DE VIVO; Antonio, ORTEGA MARTINEZ JOSE; Manuel, ARENCIBIA JIMENEZ JOSE; Minarini, Anna; Cl...audia, Sissi | 2016-01-01 | - | - | 6.01 Brevetto | - |
A kinetic study of new polyamine analogs oxidized by bovine serum amine oxidase . | S Saccoccio; Minarini A; A Milelli; V Tumiatti; G Tempera; N Viceconte; R Stevanato; E Agostinelli | 2011-01-01 | - | (sine nomine) | 4.02 Riassunto (Abstract) | - |
Affinity and selectivity at M2 and M3 muscarinic receptor subtypes of cyclic and open oxygenated analogues of 4-DAMP | Tumiatti V.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R.; Bolognesi M.L. | 1992-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |
Alzheimer's disease: new approaches to drug discovery. | Bolognesi M.L.; Matera R.; Minarini A.; Rosini M.; Melchiorre C. | 2009-01-01 | CURRENT OPINION IN CHEMICAL BIOLOGY | - | 1.01 Articolo in rivista | - |
An optimized polyamine moiety boosts the potency of human type II topoisomerase poisons as quantified by comparative analysis centered on the clinical candidate F14512 | Palermo, G.; Minniti, E.; Greco, M.L.; Riccardi, L.; Simoni, E.; Convertino, M.; Marchetti, C.; R...osini, M.; Sissi, C.; Minarini, A.; De Vivo, M. | 2015-01-01 | CHEMICAL COMMUNICATIONS | - | 1.01 Articolo in rivista | 84. Chem. Comm. 2015.pdf |
Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines | Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Sp...ampinato S.; Tumiatti V.; Melchiorre C. | 2001-01-01 | BRITISH JOURNAL OF PHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Antidepressivi e antipsicotici | Minarini, Anna; Melchiorre, Carlo | 2015-01-01 | - | CEA- Casa Editrice Ambrosiana | 2.01 Capitolo / saggio in libro | - |
Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach | Di Paolo, Maria Luisa; Cozza, Giorgio; Milelli, Andrea; Zonta, Francesca; Sarno, Stefania; Minnit...i, Elirosa; Ursini, Fulvio; Rosini, Michela; Minarini, Anna | 2019-01-01 | THE FEBS JOURNAL | - | 1.01 Articolo in rivista | - |
Benextramine derivatives as probes to target human monoamine oxidases | Maria Luisa Di Paolo; Andrea Milelli; Giorgio Cozza; Monica Rossetto; Michela Rosini; Anna Minarini | 2015-01-01 | AMINO ACIDS | - | 1.06 Abstract in rivista | - |
Beta-secretase monolithic micro-IMER (immobilized enzyme reactor) for on-line HPLC screening of quinone-bearing polyamine inhibitors. | Mancini F.; Bolognesi ML.; Minarini A.; Melchiorre C.; Andrisano V. | 2007-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Bovine Serum Amine Oxidase and Polyamine Analogues: Chemical Synthesis and Biological Evaluation Integrated with Molecular Docking and 3-D QSAR Studies | Ragno, Rino; Minarini, Anna; Proia, Eleonora; Lorenzo, Antonini; Milelli, Andrea; Tumiatti, Vince...nzo; Fiore, Marco; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Di Paolo, Maria Luisa; Agostinelli, Enzo | 2022-01-01 | JOURNAL OF CHEMICAL INFORMATION AND MODELING | - | 1.01 Articolo in rivista | - |
Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate. | Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E...; Lodola, A; Mor, M; Milelli, A; Minarini, A. | 2016-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Cystamine-tacrine dimer: A new multi-target-directed ligand as potential therapeutic agent for Alzheimer's disease treatment. | Minarini A.; Milelli A.; Tumiatti V.; Rosini M.; Simoni E.; Bolognesi M.L.; Andrisano V.; Bartoli...ni M.; Motori E.; Angeloni C.; Hrelia S. | 2012-01-01 | NEUROPHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Cystamine-tacrine dimer: a new multi-target-directed ligand as potential therapeutic agent for Alzheimer’s disease treatment | A. Minarini; A. Milelli; V. Tumiatti; E. Simoni; M. L. Bolognesi; V. Andrisano; M. Bartolini; E. ...Motori; C. Angeloni ; S. Hrelia; C.Melchiorre | 2011-01-01 | - | 2011 Università del Salento – Coordinamento SIBA- | 4.02 Riassunto (Abstract) | - |
Cytotoxicity of methoctramine and methoctramine-related polyamines. | Zini M.; Passariello C.L.; Gottardi D.; Cetrullo S.; Flamigni F.; Pignatti C.; Minarini A.; Tumia...tti V.; Milelli A.; Melchiorre C.; Stefanelli C. | 2009-01-01 | CHEMICO-BIOLOGICAL INTERACTIONS | - | 1.01 Articolo in rivista | - |
Cytotoxicity of Methoctramine and related Spermine analogues | A. Minarini; V. Tumiatti; F. Flamigni; M. Zini; C. Stefanelli | 2007-01-01 | - | CSU Università degli Studi di Roma La Sapienza | 4.02 Riassunto (Abstract) | - |
Cytotoxicity of methoctramine-related polyamines | V. Tumiatti; A. Minarini; A. Milelli; C. Cappadone; M. Zini; C. Stefanelli | 2011-01-01 | - | SN | 4.02 Riassunto (Abstract) | - |
Design and synthesis of new multitarget agents for the study of neuroinflammation in Alzheimer's disease | Giambattista Marotta, Rita Maria Concetta Di Martino, Debora Russo, Ilaria Penna, Michela Rosini,... Jose Antonio Ortega, Anna Minarini | 2021-01-01 | - | - | 4.03 Poster | - |
Design, synthesis and biological activity of some 4-DAMP- related compounds | Tumiatti V.; Santi S.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R. | 1995-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |