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Mostrati risultati da 41 a 60 di 155
Titolo Autore(i) Anno Periodico Editore Tipo File
Methoctramine effects on nicotinic acetylcholine receptor kinetics E. Nurowska; V. Tumiatti; A. Minarini; F. Ruzzier 2006-01-01 ACTA PHYSIOLOGICA - 4.02 Riassunto (Abstract) -
One-molecule-multiple-target strategy: a novel multifunctional molecule designed to block EGF-r and to exert pro-apoptotic effects M.L. Bolognesi;
A. Antonello;
A. Tarozzi;
M. Rosini;
A. Minarini;
V. Tumiatti; P. Hrelia;
C...
. Melchiorre.
2006-01-01 - s.n 4.02 Riassunto (Abstract) -
Recent advances in the design and synthesis of prazosin derivatives A. Minarini;
M.L. Bolognesi;
V. Tumiatti;
C. Melchiorre.
2006-01-01 EXPERT OPINION ON DRUG DISCOVERY - 1.01 Articolo in rivista -
Progress in acetylcholinesterase inhibitors for Alzheimer's disease M.L. Bolognesi; A. Minarini; V. Tumiatti; C. Melchiorre 2006-01-01 EXPERT OPINION ON THERAPEUTIC PATENTS - 1.01 Articolo in rivista -
Lipoic acid, a lead structure for multi-target-directed drugs for neurodegeneration M.L. Bolognesi; A. Minarini; V. Tumiatti; C. Melchiorre 2006-01-01 MINI-REVIEWS IN MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Cytotoxicity of Methoctramine and related Spermine analogues A. Minarini; V. Tumiatti; F. Flamigni; M. Zini; C. Stefanelli 2007-01-01 - CSU Università degli Studi di Roma La Sapienza 4.02 Riassunto (Abstract) -
Beta-secretase monolithic micro-IMER (immobilized enzyme reactor) for on-line HPLC screening of quinone-bearing polyamine inhibitors. Mancini F.; Bolognesi ML.; Minarini A.; Melchiorre C.; Andrisano V. 2007-01-01 - s.n 4.02 Riassunto (Abstract) -
Progettazione e sintesi di derivati poliamminici per il trattamento della malattia di Alzheimer V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; V. Andrisano; M. Bartolini; F. ...Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre 2007-01-01 - s.n 4.01 Contributo in Atti di convegno -
Memoquine derivatives as potent inhibitors of AChE-induced amyloid-beta aggregation Bolognesi ML; Cavalli A; Andrisano V; Bartolini M; Minarini A; Melchiorre C 2007-01-01 - s.n 4.01 Contributo in Atti di convegno -
Quinone-bearing polyamines are AChE inhibitors endowed with multifunctional properties M.L. Bolognesi; R. Banzi; A. Cavalli; A. Minarini; M. Bartolini; V. Andrisano; M. Recanatini; C. ...Melchiorre 2007-01-01 - s.n 4.02 Riassunto (Abstract) -
Recent advances in alpha1-adrenoreceptor antagonists as pharmacological tools and therapeutic agents. Rosini M; Bolognesi ML; Giardina D; Minarini A; Tumiatti V; Melchiorre C. 2007-01-01 CURRENT TOPICS IN MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
New quinazoline compounds as non-peptidomimetic BACE-1 inhibitors in the treatment of Alzheimer's disease Matera R; Minarini A; Rosini M; Andrisano V; Mancini F; Melchiorre C. 2007-01-01 - s.n 4.01 Contributo in Atti di convegno -
Novel Class of Quinone-Bearing Polyamines as Multi-Target-Directed Ligands To Combat Alzheimer's Disease Bolognesi ML; Banzi R; Bartolini M; Cavalli A; Tarozzi A; Andrisano V; Minarini A; Rosini M; Tumi...atti V; Bergamini C; Fato R; Lenaz G; Hrelia P; Cattaneo A; Recanatini M; Melchiorre C. 2007-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Structure-activity relationships of methoctramine-related polyamines as muscarinic antagonist: Effect of replacing the inner polymethylene chain with cyclic moieties V. Tumiatti; A. Minarini; A. Milelli; M. Rosini; M. Buccioni; G. Marucci; C. Ghelardini; C. Bellu...cci; C. Melchiorre 2007-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
From dual binding site acetylcholinesterase inhibitors to multi-target-directed ligands (MTDLs): a step forward in the treatment of Alzheimer's disease M. L. Bolognesi; A. Minarini; M. Rosini; V. Tumiatti; C. Melchiorre 2008-01-01 MINI-REVIEWS IN MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Structure-Activity Relationships of Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone. 4. Futher Investigation on the Inner Spacer. V. Tumiatti; A. Milelli; A. Minarini; M. Rosini; M. L. Bolognesi; M. Micco; V. Andrisano; M. Bart...olini; F. Mancini; M. Recanatini; A. Cavalli; C. Melchiorre 2008-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Multi-target-Directed Ligands To Combat Neurodegenerative Diseases A. Cavalli; M. L. Bolognesi; A. Minarini; M.Rosini; V. Tumiatti; M. Recanatini; C. Melchiorre 2008-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Structure-Activity Relationships of New Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; M. Micco; V. Andrisano; M. Bart...olini; F. Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre 2008-01-01 - s.n 4.02 Riassunto (Abstract) -
Synthesis of monomeric derivatives to probe Memoquin bivalent interactions ML. Bolognesi; A. Minarini; M. Bartolini; A. Cavalli; F. Mancini; V. Andrisano; M. Rosini; V. Tum...iatti; C. Melchiorre 2008-01-01 - s.n 4.02 Riassunto (Abstract) -
Design, synthesis, and biological evaluation of pirenzepine analogs bearing a 1,2-cyclohexanediamine and a perhydroquinoxaline units in exchange for the piperazine ring as antimuscarinics A. Minarini; G. Marucci; C. Bellucci; G. Giorgi; V. Tumiatti; M. L. Bolognesi; R. Matera; M. Rosi...ni; C. Melchiorre 2008-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Mostrati risultati da 41 a 60 di 155
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