MILELLI, ANDREA

MILELLI, ANDREA  

DIPARTIMENTO DI SCIENZE PER LA QUALITA' DELLA VITA  

Docenti di ruolo di IIa fascia  

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Risultati 1 - 20 di 86 (tempo di esecuzione: 0.04 secondi).
Titolo Autore(i) Anno Periodico Editore Tipo File
First in Class Dual Non-ATP-Competitive Glycogen Synthase Kinase 3β/Histone Deacetylase Inhibitors as a Potential Therapeutic to Treat Alzheimer’s Disease Santini A.; Tassinari E.; Poeta E.; Loi M.; Ciani E.; Trazzi S.; Piccarducci R.; Daniele S.; Mart...ini C.; Pagliarani B.; Tarozzi A.; Bersani M.; Spyrakis F.; Danková D.; Olsen C.A.; Soldati R.; Tumiatti V.; Montanari S.; De Simone A.; Milelli A. 2024-01-01 ACS CHEMICAL NEUROSCIENCE - 1.01 Articolo in rivista acs-cn.pdf
Integrating a quinone substructure into histone deacetylase inhibitors to cope with Alzheimer's disease and cancer Guardigni M.; Greco G.; Poeta E.; Santini A.; Tassinari E.; Bergamini C.; Zalambani C.; De Simone... A.; Andrisano V.; Uliassi E.; Monti B.; Bolognesi M.L.; Fimognari C.; Milelli A. 2024-01-01 RSC MEDICINAL CHEMISTRY - 1.01 Articolo in rivista d4md00175c.pdfd4md00175c1.pdf
From Monoamine Oxidase Inhibition to Antiproliferative Activity: New Biological Perspectives for Polyamine Analogs Nordio G.; Piazzola F.; Cozza G.; Rossetto M.; Cervelli M.; Minarini A.; Basagni F.; Tassinari E....; Dalla Via L.; Milelli A.; Di Paolo M.L. 2023-01-01 MOLECULES - 1.01 Articolo in rivista molecules-28-06329-v3.pdfmolecules-2562834-supplementary.pdf
PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease Guardigni M.; Pruccoli L.; Santini A.; Simone A.D.; Bersani M.; Spyrakis F.; Frabetti F.; Uliassi... E.; Andrisano V.; Pagliarani B.; Fernández-Gómez P.; Palomo V.; Bolognesi M.L.; Tarozzi A.; Milelli A. 2023-01-01 ACS CHEMICAL NEUROSCIENCE - 1.01 Articolo in rivista acschemneuro.3c00096.pdf
Targeted Protein Degradation for Infectious Diseases: from Basic Biology to Drug Discovery Rocío Marisol Espinoza Chávez; Salerno A.; Liuzzi A.; Ilari A.; Milelli A.; Uliassi E.; Bolognesi... M.L. 2023-01-01 ACS BIO & MED CHEM AU - 1.01 Articolo in rivista acsbiomedchemau.2c00063.pdf
Asymmetric Organocatalysis: A Survival Guide to Medicinal Chemists EFRAIM REYES; Liher Prieto; ANDREA MILELLI 2022-01-01 MOLECULES - 1.01 Articolo in rivista molecules-28-00271 (1).pdf
Bovine Serum Amine Oxidase and Polyamine Analogues: Chemical Synthesis and Biological Evaluation Integrated with Molecular Docking and 3-D QSAR Studies Ragno, Rino; Minarini, Anna; Proia, Eleonora; Lorenzo, Antonini; Milelli, Andrea; Tumiatti, Vince...nzo; Fiore, Marco; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Di Paolo, Maria Luisa; Agostinelli, Enzo 2022-01-01 JOURNAL OF CHEMICAL INFORMATION AND MODELING - 1.01 Articolo in rivista Accepted.20220504_con link.pdfSI JCIM 2022.pdfci2c00559_si_002.xlsx
Enriching Proteolysis Targeting Chimeras with a Second Modality: When Two Are Better Than One Salerno, Alessandra; Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Testi, Eleonora; Gua...rdigni, Melissa; Roberti, Marinella; Milelli, Andrea; Bolognesi, Maria Laura 2022-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista acs.jmedchem.2c00302.pdf
PROTAC-INDUCED GLYCOGEN SYNTHASE KINASE 3B DEGRADATION Santini, A.; Pruccoli, L.; Guardigni, M.; De Simone, A.; Spyrakis, F.; Frabetti, F.; Andrisano, V....; Bolognesi, M. L.; Tarozzi, A.; Milelli, A. 2022-01-01 - - 4.03 Poster -
Glycogen Synthase Kinase 3β: A New Gold Rush in Anti-Alzheimer’s Disease Multitarget Drug Discovery? Angela De Simone,
Vincenzo Tumiatti,
VIncenza Andrisano,
Andrea Milelli
2021-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista acs.jmedchem.0c00931.pdf
Treatment with a GSK-3β/HDAC Dual Inhibitor Restores Neuronal Survival and Maturation in an In Vitro and In Vivo Model of CDKL5 Deficiency Disorder Loi, Manuela; Gennaccaro, Laura; Fuchs, Claudia; Trazzi, Stefania; Medici, Giorgio; Galvani, Gius...eppe; Mottolese, Nicola; Tassinari, Marianna; Giorgini, Roberto Rimondini; Milelli, Andrea; Ciani, Elisabetta 2021-01-01 INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES - 1.01 Articolo in rivista Loi et al 2021.pdfijms-1212824-supplementary.pdf
Targeting topoisomerase II with trypthantrin derivatives: Discovery of 7-((2-(dimethylamino)ethyl)amino)indolo[2,1-b]quinazoline-6,12-dione as an antiproliferative agent and to treat cancer Catanzaro E.; Betari N.; Arencibia J.M.; Montanari S.; Sissi C.; De Simone A.; Vassura I.; Santin...i A.; Andrisano V.; Tumiatti V.; De Vivo M.; Krysko D.V.; Rocchi M.B.L.; Fimognari C.; Milelli A. 2020-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista Draft_revised_Milelli no copertina.pdf
Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach Di Paolo, Maria Luisa; Cozza, Giorgio; Milelli, Andrea; Zonta, Francesca; Sarno, Stefania; Minnit...i, Elirosa; Ursini, Fulvio; Rosini, Michela; Minarini, Anna 2019-01-01 THE FEBS JOURNAL - 1.01 Articolo in rivista -
COMPOSTI ISOTIOCIANATI E ISOSELENCIANATI Fimognari C, Sestili P, Milelli A 2019-01-01 - - 6.01 Brevetto -
Correction: Discovery of the First-in-Class GSK-3β/HDAC Dual Inhibitor as Disease-Modifying Agent to Combat Alzheimer's Disease (ACS Medicinal Chemistry Letters (2019) 10: 4 (469−474) DOI: 10.1021/acsmedchemlett.8b00507) De Simone A.; La Pietra V.; Betari N.; Petragnani N.; Conte M.; Daniele S.; Pietrobono D.; Martin...i C.; Petralla S.; Casadei R.; Davani L.; Frabetti F.; Russomanno P.; Novellino E.; Montanari S.; Tumiatti V.; Ballerini P.; Sarno F.; Nebbioso A.; Altucci L.; Monti B.; Andrisano V.; Milelli A. 2019-01-01 ACS MEDICINAL CHEMISTRY LETTERS - 1.01 Articolo in rivista -
Deuterium Incorporation Protects Cells from Oxidative Damage Sestili P.; Brigotti M.; Calcabrini C.; Turrini E.; Arfilli V.; Carnicelli D.; Lucarini M.; Mazza...nti A.; Milelli A.; Righi V.; Fimognari C. 2019-01-01 OXIDATIVE MEDICINE AND CELLULAR LONGEVITY - 1.01 Articolo in rivista SestiliEtAl_2019_OxidativeMedCellLong.pdf
Discovery of the First-in-Class GSK-3β/HDAC Dual Inhibitor as Disease-Modifying Agent To Combat Alzheimer's Disease. De Simone A, La Pietra V, Betari N, Petragnani N, Conte M, Daniele S, Pietrobono D, Martini C, Pe...tralla S, Casadei R, Davani L, Frabetti F, Russomanno P, Novellino E, Montanari S, Tumiatti V, Ballerini P, Sarno F, Nebbioso A, Altucci L, Monti B, Andrisano V, Milelli A. 2019-01-01 ACS MEDICINAL CHEMISTRY LETTERS - 1.01 Articolo in rivista AM11585-685764.pdf
Distinct biological responses of metastatic castration resistant prostate cancer cells upon exposure to G-quadruplex interacting naphthalenediimide derivatives Recagni M.; Greco M.L.; Milelli A.; Minarini A.; Zaffaroni N.; Folini M.; Sissi C. 2019-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Exploring the activity of polyamine analogues on polyamine and spermine oxidase: methoctramine, a potent and selective inhibitor of polyamine oxidase Di Paolo, Maria Luisa; Cervelli, Manuela; Mariottini, Paolo; Leonetti, Alessia; Polticelli, Fabio...; Rosini, Michela; Milelli, Andrea; Basagni, Filippo; Venerando, Rina; Agostinelli, Enzo; Minarini, Anna 2019-01-01 JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY - 1.01 Articolo in rivista 99. J.Enz. Inhib. Med Chem 2019.pdf
Histone Deacetylase Inhibitors as Multitarget Ligands: New Players in Alzheimer's Disease Drug Discovery? De Simone Angela; Milelli Andrea 2019-01-01 CHEMMEDCHEM - 1.01 Articolo in rivista -