MILELLI, ANDREA
MILELLI, ANDREA
DIPARTIMENTO DI SCIENZE PER LA QUALITA' DELLA VITA
Docenti di ruolo di IIa fascia
"Non-canonical” structures of Braf promoter as novel target in anticancer therapy
2015 Maria Laura Greco; Marco Folini; Andrea Milelli; Anna Minarini; Claudia Sissi
- Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors.
2016 Angela, De Simone; Andrea, Milelli; Marina, Naldi; Vincenza, Andrisano
A kinetic study of new polyamine analogs oxidized by bovine serum amine oxidase .
2011 S Saccoccio; Minarini A; A Milelli; V Tumiatti; G Tempera; N Viceconte; R Stevanato; E Agostinelli
Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors.
2016 De Simone, A; Milelli, A; Naldi, M; Andrisano, V.
Application of an ESI-QTOF method for the detailed characterization of GSK-3β inhibitors
2017 De Simone, Angela; Fiori, Jessica; Naldi, Marina; D'Urzo, Annalisa; Tumiatti, Vincenzo; Milelli, Andrea; Andrisano, Vincenza
Application of ESI-MS method for detailed characterization of GSK-3β inhibitors by monitoring GSM peptide phosphorylation.Angelini Farmaceutici.
2016 De Simone, A; Naldi, M; Milelli, A; Andrisano, V
Asymmetric 1,4-addition of oxazolones to nitroalkenes by bifunctional cinchona alkaloid thiourea organocatalysts: synthesis of alpha,alpha-disubstituted alpha-amino acids.
2008 ALEMÁN J; MILELLI A; CABRERA S; REYES E; JØRGENSEN KA
Asymmetric Organocatalysis: A Survival Guide to Medicinal Chemists
2022 EFRAIM REYES; Liher Prieto; ANDREA MILELLI
Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach
2019 Di Paolo, Maria Luisa; Cozza, Giorgio; Milelli, Andrea; Zonta, Francesca; Sarno, Stefania; Minniti, Elirosa; Ursini, Fulvio; Rosini, Michela; Minarini, Anna
Benextramine derivatives as probes to target human monoamine oxidases
2015 Maria Luisa Di Paolo; Andrea Milelli; Giorgio Cozza; Monica Rossetto; Michela Rosini; Anna Minarini
Bis(7)-tacrine Derivatives as Multitarget-Directed Ligands: Focus on Anticholinesterase and Antiamyloid Activities
2010 Bolognesi ML; Bartolini M ; Mancini F ; Chiriano G ; Ceccarini L; Rosini M; Milelli A; Tumiatti V; Andrisano V; Melchiorre C
Bovine Serum Amine Oxidase and Polyamine Analogues: Chemical Synthesis and Biological Evaluation Integrated with Molecular Docking and 3-D QSAR Studies
2022 Ragno, Rino; Minarini, Anna; Proia, Eleonora; Lorenzo, Antonini; Milelli, Andrea; Tumiatti, Vincenzo; Fiore, Marco; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Di Paolo, Maria Luisa; Agostinelli, Enzo
Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate.
2016 Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E; Lodola, A; Mor, M; Milelli, A; Minarini, A.
COMPOSTI ISOTIOCIANATI E ISOSELENCIANATI
2019 Fimognari C, Sestili P, Milelli A
Correction: Discovery of the First-in-Class GSK-3β/HDAC Dual Inhibitor as Disease-Modifying Agent to Combat Alzheimer's Disease (ACS Medicinal Chemistry Letters (2019) 10: 4 (469−474) DOI: 10.1021/acsmedchemlett.8b00507)
2019 De Simone A.; La Pietra V.; Betari N.; Petragnani N.; Conte M.; Daniele S.; Pietrobono D.; Martini C.; Petralla S.; Casadei R.; Davani L.; Frabetti F.; Russomanno P.; Novellino E.; Montanari S.; Tumiatti V.; Ballerini P.; Sarno F.; Nebbioso A.; Altucci L.; Monti B.; Andrisano V.; Milelli A.
Cystamine-tacrine dimer: A new multi-target-directed ligand as potential therapeutic agent for Alzheimer's disease treatment.
2012 Minarini A.; Milelli A.; Tumiatti V.; Rosini M.; Simoni E.; Bolognesi M.L.; Andrisano V.; Bartolini M.; Motori E.; Angeloni C.; Hrelia S.
Cystamine-tacrine dimer: a new multi-target-directed ligand as potential therapeutic agent for Alzheimer’s disease treatment
2011 A. Minarini; A. Milelli; V. Tumiatti; E. Simoni; M. L. Bolognesi; V. Andrisano; M. Bartolini; E. Motori; C. Angeloni ; S. Hrelia; C.Melchiorre
Cytotoxicity of methoctramine and methoctramine-related polyamines.
2009 Zini M.; Passariello C.L.; Gottardi D.; Cetrullo S.; Flamigni F.; Pignatti C.; Minarini A.; Tumiatti V.; Milelli A.; Melchiorre C.; Stefanelli C.
Cytotoxicity of methoctramine-related polyamines
2011 V. Tumiatti; A. Minarini; A. Milelli; C. Cappadone; M. Zini; C. Stefanelli
Design, synthesis and biological evaluation of new naphtalene diimides bearing isothiocyanate functionality
2012 A. Minarini; A. Milelli; V. Tumiatti; L. Ferruzzi; M. R. Marton; E. Turrini; P. Hrelia; C. Fimognari
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
"Non-canonical” structures of Braf promoter as novel target in anticancer therapy | Maria Laura Greco; Marco Folini; Andrea Milelli; Anna Minarini; Claudia Sissi | 2015-01-01 | - | - | 4.03 Poster | - |
- Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors. | Angela, De Simone; Andrea, Milelli; Marina, Naldi; Vincenza, Andrisano | 2016-01-01 | - | - | 4.03 Poster | - |
A kinetic study of new polyamine analogs oxidized by bovine serum amine oxidase . | S Saccoccio; Minarini A; A Milelli; V Tumiatti; G Tempera; N Viceconte; R Stevanato; E Agostinelli | 2011-01-01 | - | (sine nomine) | 4.02 Riassunto (Abstract) | - |
Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors. | De Simone, A; Milelli, A; Naldi, M; Andrisano, V. | 2016-01-01 | - | - | 4.03 Poster | - |
Application of an ESI-QTOF method for the detailed characterization of GSK-3β inhibitors | De Simone, Angela; Fiori, Jessica; Naldi, Marina; D'Urzo, Annalisa; Tumiatti, Vincenzo; Milelli, ...Andrea; Andrisano, Vincenza | 2017-01-01 | JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS | - | 1.01 Articolo in rivista | - |
Application of ESI-MS method for detailed characterization of GSK-3β inhibitors by monitoring GSM peptide phosphorylation.Angelini Farmaceutici. | De Simone, A; Naldi, M; Milelli, A; Andrisano, V | 2016-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
Asymmetric 1,4-addition of oxazolones to nitroalkenes by bifunctional cinchona alkaloid thiourea organocatalysts: synthesis of alpha,alpha-disubstituted alpha-amino acids. | ALEMÁN J; MILELLI A; CABRERA S; REYES E; JØRGENSEN KA | 2008-01-01 | CHEMISTRY-A EUROPEAN JOURNAL | - | 1.01 Articolo in rivista | - |
Asymmetric Organocatalysis: A Survival Guide to Medicinal Chemists | EFRAIM REYES; Liher Prieto; ANDREA MILELLI | 2022-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-28-00271 (1).pdf |
Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach | Di Paolo, Maria Luisa; Cozza, Giorgio; Milelli, Andrea; Zonta, Francesca; Sarno, Stefania; Minnit...i, Elirosa; Ursini, Fulvio; Rosini, Michela; Minarini, Anna | 2019-01-01 | THE FEBS JOURNAL | - | 1.01 Articolo in rivista | - |
Benextramine derivatives as probes to target human monoamine oxidases | Maria Luisa Di Paolo; Andrea Milelli; Giorgio Cozza; Monica Rossetto; Michela Rosini; Anna Minarini | 2015-01-01 | AMINO ACIDS | - | 1.06 Abstract in rivista | - |
Bis(7)-tacrine Derivatives as Multitarget-Directed Ligands: Focus on Anticholinesterase and Antiamyloid Activities | Bolognesi ML; Bartolini M ; Mancini F ; Chiriano G ; Ceccarini L; Rosini M; Milelli A; Tumiatti V...; Andrisano V; Melchiorre C | 2010-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
Bovine Serum Amine Oxidase and Polyamine Analogues: Chemical Synthesis and Biological Evaluation Integrated with Molecular Docking and 3-D QSAR Studies | Ragno, Rino; Minarini, Anna; Proia, Eleonora; Lorenzo, Antonini; Milelli, Andrea; Tumiatti, Vince...nzo; Fiore, Marco; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Di Paolo, Maria Luisa; Agostinelli, Enzo | 2022-01-01 | JOURNAL OF CHEMICAL INFORMATION AND MODELING | - | 1.01 Articolo in rivista | - |
Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate. | Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E...; Lodola, A; Mor, M; Milelli, A; Minarini, A. | 2016-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
COMPOSTI ISOTIOCIANATI E ISOSELENCIANATI | Fimognari C, Sestili P, Milelli A | 2019-01-01 | - | - | 6.01 Brevetto | - |
Correction: Discovery of the First-in-Class GSK-3β/HDAC Dual Inhibitor as Disease-Modifying Agent to Combat Alzheimer's Disease (ACS Medicinal Chemistry Letters (2019) 10: 4 (469−474) DOI: 10.1021/acsmedchemlett.8b00507) | De Simone A.; La Pietra V.; Betari N.; Petragnani N.; Conte M.; Daniele S.; Pietrobono D.; Martin...i C.; Petralla S.; Casadei R.; Davani L.; Frabetti F.; Russomanno P.; Novellino E.; Montanari S.; Tumiatti V.; Ballerini P.; Sarno F.; Nebbioso A.; Altucci L.; Monti B.; Andrisano V.; Milelli A. | 2019-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
Cystamine-tacrine dimer: A new multi-target-directed ligand as potential therapeutic agent for Alzheimer's disease treatment. | Minarini A.; Milelli A.; Tumiatti V.; Rosini M.; Simoni E.; Bolognesi M.L.; Andrisano V.; Bartoli...ni M.; Motori E.; Angeloni C.; Hrelia S. | 2012-01-01 | NEUROPHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Cystamine-tacrine dimer: a new multi-target-directed ligand as potential therapeutic agent for Alzheimer’s disease treatment | A. Minarini; A. Milelli; V. Tumiatti; E. Simoni; M. L. Bolognesi; V. Andrisano; M. Bartolini; E. ...Motori; C. Angeloni ; S. Hrelia; C.Melchiorre | 2011-01-01 | - | 2011 Università del Salento – Coordinamento SIBA- | 4.02 Riassunto (Abstract) | - |
Cytotoxicity of methoctramine and methoctramine-related polyamines. | Zini M.; Passariello C.L.; Gottardi D.; Cetrullo S.; Flamigni F.; Pignatti C.; Minarini A.; Tumia...tti V.; Milelli A.; Melchiorre C.; Stefanelli C. | 2009-01-01 | CHEMICO-BIOLOGICAL INTERACTIONS | - | 1.01 Articolo in rivista | - |
Cytotoxicity of methoctramine-related polyamines | V. Tumiatti; A. Minarini; A. Milelli; C. Cappadone; M. Zini; C. Stefanelli | 2011-01-01 | - | SN | 4.02 Riassunto (Abstract) | - |
Design, synthesis and biological evaluation of new naphtalene diimides bearing isothiocyanate functionality | A. Minarini; A. Milelli; V. Tumiatti; L. Ferruzzi; M. R. Marton; E. Turrini; P. Hrelia; C. Fimognari | 2012-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |