CRIS Current Research Information System

MILELLI, ANDREA

MILELLI, ANDREA  

FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE  

Docenti di ruolo di IIa fascia  

Mostra records
Risultati 1 - 20 di 92 (tempo di esecuzione: 0.023 secondi).
Titolo Autore(i) Anno Periodico Editore Tipo File
AR-A014418-based dual Glycogen Synthase Kinase 3β/Histone Deacetylase inhibitors as potential therapeutics for Alzheimer's disease Santini, Alan; Tassinari, Elisa; Altomare, Alessandra; Loi, Manuela; Ciani, Elisabetta; Trazzi, S...tefania; Piccarducci, Rebecca; Daniele, Simona; Martini, Claudia; Pagliarani, Barbara; Tarozzi, Andrea; Bersani, Matteo; Spyrakis, Francesca; Danková, Daniela; Poeta, Eleonora; Raimondi, Simone; Davani, Lara; Aldini, Giancarlo; Andrisano, Vincenza; De Simone, Angela; Milelli, Andrea 2025-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista AR-A014418-based dual Glycogen Synthase Kinase 3β_Histone Deacetylase inhibitors as potential therapeutics for Alzheimer_s disease.pdf; 1-s2.0-S0223523425006038-mmc1.docx
Design, synthesis and pharmacological evaluation of multitarget GPR40 agonists/HDAC6 inhibitors for Alzheimer's disease Pinheiro, P. D. S. M.; De Chirico, F.; Loi, M.; Trazzi, S.; Ciani, E.; Rodrigues, D. A.; Alves, M.... A.; Lima, L. M.; Milelli, A.; Monti, B.; Manssour Fraga, C. A.; Bolognesi, M. L. 2025-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Leveraging targeted kinase degradation as a novel therapeutic strategy for Alzheimer's disease Tassinari, Elisa; Milelli, Andrea 2025-01-01 RSC MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Targeting Tau Protein with Proximity Inducing Modulators: A New Frontier to Combat Tauopathies Uliassi, E.; Bolognesi, M. L.; Milelli, A. 2025-01-01 ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE - 1.01 Articolo in rivista DraftRev_Clean.pdf
Topoisomerase II inhibitors in oncology: an updated patent review (2016-present) Turrini, Eleonora; Maffei, Francesca; Milelli, Andrea; Fimognari, Carmela 2025-01-01 EXPERT OPINION ON THERAPEUTIC PATENTS - 1.01 Articolo in rivista Expert Opinion on Therapeutic patents_topo II inhibitors_revised.pdf
First in Class Dual Non-ATP-Competitive Glycogen Synthase Kinase 3β/Histone Deacetylase Inhibitors as a Potential Therapeutic to Treat Alzheimer’s Disease Santini, A.; Tassinari, E.; Poeta, E.; Loi, M.; Ciani, E.; Trazzi, S.; Piccarducci, R.; Daniele, ...S.; Martini, C.; Pagliarani, B.; Tarozzi, A.; Bersani, M.; Spyrakis, F.; Danková, D.; Olsen, C. A.; Soldati, R.; Tumiatti, V.; Montanari, S.; De Simone, A.; Milelli, A. 2024-01-01 ACS CHEMICAL NEUROSCIENCE - 1.01 Articolo in rivista acs-cn.pdf
Integrating a quinone substructure into histone deacetylase inhibitors to cope with Alzheimer's disease and cancer Guardigni M.; Greco G.; Poeta E.; Santini A.; Tassinari E.; Bergamini C.; Zalambani C.; De Simone... A.; Andrisano V.; Uliassi E.; Monti B.; Bolognesi M.L.; Fimognari C.; Milelli A. 2024-01-01 RSC MEDICINAL CHEMISTRY - 1.01 Articolo in rivista d4md00175c.pdf; d4md00175c1.pdf
New rhodol-sulforaphane conjugates as innovative isothiocyanate-based cytotoxic agents for cancer cells Milelli, A.; Catanzaro, E.; Greco, G.; Calcabrini, C.; Turrini, E.; Maffei, F.; Burattini, S.; Gu...ardigni, M.; Sissi, C.; Schnekenburger, M.; Diederich, M.; Sestili, P.; Fimognari, C. 2024-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista MG_paper Eur J Med Chem_Revised_UNmarked.pdf
From Monoamine Oxidase Inhibition to Antiproliferative Activity: New Biological Perspectives for Polyamine Analogs Nordio G.; Piazzola F.; Cozza G.; Rossetto M.; Cervelli M.; Minarini A.; Basagni F.; Tassinari E....; Dalla Via L.; Milelli A.; Di Paolo M.L. 2023-01-01 MOLECULES - 1.01 Articolo in rivista molecules-28-06329-v3.pdf; molecules-2562834-supplementary.pdf
PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease Guardigni M.; Pruccoli L.; Santini A.; Simone A.D.; Bersani M.; Spyrakis F.; Frabetti F.; Uliassi... E.; Andrisano V.; Pagliarani B.; Fernández-Gómez P.; Palomo V.; Bolognesi M.L.; Tarozzi A.; Milelli A. 2023-01-01 ACS CHEMICAL NEUROSCIENCE - 1.01 Articolo in rivista acschemneuro.3c00096.pdf
Targeted Protein Degradation for Infectious Diseases: from Basic Biology to Drug Discovery Rocío Marisol Espinoza Chávez; Salerno A.; Liuzzi A.; Ilari A.; Milelli A.; Uliassi E.; Bolognesi... M.L. 2023-01-01 ACS BIO & MED CHEM AU - 1.01 Articolo in rivista acsbiomedchemau.2c00063.pdf
Asymmetric Organocatalysis: A Survival Guide to Medicinal Chemists EFRAIM REYES; Liher Prieto; ANDREA MILELLI 2022-01-01 MOLECULES - 1.01 Articolo in rivista molecules-28-00271 (1).pdf
Bovine Serum Amine Oxidase and Polyamine Analogues: Chemical Synthesis and Biological Evaluation Integrated with Molecular Docking and 3-D QSAR Studies Ragno, Rino; Minarini, Anna; Proia, Eleonora; Lorenzo, Antonini; Milelli, Andrea; Tumiatti, Vince...nzo; Fiore, Marco; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Di Paolo, Maria Luisa; Agostinelli, Enzo 2022-01-01 JOURNAL OF CHEMICAL INFORMATION AND MODELING - 1.01 Articolo in rivista Accepted.20220504_con link.pdf; SI JCIM 2022.pdf; ci2c00559_si_002.xlsx
Enriching Proteolysis Targeting Chimeras with a Second Modality: When Two Are Better Than One Salerno, Alessandra; Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Testi, Eleonora; Gua...rdigni, Melissa; Roberti, Marinella; Milelli, Andrea; Bolognesi, Maria Laura 2022-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista acs.jmedchem.2c00302.pdf
PROTAC-INDUCED GLYCOGEN SYNTHASE KINASE 3B DEGRADATION Santini, A.; Pruccoli, L.; Guardigni, M.; De Simone, A.; Spyrakis, F.; Frabetti, F.; Andrisano, V....; Bolognesi, M. L.; Tarozzi, A.; Milelli, A. 2022-01-01 - - 4.03 Poster -
Glycogen Synthase Kinase 3β: A New Gold Rush in Anti-Alzheimer’s Disease Multitarget Drug Discovery? Angela De Simone,
Vincenzo Tumiatti,
VIncenza Andrisano,
Andrea Milelli 		2021-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista acs.jmedchem.0c00931.pdf
Treatment with a GSK-3β/HDAC Dual Inhibitor Restores Neuronal Survival and Maturation in an In Vitro and In Vivo Model of CDKL5 Deficiency Disorder Loi, Manuela; Gennaccaro, Laura; Fuchs, Claudia; Trazzi, Stefania; Medici, Giorgio; Galvani, Gius...eppe; Mottolese, Nicola; Tassinari, Marianna; Giorgini, Roberto Rimondini; Milelli, Andrea; Ciani, Elisabetta 2021-01-01 INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES - 1.01 Articolo in rivista Loi et al 2021.pdf; ijms-1212824-supplementary.pdf
Targeting topoisomerase II with trypthantrin derivatives: Discovery of 7-((2-(dimethylamino)ethyl)amino)indolo[2,1-b]quinazoline-6,12-dione as an antiproliferative agent and to treat cancer Catanzaro E.; Betari N.; Arencibia J.M.; Montanari S.; Sissi C.; De Simone A.; Vassura I.; Santin...i A.; Andrisano V.; Tumiatti V.; De Vivo M.; Krysko D.V.; Rocchi M.B.L.; Fimognari C.; Milelli A. 2020-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista Draft_revised_Milelli no copertina.pdf
Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach Di Paolo, Maria Luisa; Cozza, Giorgio; Milelli, Andrea; Zonta, Francesca; Sarno, Stefania; Minnit...i, Elirosa; Ursini, Fulvio; Rosini, Michela; Minarini, Anna 2019-01-01 THE FEBS JOURNAL - 1.01 Articolo in rivista -
COMPOSTI ISOTIOCIANATI E ISOSELENCIANATI Fimognari, C; Sestili, P; Milelli, A 2019-01-01 - - 6.01 Brevetto -