BAGNOLINI, GRETA

BAGNOLINI, GRETA  

FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE  

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Risultati 1 - 20 di 25 (tempo di esecuzione: 0.005 secondi).
Titolo Autore(i) Anno Periodico Editore Tipo File
Design and synthesis of small molecules targeting pre-miRNA21 toward the development of ribonuclease targeting chimeras (RIBOTACs) to regulate the oncogenic miRNA21 Sdei, F.; Bagnolini, G.; Falchi, F.; Sosic, A.; Fabbian, S.; Duca, M.; Bolognesi, M. L. 2025-01-01 - - 4.01 Contributo in Atti di convegno -
Investigating synthetic lethality and PARP inhibitor resistance in pancreatic cancer through enantiomer differential activity Masi, Mirco; Poppi, Laura; Previtali, Viola; Nelson, Shannon R; Wynne, Kieran; Varignani, Giulia;... espandi Falchi, Federico; Veronesi, Marina; Albanesi, Ennio; Tedesco, Daniele; De Franco, Francesca; Ciamarone, Andrea; Myers, Samuel H; Ortega, Jose Antonio; Bagnolini, Greta; Ferrandi, Giovanni; Farabegoli, Fulvia; Tirelli, Nicola; Di Stefano, Giuseppina; Oliviero, Giorgio; Walsh, Naomi; Roberti, Marinella; Girotto, Stefania; Cavalli, Andrea 2025-01-01 CELL DEATH DISCOVERY - 1.01 Articolo in rivista Masi_et_al-2025-Cell_Death_Discovery.pdf41420_2025_2382_MOESM3_ESM.xlsx41420_2025_2382_MOESM2_ESM.pdf41420_2025_2382_MOESM1_ESM.docx
A journey through targeting BRCA2-RAD51 protein-protein interaction to establish synthetic lethality as paradigm for anticancer drug discovery Bagnolini G., Poppi L., Previtali V., Ferrandi G., Rinaldi F., Girotto S., Hirsch A.K.H., Roberti... espandi M., Cavalli A. 2024-01-01 - - 4.01 Contributo in Atti di convegno -
Design and synthesis of RAD51-BRCA2 disruptors to inhibit homologous recombination and achieve synthetic lethality in pancreatic cancer cells Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Previtali, Viola; Roberti, Marinella; Cavalli... espandi, Andrea 2024-01-01 - - 4.03 Poster -
Design and synthesis of RAD51-BRCA2 protein-protein interaction disruptors to trigger synthetic lethality with Olaparib in pancreatic cancer cells Ferrandi, Giovanni; Poppi, Laura; Bagnolini, Greta; Falchi, Federico; Previtali, Viola; Girotto, ... espandiStefania; Roberti, Marinella; Cavalli, Andrea 2024-01-01 - - 4.03 Poster -
Design and synthesis of small molecules binders of pre-miRNA21 toward the regulation of oncogenic miRNA21 Sdei, Federico; Bagnolini, Greta; Ghezzo, M.; Sosic, Alice; Sissi, Claudia; Bolognesi, MARIA LAURA 2024-01-01 - - 4.03 Poster -
DESIGN AND SYNTHESIS OF SMALL MOLECULES TARGETING PRE-MIRNA21 TOWARD THE DEVELOPMENT OF RIBONUCLEASE TARGETING CHIMERAS (RIBOTACS) TO REGULATE THE ONCOGENIC MIRNA21 Sdei, F.; Bagnolini, G.; Falchi, F.; Sosic, A.; Bolognesi, M. L. 2024-01-01 - - 4.01 Contributo in Atti di convegno -
Differential enantiomers activity of ARN24089 to achieve synthetic lethality in pancreatic cancer Previtali, Viola; Masi, Mirco; Poppi, Laura; Varignani, Giulia; Falchi, Federico; Tedesco, Daniel... espandie; Wynne, Kieran; Oliviero, Giorgio; Bagnolini, Greta; Farabegoli, Fulvia; DI STEFANO, Giuseppina; Girotto, Stefania; Roberti, Marinella; Cavalli, Andrea 2024-01-01 - - 4.03 Poster -
New Horizons of Synthetic Lethality in Cancer: Current Development and Future Perspectives Previtali, Viola; Bagnolini, Greta; Ciamarone, Andrea; Ferrandi, Giovanni; Rinaldi, Francesco; My... espandiers, Samuel Harry; Roberti, Marinella; Cavalli, Andrea 2024-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista New Horizons of Synthetic Lethality in Cancer_ Current Development and Future Perspectives.pdf
Targeting RNA degradation with small molecules: design and synthesis of selective RNA binders and development of ribonuclease targeting chimeras (RIBOTACs) Sdei, Federico; Bagnolini, Greta; Falchi, Federico; Ghezzo, M.; Sosic, Alice; Sissi, Claudia; Rob... espandierti, Marinella; Bolognesi, MARIA LAURA 2024-01-01 - - 4.03 Poster -
An 19F NMR fragment-based approach for the discovery and development of BRCA2-RAD51 inhibitors to pursuit synthetic lethality in combination with PARP inhibition in pancreatic cancer Myers, S. H.; Poppi, L.; Rinaldi, F.; Veronesi, M.; Ciamarone, A.; Previtali, V.; Bagnolini, G.; ... espandiSchipani, F.; Ortega Martínez, J. A.; Girotto, S.; Di Stefano, G.; Farabegoli, F.; Walsh, N.; De Franco, F.; Roberti, M.; Cavalli, A. 2023-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista 1-s2.0-S0223523423010814-mmc1.docx1-s2.0-S0223523423010814-main.pdf
Design and synthesis of RAD51-BRCA disruptors to inhibit homologous recombination and achieve synthetic lethality in cancer cells Ferrandi, Giovanni; Bagnolini, Greta; Roberti, Marinella; Cavalli, Andrea 2023-01-01 - - 4.03 Poster -
Recognizing the power of machine learning and other computational methods to accelerate progress in small molecule targeting of RNA Bagnolini, G; Luu, Tb; Hargrove, Ae 2023-01-01 RNA - 1.01 Articolo in rivista -
Triggering RNA degradation with small molecules: development of RIBOnuclease TArgeting Chimeras (RIBOTACs) Bagnolini, G.; Falchi, F.; Sdei, F.; Roberti, M.; Sosic, A.; Sissi, C.; Bolognesi, M. L. 2023-01-01 - - 4.03 Poster -
Identification of RAD51-BRCA2 Inhibitors Using N-Acylhydrazone-Based Dynamic Combinatorial Chemistry Bagnolini, G.; Balboni, B.; Schipani, F.; Gioia, D.; Veronesi, M.; De Franco, F.; Kaya, C.; Jumde... espandi, R. P.; Ortega, J. A.; Girotto, S.; Hirsch, A. K. H.; Roberti, M.; Cavalli, A. 2022-01-01 ACS MEDICINAL CHEMISTRY LETTERS - 1.01 Articolo in rivista acsmedchemlett._2022.pdf
Identification of RAD51-BRCA2 inhibitors using N-acylhydrazone-based dynamic combinatorial chemistry Bagnolini, Greta; Balboni, Beatrice; Schipani, Fabrizio; Gioia, Dario; Veronesi, Marina; De Franc... espandio, Francesca; Kaya, Cansu; Jumde, Ravindra P.; Antonio Ortega, Jose; Girotto, Stefania; Hirsch, Anna K. H.; Roberti, Marinella; Cavalli, Andrea 2022-01-01 - - 4.01 Contributo in Atti di convegno -
Insights into the activity of ARN24089, a new RAD51-BRCA2 disruptor that inhibits homologous recombination and achieves synthetic lethality in pancreatic cancer Previtali V., Myers S. H., Bagnolini G., Poppi L., Rinaldi F., Schipani F., Ortega J. A., De Fran... espandico F., Pellicciari R., Girotto S., Oliviero G., Walsh N., Valenti G., Tirelli N., Di Stefano G., Roberti M., Cavalli A. 2022-01-01 - - 4.02 Riassunto (Abstract) -
Inhibition of Urease, a Ni-Enzyme: The Reactivity of a Key Thiol With Mono- and Di-Substituted Catechols Elucidated by Kinetic, Structural, and Theoretical Studies Mazzei L.; Contaldo U.; Musiani F.; Cianci M.; Bagnolini G.; Roberti M.; Ciurli S. 2021-01-01 ANGEWANDTE CHEMIE. INTERNATIONAL EDITION - 1.01 Articolo in rivista Manuscript.pdfSupplementary Information.pdf
Dihydroquinoline pyrazoline-based compound as a new RAD51-BRCA2 protein-protein disruptor to trigger synthetic lethality in pancreatic cancer Bagnolini, Greta; Manerba, Marcella; Balboni, Andrea; Antonio Ortega, Jose; Gioia, Dario; De Fran... espandico, Francesca; Roberti, Marinella; Cavalli, Andrea 2020-01-01 - - 4.03 Poster -
Synthetic Lethality in Pancreatic Cancer: Discovery of a New RAD51-BRCA2 Small Molecule Disruptor That Inhibits Homologous Recombination and Synergizes with Olaparib Bagnolini G.; Milano D.; Manerba M.; Schipani F.; Ortega J.A.; Gioia D.; Falchi F.; Balboni A.; F... espandiarabegoli F.; De Franco F.; Robertson J.; Pellicciari R.; Pallavicini I.; Peri S.; Minucci S.; Girotto S.; Di Stefano G.; Roberti M.; Cavalli A. 2020-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista ASAP_acs.jmedchem.9b01526.pdf