MORIGI, RITA
MORIGI, RITA
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di IIa fascia
Identification of MBT3T as a new effective therapeutic option in imatinib-resistant gastrointestinal stromal tumors (GISTs)
2026 Ravegnini, Gloria; Esposito, Daniele; Gorini, Francesca; Marforio, Tainah Dorina; Coschina, Emma; Benuzzi, Eva; Simone, Antonella; Samaha, Ahmed; Di Vito, Aldo; Rossi, Martina; Hrelia, Patrizia; Locatelli, Alessandra; Calvaresi, Matteo; Facchinello, Nicola; Morigi, Rita; Angelini, Sabrina
Effects of hydrazone-based G-quadruplex ligands on FANCJ/BRIP1-depleted cancer cells and a Caenorhabditis elegans dog-1-/- strain
2025 Germoglio, Marcello; D'Aria, Federica; Cortone, Giuseppe; Prodomo, Antonello; Mahtab, Mohammad; Morigi, Rita; Amato, Jussara; Pisani, Francesca M; Giancola, Concetta
Molecular Tools for Precision Targeting and Detection of G-Quadruplex Structures
2025 Esposito, Daniele; Locatelli, Alessandra; Morigi, Rita
Identification of a new bisindolinone arresting IGROV1 cells proliferation
2024 Morigi R.; Zalambani C.; Farruggia G.; Verardi L.; Esposito D.; Leoni A.; Borsetti F.; Voltattorni M.; Zambonin L.; Pincigher L.; Calonghi N.; Locatelli A.
Isatin Bis-Imidathiazole Hybrids Identified as FtsZ Inhibitors with On-Target Activity Against Staphylococcus aureus
2024 Morigi, Rita; Esposito, Daniele; Calvaresi, Matteo; Marforio, TAINAH DORINA; Gentilomi, GIOVANNA ANGELA; Bonvicini, Francesca; Locatelli, Alessandra
Balancing Affinity, Selectivity, and Cytotoxicity of Hydrazone-Based G-Quadruplex Ligands for Activation of Interferon β Genes in Cancer Cells
2022 Marzano S.; Miglietta G.; Morigi R.; Marinello J.; Arleo A.; Procacci M.; Locatelli A.; Leoni A.; Pagano B.; Randazzo A.; Amato J.; Capranico G.
Isatin Bis-Indole and Bis-Imidazothiazole Hybrids: Synthesis and Antimicrobial Activity
2022 Francesca Bonvicini, Alessandra Locatelli, Rita Morigi, Alberto Leoni, Giovanna Angela Gentilomi
Synthesis, in vitro cytotoxicity, molecular docking and ADME study of some indolin-2-one linked 1,2,3-triazole derivatives
2022 Das A.; Greco G.; Kumar S.; Catanzaro E.; Morigi R.; Locatelli A.; Schols D.; Alici H.; Tahtaci H.; Ravindran F.; Fimognari C.; Karki S.S.
Synthesis and biological evaluation of new bis-indolinone derivatives endowed with cytotoxic activity
2021 Morigi R.; Catanzaro E.; Locatelli A.; Calcabrini C.; Pellicioni V.; Leoni A.; Fimognari C.
Indole derivative interacts with estrogen receptor beta and inhibits human ovarian cancer cell growth
2020 Verardi L.; Fiori J.; Andrisano V.; Locatelli A.; Morigi R.; Naldi M.; Bertucci C.; Strocchi E.; Boga C.; Micheletti G.; Calonghi N.
Monohydrazone Based G-Quadruplex Selective Ligands Induce DNA Damage and Genome Instability in Human Cancer Cells
2020 Amato J.; Miglietta G.; Morigi R.; Iaccarino N.; Locatelli A.; Leoni A.; Novellino E.; Pagano B.; Capranico G.; Randazzo A.
Synthesis and biological evaluation of thiazole derivatives on basic defects underlying cystic fibrosis.
2020 Pesce, Emanuela; Pedemonte, Nicoletta; Leoni, Alberto; Locatelli, Alessandra; Morigi, Rita
Capitolo 7 - Titolazioni Complessometriche
2019 Rita Morigi
DNA damage and genome instability by G-quadruplex ligands are mediated by R loops in human cancer cells
2019 De Magis, Alessio; Manzo, Stefano G.; Russo, Marco; Marinello, Jessica; Morigi, Rita; Sordet, Olivier; Capranico, Giovanni*
Synthesis of 3-(Imidazo[2,1-b]thiazol-6-yl)-2H-chromen-2-one derivatives and study of their antiviral activity against parvovirus B19
2019 Conti, Ilaria; Morigi, Rita; Locatelli, Alessandra*; Rambaldi, Mirella; Bua, Gloria; Gallinella, Giorgio; Leoni, Alberto
Synthesis, in vitro and in vivo biological evaluation of substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones as new potent anticancer agents
2019 Morigi, R., Locatelli, A., Leoni, A., Rambaldi, M., Bortolozzi, R., Mattiuzzo, E., Ronca, R., Maccarinelli, F., Hamel, E., Bai, R., Brancale, A., Viola, G.
Genome instability by G-quadruplex ligands are mediated by R-loops in human cancer cells
2018 Alessio De Magis, Stefano G. Manzo, Jessica Marinello, Marco Russo, Olivier Sordet, Rita Morigi, Giovanni Capranico
Investigation on the effects of antimicrobial imidazo[2,1-b]thiazole derivatives on the genitourinary microflora
2018 Morigi, Rita; Vitali, Beatrice; Prata, Cecilia; Palomino, Rogers A. A; Graziadio, Alessandra; Locatelli, Alessandra; Rambaldi, Mirella; Leoni, Alberto
R loop-driven genome instability by G-quadruplex binders in BRCA2-silenced human cancer cells.
2018 A. De Magis, S. G. Manzo, M. Russo, J. Marinello, O. Sordet, R. Morigi, G. Capranico.
Targeting human telomeric and promoter G-quardruplexes: synthesis, biophysical and biological studies of new guanylhydrazones as potential antitumor agents
2018 R. Morigi, J. Amato, N. Iaccarino, B. Pagano, A. Locatelli, A. Leoni, M. Rambaldi, G. Miglietta, J. Marinello, G. Capranico, E. Novellino, A. Randazzo
| Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
|---|---|---|---|---|---|---|
| Identification of MBT3T as a new effective therapeutic option in imatinib-resistant gastrointestinal stromal tumors (GISTs) | Ravegnini, Gloria; Esposito, Daniele; Gorini, Francesca; Marforio, Tainah Dorina; Coschina, Emma;... Benuzzi, Eva; Simone, Antonella; Samaha, Ahmed; Di Vito, Aldo; Rossi, Martina; Hrelia, Patrizia; Locatelli, Alessandra; Calvaresi, Matteo; Facchinello, Nicola; Morigi, Rita; Angelini, Sabrina | 2026-01-01 | JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH | - | 1.01 Articolo in rivista | - |
| Effects of hydrazone-based G-quadruplex ligands on FANCJ/BRIP1-depleted cancer cells and a Caenorhabditis elegans dog-1-/- strain | Germoglio, Marcello; D'Aria, Federica; Cortone, Giuseppe; Prodomo, Antonello; Mahtab, Mohammad; M...origi, Rita; Amato, Jussara; Pisani, Francesca M; Giancola, Concetta | 2025-01-01 | NAR CANCER | - | 1.01 Articolo in rivista | zcaf004.pdf; zcaf004_supplemental_file.pdf |
| Molecular Tools for Precision Targeting and Detection of G-Quadruplex Structures | Esposito, Daniele; Locatelli, Alessandra; Morigi, Rita | 2025-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-30-04099.pdf |
| Identification of a new bisindolinone arresting IGROV1 cells proliferation | Morigi R.; Zalambani C.; Farruggia G.; Verardi L.; Esposito D.; Leoni A.; Borsetti F.; Voltattorn...i M.; Zambonin L.; Pincigher L.; Calonghi N.; Locatelli A. | 2024-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | 1-s2.0-S0223523424002459-main.pdf; 1-s2.0-S0223523424002459-mmc1.docx |
| Isatin Bis-Imidathiazole Hybrids Identified as FtsZ Inhibitors with On-Target Activity Against Staphylococcus aureus | Morigi, Rita; Esposito, Daniele; Calvaresi, Matteo; Marforio, TAINAH DORINA; Gentilomi, GIOVANNA ...ANGELA; Bonvicini, Francesca; Locatelli, Alessandra | 2024-01-01 | ANTIBIOTICS | - | 1.01 Articolo in rivista | 2024_Antibiotics.pdf; 2024_Antibiotics-3244517-supplementary.pdf |
| Balancing Affinity, Selectivity, and Cytotoxicity of Hydrazone-Based G-Quadruplex Ligands for Activation of Interferon β Genes in Cancer Cells | Marzano S.; Miglietta G.; Morigi R.; Marinello J.; Arleo A.; Procacci M.; Locatelli A.; Leoni A.;... Pagano B.; Randazzo A.; Amato J.; Capranico G. | 2022-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | JMC.pdf; jm2c00772_si_002.pdf |
| Isatin Bis-Indole and Bis-Imidazothiazole Hybrids: Synthesis and Antimicrobial Activity | Francesca Bonvicini, Alessandra Locatelli, Rita Morigi, Alberto Leoni, Giovanna Angela Gentilomi | 2022-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-27-05781.pdf |
| Synthesis, in vitro cytotoxicity, molecular docking and ADME study of some indolin-2-one linked 1,2,3-triazole derivatives | Das A.; Greco G.; Kumar S.; Catanzaro E.; Morigi R.; Locatelli A.; Schols D.; Alici H.; Tahtaci H....; Ravindran F.; Fimognari C.; Karki S.S. | 2022-01-01 | COMPUTATIONAL BIOLOGY AND CHEMISTRY | - | 1.01 Articolo in rivista | Synthesis, in vitro cytotoxicity, molecular docking and ADME study of some indolin-2-one linked 1,2,3-triazole derivatives.pdf |
| Synthesis and biological evaluation of new bis-indolinone derivatives endowed with cytotoxic activity | Morigi R.; Catanzaro E.; Locatelli A.; Calcabrini C.; Pellicioni V.; Leoni A.; Fimognari C. | 2021-01-01 | MOLECULES | - | 1.01 Articolo in rivista | Synthesis and Biological Evaluation of New Bis-Indolinone Derivatives Endowed with Cytotoxic Activity.pdf |
| Indole derivative interacts with estrogen receptor beta and inhibits human ovarian cancer cell growth | Verardi L.; Fiori J.; Andrisano V.; Locatelli A.; Morigi R.; Naldi M.; Bertucci C.; Strocchi E.; ...Boga C.; Micheletti G.; Calonghi N. | 2020-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-25-04438-v2.pdf |
| Monohydrazone Based G-Quadruplex Selective Ligands Induce DNA Damage and Genome Instability in Human Cancer Cells | Amato J.; Miglietta G.; Morigi R.; Iaccarino N.; Locatelli A.; Leoni A.; Novellino E.; Pagano B.;... Capranico G.; Randazzo A. | 2020-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Monohydrazone-Based-GQuadruplex-Selective-Ligands-Induce-DNA-Damage-and-Genome-Instability-in-Human-Cancer-Cells2020Journal-of-Medicinal-Chemistry.pdf |
| Synthesis and biological evaluation of thiazole derivatives on basic defects underlying cystic fibrosis. | Pesce, Emanuela; Pedemonte, Nicoletta; Leoni, Alberto; Locatelli, Alessandra; Morigi, Rita | 2020-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | Post-print BMCL 2020 30 127473.pdf; Synthesis and biological evaluation of thiazole derivatives on basic defects underlying cystic fibrosis..pdf |
| Capitolo 7 - Titolazioni Complessometriche | Rita Morigi | 2019-01-01 | - | EdiSES | 2.01 Capitolo / saggio in libro | - |
| DNA damage and genome instability by G-quadruplex ligands are mediated by R loops in human cancer cells | De Magis, Alessio; Manzo, Stefano G.; Russo, Marco; Marinello, Jessica; Morigi, Rita; Sordet, Oli...vier; Capranico, Giovanni* | 2019-01-01 | PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA | - | 1.01 Articolo in rivista | - |
| Synthesis of 3-(Imidazo[2,1-b]thiazol-6-yl)-2H-chromen-2-one derivatives and study of their antiviral activity against parvovirus B19 | Conti, Ilaria; Morigi, Rita; Locatelli, Alessandra*; Rambaldi, Mirella; Bua, Gloria; Gallinella, ...Giorgio; Leoni, Alberto | 2019-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-24-01037.pdf |
| Synthesis, in vitro and in vivo biological evaluation of substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones as new potent anticancer agents | Morigi, R., Locatelli, A., Leoni, A., Rambaldi, M., Bortolozzi, R., Mattiuzzo, E., Ronca, R., Mac...carinelli, F., Hamel, E., Bai, R., Brancale, A., Viola, G. | 2019-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | EJMC 166, 2019, 514 530 Post print .pdf |
| Genome instability by G-quadruplex ligands are mediated by R-loops in human cancer cells |
Alessio De Magis, Stefano G. Manzo, Jessica Marinello, Marco Russo, Olivier Sordet, Rita Morigi,... Giovanni Capranico |
2018-01-01 | - | - | 4.02 Riassunto (Abstract) | - |
| Investigation on the effects of antimicrobial imidazo[2,1-b]thiazole derivatives on the genitourinary microflora | Morigi, Rita; Vitali, Beatrice; Prata, Cecilia; Palomino, Rogers A. A; Graziadio, Alessandra; Loc...atelli, Alessandra; Rambaldi, Mirella; Leoni, Alberto | 2018-01-01 | MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
| R loop-driven genome instability by G-quadruplex binders in BRCA2-silenced human cancer cells. | A. De Magis, S. G. Manzo, M. Russo, J. Marinello, O. Sordet, R. Morigi, G. Capranico. | 2018-01-01 | CANCER RESEARCH | - | 4.03 Poster | - |
| Targeting human telomeric and promoter G-quardruplexes: synthesis, biophysical and biological studies of new guanylhydrazones as potential antitumor agents | R. Morigi, J. Amato, N. Iaccarino, B. Pagano, A. Locatelli, A. Leoni, M. Rambaldi, G. Miglietta, ...J. Marinello, G. Capranico, E. Novellino, A. Randazzo | 2018-01-01 | - | - | 4.02 Riassunto (Abstract) | - |