Sfoglia per Autore
Synthetic small molecule Cdc25 phosphatases inhibitors
2008 L. Garuti;| M. Roberti|; D. Pizzirani
Identification of biphenyl-based hybrid molecules able to decrease the intracellular level of Bcl-2 protein in Bcl-2 overexpressing leukemia cells
2009 Pizzirani D.; Roberti M.; Grimaudo S.; Di Cristina A.; Pipitone R.M.; Tolomeo M.; Recanatini M.
Small molecule aurora kinases inhibitors
2009 L. Garuti; M.Roberti; G. Bottegoni
Docking ligands on protein surfaces: the case study of prion protein.
2009 Kranjc A.; Bongarzone S.; Rossetti G.; Biarnes X.; Cavalli A.; Bolognesi M. L.; Roberti M.; Legname G.; Carloni P.
Parallel Synthesis, Evaluation, and Preliminary Structure-Activity Relationship of 2,5-Diamino-1,4-benzoquinones as a Novel Class of Bivalent Anti-Prion Compound.
2010 Bongarzone S; Tran HN; Cavalli A; Roberti M; Carloni P; Legname G; Bolognesi ML.
Multiple Ligand Strategy in anticancer drug discovery
2010 Roberti M; Bottegoni G.; Recanatini M.
Non-ATP competitive protein kinase inhibitors
2010 L. Garuti; M. Roberti; G. Bottegoni
Thermal and catalytic reactions of ethyl diazopiruvate with [60]fullerene
2010 M. Roberti; B. Natalini; V. Andrisano; R. Seraglia; A. Gioiello; R. Pellicciari
Irreversible protein kinase inhibitors
2011 L. Garuti; M. Roberti; G. Bottegoni
Sequential Virtual Screening Approach to the Identification of Small Organic Molecules as Potential BACE-1 Inhibitors
2011 Chiriano G.; Sartini A.; Mancini F.; Andrisano V.; Bolognesi M. L.; Roberti M.; Recanatini M.; Carloni P.; Cavalli A.
Hybrid Lipoic Acid Derivatives to Attack Prion Disease on Multiple Fronts
2011 Bongarzone S; Tran HN; Cavalli A; Roberti M; Rosini M; Carloni P; Legname G; Bolognesi ML
Galloflavin, a new lactate dehydrogenase inhibitor, induces the death of human breast cancer cells with different glycolytic attitude by affecting distinct signaling pathways.
2012 Farabegoli F.; Vettraino M.; Manerba M.; Fiume L.; Roberti M.; Di Stefano G.
Galloflavin (CAS 568-80-9), a novel inhibitor of lactate dehydrogenase.
2012 Manerba M.; Vettraino M.; Fiume L.; Di Stefano G.; Sartini A.; Giacomini E.; Buonfiglio R.; Roberti M.; Recanatini M.
Polo-like kinases inhibitors
2012 L. Garuti; M. Roberti; G. Bottegoni
A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation
2012 G. P. Chiriano; A. De Simone; F. Mancini; D. I. Perez; A. Cavalli; M. L. Bolognesi; G. Legname; A. Martinez; V. Andrisano; P. Carloni; M. Roberti
Computational design and discovery of "minimally structured" hERG blockers.
2012 Cavalli A.; Buonfiglio R.; Ianni C.; Masetti M.; Ceccarini L.; Caves R.; Chang M.W.; Mitcheson J.S.; Roberti M.; Recanatini M.
TTAS a New Stilbene Derivative that Induces Apoptosis in Leishmania Infantum
2013 M. Tolomeo; M. Roberti; L. Scapozza; C. Tarantelli; E. Giacomini; L. Titone; L. Saporito; P. Di Carlo; C. Colomba
A natural-like synthetic small molecule impairs bcr-abl signaling cascades and induces megakaryocyte differentiation in erythroleukemia cells
2013 Turroni S.; Tolomeo M.; Mamone G.; Picariello G.; Giacomini E.; Brigidi P.; Roberti M.; Grimaudo S.; Pipitone R.M.; Di Cristina A.; Recanatini M.
Benzimidazole derivatives as kinase inhibitors
2014 Garuti L; Roberti M; Bottegoni G.
Multitarget Drug Design Strategy: Quinone–Tacrine Hybrids Designed To Block Amyloid-β Aggregation and To Exert Anticholinesterase and Antioxidant Effects
2014 Eugenie Nepovimova;Elisa Uliassi;Jan Korabecny;Luis Emiliano Peña-Altamira;Sarah Samez;Alessandro Pesaresi;Gregory E. Garcia;Manuela Bartolini;Vincenza Andrisano;Christian Bergamini;Romana Fato;Doriano Lamba;Marinella Roberti;Kamil Kuca;Barbara Monti;Maria Laura Bolognesi
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Synthetic small molecule Cdc25 phosphatases inhibitors | L. Garuti;| M. Roberti|; D. Pizzirani | 2008-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Identification of biphenyl-based hybrid molecules able to decrease the intracellular level of Bcl-2 protein in Bcl-2 overexpressing leukemia cells | Pizzirani D.; Roberti M.; Grimaudo S.; Di Cristina A.; Pipitone R.M.; Tolomeo M.; Recanatini M. | 2009-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Small molecule aurora kinases inhibitors | L. Garuti; M.Roberti; G. Bottegoni | 2009-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Docking ligands on protein surfaces: the case study of prion protein. | Kranjc A.; Bongarzone S.; Rossetti G.; Biarnes X.; Cavalli A.; Bolognesi M. L.; Roberti M.; Legna...me G.; Carloni P. | 2009-01-01 | JOURNAL OF CHEMICAL THEORY AND COMPUTATION | - | 1.01 Articolo in rivista | - |
Parallel Synthesis, Evaluation, and Preliminary Structure-Activity Relationship of 2,5-Diamino-1,4-benzoquinones as a Novel Class of Bivalent Anti-Prion Compound. | Bongarzone S; Tran HN; Cavalli A; Roberti M; Carloni P; Legname G; Bolognesi ML. | 2010-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Multiple Ligand Strategy in anticancer drug discovery | Roberti M; Bottegoni G.; Recanatini M. | 2010-01-01 | - | Simona Rapposelli | 2.01 Capitolo / saggio in libro | - |
Non-ATP competitive protein kinase inhibitors | L. Garuti; M. Roberti; G. Bottegoni | 2010-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Thermal and catalytic reactions of ethyl diazopiruvate with [60]fullerene | M. Roberti; B. Natalini; V. Andrisano; R. Seraglia; A. Gioiello; R. Pellicciari | 2010-01-01 | TETRAHEDRON | - | 1.01 Articolo in rivista | - |
Irreversible protein kinase inhibitors | L. Garuti; M. Roberti; G. Bottegoni | 2011-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Sequential Virtual Screening Approach to the Identification of Small Organic Molecules as Potential BACE-1 Inhibitors | Chiriano G.; Sartini A.; Mancini F.; Andrisano V.; Bolognesi M. L.; Roberti M.; Recanatini M.; Ca...rloni P.; Cavalli A. | 2011-01-01 | CHEMICAL BIOLOGY & DRUG DESIGN | - | 1.01 Articolo in rivista | - |
Hybrid Lipoic Acid Derivatives to Attack Prion Disease on Multiple Fronts | Bongarzone S; Tran HN; Cavalli A; Roberti M; Rosini M; Carloni P; Legname G; Bolognesi ML | 2011-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
Galloflavin, a new lactate dehydrogenase inhibitor, induces the death of human breast cancer cells with different glycolytic attitude by affecting distinct signaling pathways. | Farabegoli F.; Vettraino M.; Manerba M.; Fiume L.; Roberti M.; Di Stefano G. | 2012-01-01 | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | - | 1.01 Articolo in rivista | - |
Galloflavin (CAS 568-80-9), a novel inhibitor of lactate dehydrogenase. | Manerba M.; Vettraino M.; Fiume L.; Di Stefano G.; Sartini A.; Giacomini E.; Buonfiglio R.; Rober...ti M.; Recanatini M. | 2012-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
Polo-like kinases inhibitors | L. Garuti; M. Roberti; G. Bottegoni | 2012-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation | G. P. Chiriano; A. De Simone; F. Mancini; D. I. Perez; A. Cavalli; M. L. Bolognesi; G. Legname; A.... Martinez; V. Andrisano; P. Carloni; M. Roberti | 2012-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Computational design and discovery of "minimally structured" hERG blockers. | Cavalli A.; Buonfiglio R.; Ianni C.; Masetti M.; Ceccarini L.; Caves R.; Chang M.W.; Mitcheson J....S.; Roberti M.; Recanatini M. | 2012-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
TTAS a New Stilbene Derivative that Induces Apoptosis in Leishmania Infantum | M. Tolomeo; M. Roberti; L. Scapozza; C. Tarantelli; E. Giacomini; L. Titone; L. Saporito; P. Di C...arlo; C. Colomba | 2013-01-01 | EXPERIMENTAL PARASITOLOGY | - | 1.01 Articolo in rivista | - |
A natural-like synthetic small molecule impairs bcr-abl signaling cascades and induces megakaryocyte differentiation in erythroleukemia cells | Turroni S.; Tolomeo M.; Mamone G.; Picariello G.; Giacomini E.; Brigidi P.; Roberti M.; Grimaudo ...S.; Pipitone R.M.; Di Cristina A.; Recanatini M. | 2013-01-01 | PLOS ONE | - | 1.01 Articolo in rivista | PLoS_One_2013.pdf |
Benzimidazole derivatives as kinase inhibitors | Garuti L; Roberti M; Bottegoni G. | 2014-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Multitarget Drug Design Strategy: Quinone–Tacrine Hybrids Designed To Block Amyloid-β Aggregation and To Exert Anticholinesterase and Antioxidant Effects | Eugenie Nepovimova;Elisa Uliassi;Jan Korabecny;Luis Emiliano Peña-Altamira;Sarah Samez;Alessandro... Pesaresi;Gregory E. Garcia;Manuela Bartolini;Vincenza Andrisano;Christian Bergamini;Romana Fato;Doriano Lamba;Marinella Roberti;Kamil Kuca;Barbara Monti;Maria Laura Bolognesi | 2014-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
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