Sfoglia per Autore
Novel antiproliferative chimeric compounds with marked histone deacetylase inhibitory activity.
2014 Giacomini E;Nebbioso A;Ciotta A;Ianni C;Falchi F;Roberti M;Tolomeo M;Grimaudo S;Cristina AD;Pipitone RM;Altucci L;Recanatini M
Berberine and its metabolites: Relationship between physicochemical properties and plasma levels after administration to human subjects
2014 Spinozzi, S.; Colliva, C.; Camborata, C.; Roberti, M.; Ianni, C.; Neri, F.; Calvarese, C.; Lisotti, A.; Mazzella, G.; Roda, A.
Lactate dehydrogenase inhibitors sensitize lymphoma cells to cisplatin without enhancing the drug effects on immortalized normal lymphocytes.
2015 M. Manerba; L. Di Ianni; L. Fiume; M. Roberti; M. Recanatini; G. Di Stefano
Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors
2015 Sebastiano Rupiani; Rosa Buonfiglio; Marcella Manerba; Lorenza Di Ianni; Marina Vettraino; Elisa Giacomini; Matteo Masetti; Federico Falchi; Giuseppina Di Stefano; Marinella Roberti; Maurizio Recanatini
Multi-kinase inhibitors
2015 Garuti L; Roberti M; Bottegoni G
Capitolo 2. Proprietà chimico-fisiche e attività biologica
2015 Bolognesi, Maria Laura; Roberti, Marinella
A ligand-based virtual screening approach to identify small molecules as hERG channel activators
2015 Giacomini, E.; Buonfiglio, R.; Masetti, M.; Wang, Y.; Tseng, G.-N.; Roberti, M.; Recanatini, M.
In vitro antileishmanial activity of trans-stilbene and terphenyl compounds
2016 Castelli, G; Bruno, F; Vitale, F; Roberti, M; Colomba, C; Giacomini, E; Guidotti, L; Cascio, A; Tolomeo, M
The use of stilbene scaffold in medicinal chemistry and multi-target drug design
2016 Giacomini, Elisa; Rupiani, Sebastiano; Guidotti, Laura; Recanatini, Maurizio; Roberti, Marinella
Diaryl Urea: A Privileged Structure in Anticancer Agents
2016 Garuti, Laura; Roberti, Marinella; Ferraro, Mariarosaria; Bottegoni, Giovanni
Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A
2016 Rupiani, Sebastiano; Guidotti, Laura; Manerba, Marcella; Di Ianni, Lorenza; Giacomini, Elisa; Falchi, Federico; Di Stefano, Giuseppina; Roberti, Marinella; Recanatini, Maurizio
Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease
2017 Jeřábek, Jakub; Uliassi, Elisa; Guidotti, Laura; Korábečný, Jan; Soukup, Ondřej; Sepsova, Vendula; Hrabinova, Martina; Kuča, Kamil; Bartolini, Manuela; Peña-Altamira, Luis Emiliano; Petralla, Sabrina; Monti, Barbara; Roberti, Marinella; Bolognesi, Maria Laura
LDH inhibition impacts on heat shock response and induces senescence of hepatocellular carcinoma cells
2017 Manerba, Marcella; Di Ianni, Lorenza; Govoni, Marzia; Roberti, Marinella; Recanatini, Maurizio; Di Stefano, Giuseppina
Synthetic Lethality Triggered by Combining Olaparib with BRCA2-Rad51 Disruptors
2017 Falchi, Federico; Giacomini, Elisa; Masini, Tiziana; Boutard, Nicolas; Di Ianni, Lorenza; Manerba, Marcella; Farabegoli, Fulvia; Rossini, Lara; Robertson, Janet; Minucci, Saverio; Pallavicini, Isabella; Di Stefano, Giuseppina; Roberti, Marinella; Pellicciari, Roberto; Cavalli, Andrea
Lactate dehydrogenase inhibitors can reverse inflammation induced changes in colon cancer cells
2017 Manerba, Marcella; Di Ianni, Lorenza; Govoni, Marzia; Roberti, Marinella; Recanatini, Maurizio; Di Stefano, Giuseppina
Combined analytical approaches to define biodistribution and biological activity of semi-synthetic berberrubine, the active metabolite of natural berberine
2018 Porru, Emanuele; Franco, Placido; Calabria, Donato; Spinozzi, Silvia; Roberti, Marinella; Caliceti, Cristiana; Roda, Aldo
Effects of trans-stilbene and terphenyl compounds on different strains of Leishmania and on cytokines production from infected macrophages
2018 Bruno, Federica; Castelli, Germano; Vitale, Fabrizio; Giacomini, Elisa; Roberti, Marinella; Colomba, Claudia; Cascio, Antonio; Tolomeo, Manlio*
Characterisation of bioactive compounds in wine by-products: toward the valorisation of sustainable resources
2019 Camilla Marasca, Irene Brusa, Chiara Cabrelle, Michele Protti, Matteo Micucci, Laura Mercolini, Marinella Roberti, Roberta Budriesi, Maurizio Recanatini
Rad51/Brca2 Disruptors Inhibit Homologous Recombination and Synergize with Olaparib in Pancreatic Cancer Cells
2019 Marinella Roberti, Fabrizio Schipani, Greta Bagnolini, Domenico Milano, Elisa Giacomini, Federico Falchi, Andrea Balboni, Marcella Manerba, Fulvia Farabegoli, Francesca De Franco, Janet Robertson, Saverio Minucci, Isabella Pallavicini, Giuseppina Di Stefano, Stefania Girotto, Roberto Pellicciari, and Andrea Cavalli
A Focused Library of Psychotropic Analogues with Neuroprotective and Neuroregenerative Potential
2019 Uliassi, Elisa; Pena-Altamira, Luis Emiliano; Morales, Aixa V.; Massenzio, Francesca; Petralla, Sabrina; Rossi, Michele; Roberti, Marinella; Martinez Gonzalez, Loreto; Martinez, Ana; Monti, Barbara; Bolognesi, Maria Laura*
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Novel antiproliferative chimeric compounds with marked histone deacetylase inhibitory activity. | Giacomini E;Nebbioso A;Ciotta A;Ianni C;Falchi F;Roberti M;Tolomeo M;Grimaudo S;Cristina AD;Pipit...one RM;Altucci L;Recanatini M | 2014-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
Berberine and its metabolites: Relationship between physicochemical properties and plasma levels after administration to human subjects | Spinozzi, S.; Colliva, C.; Camborata, C.; Roberti, M.; Ianni, C.; Neri, F.; Calvarese, C.; Lisott...i, A.; Mazzella, G.; Roda, A. | 2014-01-01 | JOURNAL OF NATURAL PRODUCTS | - | 1.01 Articolo in rivista | - |
Lactate dehydrogenase inhibitors sensitize lymphoma cells to cisplatin without enhancing the drug effects on immortalized normal lymphocytes. | M. Manerba; L. Di Ianni; L. Fiume; M. Roberti; M. Recanatini; G. Di Stefano | 2015-01-01 | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | - | 1.01 Articolo in rivista | REVISED TEXT-1.pdf |
Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors | Sebastiano Rupiani; Rosa Buonfiglio; Marcella Manerba; Lorenza Di Ianni; Marina Vettraino; Elisa ...Giacomini; Matteo Masetti; Federico Falchi; Giuseppina Di Stefano; Marinella Roberti; Maurizio Recanatini | 2015-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Multi-kinase inhibitors | Garuti L; Roberti M; Bottegoni G | 2015-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Capitolo 2. Proprietà chimico-fisiche e attività biologica | Bolognesi, Maria Laura; Roberti, Marinella | 2015-01-01 | - | Casa Editrice Ambrosiana | 2.01 Capitolo / saggio in libro | - |
A ligand-based virtual screening approach to identify small molecules as hERG channel activators | Giacomini, E.; Buonfiglio, R.; Masetti, M.; Wang, Y.; Tseng, G.-N.; Roberti, M.; Recanatini, M. | 2015-01-01 | COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING | - | 1.01 Articolo in rivista | - |
In vitro antileishmanial activity of trans-stilbene and terphenyl compounds | Castelli, G; Bruno, F; Vitale, F; Roberti, M; Colomba, C; Giacomini, E; Guidotti, L; Cascio, A; T...olomeo, M | 2016-01-01 | EXPERIMENTAL PARASITOLOGY | - | 1.01 Articolo in rivista | - |
The use of stilbene scaffold in medicinal chemistry and multi-target drug design | Giacomini, Elisa; Rupiani, Sebastiano; Guidotti, Laura; Recanatini, Maurizio; Roberti, Marinella | 2016-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Diaryl Urea: A Privileged Structure in Anticancer Agents | Garuti, Laura; Roberti, Marinella; Ferraro, Mariarosaria; Bottegoni, Giovanni | 2016-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A | Rupiani, Sebastiano; Guidotti, Laura; Manerba, Marcella; Di Ianni, Lorenza; Giacomini, Elisa; Fal...chi, Federico; Di Stefano, Giuseppina; Roberti, Marinella; Recanatini, Maurizio | 2016-01-01 | ORGANIC & BIOMOLECULAR CHEMISTRY | - | 1.01 Articolo in rivista | - |
Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease | Jeřábek, Jakub; Uliassi, Elisa; Guidotti, Laura; Korábečný, Jan; Soukup, Ondřej; Sepsova, Vendula...; Hrabinova, Martina; Kuča, Kamil; Bartolini, Manuela; Peña-Altamira, Luis Emiliano; Petralla, Sabrina; Monti, Barbara; Roberti, Marinella; Bolognesi, Maria Laura | 2017-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
LDH inhibition impacts on heat shock response and induces senescence of hepatocellular carcinoma cells | Manerba, Marcella; Di Ianni, Lorenza; Govoni, Marzia; Roberti, Marinella; Recanatini, Maurizio; D...i Stefano, Giuseppina | 2017-01-01 | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | - | 1.01 Articolo in rivista | Bozza finale_PHASCI_4029_final.pdf |
Synthetic Lethality Triggered by Combining Olaparib with BRCA2-Rad51 Disruptors | Falchi, Federico; Giacomini, Elisa; Masini, Tiziana; Boutard, Nicolas; Di Ianni, Lorenza; Manerba..., Marcella; Farabegoli, Fulvia; Rossini, Lara; Robertson, Janet; Minucci, Saverio; Pallavicini, Isabella; Di Stefano, Giuseppina; Roberti, Marinella; Pellicciari, Roberto; Cavalli, Andrea | 2017-01-01 | ACS CHEMICAL BIOLOGY | - | 1.01 Articolo in rivista | - |
Lactate dehydrogenase inhibitors can reverse inflammation induced changes in colon cancer cells | Manerba, Marcella; Di Ianni, Lorenza; Govoni, Marzia; Roberti, Marinella; Recanatini, Maurizio; D...i Stefano, Giuseppina | 2017-01-01 | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | - | 1.01 Articolo in rivista | manerba_2107.pdf |
Combined analytical approaches to define biodistribution and biological activity of semi-synthetic berberrubine, the active metabolite of natural berberine | Porru, Emanuele; Franco, Placido; Calabria, Donato; Spinozzi, Silvia; Roberti, Marinella; Calicet...i, Cristiana; Roda, Aldo | 2018-01-01 | ANALYTICAL AND BIOANALYTICAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Effects of trans-stilbene and terphenyl compounds on different strains of Leishmania and on cytokines production from infected macrophages | Bruno, Federica; Castelli, Germano; Vitale, Fabrizio; Giacomini, Elisa; Roberti, Marinella; Colom...ba, Claudia; Cascio, Antonio; Tolomeo, Manlio* | 2018-01-01 | EXPERIMENTAL PARASITOLOGY | - | 1.01 Articolo in rivista | - |
Characterisation of bioactive compounds in wine by-products: toward the valorisation of sustainable resources | Camilla Marasca, Irene Brusa, Chiara Cabrelle, Michele Protti, Matteo Micucci, Laura Mercolini, M...arinella Roberti, Roberta Budriesi, Maurizio Recanatini | 2019-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
Rad51/Brca2 Disruptors Inhibit Homologous Recombination and Synergize with Olaparib in Pancreatic Cancer Cells | Marinella Roberti, Fabrizio Schipani, Greta Bagnolini, Domenico Milano, Elisa Giacomini, Federico... Falchi, Andrea Balboni, Marcella Manerba, Fulvia Farabegoli, Francesca De Franco, Janet Robertson, Saverio Minucci, Isabella Pallavicini, Giuseppina Di Stefano, Stefania Girotto, Roberto Pellicciari, and Andrea Cavalli | 2019-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A Focused Library of Psychotropic Analogues with Neuroprotective and Neuroregenerative Potential | Uliassi, Elisa; Pena-Altamira, Luis Emiliano; Morales, Aixa V.; Massenzio, Francesca; Petralla, S...abrina; Rossi, Michele; Roberti, Marinella; Martinez Gonzalez, Loreto; Martinez, Ana; Monti, Barbara; Bolognesi, Maria Laura* | 2019-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | - |
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