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Mostrati risultati da 21 a 40 di 182
Titolo Autore(i) Anno Periodico Editore Tipo File
Synthesis and biological profile at muscarinic M2 and M3 receptor subtypes of some analogs of diphenidol Varoli L.; Burnelli S.; Budriesi R.; Guarnieri A.; Chiarini A.; Recanatini M. 1996-01-01 MEDICINAL CHEMISTRY RESEARCH - 1.01 Articolo in rivista -
Study of lipophilic character of serotonergic ligands Biagi G.L.; Barbaro A.M.; Sapone A.; Borea P.A.; Varani K.; Recanatini M. 1996-01-01 JOURNAL OF CHROMATOGRAPHY A - 1.01 Articolo in rivista -
A comparative QSAR analysis of acetylcholinesterase inhibitors currently studied for the treatment of Alzheimer's disease Recanatini M.; Cavalli A.; Hansch C. 1997-01-01 CHEMICO-BIOLOGICAL INTERACTIONS - 1.01 Articolo in rivista -
Comparative molecular field analysis of non-steroidal aromatase inhibitors: An extended model for two different structural classes Recanatini M.; Cavalli A. 1998-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Comparative molecular field analysis (CoMFA) of a series of selective adenosine receptor A(2A) antagonists Baraldi P.G.; Borea P.A.; Bergonzoni M.; Cacciari B.; Ongini E.; Recanatini M.; Spalluto G. 1999-01-01 DRUG DEVELOPMENT RESEARCH - 1.01 Articolo in rivista -
WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for α1-adrenoreceptor subtypes and 5-HT(1A) receptors Bolognesi M.L.; Budriesi R.; Cavalli A.; Chiarini A.; Gotti R.; Leonardi A.; Minarini A.; Poggesi... E.; Recanatini M.; Rosini M.; Tumiatti V.; Melchiorre C. 1999-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Linking CoMFA and protein homology models of enzyme-inhibitor interactions: An application to non-steroidal aromatase inhibitors Cavalli A.; Greco G.; Novellino E.; Recanatini M. 2000-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
SAR of 9-amino-1,2,3-4-tetrahydroacridine-based acetylcholinesterase inhibitors: Synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues Recanatini M.; Cavalli A.; Belluti F.; Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Valenti P.; Andris...ano V.; Bartolini M.; Cavrini V. 2000-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Design, synthesis and binding at cloned muscarinic receptors of N-[5-(1'-substituted-acetoxymethyl)-3-oxadiazolyl] and N-[4-(1'-substituted-acetoxymethyl)-2-dioxolanyl] dialkyl amines Manfredini S.; Lampronti I.; Vertuani S.; Solaroli N.; Recanatini M.; Bryan D.; Mckinney M. 2000-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: Molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives Rampa A.; Bisi A.; Belluti F.; Gobbi S.; Valenti P.; Andrisano V.; Cavrini V.; Cavalli A.; Recana...tini M. 2000-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
A new class of nonsteroidal aromatase inhibitors: Design and synthesis of chromone and xanthone derivatives and inhibition of the P450 enzymes aromatase and 17α-hydroxylase/C17,20-lyase Recanatini M.; Hartmann R.W.; Bisi A.; Cavalli A.; Belluti F.; Gobbi S.; Rampa A.; Valenti P.; Pa...lzer M.; Palusczak A. 2001-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Caval...li A.; Recanatini M.; Valenti P. 2001-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Three-dimensional model of the cyclin-dependent kinase 1 (CDK1): Ab initio active site parameters for molecular dynamics studies of CDKs Cavalli A.; Dezi C.; Folkers G.; Scapozza L.; Recanatini M. 2001-01-01 PROTEINS - 1.01 Articolo in rivista -
Safety of non-antiarrhythmic drugs that prolong the QT interval or induce torsade de pointes: An overview De Ponti F.; Poluzzi E.; Cavalli A.; Recanatini M.; Montanaro N. 2002-01-01 DRUG SAFETY - 1.01 Articolo in rivista -
Toward a pharmacophore for drugs inducing the long QT syndrome: Insights from a CoMFA study of HERG K+ channel blockers Cavalli A.; Poluzzi E.; De Ponti F.; Recanatini M. 2002-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Acetylcholinesterase inhibitors in the context of therapeutic strategies to combat alzheimer's disease Recanatini M.; Cavalli A. 2002-01-01 EXPERT OPINION ON THERAPEUTIC PATENTS - 1.01 Articolo in rivista -
Nonsteroidal aromatase inhibitors: Recent advances Recanatini M.; Cavalli A.; Valenti P. 2002-01-01 MEDICINAL RESEARCH REVIEWS - 1.01 Articolo in rivista -
Looking for selectivity among cytochrome P450s inhibitors Cavalli A.; Recanatini M. 2002-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valen...ti P.; Recanatini M. 2003-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Density functional study of the enzymatic reaction catalyzed by a cyclin-dependent kinase Cavalli A.; De Vivo M.; Recanatini M. 2003-01-01 CHEMICAL COMMUNICATIONS - 1.01 Articolo in rivista -
Mostrati risultati da 21 a 40 di 182
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