Sfoglia per Autore
Process for preparation of 1,4-benzoquinone-2,5-diamines by reaction of amines with 1,4-benzoquinones bearing leaving groups at the 2- and 5-positions
2006 M.L. Bolognesi; R. Banzi; A. Minarini; C. Melchiorre
Methoctramine analogues inhibit capsaicin induced currents in dorsal root ganglia and Xenopus oocytes expressing TRPV1
2006 Mellor IR; Rosini M; Minarini A; Tumiatti V; Melchiorre C
Methoctramine effects on nicotinic acetylcholine receptor kinetics
2006 E. Nurowska; V. Tumiatti; A. Minarini; F. Ruzzier
Progettazione e sintesi di poliammine a potenziale attività antitumorale
2006 Tumiatti V; Milelli A; Minarini A; Bolognesi M; Baiocchi D; Roncuzzi L; Gasperi-Campani A; Melchiorre C
One-molecule-multiple-target strategy: a novel multifunctional molecule designed to block EGF-r and to exert pro-apoptotic effects
2006 M.L. Bolognesi; A. Antonello; A. Tarozzi; M. Rosini; A. Minarini; V. Tumiatti; P. Hrelia; C. Melchiorre.
Cytotoxicity of Methoctramine and related Spermine analogues
2007 A. Minarini; V. Tumiatti; F. Flamigni; M. Zini; C. Stefanelli
Quinone-bearing polyamines are AChE inhibitors endowed with multifunctional properties
2007 M.L. Bolognesi; R. Banzi; A. Cavalli; A. Minarini; M. Bartolini; V. Andrisano; M. Recanatini; C. Melchiorre
Progettazione e sintesi di derivati poliamminici per il trattamento della malattia di Alzheimer
2007 V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; V. Andrisano; M. Bartolini; F. Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre
Memoquine derivatives as potent inhibitors of AChE-induced amyloid-beta aggregation
2007 Bolognesi ML; Cavalli A; Andrisano V; Bartolini M; Minarini A; Melchiorre C
Beta-secretase monolithic micro-IMER (immobilized enzyme reactor) for on-line HPLC screening of quinone-bearing polyamine inhibitors.
2007 Mancini F.; Bolognesi ML.; Minarini A.; Melchiorre C.; Andrisano V.
Novel Class of Quinone-Bearing Polyamines as Multi-Target-Directed Ligands To Combat Alzheimer's Disease
2007 Bolognesi ML; Banzi R; Bartolini M; Cavalli A; Tarozzi A; Andrisano V; Minarini A; Rosini M; Tumiatti V; Bergamini C; Fato R; Lenaz G; Hrelia P; Cattaneo A; Recanatini M; Melchiorre C.
Recent advances in alpha1-adrenoreceptor antagonists as pharmacological tools and therapeutic agents.
2007 Rosini M; Bolognesi ML; Giardina D; Minarini A; Tumiatti V; Melchiorre C.
New quinazoline compounds as non-peptidomimetic BACE-1 inhibitors in the treatment of Alzheimer's disease
2007 Matera R; Minarini A; Rosini M; Andrisano V; Mancini F; Melchiorre C.
Structure-activity relationships of methoctramine-related polyamines as muscarinic antagonist: Effect of replacing the inner polymethylene chain with cyclic moieties
2007 V. Tumiatti; A. Minarini; A. Milelli; M. Rosini; M. Buccioni; G. Marucci; C. Ghelardini; C. Bellucci; C. Melchiorre
Synthesis of monomeric derivatives to probe Memoquin bivalent interactions
2008 ML. Bolognesi; A. Minarini; M. Bartolini; A. Cavalli; F. Mancini; V. Andrisano; M. Rosini; V. Tumiatti; C. Melchiorre
Progress in acetylcholinesterase inhibitors for Alzheimer's disease: an update
2008 V. Tumiatti; M. L. Bolognesi; A. Minarini; M. Rosini; A. Milelli; R. Matera; C. Melchiorre
Structure-Activity Relationships of New Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone
2008 V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; M. Micco; V. Andrisano; M. Bartolini; F. Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre
Structure-Activity Relationships of Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone. 4. Futher Investigation on the Inner Spacer.
2008 V. Tumiatti; A. Milelli; A. Minarini; M. Rosini; M. L. Bolognesi; M. Micco; V. Andrisano; M. Bartolini; F. Mancini; M. Recanatini; A. Cavalli; C. Melchiorre
Design, synthesis, and biological evaluation of pirenzepine analogs bearing a 1,2-cyclohexanediamine and a perhydroquinoxaline units in exchange for the piperazine ring as antimuscarinics
2008 A. Minarini; G. Marucci; C. Bellucci; G. Giorgi; V. Tumiatti; M. L. Bolognesi; R. Matera; M. Rosini; C. Melchiorre
Inhibition of Acetylcholinesterase, Beta-Amyloid Aggregation, and NMDA Receptors in Alzheimer's Disease: A Promising Direction for the Multi-target-Directed Ligands Gold Rush
2008 M. Rosini; E. Simoni; M. Bartolini; A. Cavalli; L. Ceccarini; N. Pascu; D. W. McClymont; A. Tarozzi; M. L. Bolognesi; A. Minarini; V. Tumiatti; V. Andrisano; I. R. Mellor; C. Melchiorre
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Process for preparation of 1,4-benzoquinone-2,5-diamines by reaction of amines with 1,4-benzoquinones bearing leaving groups at the 2- and 5-positions |
M.L. Bolognesi; R. Banzi; A. Minarini; C. Melchiorre |
2006-01-01 | - | - | 6.01 Brevetto | - |
Methoctramine analogues inhibit capsaicin induced currents in dorsal root ganglia and Xenopus oocytes expressing TRPV1 | Mellor IR; Rosini M; Minarini A; Tumiatti V; Melchiorre C | 2006-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Methoctramine effects on nicotinic acetylcholine receptor kinetics | E. Nurowska; V. Tumiatti; A. Minarini; F. Ruzzier | 2006-01-01 | ACTA PHYSIOLOGICA | - | 4.02 Riassunto (Abstract) | - |
Progettazione e sintesi di poliammine a potenziale attività antitumorale | Tumiatti V; Milelli A; Minarini A; Bolognesi M; Baiocchi D; Roncuzzi L; Gasperi-Campani A; Melchi...orre C | 2006-01-01 | - | Società di chimica Italiana | 4.02 Riassunto (Abstract) | - |
One-molecule-multiple-target strategy: a novel multifunctional molecule designed to block EGF-r and to exert pro-apoptotic effects |
M.L. Bolognesi; A. Antonello; A. Tarozzi; M. Rosini; A. Minarini; V. Tumiatti; P. Hrelia; C.... Melchiorre. |
2006-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Cytotoxicity of Methoctramine and related Spermine analogues | A. Minarini; V. Tumiatti; F. Flamigni; M. Zini; C. Stefanelli | 2007-01-01 | - | CSU Università degli Studi di Roma La Sapienza | 4.02 Riassunto (Abstract) | - |
Quinone-bearing polyamines are AChE inhibitors endowed with multifunctional properties | M.L. Bolognesi; R. Banzi; A. Cavalli; A. Minarini; M. Bartolini; V. Andrisano; M. Recanatini; C. ...Melchiorre | 2007-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Progettazione e sintesi di derivati poliamminici per il trattamento della malattia di Alzheimer | V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; V. Andrisano; M. Bartolini; F. ...Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Memoquine derivatives as potent inhibitors of AChE-induced amyloid-beta aggregation | Bolognesi ML; Cavalli A; Andrisano V; Bartolini M; Minarini A; Melchiorre C | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Beta-secretase monolithic micro-IMER (immobilized enzyme reactor) for on-line HPLC screening of quinone-bearing polyamine inhibitors. | Mancini F.; Bolognesi ML.; Minarini A.; Melchiorre C.; Andrisano V. | 2007-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Novel Class of Quinone-Bearing Polyamines as Multi-Target-Directed Ligands To Combat Alzheimer's Disease | Bolognesi ML; Banzi R; Bartolini M; Cavalli A; Tarozzi A; Andrisano V; Minarini A; Rosini M; Tumi...atti V; Bergamini C; Fato R; Lenaz G; Hrelia P; Cattaneo A; Recanatini M; Melchiorre C. | 2007-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Recent advances in alpha1-adrenoreceptor antagonists as pharmacological tools and therapeutic agents. | Rosini M; Bolognesi ML; Giardina D; Minarini A; Tumiatti V; Melchiorre C. | 2007-01-01 | CURRENT TOPICS IN MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
New quinazoline compounds as non-peptidomimetic BACE-1 inhibitors in the treatment of Alzheimer's disease | Matera R; Minarini A; Rosini M; Andrisano V; Mancini F; Melchiorre C. | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Structure-activity relationships of methoctramine-related polyamines as muscarinic antagonist: Effect of replacing the inner polymethylene chain with cyclic moieties | V. Tumiatti; A. Minarini; A. Milelli; M. Rosini; M. Buccioni; G. Marucci; C. Ghelardini; C. Bellu...cci; C. Melchiorre | 2007-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Synthesis of monomeric derivatives to probe Memoquin bivalent interactions | ML. Bolognesi; A. Minarini; M. Bartolini; A. Cavalli; F. Mancini; V. Andrisano; M. Rosini; V. Tum...iatti; C. Melchiorre | 2008-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Progress in acetylcholinesterase inhibitors for Alzheimer's disease: an update | V. Tumiatti; M. L. Bolognesi; A. Minarini; M. Rosini; A. Milelli; R. Matera; C. Melchiorre | 2008-01-01 | EXPERT OPINION ON THERAPEUTIC PATENTS | - | 1.01 Articolo in rivista | - |
Structure-Activity Relationships of New Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone | V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; M. Micco; V. Andrisano; M. Bart...olini; F. Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre | 2008-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Structure-Activity Relationships of Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone. 4. Futher Investigation on the Inner Spacer. | V. Tumiatti; A. Milelli; A. Minarini; M. Rosini; M. L. Bolognesi; M. Micco; V. Andrisano; M. Bart...olini; F. Mancini; M. Recanatini; A. Cavalli; C. Melchiorre | 2008-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Design, synthesis, and biological evaluation of pirenzepine analogs bearing a 1,2-cyclohexanediamine and a perhydroquinoxaline units in exchange for the piperazine ring as antimuscarinics | A. Minarini; G. Marucci; C. Bellucci; G. Giorgi; V. Tumiatti; M. L. Bolognesi; R. Matera; M. Rosi...ni; C. Melchiorre | 2008-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Inhibition of Acetylcholinesterase, Beta-Amyloid Aggregation, and NMDA Receptors in Alzheimer's Disease: A Promising Direction for the Multi-target-Directed Ligands Gold Rush | M. Rosini; E. Simoni; M. Bartolini; A. Cavalli; L. Ceccarini; N. Pascu; D. W. McClymont; A. Taroz...zi; M. L. Bolognesi; A. Minarini; V. Tumiatti; V. Andrisano; I. R. Mellor; C. Melchiorre | 2008-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
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