The synthetic approach to methyl N-(tert-butoxycarbonyl)- S-(3-thienyl)-L-cysteinate (1) and methyl N-(tert-butoxycarbonyl)- S-[2-(3-thienyl)ethyl]-L-cysteinate (2) through tosylate intermediates is reported and discussed. These compounds, which combine the properties of the cysteine side-chain with those of the thiophene ring represent both potential bioactive molecules and interesting synthons for the development of new materials.
Synthesis of two novel cysteine functionalized thiophenes / R. Cagnoli; M. Lanzi; A. Mucci; F. Parenti; L. Schenetti. - In: SYNTHESIS. - ISSN 0039-7881. - STAMPA. - 2:(2005), pp. 267-271. [10.1055/s-2004-834930]
Synthesis of two novel cysteine functionalized thiophenes
LANZI, MASSIMILIANO;
2005
Abstract
The synthetic approach to methyl N-(tert-butoxycarbonyl)- S-(3-thienyl)-L-cysteinate (1) and methyl N-(tert-butoxycarbonyl)- S-[2-(3-thienyl)ethyl]-L-cysteinate (2) through tosylate intermediates is reported and discussed. These compounds, which combine the properties of the cysteine side-chain with those of the thiophene ring represent both potential bioactive molecules and interesting synthons for the development of new materials.I documenti in IRIS sono protetti da copyright e tutti i diritti sono riservati, salvo diversa indicazione.