MAZZEI, LUCA
MAZZEI, LUCA
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Ricercatori a tempo determinato
An isothermal calorimetry assay for determining steady state kinetic and Ensitrelvir inhibition parameters for SARS-CoV-2 3CL-protease
2024 Mazzei, L.; Ranieri, S.; Silvestri, D.; Greene-Cramer, R.; Cioffi, C.; Montelione, G. T.; Ciurli, S.
Exploring the conformational space of the mobile flap in Sporosarcina pasteurii urease by cryo-electron microscopy
2024 Mazzei, L.; Tria, G.; Ciurli, S.; Cianci, M.
Is bismuth(iii) able to inhibit the activity of urease? Puzzling results in the quest for soluble urease complexes for agrochemical and medicinal applications
2024 Contini, L.; Paul, A.; Mazzei, L.; Ciurli, S.; Roncarati, D.; Braga, D.; Grepioni, F.
Kinetic and structural details of urease inactivation by thiuram disulphides
2024 Mazzei L.; Paul A.; Cianci M.; Devodier M.; Mandelli D.; Carloni P.; Ciurli S.
Metal selectivity and translocation mechanism characterization in proteoliposomes of the transmembrane NiCoT transporter NixA from Helicobacter pylori
2024 Hernandez J.A.; Micus P.S.; Sunga S.A.L.; Mazzei L.; Ciurli S.; Meloni G.
Determination and Kinetic Characterization of a New Potential Inhibitor for AmsI Protein Tyrosine Phosphatase from the Apple Pathogen Erwinia amylovora
2023 Albani S.; Polsinelli I.; Mazzei L.; Musiani F.; Benini S.
Optimized Ebselen-Based Inhibitors of Bacterial Ureases with Nontypical Mode of Action
2023 Macegoniuk K.; Tabor W.; Mazzei L.; Cianci M.; Giurg M.; Olech K.; Burda-Grabowska M.; Kaleta R.; Grabowiecka A.; Mucha A.; Ciurli S.; Berlicki L.
Protocol for production and purification of SARS-CoV-2 3CLpro
2023 Mazzei L.; Greene-Cramer R.; Bafna K.; Jovanovic A.; De Falco A.; Acton T.B.; Royer C.A.; Ciurli S.; Montelione G.T.
Water-Soluble Pyrolysis Products as Novel Urease Inhibitors Safe for Plants and Soil Fauna
2023 Samori', C.; Mazzei, L.; Guidi, E.; Buscaroli, A.; Pasteris, A.; Rombola', A.; Zannoni, D.; Galletti, P.
Inhibition of Urease by Hydroquinones: A Structural and Kinetic Study
2022 Mazzei L.; Cianci M.; Ciurli S.
Steps towards a nature inspired inorganic crystal engineering
2022 Grepioni, Fabrizia; Casali, Lucia; Fiore, Cecilia; Mazzei, Luca; Sun, Renren; Shemchuk, Oleksii; Braga, Dario
Thiocarbamoyl Disulfides as Inhibitors of Urease and Ammonia Monooxygenase: Crystal Engineering for Novel Materials
2022 Casali, L; Mazzei, L; Sun, RR; Chierotti, MR; Gobetto, R; Braga, D; Grepioni, F; Ciurli, S
Correction to: The structure-based reaction mechanism of urease, a nickel dependent enzyme: tale of a long debate (JBIC Journal of Biological Inorganic Chemistry, (2020), 25, 6, (829-845), 10.1007/s00775-020-01808-w)
2021 Mazzei L.; Musiani F.; Ciurli S.
Inhibition of Urease, a Ni-Enzyme: The Reactivity of a Key Thiol With Mono- and Di-Substituted Catechols Elucidated by Kinetic, Structural, and Theoretical Studies
2021 Mazzei L.; Contaldo U.; Musiani F.; Cianci M.; Bagnolini G.; Roberti M.; Ciurli S.
Kinetic and structural analysis of the inactivation of urease by mixed-ligand phosphine halide Ag(I) complexes
2021 Luca Mazzei, Damiano Cirri, Michele Cianci, Luigi Messori, Stefano Ciurli
Medicinal Au(I) compounds targeting urease as prospective antimicrobial agents: unveiling the structural basis for enzyme inhibition
2021 Luca Mazzei, Lara Massei, Michele Cianci, Luigi Messori, Stefano Ciurli
Structure, dynamics, and function of SrnR, a transcription factor for nickel-dependent gene expression
2021 Mazzei L.; Musiani F.; Zerko S.; Kozminski W.; Cianci M.; Beniamino Y.; Ciurli S.; Zambelli B.
Urease
2021 Mazzei, Luca; Ciurli, Stefano
Intrinsic disorder in the nickel-dependent urease network
2020 Zambelli, Barbara; Mazzei, Luca; Ciurli, Stefano
The structure-based reaction mechanism of urease, a nickel dependent enzyme: tale of a long debate
2020 Mazzei L.; Musiani F.; Ciurli S.