DI MARTINO, RITA MARIA CONCETTA
DI MARTINO, RITA MARIA CONCETTA
Collaboratori
Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold
2023 De Lorenzi, Ersilia; Seghetti, Francesca; Tarozzi, Andrea; Pruccoli, Letizia; Contardi, Cecilia; Serra, Massimo; Bisi, Alessandra; Gobbi, Silvia; Vistoli, Giulio; Gervasoni, Silvia; Argentini, Carla; Ghirardo, Giulia; Guarato, Giulia; Orso, Genny; Belluti, Federica; Di Martino, Rita Maria Concetta; Zusso, Morena
Modulation of Amyloid β-induced Microglia Activation and Neuronal Cell Death by Curcumin and Analogues
2022 De Lorenzi E.; Contardi C.; Serra M.; Bisceglia F.; Franceschini D.; Pagetta A.; Zusso M.; Di Martino R.M.C.; Seghetti F.; Belluti F.
Gsk‐3β, fyn, and dyrk1a: Master regulators in neurodegenerative pathways
2021 Demuro S.; Di Martino R.M.C.; Ortega J.A.; Cavalli A.
Curcumin-1,2,3-triazole conjugation for targeting the cancer apoptosis machinery.
2020 Seghetti F., Di Martino R.M.C., Catanzaro E., Bisi A., Gobbi S., Rampa A., Canonico B., Montanari M., Krysko D.V., Papa S., Fimognari C., Belluti F.
Multitarget Compounds for Bipolar Disorder: From Rational Design to Preliminary Pharmacokinetic Evaluation
2020 Di Martino, R. M. C.; Bottegoni, G.; Seghetti, F.; Russo, D.; Penna, I.; De Simone, A.; Ottonello, G.; Mandrup Bertozzi, S.; Armirotti, A.; Bandiera, T.; Belluti, F.; Cavalli, A.
Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson's Disease
2020 Rita Maria Concetta Di Martino; Letizia Pruccoli; Alessandra Bisi; Silvia Gobbi; Angela Rampa; Ana Martinez; Concepción Pérez; Loreto Martinez-Gonzalez; Maria Paglione; Elia Di Schiavi; Francesca Seghetti; Andrea Tarozzi; Federica Belluti
Investigating Drug-Target Residence Time in Kinases through Enhanced Sampling Simulations
2019 Gobbo D.; Piretti V.; Di Martino R.M.C.; Tripathi S.K.; Giabbai B.; Storici P.; Demitri N.; Girotto S.; Decherchi S.; Cavalli A.
Identification of chalcone-based antileishmanial agents targeting trypanothione reductase
2018 Ortalli, Margherita; Ilari, Andrea; Colotti, Gianni; De Ionna, Ilenia; Battista, Theo; Bisi, Alessandra; Gobbi, Silvia; Rampa, Angela; Di Martino, Rita M.C.; Gentilomi, Giovanna A.; Varani, Stefania; Belluti, Federica*
Phenolic 1,3-diketones attenuate lipopolysaccharide-induced inflammatory response by an alternative magnesium-mediated mechanism
2017 Zusso, Morena; Mercanti, Giulia; Belluti, Federica; Di Martino, Rita Maria Concetta; Pagetta, Andrea; Marinelli, Carla; Brun, Paola; Ragazzi, Eugenio; Rita, Lo; Stifani, Stefano; Giusti, Pietro; Moro, Stefano
Recent progress on curcumin-based therapeutics: a patent review (2012-2016). Part I: Curcumin
2017 Di Martino, Rita Maria Concetta; Luppi, Barbara; Bisi, Alessandra; Gobbi, Silvia; Rampa, Angela; Abruzzo, Angela; Belluti, Federica
Recent progress on curcumin-based therapeutics: a patent review (2012-2016). Part II: curcumin derivatives in cancer and neurodegeneration
2017 Di Martino, Rita Maria Concetta; Bisi, Alessandra; Rampa, Angela; Gobbi, Silvia; Belluti, Federica
Naturally inspired molecules as multifunctional agents for Alzheimer's disease treatment
2016 Rampa, Angela; Tarozzi, Andrea; Mancini, Francesca; Pruccoli, Letizia; Di Martino, Rita Maria Concetta; Gobbi, Silvia; Bisi, Alessandra; De Simone, Angela; Palomba, Francesco; Zaccheroni, Nelsi; Belluti, Federica
Versatility of the Curcumin Scaffold: Discovery of Potent and Balanced Dual BACE-1 and GSK-3β Inhibitors
2016 Di Martino, Rita Maria Concetta; De Simone, Angela; Andrisano, Vincenza; Bisignano, Paola; Bisi, Alessandra; Gobbi, Silvia; Rampa, Angela; Fato, Romana; Bergamini, Christian; Perez, Daniel I.; Martinez, Ana; Bottegoni, Giovanni; Cavalli, Andrea; Belluti, Federica
From AChE to BACE1 inhibitors: The role of the amine on the indanone scaffold
2015 Angela, Rampa; Francesca, Mancini; Angela, De Simone; Federico, Falchi; Federica, Belluti; Rita Maria, Concetta Di Martino; Silvia, Gobbi; Vincenza, Andrisano; Andrea, Tarozzi; Manuela, Bartolini; Andrea, Cavalli; Alessandra, Bisi
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold | De Lorenzi, Ersilia; Seghetti, Francesca; Tarozzi, Andrea; Pruccoli, Letizia; Contardi, Cecilia; ...Serra, Massimo; Bisi, Alessandra; Gobbi, Silvia; Vistoli, Giulio; Gervasoni, Silvia; Argentini, Carla; Ghirardo, Giulia; Guarato, Giulia; Orso, Genny; Belluti, Federica; Di Martino, Rita Maria Concetta; Zusso, Morena | 2023-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold.pdf; 1-s2.0-S0223523423002635-mmc1.pdf |
Modulation of Amyloid β-induced Microglia Activation and Neuronal Cell Death by Curcumin and Analogues | De Lorenzi E.; Contardi C.; Serra M.; Bisceglia F.; Franceschini D.; Pagetta A.; Zusso M.; Di Mar...tino R.M.C.; Seghetti F.; Belluti F. | 2022-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | ijms-23-04381-v3.pdf |
Gsk‐3β, fyn, and dyrk1a: Master regulators in neurodegenerative pathways | Demuro S.; Di Martino R.M.C.; Ortega J.A.; Cavalli A. | 2021-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | Demuroetal2021.pdf |
Curcumin-1,2,3-triazole conjugation for targeting the cancer apoptosis machinery. | Seghetti F., Di Martino R.M.C., Catanzaro E., Bisi A., Gobbi S., Rampa A., Canonico B., Montanari... M., Krysko D.V., Papa S., Fimognari C., Belluti F. | 2020-01-01 | MOLECULES | - | 1.01 Articolo in rivista | Molecules_2020_Curcumins.pdf |
Multitarget Compounds for Bipolar Disorder: From Rational Design to Preliminary Pharmacokinetic Evaluation | Di Martino, R. M. C.; Bottegoni, G.; Seghetti, F.; Russo, D.; Penna, I.; De Simone, A.; Ottonello..., G.; Mandrup Bertozzi, S.; Armirotti, A.; Bandiera, T.; Belluti, F.; Cavalli, A. | 2020-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | Post print.pdf |
Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson's Disease | Rita Maria Concetta Di Martino; Letizia Pruccoli; Alessandra Bisi; Silvia Gobbi; Angela Rampa; An...a Martinez; Concepción Pérez; Loreto Martinez-Gonzalez; Maria Paglione; Elia Di Schiavi; Francesca Seghetti; Andrea Tarozzi; Federica Belluti | 2020-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | Nrf2 Inducer for the Treatment of Parkinson’s Disease.pdf |
Investigating Drug-Target Residence Time in Kinases through Enhanced Sampling Simulations | Gobbo D.; Piretti V.; Di Martino R.M.C.; Tripathi S.K.; Giabbai B.; Storici P.; Demitri N.; Girot...to S.; Decherchi S.; Cavalli A. | 2019-01-01 | JOURNAL OF CHEMICAL THEORY AND COMPUTATION | - | 1.01 Articolo in rivista | - |
Identification of chalcone-based antileishmanial agents targeting trypanothione reductase | Ortalli, Margherita; Ilari, Andrea; Colotti, Gianni; De Ionna, Ilenia; Battista, Theo; Bisi, Ales...sandra; Gobbi, Silvia; Rampa, Angela; Di Martino, Rita M.C.; Gentilomi, Giovanna A.; Varani, Stefania; Belluti, Federica* | 2018-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | ortalli2018.pdf |
Phenolic 1,3-diketones attenuate lipopolysaccharide-induced inflammatory response by an alternative magnesium-mediated mechanism | Zusso, Morena; Mercanti, Giulia; Belluti, Federica; Di Martino, Rita Maria Concetta; Pagetta, And...rea; Marinelli, Carla; Brun, Paola; Ragazzi, Eugenio; Rita, Lo; Stifani, Stefano; Giusti, Pietro; Moro, Stefano | 2017-01-01 | BRITISH JOURNAL OF PHARMACOLOGY | - | 1.01 Articolo in rivista | phenolic.accept.pdf |
Recent progress on curcumin-based therapeutics: a patent review (2012-2016). Part I: Curcumin | Di Martino, Rita Maria Concetta; Luppi, Barbara; Bisi, Alessandra; Gobbi, Silvia; Rampa, Angela; ...Abruzzo, Angela; Belluti, Federica | 2017-01-01 | EXPERT OPINION ON THERAPEUTIC PATENTS | - | 1.01 Articolo in rivista | - |
Recent progress on curcumin-based therapeutics: a patent review (2012-2016). Part II: curcumin derivatives in cancer and neurodegeneration | Di Martino, Rita Maria Concetta; Bisi, Alessandra; Rampa, Angela; Gobbi, Silvia; Belluti, Federica | 2017-01-01 | EXPERT OPINION ON THERAPEUTIC PATENTS | - | 1.01 Articolo in rivista | - |
Naturally inspired molecules as multifunctional agents for Alzheimer's disease treatment | Rampa, Angela; Tarozzi, Andrea; Mancini, Francesca; Pruccoli, Letizia; Di Martino, Rita Maria Con...cetta; Gobbi, Silvia; Bisi, Alessandra; De Simone, Angela; Palomba, Francesco; Zaccheroni, Nelsi; Belluti, Federica | 2016-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-21-00643.pdf |
Versatility of the Curcumin Scaffold: Discovery of Potent and Balanced Dual BACE-1 and GSK-3β Inhibitors | Di Martino, Rita Maria Concetta; De Simone, Angela; Andrisano, Vincenza; Bisignano, Paola; Bisi, ...Alessandra; Gobbi, Silvia; Rampa, Angela; Fato, Romana; Bergamini, Christian; Perez, Daniel I.; Martinez, Ana; Bottegoni, Giovanni; Cavalli, Andrea; Belluti, Federica | 2016-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | AM11585-579953.pdf |
From AChE to BACE1 inhibitors: The role of the amine on the indanone scaffold | Angela, Rampa; Francesca, Mancini; Angela, De Simone; Federico, Falchi; Federica, Belluti; Rita M...aria, Concetta Di Martino; Silvia, Gobbi; Vincenza, Andrisano; Andrea, Tarozzi; Manuela, Bartolini; Andrea, Cavalli; Alessandra, Bisi | 2015-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |