BISI, ALESSANDRA
BISI, ALESSANDRA
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di IIa fascia
Chalcones induce apoptosis, autophagy and reduce spreading in osteosarcoma 3D models
2024 Rossi M.; Pellegrino C.; Rydzyk M.M.; Farruggia G.; de Biase D.; Cetrullo S.; D'Adamo S.; Bisi A.; Blasi P.; Malucelli E.; Cappadone C.; Gobbi S.
Chromone-based small molecules for multistep shutdown of arachidonate pathway: Simultaneous inhibition of COX-2, 15-LOX and mPGES-1 enzymes
2024 Elzahhar P.A.; Orioli R.; Hassan N.W.; Gobbi S.; Belluti F.; Labib H.F.; El-Yazbi A.F.; Nassra R.; Belal A.S.F.; Bisi A.
Naturally Inspired Coumarin Derivatives in Alzheimer’s Disease Drug Discovery: Latest Advances and Current Challenges
2024 Orioli R.; Belluti F.; Gobbi S.; Rampa A.; Bisi A.
Switching from Aromatase Inhibitors to Dual Targeting Flavonoid-Based Compounds for Breast Cancer Treatment
2023 Gobbi S.; Martini S.; Rozza R.; Spinello A.; Caciolla J.; Rampa A.; Belluti F.; Zaffaroni N.; Magistrato A.; Bisi A.
Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold
2023 De Lorenzi, Ersilia; Seghetti, Francesca; Tarozzi, Andrea; Pruccoli, Letizia; Contardi, Cecilia; Serra, Massimo; Bisi, Alessandra; Gobbi, Silvia; Vistoli, Giulio; Gervasoni, Silvia; Argentini, Carla; Ghirardo, Giulia; Guarato, Giulia; Orso, Genny; Belluti, Federica; Di Martino, Rita Maria Concetta; Zusso, Morena
Hitting drug-resistant malaria infection with triazole-linked flavonoid–chloroquine hybrid compounds
2022 Seghetti, Francesca; Belluti, Federica; Rampa, Angela; Gobbi, Silvia; Legac, Jenny; Parapini, Silvia; Basilico, Nicoletta; Bisi, Alessandra
Interplay Between Endocannabinoid System and Neurodegeneration: Focus on Polypharmacology
2022 Seghetti F.; Gobbi S.; Belluti F.; Rampa A.; Bisi A.
Natural-like Chalcones with Antitumor Activity on Human MG63 Osteosarcoma Cells
2022 Rossi, Martina; Cappadone, Concettina; Picone, Giovanna; Bisi, Alessandra; Farruggia, Giovanna; Belluti, Federica; Blasi, Paolo; Gobbi, Silvia; Malucelli, Emil
Single-digit nanomolar inhibitors lock the aromatase active site via a dualsteric targeting strategy
2022 Caciolla J.; Martini S.; Spinello A.; Belluti F.; Bisi A.; Zaffaroni N.; Magistrato A.; Gobbi S.
Targeting neuronal calcium channels and GSK3β for Alzheimer's disease with naturally-inspired Diels-Alder adducts
2022 Bisi, A.; Feoli, A.; Trezza, A.; Viejo, L.; Formaggio, F.; Bartolini, M.; Belluti, F.; Gobbi, S.; Spiga, O.; Caprini, M.; de los Rios, C.; Castellano, S.; Rampa, A.
Balanced dual acting compounds targeting aromatase and estrogen receptor α as an emerging therapeutic opportunity to counteract estrogen responsive breast cancer
2021 Caciolla, J.; Martini, S.; Spinello, A.; Pavlin, M.; Turrini, E.; Simonelli, F.; Belluti, F.; Rampa, A.; Bisi, A.; Fimognari, C.; Zaffaroni, N.; Gobbi, S.; Magistrato, A.
Flavonoid-inspired vascular disrupting agents: Exploring flavone-8-acetic acid and derivatives in the new century
2021 Gobbi S.; Belluti F.; Rampa A.; Bisi A.
Improved eradication efficacy of a combination of newly identified antimicrobial agents in C. albicans and S. aureus mixed-species biofilm
2021 Bonvicini F.; Belluti F.; Bisi A.; Gobbi S.; Manet I.; Gentilomi G.A.
Multifaceted activity of polyciclic MDR revertant agents in drug-resistant leukemic cells: Role of the spacer
2021 Caciolla J.; Picone G.; Farruggia G.; Valenti D.; Rampa A.; Malucelli E.; Belluti F.; Trezza A.; Spiga O.; Iotti S.; Gobbi S.; Cappadone C.; Bisi A.
New Coumarin derivatives as cholinergic and cannabinoid system modulators
2021 Montanari S.; Allara M.; Scalvini L.; Kostrzewa M.; Belluti F.; Gobbi S.; Naldi M.; Rivara S.; Bartolini M.; Ligresti A.; Bisi A.; Rampa A.
Tackling Alzheimer's Disease with Existing Drugs:A Promising Strategy for Bypassing Obstacles
2021 Rampa, Angela; Gobbi, Silvia; Belluti, Federica; Bisi, Alessandra
Curcumin-1,2,3-triazole conjugation for targeting the cancer apoptosis machinery.
2020 Seghetti F., Di Martino R.M.C., Catanzaro E., Bisi A., Gobbi S., Rampa A., Canonico B., Montanari M., Krysko D.V., Papa S., Fimognari C., Belluti F.
Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson's Disease
2020 Rita Maria Concetta Di Martino; Letizia Pruccoli; Alessandra Bisi; Silvia Gobbi; Angela Rampa; Ana Martinez; Concepción Pérez; Loreto Martinez-Gonzalez; Maria Paglione; Elia Di Schiavi; Francesca Seghetti; Andrea Tarozzi; Federica Belluti
Reconsidering Aromatase for Breast Cancer Treatment: New Roles for an Old Target
2020 Caciolla J.; Bisi A.; Belluti F.; Rampa A.; Gobbi S.
Targeting Orthosteric and Allosteric Pockets of Aromatase via Dual-Mode Novel Azole Inhibitors
2020 Caciolla, J.; Spinello, A.; Martini, S.; Bisi, A.; Zaffaroni, N.; Gobbi, S.; Magistrato, A.