BARTOLINI, MANUELA
BARTOLINI, MANUELA
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di Ia fascia
Chromatographia
In corso di stampa M. Bartolini
Cholinesterase Inhibition for the Treatment of Neurodegenerative Diseases: Assay Methodologies and Reference Compounds
2025 Bartolini, M.
Isofagomine-coumarin hybrids: bridging cancer and Alzheimer's disease
2025 Santos Evangelista, T. C.; González-Bakker, A.; Puerta, A.; Poeta, E.; Monti, B.; Naldi, M.; Bolognesi, M. L.; Bartolini, M.; Vaaland Holmgard, I. C.; Butt, A.; Padrón, J. M.; Fernández-Bolaños, J. G.; Sydnes, M. O.; Lindbäck, E.; López, Ó.
Multi-Target Glitazones for Modulating Peroxisome Proliferator-Activated Receptor-γ, Cyclooxygenase-2, and Carbonic Anhydrases for the Management of Metabolic Dysfunction
2025 Elzahhar, Perihan A.; Nematalla, Hisham A.; Abouayana, Malak A.; El Ashry, El Sayed H.; Balbaa, Mahmoud; Petreni, Andrea; Nassra, Rasha; Yassin, Hend A.; Kamel, Yasmine N.; Elrewiny, Mohamed A.; Agami, Mahmoud A.; Makkar, Monica; Sai, Minh; Merk, Daniel; Labib, Hala F.; Spagnuolo, Rosaria; Naldi, Marina; Bartolini, Manuela; El-Hawash, Soad A.; Supuran, Claudiu T.; Belal, Ahmed S. F.; El-Yazbi, Ahmed F.
Association between Albumin Alterations and Renal Function in Patients with Type 2 Diabetes Mellitus
2024 Nugnes, M.; Baldassarre, M.; Ribichini, D.; Tedesco, D.; Capelli, I.; Vetrano, D.; Marchignoli, F.; Brodosi, L.; Pompili, E.; Petroni, M. L.; La Manna, G.; Marchesini, G.; Naldi, M.; Bartolini, M.
Exploiting the pyrazole scaffold for multipotent agents in Alzheimer’s disease
2024 Orioli, Rebecca; Feoli, Alessandra; Gobbi, Silvia; Belluti, Federica; Bartolini, Manuela; Castellano, Sabrina; Bisi, Alessandra
HSA-nanobinders crafted from bioresponsive prodrugs for combined cancer chemoimmunotherapy–an in vitro exploration
2024 Tubertini M.; Menilli L.; Milani C.; Martini C.; Navacchia M.L.; Nugnes M.; Bartolini M.; Naldi M.; Tedesco D.; Martella E.; Guerrini A.; Ferroni C.; Moret F.; Varchi G.
Novel multifunctional tacrine–donepezil hybrids against Alzheimer's disease: Design synthesis and bioactivity studies
2024 Bayraktar, Gülşah; Bartolini, Manuela; Bolognesi, Maria Laura; Erdoğan, Mumin Alper; Armağan, Güliz; Bayır, Ece; Şendemir, Aylin; Bagetta, Donatella; Alcaro, Stefano; Alptüzün, Vildan
Stepwise Structural Simplification of the Dihydroxyanthraquinone Moiety of a Multitarget Rhein-Based Anti-Alzheimer Lead to Improve Drug Metabolism and Pharmacokinetic Properties
2024 Pont, Caterina; Sampietro, Anna; Pérez-Areales, F. Javier; Cristiano, Nunzia; Albalat, Agustí; Pérez, Belén; Bartolini, Manuela; De Simone, Angela; Andrisano, Vincenza; Barenys, Marta; Teixidó, Elisabet; Sabaté, Raimon; Loza, M. Isabel; Brea, José; Muñoz-Torrero, Diego
The novel SMYD3 inhibitor EM127 impairs DNA repair response to chemotherapy-induced DNA damage and reverses cancer chemoresistance
2024 Sanese, Paola; De Marco, Katia; Lepore Signorile, Martina; La Rocca, Francesca; Forte, Giovanna; Latrofa, Marialaura; Fasano, Candida; Disciglio, Vittoria; Di Nicola, Elisabetta; Pantaleo, Antonino; Bianco, Giusy; Spilotro, Vito; Ferroni, Claudia; Tubertini, Matilde; Labarile, Nicoletta; De Marinis, Lucia; Armentano, Raffaele; Gigante, Gianluigi; Lantone, Valerio; Lantone, Giuliano; Naldi, Marina; Bartolini, Manuela; Varchi, Greta; Del Rio, Alberto; Grossi, Valentina; Simone, Cristiano
Exopolysaccharides from vaginal lactobacilli modulate microbial biofilms
2023 Giordani B.; Naldi M.; Croatti V.; Parolin C.; Erdogan U.; Bartolini M.; Vitali B.
Exopolysaccharides released by vaginal Lactobacillus strains: chemical characterization and modulation of biofilm formation.
2023 Carola Parolin, Barbara Giordani, Marina Naldi, Ülfet Erdoğan, Vanessa Croatti, Manuela Bartolini, Beatrice Vitali
Galantamine-memantine hybrids for Alzheimer's disease: The influence of linker rigidity in biological activity and pharmacokinetic properties
2023 Basagni, Filippo; Ortega, Jose A; Bertozzi, Sine M; Armirotti, Andrea; Summa, Maria; Bertorelli, Rosalia; Bartolini, Manuela; Mellor, Ian R; Bedeschi, Martina; Bottegoni, Giovanni; Lembo, Vittorio; Minarini, Anna; Cavalli, Andrea; Rosini, Michela
Impact of Lactobacillus exopolysaccharides on vaginal microbial biofilms
2023 Beatrice Vitali, Barbara Giordani, Marina Naldi, Ülfet Erdoğan, Vanessa Croatti, Manuela Bartolini, Carola Parolin
Microsampling and enantioselective liquid chromatography coupled to mass spectrometry for chiral bioanalysis of novel psychoactive substances
2023 Protti, Michele; Varfaj, Ina; Carotti, Andrea; Tedesco, Daniele; Bartolini, Manuela; Favilli, Alessandro; Gerli, Sandro; Mercolini, Laura; Sardella, Roccaldo
Quinolinetrione-tacrine hybrids as multi-target-directed ligands against Alzheimer's disease
2023 Uliassi, E; Bergamini, C; Rizzardi, N; Naldi, M; Cores, A; Bartolini, M; Menéndez, JC; Bolognesi, ML
Discovery and in Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's Disease
2022 Codony S.; Pont C.; Grinan-Ferre C.; Di Pede-Mattatelli A.; Calvo-Tusell C.; Feixas F.; Osuna S.; Jarne-Ferrer J.; Naldi M.; Bartolini M.; Loza M.I.; Brea J.; Perez B.; Bartra C.; Sanfeliu C.; Juarez-Jimenez J.; Morisseau C.; Hammock B.D.; Pallas M.; Vazquez S.; Munoz-Torrero D.
Discovery of Dual Aβ/Tau Inhibitors and Evaluation of Their Therapeutic Effect on a Drosophila Model of Alzheimer's Disease
2022 Gandini, Annachiara; Gonçalves, Ana Elisa; Strocchi, Silvia; Albertini, Claudia; Janočková, Jana; Tramarin, Anna; Grifoni, Daniela; Poeta, Eleonora; Soukup, Ondrej; Muñoz-Torrero, Diego; Monti, Barbara; Sabaté, Raimon; Bartolini, Manuela; Legname, Giuseppe; Bolognesi, Maria Laura
Discovery of the 4-aminopiperidine-based compound EM127 for the site-specific covalent inhibition of SMYD3
2022 Parenti, Md; Naldi, M; Manoni, E; Fabini, E; Cederfelt, D; Talibov, Vo; Gressani, V; Guven, U; Grossi, V; Fasano, C; Sanese, P; De Marco, K; Shtil, Aa; Kurkin, Av; Altieri, A; Danielson, Uh; Caretti, G; Simone, C; Varchi, G; Bartolini, M; Del Rio, A
HSA-Binding Prodrugs-Based Nanoparticles Endowed with Chemo and Photo-Toxicity against Breast Cancer
2022 Rapozzi V.; Moret F.; Menilli L.; Guerrini A.; Tedesco D.; Naldi M.; Bartolini M.; Gani M.; Zorzet S.; Columbaro M.; Milani C.; Martini C.; Ferroni C.; Varchi G.
| Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
|---|---|---|---|---|---|---|
| Chromatographia | M. Bartolini | 9999-01-01 | CHROMATOGRAPHIA | - | 8.01 Ruolo editoriale in rivista | - |
| Cholinesterase Inhibition for the Treatment of Neurodegenerative Diseases: Assay Methodologies and Reference Compounds | Bartolini, M. | 2025-01-01 | - | Springer Nature | 2.01 Capitolo / saggio in libro | - |
| Isofagomine-coumarin hybrids: bridging cancer and Alzheimer's disease | Santos Evangelista, T. C.; González-Bakker, A.; Puerta, A.; Poeta, E.; Monti, B.; Naldi, M.; Bolo...gnesi, M. L.; Bartolini, M.; Vaaland Holmgard, I. C.; Butt, A.; Padrón, J. M.; Fernández-Bolaños, J. G.; Sydnes, M. O.; Lindbäck, E.; López, Ó. | 2025-01-01 | CHEMICO-BIOLOGICAL INTERACTIONS | - | 1.01 Articolo in rivista | - |
| Multi-Target Glitazones for Modulating Peroxisome Proliferator-Activated Receptor-γ, Cyclooxygenase-2, and Carbonic Anhydrases for the Management of Metabolic Dysfunction | Elzahhar, Perihan A.; Nematalla, Hisham A.; Abouayana, Malak A.; El Ashry, El Sayed H.; Balbaa, M...ahmoud; Petreni, Andrea; Nassra, Rasha; Yassin, Hend A.; Kamel, Yasmine N.; Elrewiny, Mohamed A.; Agami, Mahmoud A.; Makkar, Monica; Sai, Minh; Merk, Daniel; Labib, Hala F.; Spagnuolo, Rosaria; Naldi, Marina; Bartolini, Manuela; El-Hawash, Soad A.; Supuran, Claudiu T.; Belal, Ahmed S. F.; El-Yazbi, Ahmed F. | 2025-01-01 | ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE | - | 1.01 Articolo in rivista | - |
| Association between Albumin Alterations and Renal Function in Patients with Type 2 Diabetes Mellitus | Nugnes, M.; Baldassarre, M.; Ribichini, D.; Tedesco, D.; Capelli, I.; Vetrano, D.; Marchignoli, F....; Brodosi, L.; Pompili, E.; Petroni, M. L.; La Manna, G.; Marchesini, G.; Naldi, M.; Bartolini, M. | 2024-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | Nugnes_ijms-25-03168.pdf; Nugnes_ijms-2842343-supplementary.pdf |
| Exploiting the pyrazole scaffold for multipotent agents in Alzheimer’s disease | Orioli, Rebecca; Feoli, Alessandra; Gobbi, Silvia; Belluti, Federica; Bartolini, Manuela; Castell...ano, Sabrina; Bisi, Alessandra | 2024-01-01 | - | - | 4.03 Poster | - |
| HSA-nanobinders crafted from bioresponsive prodrugs for combined cancer chemoimmunotherapy–an in vitro exploration | Tubertini M.; Menilli L.; Milani C.; Martini C.; Navacchia M.L.; Nugnes M.; Bartolini M.; Naldi M....; Tedesco D.; Martella E.; Guerrini A.; Ferroni C.; Moret F.; Varchi G. | 2024-01-01 | FRONTIERS IN CHEMISTRY | - | 1.01 Articolo in rivista | fchem-12-1378233 (1).pdf; Supplementary data.pdf |
| Novel multifunctional tacrine–donepezil hybrids against Alzheimer's disease: Design synthesis and bioactivity studies | Bayraktar, Gülşah; Bartolini, Manuela; Bolognesi, Maria Laura; Erdoğan, Mumin Alper; Armağan, Gül...iz; Bayır, Ece; Şendemir, Aylin; Bagetta, Donatella; Alcaro, Stefano; Alptüzün, Vildan | 2024-01-01 | ARCHIV DER PHARMAZIE | - | 1.01 Articolo in rivista | Archiv der Pharmazie - 2024 - Bayraktar - Novel multifunctional tacrine donepezil hybrids against Alzheimer s disease .pdf; Supplemental Material - Novel Compounds and Biological Screening Results_1.doc; Supplemental Material - Novel Compounds and Biological Screening Results_2.docx |
| Stepwise Structural Simplification of the Dihydroxyanthraquinone Moiety of a Multitarget Rhein-Based Anti-Alzheimer Lead to Improve Drug Metabolism and Pharmacokinetic Properties | Pont, Caterina; Sampietro, Anna; Pérez-Areales, F. Javier; Cristiano, Nunzia; Albalat, Agustí; Pé...rez, Belén; Bartolini, Manuela; De Simone, Angela; Andrisano, Vincenza; Barenys, Marta; Teixidó, Elisabet; Sabaté, Raimon; Loza, M. Isabel; Brea, José; Muñoz-Torrero, Diego | 2024-01-01 | PHARMACEUTICS | - | 1.01 Articolo in rivista | pharmaceutics-16-00982.pdf; pharmaceutics-3101614-supplementary.pdf |
| The novel SMYD3 inhibitor EM127 impairs DNA repair response to chemotherapy-induced DNA damage and reverses cancer chemoresistance | Sanese, Paola; De Marco, Katia; Lepore Signorile, Martina; La Rocca, Francesca; Forte, Giovanna; ...Latrofa, Marialaura; Fasano, Candida; Disciglio, Vittoria; Di Nicola, Elisabetta; Pantaleo, Antonino; Bianco, Giusy; Spilotro, Vito; Ferroni, Claudia; Tubertini, Matilde; Labarile, Nicoletta; De Marinis, Lucia; Armentano, Raffaele; Gigante, Gianluigi; Lantone, Valerio; Lantone, Giuliano; Naldi, Marina; Bartolini, Manuela; Varchi, Greta; Del Rio, Alberto; Grossi, Valentina; Simone, Cristiano | 2024-01-01 | JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH | - | 1.01 Articolo in rivista | Sanese et al J Exp Clin Cancer Res_2024_43_151-compresso.pdf; Sanese et al J Exp Clin Cancer Res_2024_43_151-supplementary_file_1.pdf; Sanese_et_al_supplementary_dfile_2_13046_2024_3078_MOESM2_ESM.xlsx |
| Exopolysaccharides from vaginal lactobacilli modulate microbial biofilms | Giordani B.; Naldi M.; Croatti V.; Parolin C.; Erdogan U.; Bartolini M.; Vitali B. | 2023-01-01 | MICROBIAL CELL FACTORIES | - | 1.01 Articolo in rivista | Giordani 2023_EPS.pdf; 12934_2023_2053_MOESM1_ESM.pdf |
| Exopolysaccharides released by vaginal Lactobacillus strains: chemical characterization and modulation of biofilm formation. | Carola Parolin, Barbara Giordani, Marina Naldi, Ülfet Erdoğan, Vanessa Croatti, Manuela Bartolini..., Beatrice Vitali | 2023-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
| Galantamine-memantine hybrids for Alzheimer's disease: The influence of linker rigidity in biological activity and pharmacokinetic properties | Basagni, Filippo; Ortega, Jose A; Bertozzi, Sine M; Armirotti, Andrea; Summa, Maria; Bertorelli, ...Rosalia; Bartolini, Manuela; Mellor, Ian R; Bedeschi, Martina; Bottegoni, Giovanni; Lembo, Vittorio; Minarini, Anna; Cavalli, Andrea; Rosini, Michela | 2023-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Eur. J. Med.Chem. 2023.pdf; 1-s2.0-S0223523423007705-mmc1.docx |
| Impact of Lactobacillus exopolysaccharides on vaginal microbial biofilms |
Beatrice Vitali, Barbara Giordani, Marina Naldi, Ülfet Erdoğan, Vanessa Croatti, Manuela Bartolin...i, Carola Parolin |
2023-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
| Microsampling and enantioselective liquid chromatography coupled to mass spectrometry for chiral bioanalysis of novel psychoactive substances | Protti, Michele; Varfaj, Ina; Carotti, Andrea; Tedesco, Daniele; Bartolini, Manuela; Favilli, Ale...ssandro; Gerli, Sandro; Mercolini, Laura; Sardella, Roccaldo | 2023-01-01 | TALANTA | - | 1.01 Articolo in rivista | Protti_et_al_Talanta_257(2023)124332.pdf; 1-s2.0-S0039914023000838-mmc1.docx |
| Quinolinetrione-tacrine hybrids as multi-target-directed ligands against Alzheimer's disease | Uliassi, E; Bergamini, C; Rizzardi, N; Naldi, M; Cores, A; Bartolini, M; Menéndez, JC; Bolognesi, ML | 2023-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | 1-s2.0-S0968089623002675-main.pdf; 1-s2.0-S0968089623002675-mmc1.docx |
| Discovery and in Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's Disease | Codony S.; Pont C.; Grinan-Ferre C.; Di Pede-Mattatelli A.; Calvo-Tusell C.; Feixas F.; Osuna S.;... Jarne-Ferrer J.; Naldi M.; Bartolini M.; Loza M.I.; Brea J.; Perez B.; Bartra C.; Sanfeliu C.; Juarez-Jimenez J.; Morisseau C.; Hammock B.D.; Pallas M.; Vazquez S.; Munoz-Torrero D. | 2022-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | 2022_acs.jmedchem.1c02150.pdf |
| Discovery of Dual Aβ/Tau Inhibitors and Evaluation of Their Therapeutic Effect on a Drosophila Model of Alzheimer's Disease | Gandini, Annachiara; Gonçalves, Ana Elisa; Strocchi, Silvia; Albertini, Claudia; Janočková, Jana;... Tramarin, Anna; Grifoni, Daniela; Poeta, Eleonora; Soukup, Ondrej; Muñoz-Torrero, Diego; Monti, Barbara; Sabaté, Raimon; Bartolini, Manuela; Legname, Giuseppe; Bolognesi, Maria Laura | 2022-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | acschemneuro.2c00357.pdf; cn2c00357_si_001.pdf |
| Discovery of the 4-aminopiperidine-based compound EM127 for the site-specific covalent inhibition of SMYD3 | Parenti, Md; Naldi, M; Manoni, E; Fabini, E; Cederfelt, D; Talibov, Vo; Gressani, V; Guven, U; Gr...ossi, V; Fasano, C; Sanese, P; De Marco, K; Shtil, Aa; Kurkin, Av; Altieri, A; Danielson, Uh; Caretti, G; Simone, C; Varchi, G; Bartolini, M; Del Rio, A | 2022-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Parenti et al_EJMC_2022_post_print.pdf |
| HSA-Binding Prodrugs-Based Nanoparticles Endowed with Chemo and Photo-Toxicity against Breast Cancer | Rapozzi V.; Moret F.; Menilli L.; Guerrini A.; Tedesco D.; Naldi M.; Bartolini M.; Gani M.; Zorze...t S.; Columbaro M.; Milani C.; Martini C.; Ferroni C.; Varchi G. | 2022-01-01 | CANCERS | - | 1.01 Articolo in rivista | Rapozzi et al_cancers-14-00877.pdf |