PIAZZI, LORNA

PIAZZI, LORNA  

DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE  

Assegnisti  

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Risultati 1 - 20 di 36 (tempo di esecuzione: 0.021 secondi).
Titolo Autore(i) Anno Periodico Editore Tipo File
1,4-dihydropyridine derivatives as calcium channel modulators: the role of 3-methoxy-flavone moiety R. Budriesi; A. Bisi; P. Ioan; A. Rampa; S. Gobbi; F. Belluti; L. Piazzi; P. Valenti; A. Chiarini 2005-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valen...ti P.; Recanatini M. 2003-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Caval...li A.; Recanatini M.; Valenti P. 2001-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Analogues of the dual acetylcholinesterase inhibitor AP2238: synthesis and SAR L. Piazzi; M. Bartolini; F. Belluti; A. Bisi; A. Cavalli; S. Gobbi; A. Rampa; P. Valenti 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
Benzofuran-Based Hybrid Compounds for the Inhibition of Cholinesterase Activity, Abeta Amyloid Aggregation, and Abeta Neurotoxicity S. Rizzo; C. Riviere; L. Piazzi; A. Bisi; S. Gobbi; M. Bartolini; V. Andrisano; F. Morroni; A. Ta...rozzi; J. P. Monti; A. Rampa 2008-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Benzophenone derivatives as Inhibitors of Acetylcholinesterase F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; M. Bartolini; A. Cavalli; P. Valenti 2005-01-01 - s.n 4.02 Riassunto (Abstract) -
CHOLINESTERASE INHIBITORS: SAR AND ENZYME INHIBITORY ACTIVITY OF 3-[omega-(BENZYLMETHYLAMINO)ALKOXY]XANTHEN-9-ONES L. Piazzi; F. Belluti; A. Bisi; S. Gobbi; S. Rizzo; M. Bartolini; V. Andrisano; M. Recanatini; A.... Rampa 2007-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Cholinesterase inhibitors: xanthostigmine derivatives blocking the acetylcholinesterase-induced beta-amyloid aggregation. Belluti F.; Rampa A.; Piazzi L.; Bisi A.; Gobbi S.; Bartolini M.; Andrisano V.; Cavalli A.; Recan...atini M.; Valenti P. 2005-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Complementary medicinal chemistry-driven strategies toward new antitrypanosomal and antileishmanial lead drug candidates Cavalli A; Lizzi F ; Bongarzone S ; Belluti F; Piazzi L ; Bolognesi ML 2010-01-01 FEMS IMMUNOLOGY AND MEDICAL MICROBIOLOGY - 1.01 Articolo in rivista -
Derivati a struttura benzofenonica come inibitori dell'acetilcolinesterasi F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; V. Andrisano; M. Bartolini; A. Cavalli; M. Re...canatini; P. Valenti 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
Design, synthesis, and evaluation of benzophenone derivatives as novel acetylcholinesterase inhibitors F. Belluti; L. Piazzi; A. Bisi; S. Gobbi; M. Bartolini;
A. Cavalli; P. Valenti; A. Rampa
2009-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Development of a Focused Library of Triazole-Linked Privileged-Structure-Based Conjugates Leading to the Discovery of Novel Phenotypic Hits against Protozoan Parasitic Infections Uliassi, Elisa; Piazzi, Lorna; Belluti, Federica; Mazzanti, Andrea; Kaiser, Marcel; Brun, Reto; M...oraes, Carolina B.; Freitas-Junior, Lucio H.; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Borsari, Chiara; Costi, Maria Paola; Bolognesi, Maria Laura* 2018-01-01 CHEMMEDCHEM - 1.01 Articolo in rivista -
Enantioselective nonsteroidal aromatase inhibitors identified through a multidisciplinary medicinal chemistry approach Cavalli A.; Bisi A.; Bertucci C.; Rosini C.; Paluszcak A.; Gobbi S.; Giorgio E.; Rampa A.; Bellut...i F.; Piazzi L.; Valenti P.; Hartmann R.W.; Recanatini M. 2005-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Extensive SAR and computational studies of 3-{4-[(benzylmethylamino)methyl]phenyl}-6,7-dimethoxy-2H-2-chromenone (AP2238) derivatives. Piazzi L.; Cavalli A.; Belluti F.; Bisi A.; Gobbi S.; Rizzo S.; Bartolini M.; Andrisano V.; Recan...atini M.; Rampa A. 2007-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
High-throughput screening of beta-secretase inhibitors by multiwell FRET assay F.Mancini; F.Belluti; L.Piazzi; A.Rampa; M.Bartolini; V.Andrisano 2008-01-01 - s.n 4.02 Riassunto (Abstract) -
Homopterocarpanes as bridged triarylethylene analogues: synthesis and antagonistic effects in human MCF-7 breast cancer cells A. Rampa; A. Bisi; F. Belluti; S. Gobbi; L. Piazzi; P. Valenti; A. Zampiron; A. Caputo; K. Varani...; P. A. Borea; M. Carrara 2005-01-01 IL FARMACO - 1.01 Articolo in rivista -
Hybrid drugs for Alzheimer's disease: new indanone derivatives bearing a pharmacophoric fragment of AP2238 Rampa A.; Belluti F.; Gobbi S.; Piazzi L.; Bartolini M.; Bisi A. 2007-01-01 - s.n 4.02 Riassunto (Abstract) -
Imidazolylmethylbenzophenones as highly potent aromatase inhibitors. Gobbi S.; Cavalli A.; Negri M.; Schewe K.E.; Belluti F.; Piazzi L.; Hartmann R.W.; Recanatini M.;... Bisi A. 2007-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Imidazolylmethylxanthones as potent inhibitors of cytochrome P450 aromatase S. Gobbi; A. Bisi; A. Cavalli; F. Belluti; L. Piazzi; A. Rampa; K. Schede; R. W. Hartmann 2008-01-01 - s.n 4.02 Riassunto (Abstract) -
In vitro biological activity of new analogues of flavon-8-acetic acid M. Carrara; A. Zampiron; M. Barbera; A. Caputo; S. Gobbi; F. Belluti; A. Bisi; L. Piazzi; A. Ramp...a; P. Valenti 2004-01-01 - s.n 4.02 Riassunto (Abstract) -