Sfoglia per Autore
Introduction of hydroxyl- or keto- functionalities into the side chain of azetidin-2-ones via allylic bromide rearrangement, followed by supported reagent substitution
2005 F. Benfatti; G. Cardillo; S. Fabbroni; L. Gentilucci; R. Perciaccante; A. Tolomelli
Functionalizations of the C3 side chain of densely substituted azetidin-2-ones
2005 F. Benfatti; G. Cardillo; L. Gentilucci; R. Perciaccante; A. Tolomelli
Zinc Metal-Promoted Nucleophilic Addition of Azetidin-2-ones to Aldehydes and Nitriles
2005 F. Benfatti; G. Cardillo; S. Fabbroni; L. Gentilucci; R. Perciaccante; F. Piccinelli; A. Tolomelli
Short peptidomimetics containing heterocyclic scaffolds as alpha-v-beta-3 integrins ligands.
2005 G. Cardillo; A. Tolomelli; F. Benfatti; R. Perciaccante; L. Gentilucci; F. Squassabia
An investigation of the reactivity of MCPBA and alpha-bromoalkenes under traditional or microwave-assisted conditions: Selective formation of epoxides or allylic bromides.
2005 F. Benfatti; G. Cardillo; L. Gentilucci; R. Perciaccante; A. Tolomelli
Stereoselective synthesis of a new class of spiro-beta-lactams via epoxide ring opening
2005 F. Benfatti; G. Cardillo; L. Gentilucci; R. Perciaccante; A. Tolomelli
Stereoselective synthesis of a new class of spiro-beta-lactams via epoxide ring opening
2005 G. Cardillo; A. Tolomelli; F. Benfatti; R. Perciaccante; L. Gentilucci
Synthesis and Biological Evaluation of Azido- and Aziridino-hydroxyl-beta -lactams through Stereo- and Regioselective Epoxide Ring Opening.
2006 F.Benfatti; G.Cardillo; L. Gentilucci; R. Perciaccante; A. Tolomelli; A. Catapano
Synthesis of Enantiomerically Pure alpha-v-beta-3 Integrin ligands Based on a 5,6-Dihydropyridin-2-one Scaffold.
2006 F. Benfatti; G. Cardillo; S. Fabbroni; L. Gentilucci; R. Perciaccante; A. Tolomelli; M. Baiula; S.Spampinato
Enzymatic Resolution of Ethyl 3-Hydroxy-2(1'substituted-methylidene)-butyrate by Pseudomonas Cepacia Lipase Catalyzed Acetylation
2007 F. Benfatti; G. Cardillo ; L. Gentilucci; E. Mosconi ; A. Tolomelli
A microwave-enhanced, Lewis acid-catalyzed synthesis of 1,3-dioxolanes and oxazolines from epoxides
2007 Benfatti F. ; Cardillo G. ; Gentilucci L.; Tolomelli A .; Monari M. ;Piccinelli F.
Synthesis of four-membered ring spiro-beta -lactams by epoxide ring-opening.
2007 F. Benfatti; G. Cardillo; L. Gentilucci; A. Tolomelli
Synthesis and biological evaluation of unprecedented classes of spiro-beta-lactams and azido-beta-lactams as acyl-CoA:cholesterol acyltransferase inhibitors
2007 F. Benfatti; G. Cardillo; L. Gentilucci; A. Tolomelli
Synthesis and Biological Evaluation of Nonpeptide alpha-v-beta-3/alpha-5-beta-1 Integrin Dual Antagonists containing 5,6-Dihydropyridin-2-one Scaffolds
2007 F. Benfatti; G. Cardillo; S.Fabbroni; P. Galzerano; L. Gentilucci; R. Juris; A. Tolomelli; M. Baiula; A. Spartà; S.Spampinato
Lewis acid induced highly regioselective synthesis of a new class of substituted isoxazolidines
2008 F. Benfatti; G. Cardillo; L. Gentilucci; E. Mosconi; A. Tolomelli
Synthesis of Ethyl 5-Hydroxyisoxazolidine-4-carboxylates via Michael Addition/Intramolecular Hemiketalisation
2008 F. Benfatti; A. Bottoni; L. Gentilucci; M. Monari; E. Mosconi; M. Stenta; A. Tolomelli
Me(2)Zn mediated, tert-butylhydroperoxide promoted, catalytic enantioselective Reformatsky reaction with aldehydes
2008 P. G. Cozzi; F. Benfatti; M. Guiterez Capdevila; A. Mignogna
The cycloaddition reaction between alpha-bromo vinylketenes and imines: a combined experimental and theoretical study.
2008 F. Benfatti; A. Bottoni; G. Cardillo; S. Fabbroni; L. Gentilucci; M. Stenta; A. Tolomelli
Synthesis and Biological Evaluation of Nonpeptide alpha-v-beta-3/alpha-5-beta-1 Integrin Dual Antagonists
2008 A. Tolomelli; F. Benfatti; G. Cardillo; L. Gentilucci; E. Mosconi
Synthesis of dehydro-beta-amino esters via highly regioselective amination of allylic carbonates
2008 F. Benfatti; G. Cardillo; L. Gentilucci; E. Mosconi; A. Tolomelli
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