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Mostrati risultati da 81 a 100 di 112
Titolo Autore(i) Anno Periodico Editore Tipo File
Chalcone-based carbamates for Alzheimer's disease treatment Rampa, Angela; Montanari, Serena; Pruccoli, Letizia; Bartolini, Manuela; Falchi, Federico; Feoli,... Alessandra; Cavalli, Andrea; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra 2017-01-01 FUTURE MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Drifting of heme-coordinating group in imidazolylmethylxanthones leading to improved selective inhibition of CYP11B1 Gobbi, Silvia; Qingzhong, Hu; Zimmer, Christina; Belluti, Federica; Rampa, Angela; Hartmann, Rolf... W.; Bisi, Alessandra 2017-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Coumarin derivatives as potential antitumor agents: Growth inhibition, apoptosis induction and multidrug resistance reverting activity Alessandra Bisi; Concettina Cappadone; Rampa Angela; Farruggia Giovanna; Sargenti Azzurra; Bellut...i Federica; Rita M.C. Di Martino; Malucelli, Emil; Meluzzi Alessia; Iotti Stefano; Silvia Gobbi 2017-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
A Computational Assay of Estrogen Receptor α Antagonists Reveals the Key Common Structural Traits of Drugs Effectively Fighting Refractory Breast Cancers Pavlin, Matic; Spinello, Angelo; Pennati, Marzia; Zaffaroni, Nadia; Gobbi, Silvia; Bisi, Alessand...ra; Colombo, Giorgio; Magistrato, Alessandra 2018-01-01 SCIENTIFIC REPORTS - 1.01 Articolo in rivista s41598-017-17364-4.pdf
Identification of chalcone-based antileishmanial agents targeting trypanothione reductase Ortalli, Margherita; Ilari, Andrea; Colotti, Gianni; De Ionna, Ilenia; Battista, Theo; Bisi, Ales...sandra; Gobbi, Silvia; Rampa, Angela; Di Martino, Rita M.C.; Gentilomi, Giovanna A.; Varani, Stefania; Belluti, Federica* 2018-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista ortalli2018.pdf
Exploiting the chalcone scaffold to develop multifunctional agents for Alzheimer’s disease Rampa, Angela*; Bartolini, Manuela; Pruccoli, Letizia; Naldi, Marina; Iriepa, Isabel; Moraleda, I...gnacio; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra 2018-01-01 MOLECULES - 1.01 Articolo in rivista molecules-23-01902-v3.pdf
Cardiovascular profile of xanthone-based 1,4 dihydropyridines bearing a lidoflazine pharmacophore fragment Bisi, Alessandra*; Micucci, Matteo; Gobbi, Silvia; Belluti, Federica; Budriesi, Roberta; Rampa, A...ngela 2018-01-01 MOLECULES - 1.01 Articolo in rivista molecules-23-03088.pdf
Functionalization of the chalcone scaffold for the discovery of novel lead compounds targeting fungal infections Bonvicini F.; Gentilomi G.A.; Bressan F.; Gobbi S.; Rampa A.; Bisi A.; Belluti F. 2019-01-01 MOLECULES - 1.01 Articolo in rivista molecules-24-00372.pdf
Targeting the Bacterial Membrane with a New Polycyclic Privileged Structure: A Powerful Tool To Face Staphylococcus aureus Infections Bonvicini F.; Manet I.; Belluti F.; Gobbi S.; Rampa A.; Gentilomi G.A.; Bisi A. 2019-01-01 ACS INFECTIOUS DISEASES - 1.01 Articolo in rivista -
Identification of a new tamoxifen-xanthene hybrid as pro-apoptotic anticancer agent Catanzaro E.; Seghetti F.; Calcabrini C.; Rampa A.; Gobbi S.; Sestili P.; Turrini E.; Maffei F.; ...Hrelia P.; Bisi A.; Belluti F.; Fimognari C. 2019-01-01 BIOORGANIC CHEMISTRY - 1.01 Articolo in rivista -
Benzophenones as xanthone-open model CYP11B1 inhibitors potentially useful for promoting wound healing Gobbi S.; Hu Q.; Foschi G.; Catanzaro E.; Belluti F.; Rampa A.; Fimognari C.; Hartmann R.W.; Bisi A. 2019-01-01 BIOORGANIC CHEMISTRY - 1.01 Articolo in rivista -
Polycyclic maleimide-based derivatives as first dual modulators of neuronal calcium channels and GSK-3β for Alzheimer's disease treatment Bisi, Alessandra; Arribas, Raquel L.; Micucci, Matteo; Budriesi, Roberta; Feoli, Alessandra; Cast...ellano, Sabrina; Belluti, Federica; Gobbi, Silvia; de los Rios, Cristobal; Rampa, Angela* 2019-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Discovery of novel benzofuran-based compounds with neuroprotective and immunomodulatory properties for Alzheimer's disease treatment Montanari S.; Mahmoud A.M.; Pruccoli L.; Rabbito A.; Naldi M.; Petralla S.; Moraleda I.; Bartolin...i M.; Monti B.; Iriepa I.; Belluti F.; Gobbi S.; Di Marzo V.; Bisi A.; Tarozzi A.; Ligresti A.; Rampa A. 2019-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista benzo AM .pdf
Polycyclic Maleimide-based Scaffold as New Privileged Structure for Navigating the Cannabinoid System Opportunities Bisi A.; Mokhtar Mahmoud A.; Allara M.; Naldi M.; Belluti F.; Gobbi S.; Ligresti A.; Rampa A. 2019-01-01 ACS MEDICINAL CHEMISTRY LETTERS - 1.01 Articolo in rivista -
Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson's Disease Rita Maria Concetta Di Martino; Letizia Pruccoli; Alessandra Bisi; Silvia Gobbi; Angela Rampa; An...a Martinez; Concepción Pérez; Loreto Martinez-Gonzalez; Maria Paglione; Elia Di Schiavi; Francesca Seghetti; Andrea Tarozzi; Federica Belluti 2020-01-01 ACS CHEMICAL NEUROSCIENCE - 1.01 Articolo in rivista Nrf2 Inducer for the Treatment of Parkinson’s Disease.pdfcn0c00363_si_001.pdf
Targeting Orthosteric and Allosteric Pockets of Aromatase via Dual-Mode Novel Azole Inhibitors Caciolla J.; Spinello A.; Martini S.; Bisi A.; Zaffaroni N.; Gobbi S.; Magistrato A. 2020-01-01 ACS MEDICINAL CHEMISTRY LETTERS - 1.01 Articolo in rivista -
Reconsidering Aromatase for Breast Cancer Treatment: New Roles for an Old Target Caciolla J.; Bisi A.; Belluti F.; Rampa A.; Gobbi S. 2020-01-01 MOLECULES - 1.01 Articolo in rivista Molecules review 2020.pdf
Curcumin-1,2,3-triazole conjugation for targeting the cancer apoptosis machinery. Seghetti F., Di Martino R.M.C., Catanzaro E., Bisi A., Gobbi S., Rampa A., Canonico B., Montanari... M., Krysko D.V., Papa S., Fimognari C., Belluti F. 2020-01-01 MOLECULES - 1.01 Articolo in rivista Molecules_2020_Curcumins.pdf
Balanced dual acting compounds targeting aromatase and estrogen receptor α as an emerging therapeutic opportunity to counteract estrogen responsive breast cancer Caciolla J.; Martini S.; Spinello A.; Pavlin M.; Turrini E.; Simonelli F.; Belluti F.; Rampa A.; ...Bisi A.; Fimognari C.; Zaffaroni N.; Gobbi S.; Magistrato A. 2021-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Flavonoid-inspired vascular disrupting agents: Exploring flavone-8-acetic acid and derivatives in the new century Gobbi S.; Belluti F.; Rampa A.; Bisi A. 2021-01-01 MOLECULES - 1.01 Articolo in rivista 2021 Gobbi.pdf
Mostrati risultati da 81 a 100 di 112
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