Sfoglia per Autore
Chalcone-based carbamates for Alzheimer's disease treatment
2017 Rampa, Angela; Montanari, Serena; Pruccoli, Letizia; Bartolini, Manuela; Falchi, Federico; Feoli, Alessandra; Cavalli, Andrea; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra
Drifting of heme-coordinating group in imidazolylmethylxanthones leading to improved selective inhibition of CYP11B1
2017 Gobbi, Silvia; Qingzhong, Hu; Zimmer, Christina; Belluti, Federica; Rampa, Angela; Hartmann, Rolf W.; Bisi, Alessandra
Coumarin derivatives as potential antitumor agents: Growth inhibition, apoptosis induction and multidrug resistance reverting activity
2017 Alessandra Bisi; Concettina Cappadone; Rampa Angela; Farruggia Giovanna; Sargenti Azzurra; Belluti Federica; Rita M.C. Di Martino; Malucelli, Emil; Meluzzi Alessia; Iotti Stefano; Silvia Gobbi
A Computational Assay of Estrogen Receptor α Antagonists Reveals the Key Common Structural Traits of Drugs Effectively Fighting Refractory Breast Cancers
2018 Pavlin, Matic; Spinello, Angelo; Pennati, Marzia; Zaffaroni, Nadia; Gobbi, Silvia; Bisi, Alessandra; Colombo, Giorgio; Magistrato, Alessandra
Identification of chalcone-based antileishmanial agents targeting trypanothione reductase
2018 Ortalli, Margherita; Ilari, Andrea; Colotti, Gianni; De Ionna, Ilenia; Battista, Theo; Bisi, Alessandra; Gobbi, Silvia; Rampa, Angela; Di Martino, Rita M.C.; Gentilomi, Giovanna A.; Varani, Stefania; Belluti, Federica*
Exploiting the chalcone scaffold to develop multifunctional agents for Alzheimer’s disease
2018 Rampa, Angela*; Bartolini, Manuela; Pruccoli, Letizia; Naldi, Marina; Iriepa, Isabel; Moraleda, Ignacio; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra
Cardiovascular profile of xanthone-based 1,4 dihydropyridines bearing a lidoflazine pharmacophore fragment
2018 Bisi, Alessandra*; Micucci, Matteo; Gobbi, Silvia; Belluti, Federica; Budriesi, Roberta; Rampa, Angela
Functionalization of the chalcone scaffold for the discovery of novel lead compounds targeting fungal infections
2019 Bonvicini F.; Gentilomi G.A.; Bressan F.; Gobbi S.; Rampa A.; Bisi A.; Belluti F.
Targeting the Bacterial Membrane with a New Polycyclic Privileged Structure: A Powerful Tool To Face Staphylococcus aureus Infections
2019 Bonvicini F.; Manet I.; Belluti F.; Gobbi S.; Rampa A.; Gentilomi G.A.; Bisi A.
Identification of a new tamoxifen-xanthene hybrid as pro-apoptotic anticancer agent
2019 Catanzaro E.; Seghetti F.; Calcabrini C.; Rampa A.; Gobbi S.; Sestili P.; Turrini E.; Maffei F.; Hrelia P.; Bisi A.; Belluti F.; Fimognari C.
Benzophenones as xanthone-open model CYP11B1 inhibitors potentially useful for promoting wound healing
2019 Gobbi S.; Hu Q.; Foschi G.; Catanzaro E.; Belluti F.; Rampa A.; Fimognari C.; Hartmann R.W.; Bisi A.
Polycyclic maleimide-based derivatives as first dual modulators of neuronal calcium channels and GSK-3β for Alzheimer's disease treatment
2019 Bisi, Alessandra; Arribas, Raquel L.; Micucci, Matteo; Budriesi, Roberta; Feoli, Alessandra; Castellano, Sabrina; Belluti, Federica; Gobbi, Silvia; de los Rios, Cristobal; Rampa, Angela*
Discovery of novel benzofuran-based compounds with neuroprotective and immunomodulatory properties for Alzheimer's disease treatment
2019 Montanari S.; Mahmoud A.M.; Pruccoli L.; Rabbito A.; Naldi M.; Petralla S.; Moraleda I.; Bartolini M.; Monti B.; Iriepa I.; Belluti F.; Gobbi S.; Di Marzo V.; Bisi A.; Tarozzi A.; Ligresti A.; Rampa A.
Polycyclic Maleimide-based Scaffold as New Privileged Structure for Navigating the Cannabinoid System Opportunities
2019 Bisi A.; Mokhtar Mahmoud A.; Allara M.; Naldi M.; Belluti F.; Gobbi S.; Ligresti A.; Rampa A.
Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson's Disease
2020 Rita Maria Concetta Di Martino; Letizia Pruccoli; Alessandra Bisi; Silvia Gobbi; Angela Rampa; Ana Martinez; Concepción Pérez; Loreto Martinez-Gonzalez; Maria Paglione; Elia Di Schiavi; Francesca Seghetti; Andrea Tarozzi; Federica Belluti
Targeting Orthosteric and Allosteric Pockets of Aromatase via Dual-Mode Novel Azole Inhibitors
2020 Caciolla J.; Spinello A.; Martini S.; Bisi A.; Zaffaroni N.; Gobbi S.; Magistrato A.
Reconsidering Aromatase for Breast Cancer Treatment: New Roles for an Old Target
2020 Caciolla J.; Bisi A.; Belluti F.; Rampa A.; Gobbi S.
Curcumin-1,2,3-triazole conjugation for targeting the cancer apoptosis machinery.
2020 Seghetti F., Di Martino R.M.C., Catanzaro E., Bisi A., Gobbi S., Rampa A., Canonico B., Montanari M., Krysko D.V., Papa S., Fimognari C., Belluti F.
Balanced dual acting compounds targeting aromatase and estrogen receptor α as an emerging therapeutic opportunity to counteract estrogen responsive breast cancer
2021 Caciolla J.; Martini S.; Spinello A.; Pavlin M.; Turrini E.; Simonelli F.; Belluti F.; Rampa A.; Bisi A.; Fimognari C.; Zaffaroni N.; Gobbi S.; Magistrato A.
Flavonoid-inspired vascular disrupting agents: Exploring flavone-8-acetic acid and derivatives in the new century
2021 Gobbi S.; Belluti F.; Rampa A.; Bisi A.
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Chalcone-based carbamates for Alzheimer's disease treatment | Rampa, Angela; Montanari, Serena; Pruccoli, Letizia; Bartolini, Manuela; Falchi, Federico; Feoli,... Alessandra; Cavalli, Andrea; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra | 2017-01-01 | FUTURE MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Drifting of heme-coordinating group in imidazolylmethylxanthones leading to improved selective inhibition of CYP11B1 | Gobbi, Silvia; Qingzhong, Hu; Zimmer, Christina; Belluti, Federica; Rampa, Angela; Hartmann, Rolf... W.; Bisi, Alessandra | 2017-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Coumarin derivatives as potential antitumor agents: Growth inhibition, apoptosis induction and multidrug resistance reverting activity | Alessandra Bisi; Concettina Cappadone; Rampa Angela; Farruggia Giovanna; Sargenti Azzurra; Bellut...i Federica; Rita M.C. Di Martino; Malucelli, Emil; Meluzzi Alessia; Iotti Stefano; Silvia Gobbi | 2017-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A Computational Assay of Estrogen Receptor α Antagonists Reveals the Key Common Structural Traits of Drugs Effectively Fighting Refractory Breast Cancers | Pavlin, Matic; Spinello, Angelo; Pennati, Marzia; Zaffaroni, Nadia; Gobbi, Silvia; Bisi, Alessand...ra; Colombo, Giorgio; Magistrato, Alessandra | 2018-01-01 | SCIENTIFIC REPORTS | - | 1.01 Articolo in rivista | s41598-017-17364-4.pdf |
Identification of chalcone-based antileishmanial agents targeting trypanothione reductase | Ortalli, Margherita; Ilari, Andrea; Colotti, Gianni; De Ionna, Ilenia; Battista, Theo; Bisi, Ales...sandra; Gobbi, Silvia; Rampa, Angela; Di Martino, Rita M.C.; Gentilomi, Giovanna A.; Varani, Stefania; Belluti, Federica* | 2018-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | ortalli2018.pdf |
Exploiting the chalcone scaffold to develop multifunctional agents for Alzheimer’s disease | Rampa, Angela*; Bartolini, Manuela; Pruccoli, Letizia; Naldi, Marina; Iriepa, Isabel; Moraleda, I...gnacio; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra | 2018-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-23-01902-v3.pdf |
Cardiovascular profile of xanthone-based 1,4 dihydropyridines bearing a lidoflazine pharmacophore fragment | Bisi, Alessandra*; Micucci, Matteo; Gobbi, Silvia; Belluti, Federica; Budriesi, Roberta; Rampa, A...ngela | 2018-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-23-03088.pdf |
Functionalization of the chalcone scaffold for the discovery of novel lead compounds targeting fungal infections | Bonvicini F.; Gentilomi G.A.; Bressan F.; Gobbi S.; Rampa A.; Bisi A.; Belluti F. | 2019-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-24-00372.pdf |
Targeting the Bacterial Membrane with a New Polycyclic Privileged Structure: A Powerful Tool To Face Staphylococcus aureus Infections | Bonvicini F.; Manet I.; Belluti F.; Gobbi S.; Rampa A.; Gentilomi G.A.; Bisi A. | 2019-01-01 | ACS INFECTIOUS DISEASES | - | 1.01 Articolo in rivista | - |
Identification of a new tamoxifen-xanthene hybrid as pro-apoptotic anticancer agent | Catanzaro E.; Seghetti F.; Calcabrini C.; Rampa A.; Gobbi S.; Sestili P.; Turrini E.; Maffei F.; ...Hrelia P.; Bisi A.; Belluti F.; Fimognari C. | 2019-01-01 | BIOORGANIC CHEMISTRY | - | 1.01 Articolo in rivista | - |
Benzophenones as xanthone-open model CYP11B1 inhibitors potentially useful for promoting wound healing | Gobbi S.; Hu Q.; Foschi G.; Catanzaro E.; Belluti F.; Rampa A.; Fimognari C.; Hartmann R.W.; Bisi A. | 2019-01-01 | BIOORGANIC CHEMISTRY | - | 1.01 Articolo in rivista | - |
Polycyclic maleimide-based derivatives as first dual modulators of neuronal calcium channels and GSK-3β for Alzheimer's disease treatment | Bisi, Alessandra; Arribas, Raquel L.; Micucci, Matteo; Budriesi, Roberta; Feoli, Alessandra; Cast...ellano, Sabrina; Belluti, Federica; Gobbi, Silvia; de los Rios, Cristobal; Rampa, Angela* | 2019-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Discovery of novel benzofuran-based compounds with neuroprotective and immunomodulatory properties for Alzheimer's disease treatment | Montanari S.; Mahmoud A.M.; Pruccoli L.; Rabbito A.; Naldi M.; Petralla S.; Moraleda I.; Bartolin...i M.; Monti B.; Iriepa I.; Belluti F.; Gobbi S.; Di Marzo V.; Bisi A.; Tarozzi A.; Ligresti A.; Rampa A. | 2019-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | benzo AM .pdf |
Polycyclic Maleimide-based Scaffold as New Privileged Structure for Navigating the Cannabinoid System Opportunities | Bisi A.; Mokhtar Mahmoud A.; Allara M.; Naldi M.; Belluti F.; Gobbi S.; Ligresti A.; Rampa A. | 2019-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson's Disease | Rita Maria Concetta Di Martino; Letizia Pruccoli; Alessandra Bisi; Silvia Gobbi; Angela Rampa; An...a Martinez; Concepción Pérez; Loreto Martinez-Gonzalez; Maria Paglione; Elia Di Schiavi; Francesca Seghetti; Andrea Tarozzi; Federica Belluti | 2020-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | Nrf2 Inducer for the Treatment of Parkinson’s Disease.pdf; cn0c00363_si_001.pdf |
Targeting Orthosteric and Allosteric Pockets of Aromatase via Dual-Mode Novel Azole Inhibitors | Caciolla J.; Spinello A.; Martini S.; Bisi A.; Zaffaroni N.; Gobbi S.; Magistrato A. | 2020-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
Reconsidering Aromatase for Breast Cancer Treatment: New Roles for an Old Target | Caciolla J.; Bisi A.; Belluti F.; Rampa A.; Gobbi S. | 2020-01-01 | MOLECULES | - | 1.01 Articolo in rivista | Molecules review 2020.pdf |
Curcumin-1,2,3-triazole conjugation for targeting the cancer apoptosis machinery. | Seghetti F., Di Martino R.M.C., Catanzaro E., Bisi A., Gobbi S., Rampa A., Canonico B., Montanari... M., Krysko D.V., Papa S., Fimognari C., Belluti F. | 2020-01-01 | MOLECULES | - | 1.01 Articolo in rivista | Molecules_2020_Curcumins.pdf |
Balanced dual acting compounds targeting aromatase and estrogen receptor α as an emerging therapeutic opportunity to counteract estrogen responsive breast cancer | Caciolla J.; Martini S.; Spinello A.; Pavlin M.; Turrini E.; Simonelli F.; Belluti F.; Rampa A.; ...Bisi A.; Fimognari C.; Zaffaroni N.; Gobbi S.; Magistrato A. | 2021-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Flavonoid-inspired vascular disrupting agents: Exploring flavone-8-acetic acid and derivatives in the new century | Gobbi S.; Belluti F.; Rampa A.; Bisi A. | 2021-01-01 | MOLECULES | - | 1.01 Articolo in rivista | 2021 Gobbi.pdf |
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