DIAMANTI, ELEONORA
DIAMANTI, ELEONORA
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Ricercatori a tempo determinato
A Novel Antimalarial Agent that Inhibits Protein Synthesis in Plasmodium falciparum
2025 Bravo, Patricia; Diamanti, Eleonora; Hamed, Mostafa M.; Bizzarri, Lorenzo; Wiedemar, Natalie; Passecker, Armin; Brancucci, Nicolas M. B.; Albisetti, Anna; Gumpp, Christin; Illarionov, Boris; Fischer, Markus; Witschel, Matthias; Schehl, Tobias; Hahne, Hannes; Mäser, Pascal; Rottmann, Matthias; Hirsch, Anna K. H.
Medicinal Chemistry: A Key Driver in Achieving the Global Sustainable Development Goals
2025 Martinengo, Bianca; Diamanti, Eleonora; Uliassi, Elisa; Bolognesi, Maria Laura
Overcoming the Challenges of Multi‐Target‐Directed Ligands for Alzheimer's Disease
2025 Uliassi, Elisa; Pasieka, Anna M.; Diamanti, Eleonora; Bolognesi, Maria Laura
Positive Charge in an Antimalarial Compound Unlocks Broad-Spectrum Antibacterial Activity
2025 Braun-Cornejo, Maria; Platteschorre, Mitchell; De Vries, Vincent; Bravo, Patricia; Sonawane, Vidhisha; Hamed, Mostafa M.; Haupenthal, Jörg; Reiling, Norbert; Rottmann, Matthias; Piet, Dennis; Maas, Peter; Diamanti, Eleonora; Hirsch, Anna K. H.
Targeting isoprenoid-precursor biosynthesis in Klebsiella pneumoniae: Design, synthesis and evaluation of 1-deoxy-D-xylulose 5-phosphate synthase (DXPS) inhibitors
2025 Eisa, Sidra; Lacour, Antoine; Johannsen, Sandra; Hamid, Rawia; Raj, Prateek; Heinz, Dirk W.; Hamed, Mostafa M.; Diamanti, Eleonora; Hirsch, Anna K. H.
Targeting IspD for Anti-infective and Herbicide Development: Exploring Its Role, Mechanism, and Structural Insights
2025 Willocx, Daan; Diamanti, Eleonora; Hirsch, Anna K. H.
Benign-by-Design SAHA Analogues for Human and Animal Vector-Borne Parasitic Diseases
2024 Rossi, Michele; Martinengo, Bianca; Diamanti, Eleonora; Salerno, Alessandra; Rizzardi, Nicola; Fato, Romana; Bergamini, Christian; Souza de Oliveira, Andressa; de Araújo Marques Ferreira, Thais; Andrade Holanda, Cleonice; Romeiro, Luiz Antonio Soares; Soeiro, Maria de Nazaré Correia; Nunes, Krislayne; Ferreira de Almeida Fiuza, Ludmila; Meuser Batista, Marcos; Fraga, Carlos A. M.; E. A. Alkhalaf, Hamed; Elmahallawy, Ehab Kotb; Ebiloma, Godwin U.; De Koning, Harry P.; Vittorio, Serena; Vistoli, Giulio; Blanquart, Christophe; Bertrand, Philippe; Bolognesi, Maria Laura
Expression and characterization of pantothenate energy‐coupling factor transporters as an anti‐infective drug target
2024 Shams, Atanaz; Bousis, Spyridon; Diamanti, Eleonora; Elgaher, Walid A. M.; Zeimetz, Lucie; Haupenthal, Jörg; Slotboom, Dirk J.; Hirsch, Anna K. H.
Fragment Discovery by X‐ray Crystallographic Screening Targeting the CTP Binding Site of Pseudomonas aeruginosa IspD
2024 Willocx, Daan; D'Auria, Lucia; Walsh, Danica; Scherer, Hugo; Alhayek, Alaa; Hamed, Mostafa M.; Borel, Franck; Diamanti, Eleonora; Hirsch, Anna Katharina Herta
Harnessing the 12 Green Chemistry Principles for Sustainable Antiparasitic Drugs: Toward the One Health Approach
2024 Martinengo, Bianca; Diamanti, Eleonora; Uliassi, Elisa; Bolognesi, Maria Laura
Hit optimization by dynamic combinatorial chemistry on Streptococcus pneumoniae energy-coupling factor transporter ECF-PanT
2024 Exapicheidou, Ioulia Antonia; Shams, Atanaz; Ibrahim, Hamza; Tsarenko, Aleksei; Backenköhler, Michael; Hamed, Mostafa M.; Diamanti, Eleonora; Volkamer, Andrea; Slotboom, Dirk J.; Hirsch, Anna K. H.
IspE kinase as an anti-infective target: Role of a hydrophobic pocket in inhibitor binding
2024 Hamid, Rawia; Walsh, Danica J.; Diamanti, Eleonora; Aguilar, Diana; Lacour, Antoine; Hamed, Mostafa M.; Hirsch, Anna K.H.
Target-Directed Dynamic Combinatorial Chemistry Affords Binders of Mycobacterium tuberculosis IspE
2024 Braun-Cornejo, Maria; Ornago, Camilla; Sonawane, Vidhisha; Haupenthal, Jörg; Kany, Andreas M.; Diamanti, Eleonora; Jézéquel, Gwenaëlle; Reiling, Norbert; Blankenfeldt, Wulf; Maas, Peter; Hirsch, Anna K. H.
Targeting Plasmodium falciparum IspD in the Methyl-d-erythritol Phosphate Pathway: Urea-Based Compounds with Nanomolar Potency on Target and Low-Micromolar Whole-Cell Activity
2024 Willocx, Daan; Bizzarri, Lorenzo; Alhayek, Alaa; Kannan, Deepika; Bravo, Patricia; Illarionov, Boris; Rox, Katharina; Lohse, Jonas; Fischer, Markus; Kany, Andreas M.; Hahne, Hannes; Rottmann, Matthias; Witschel, Matthias; Odom John, Audrey; Hamed, Mostafa M.; Diamanti, Eleonora; Hirsch, Anna K. H.
Targeting the Plasmodium falciparum IspE Enzyme
2024 Diamanti, Eleonora; Steinbach, Annina M.; de Carvalho, Lais P.; Ropponen, Henni-Karoliina; Lacour, Antoine; Hamid, Rawia; Eisa, Sidra; Bravo, Patricia; Bousis, Spyridon; Illarionov, Boris; Fischer, Markus; Hamed, Mostafa M.; Bach, Nina C.; Rottmann, Matthias; Held, Jana; Witschel, Matthias; Sieber, Stephan A.; Hirsch, Anna K. H.
Back in Person: Frontiers in Medicinal Chemistry 2023
2023 Gehringer, Matthias; Pape, Felix; Méndez, María; Barbie, Philipp; Unzue Lopez, Andrea; Lefranc, Julien; Klingler, Franca-Maria; Hessler, Gerhard; Langer, Thierry; Diamanti, Eleonora; Schiedel, Matthias
Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists?
2023 Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria
Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors
2023 Ropponen, Henni-Karoliina; Diamanti, Eleonora; Johannsen, Sandra; Illarionov, Boris; Hamid, Rawia; Jaki, Miriam; Sass, Peter; Fischer, Markus; Haupenthal, Jörg; Hirsch, Anna K H
Identification of inhibitors targeting the energy-coupling factor (ECF) transporters
2023 Diamanti, Eleonora; Souza, Paulo C T; Setyawati, Inda; Bousis, Spyridon; Gómez, Leticia M; Swier, Lotteke J Y M; Shams, Atanaz; Tsarenko, Aleksei; Stanek, Weronika K; Jäger, Manuel; Marrink, Siewert J; Slotboom, Dirk J; Hirsch, Anna K H
An Efficient Way to Screen Inhibitors of Energy-Coupling Factor (ECF) Transporters in a Bacterial Uptake Assay
2022 Bousis, Spyridon; Winkler, Steffen; Haupenthal, Jörg; Fulco, Francesco; Diamanti, Eleonora; Hirsch, Anna K H
| Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
|---|---|---|---|---|---|---|
| A Novel Antimalarial Agent that Inhibits Protein Synthesis in Plasmodium falciparum | Bravo, Patricia; Diamanti, Eleonora; Hamed, Mostafa M.; Bizzarri, Lorenzo; Wiedemar, Natalie; Pas...secker, Armin; Brancucci, Nicolas M. B.; Albisetti, Anna; Gumpp, Christin; Illarionov, Boris; Fischer, Markus; Witschel, Matthias; Schehl, Tobias; Hahne, Hannes; Mäser, Pascal; Rottmann, Matthias; Hirsch, Anna K. H. | 2025-01-01 | ANGEWANDTE CHEMIE. INTERNATIONAL EDITION | - | 1.01 Articolo in rivista | - |
| Medicinal Chemistry: A Key Driver in Achieving the Global Sustainable Development Goals | Martinengo, Bianca; Diamanti, Eleonora; Uliassi, Elisa; Bolognesi, Maria Laura | 2025-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
| Overcoming the Challenges of Multi‐Target‐Directed Ligands for Alzheimer's Disease | Uliassi, Elisa; Pasieka, Anna M.; Diamanti, Eleonora; Bolognesi, Maria Laura | 2025-01-01 | - | wiley | 2.01 Capitolo / saggio in libro | - |
| Positive Charge in an Antimalarial Compound Unlocks Broad-Spectrum Antibacterial Activity | Braun-Cornejo, Maria; Platteschorre, Mitchell; De Vries, Vincent; Bravo, Patricia; Sonawane, Vidh...isha; Hamed, Mostafa M.; Haupenthal, Jörg; Reiling, Norbert; Rottmann, Matthias; Piet, Dennis; Maas, Peter; Diamanti, Eleonora; Hirsch, Anna K. H. | 2025-01-01 | JACS AU | - | 1.01 Articolo in rivista | - |
| Targeting isoprenoid-precursor biosynthesis in Klebsiella pneumoniae: Design, synthesis and evaluation of 1-deoxy-D-xylulose 5-phosphate synthase (DXPS) inhibitors | Eisa, Sidra; Lacour, Antoine; Johannsen, Sandra; Hamid, Rawia; Raj, Prateek; Heinz, Dirk W.; Hame...d, Mostafa M.; Diamanti, Eleonora; Hirsch, Anna K. H. | 2025-01-01 | BIOORGANIC CHEMISTRY | - | 1.01 Articolo in rivista | - |
| Targeting IspD for Anti-infective and Herbicide Development: Exploring Its Role, Mechanism, and Structural Insights | Willocx, Daan; Diamanti, Eleonora; Hirsch, Anna K. H. | 2025-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
| Benign-by-Design SAHA Analogues for Human and Animal Vector-Borne Parasitic Diseases | Rossi, Michele; Martinengo, Bianca; Diamanti, Eleonora; Salerno, Alessandra; Rizzardi, Nicola; Fa...to, Romana; Bergamini, Christian; Souza de Oliveira, Andressa; de Araújo Marques Ferreira, Thais; Andrade Holanda, Cleonice; Romeiro, Luiz Antonio Soares; Soeiro, Maria de Nazaré Correia; Nunes, Krislayne; Ferreira de Almeida Fiuza, Ludmila; Meuser Batista, Marcos; Fraga, Carlos A. M.; E. A. Alkhalaf, Hamed; Elmahallawy, Ehab Kotb; Ebiloma, Godwin U.; De Koning, Harry P.; Vittorio, Serena; Vistoli, Giulio; Blanquart, Christophe; Bertrand, Philippe; Bolognesi, Maria Laura | 2024-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
| Expression and characterization of pantothenate energy‐coupling factor transporters as an anti‐infective drug target | Shams, Atanaz; Bousis, Spyridon; Diamanti, Eleonora; Elgaher, Walid A. M.; Zeimetz, Lucie; Haupen...thal, Jörg; Slotboom, Dirk J.; Hirsch, Anna K. H. | 2024-01-01 | PROTEIN SCIENCE | - | 1.01 Articolo in rivista | 10.1002_pro.5195.pdf |
| Fragment Discovery by X‐ray Crystallographic Screening Targeting the CTP Binding Site of Pseudomonas aeruginosa IspD | Willocx, Daan; D'Auria, Lucia; Walsh, Danica; Scherer, Hugo; Alhayek, Alaa; Hamed, Mostafa M.; Bo...rel, Franck; Diamanti, Eleonora; Hirsch, Anna Katharina Herta | 2024-01-01 | ANGEWANDTE CHEMIE. INTERNATIONAL EDITION | - | 1.01 Articolo in rivista | Angew Chem Int Ed - 2024 - Willocx - Fragment Discovery by X‐Ray Crystallographic Screening Targeting the CTP Binding Site.pdf |
| Harnessing the 12 Green Chemistry Principles for Sustainable Antiparasitic Drugs: Toward the One Health Approach | Martinengo, Bianca; Diamanti, Eleonora; Uliassi, Elisa; Bolognesi, Maria Laura | 2024-01-01 | ACS INFECTIOUS DISEASES | - | 1.01 Articolo in rivista | martinengo-et-al-2024-harnessing-the-12-green-chemistry-principles-for-sustainable-antiparasitic-drugs-toward-the-one.pdf; id4c00172_si_001.pdf |
| Hit optimization by dynamic combinatorial chemistry on Streptococcus pneumoniae energy-coupling factor transporter ECF-PanT | Exapicheidou, Ioulia Antonia; Shams, Atanaz; Ibrahim, Hamza; Tsarenko, Aleksei; Backenköhler, Mic...hael; Hamed, Mostafa M.; Diamanti, Eleonora; Volkamer, Andrea; Slotboom, Dirk J.; Hirsch, Anna K. H. | 2024-01-01 | CHEMICAL COMMUNICATIONS | - | 1.01 Articolo in rivista | - |
| IspE kinase as an anti-infective target: Role of a hydrophobic pocket in inhibitor binding | Hamid, Rawia; Walsh, Danica J.; Diamanti, Eleonora; Aguilar, Diana; Lacour, Antoine; Hamed, Mosta...fa M.; Hirsch, Anna K.H. | 2024-01-01 | STRUCTURE | - | 1.01 Articolo in rivista | - |
| Target-Directed Dynamic Combinatorial Chemistry Affords Binders of Mycobacterium tuberculosis IspE | Braun-Cornejo, Maria; Ornago, Camilla; Sonawane, Vidhisha; Haupenthal, Jörg; Kany, Andreas M.; Di...amanti, Eleonora; Jézéquel, Gwenaëlle; Reiling, Norbert; Blankenfeldt, Wulf; Maas, Peter; Hirsch, Anna K. H. | 2024-01-01 | ACS OMEGA | - | 1.01 Articolo in rivista | - |
| Targeting Plasmodium falciparum IspD in the Methyl-d-erythritol Phosphate Pathway: Urea-Based Compounds with Nanomolar Potency on Target and Low-Micromolar Whole-Cell Activity | Willocx, Daan; Bizzarri, Lorenzo; Alhayek, Alaa; Kannan, Deepika; Bravo, Patricia; Illarionov, Bo...ris; Rox, Katharina; Lohse, Jonas; Fischer, Markus; Kany, Andreas M.; Hahne, Hannes; Rottmann, Matthias; Witschel, Matthias; Odom John, Audrey; Hamed, Mostafa M.; Diamanti, Eleonora; Hirsch, Anna K. H. | 2024-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | JMedChem-2024.pdf; jm4c00212_si_001.pdf |
| Targeting the Plasmodium falciparum IspE Enzyme | Diamanti, Eleonora; Steinbach, Annina M.; de Carvalho, Lais P.; Ropponen, Henni-Karoliina; Lacour..., Antoine; Hamid, Rawia; Eisa, Sidra; Bravo, Patricia; Bousis, Spyridon; Illarionov, Boris; Fischer, Markus; Hamed, Mostafa M.; Bach, Nina C.; Rottmann, Matthias; Held, Jana; Witschel, Matthias; Sieber, Stephan A.; Hirsch, Anna K. H. | 2024-01-01 | ACS OMEGA | - | 1.01 Articolo in rivista | - |
| Back in Person: Frontiers in Medicinal Chemistry 2023 | Gehringer, Matthias; Pape, Felix; Méndez, María; Barbie, Philipp; Unzue Lopez, Andrea; Lefranc, J...ulien; Klingler, Franca-Maria; Hessler, Gerhard; Langer, Thierry; Diamanti, Eleonora; Schiedel, Matthias | 2023-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2023 - Gehringer - Back in Person Frontiers in Medicinal Chemistry 2023.pdf |
| Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists? | Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria | 2023-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2023 - Pasieka - Click Chemistry and Targeted Degradation A Winning Combination for Medicinal Chemists.pdf |
| Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors | Ropponen, Henni-Karoliina; Diamanti, Eleonora; Johannsen, Sandra; Illarionov, Boris; Hamid, Rawia...; Jaki, Miriam; Sass, Peter; Fischer, Markus; Haupenthal, Jörg; Hirsch, Anna K H | 2023-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2023 - Ropponen - Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors.pdf; downloadSupplement.pdf |
| Identification of inhibitors targeting the energy-coupling factor (ECF) transporters | Diamanti, Eleonora; Souza, Paulo C T; Setyawati, Inda; Bousis, Spyridon; Gómez, Leticia M; Swier,... Lotteke J Y M; Shams, Atanaz; Tsarenko, Aleksei; Stanek, Weronika K; Jäger, Manuel; Marrink, Siewert J; Slotboom, Dirk J; Hirsch, Anna K H | 2023-01-01 | COMMUNICATIONS BIOLOGY | - | 1.01 Articolo in rivista | s42003-023-05555-x (5).pdf; 42003_2023_5555_MOESM1_ESM.pdf; 42003_2023_5555_MOESM3_ESM.xlsx |
| An Efficient Way to Screen Inhibitors of Energy-Coupling Factor (ECF) Transporters in a Bacterial Uptake Assay | Bousis, Spyridon; Winkler, Steffen; Haupenthal, Jörg; Fulco, Francesco; Diamanti, Eleonora; Hirsc...h, Anna K H | 2022-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | ijms-23-02637.pdf; ijms-23-02637-s001.zip |