DIAMANTI, ELEONORA
DIAMANTI, ELEONORA
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Ricercatori a tempo determinato
Positive Charge in an Antimalarial Compound Unlocks Broad-Spectrum Antibacterial Activity
2025 Braun-Cornejo, Maria; Platteschorre, Mitchell; de Vries, Vincent; Bravo, Patricia; Sonawane, Vidhisha; Hamed, Mostafa M.; Haupenthal, Jörg; Reiling, Norbert; Rottmann, Matthias; Piet, Dennis; Maas, Peter; Diamanti, Eleonora; Hirsch, Anna K. H.
Targeting IspD for Anti-infective and Herbicide Development: Exploring Its Role, Mechanism, and Structural Insights
2025 Willocx, Daan; Diamanti, Eleonora; Hirsch, Anna K. H.
Benign-by-Design SAHA Analogues for Human and Animal Vector-Borne Parasitic Diseases
2024 Rossi, Michele; Martinengo, Bianca; Diamanti, Eleonora; Salerno, Alessandra; Rizzardi, Nicola; Fato, Romana; Bergamini, Christian; Souza de Oliveira, Andressa; de Araújo Marques Ferreira, Thais; Andrade Holanda, Cleonice; Romeiro, Luiz Antonio Soares; Soeiro, Maria de Nazaré Correia; Nunes, Krislayne; Ferreira de Almeida Fiuza, Ludmila; Meuser Batista, Marcos; Fraga, Carlos A. M.; E. A. Alkhalaf, Hamed; Elmahallawy, Ehab Kotb; Ebiloma, Godwin U.; De Koning, Harry P.; Vittorio, Serena; Vistoli, Giulio; Blanquart, Christophe; Bertrand, Philippe; Bolognesi, Maria Laura
Expression and characterization of pantothenate energy‐coupling factor transporters as an anti‐infective drug target
2024 Shams, Atanaz; Bousis, Spyridon; Diamanti, Eleonora; Elgaher, Walid A. M.; Zeimetz, Lucie; Haupenthal, Jörg; Slotboom, Dirk J.; Hirsch, Anna K. H.
Fragment Discovery by X‐ray Crystallographic Screening Targeting the CTP Binding Site of Pseudomonas aeruginosa IspD
2024 Willocx, Daan; D'Auria, Lucia; Walsh, Danica; Scherer, Hugo; Alhayek, Alaa; Hamed, Mostafa M.; Borel, Franck; Diamanti, Eleonora; Hirsch, Anna Katharina Herta
Harnessing the 12 Green Chemistry Principles for Sustainable Antiparasitic Drugs: Toward the One Health Approach
2024 Martinengo, Bianca; Diamanti, Eleonora; Uliassi, Elisa; Bolognesi, Maria Laura
Hit optimization by dynamic combinatorial chemistry on Streptococcus pneumoniae energy-coupling factor transporter ECF-PanT
2024 Exapicheidou, Ioulia Antonia; Shams, Atanaz; Ibrahim, Hamza; Tsarenko, Aleksei; Backenköhler, Michael; Hamed, Mostafa M.; Diamanti, Eleonora; Volkamer, Andrea; Slotboom, Dirk J.; Hirsch, Anna K. H.
IspE kinase as an anti-infective target: Role of a hydrophobic pocket in inhibitor binding
2024 Hamid, Rawia; Walsh, Danica J.; Diamanti, Eleonora; Aguilar, Diana; Lacour, Antoine; Hamed, Mostafa M.; Hirsch, Anna K.H.
Target-Directed Dynamic Combinatorial Chemistry Affords Binders of Mycobacterium tuberculosis IspE
2024 Braun-Cornejo, Maria; Ornago, Camilla; Sonawane, Vidhisha; Haupenthal, Jörg; Kany, Andreas M.; Diamanti, Eleonora; Jézéquel, Gwenaëlle; Reiling, Norbert; Blankenfeldt, Wulf; Maas, Peter; Hirsch, Anna K. H.
Targeting Plasmodium falciparum IspD in the Methyl-d-erythritol Phosphate Pathway: Urea-Based Compounds with Nanomolar Potency on Target and Low-Micromolar Whole-Cell Activity
2024 Willocx, Daan; Bizzarri, Lorenzo; Alhayek, Alaa; Kannan, Deepika; Bravo, Patricia; Illarionov, Boris; Rox, Katharina; Lohse, Jonas; Fischer, Markus; Kany, Andreas M.; Hahne, Hannes; Rottmann, Matthias; Witschel, Matthias; Odom John, Audrey; Hamed, Mostafa M.; Diamanti, Eleonora; Hirsch, Anna K. H.
Targeting the Plasmodium falciparum IspE Enzyme
2024 Diamanti, Eleonora; Steinbach, Annina M.; de Carvalho, Lais P.; Ropponen, Henni-Karoliina; Lacour, Antoine; Hamid, Rawia; Eisa, Sidra; Bravo, Patricia; Bousis, Spyridon; Illarionov, Boris; Fischer, Markus; Hamed, Mostafa M.; Bach, Nina C.; Rottmann, Matthias; Held, Jana; Witschel, Matthias; Sieber, Stephan A.; Hirsch, Anna K. H.
Back in Person: Frontiers in Medicinal Chemistry 2023
2023 Gehringer, Matthias; Pape, Felix; Méndez, María; Barbie, Philipp; Unzue Lopez, Andrea; Lefranc, Julien; Klingler, Franca-Maria; Hessler, Gerhard; Langer, Thierry; Diamanti, Eleonora; Schiedel, Matthias
Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists?
2023 Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria
Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors
2023 Ropponen, Henni-Karoliina; Diamanti, Eleonora; Johannsen, Sandra; Illarionov, Boris; Hamid, Rawia; Jaki, Miriam; Sass, Peter; Fischer, Markus; Haupenthal, Jörg; Hirsch, Anna K H
Identification of inhibitors targeting the energy-coupling factor (ECF) transporters
2023 Diamanti, Eleonora; Souza, Paulo C T; Setyawati, Inda; Bousis, Spyridon; Gómez, Leticia M; Swier, Lotteke J Y M; Shams, Atanaz; Tsarenko, Aleksei; Stanek, Weronika K; Jäger, Manuel; Marrink, Siewert J; Slotboom, Dirk J; Hirsch, Anna K H
An Efficient Way to Screen Inhibitors of Energy-Coupling Factor (ECF) Transporters in a Bacterial Uptake Assay
2022 Bousis, Spyridon; Winkler, Steffen; Haupenthal, Jörg; Fulco, Francesco; Diamanti, Eleonora; Hirsch, Anna K H
Frontiers in Medicinal Chemistry 2022 Goes Virtual
2022 Diamanti, Eleonora; Méndez, María; Ross, Tatjana; Kuttruff, Christian A; Lefranc, Julien; Klingler, Franca-Maria; von Nussbaum, Franz; Jung, Manfred; Gehringer, Matthias
Structure-Guided Optimization of Small-Molecule Folate Uptake Inhibitors Targeting the Energy-Coupling Factor Transporters
2022 Kiefer, Alexander F; Bousis, Spyridon; Hamed, Mostafa M; Diamanti, Eleonora; Haupenthal, Jörg; Hirsch, Anna K H
Targeting the IspD Enzyme in the MEP Pathway: Identification of a Novel Fragment Class
2022 Diamanti, Eleonora; Hamed, Mostafa M; Lacour, Antoine; Bravo, Patricia; Illarionov, Boris; Fischer, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H
Assessment of the rules related to gaining activity against Gram-negative bacteria
2021 Ropponen, Henni-Karoliina; Diamanti, Eleonora; Siemens, Alexandra; Illarionov, Boris; Haupenthal, Jörg; Fischer, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H