DIAMANTI, ELEONORA
DIAMANTI, ELEONORA
DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Ricercatori a tempo determinato
Harnessing the 12 Green Chemistry Principles for Sustainable Antiparasitic Drugs: Toward the One Health Approach
2024 Martinengo, Bianca; Diamanti, Eleonora; Uliassi, Elisa; Bolognesi, Maria Laura
Hit optimization by dynamic combinatorial chemistry on Streptococcus pneumoniae energy-coupling factor transporter ECF-PanT
2024 Exapicheidou, Ioulia Antonia; Shams, Atanaz; Ibrahim, Hamza; Tsarenko, Aleksei; Backenköhler, Michael; Hamed, Mostafa M.; Diamanti, Eleonora; Volkamer, Andrea; Slotboom, Dirk J.; Hirsch, Anna K. H.
Back in Person: Frontiers in Medicinal Chemistry 2023
2023 Gehringer, Matthias; Pape, Felix; Méndez, María; Barbie, Philipp; Unzue Lopez, Andrea; Lefranc, Julien; Klingler, Franca-Maria; Hessler, Gerhard; Langer, Thierry; Diamanti, Eleonora; Schiedel, Matthias
Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists?
2023 Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria
Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors
2023 Ropponen, Henni-Karoliina; Diamanti, Eleonora; Johannsen, Sandra; Illarionov, Boris; Hamid, Rawia; Jaki, Miriam; Sass, Peter; Fischer, Markus; Haupenthal, Jörg; Hirsch, Anna K H
Identification of inhibitors targeting the energy-coupling factor (ECF) transporters
2023 Diamanti, Eleonora; Souza, Paulo C T; Setyawati, Inda; Bousis, Spyridon; Gómez, Leticia M; Swier, Lotteke J Y M; Shams, Atanaz; Tsarenko, Aleksei; Stanek, Weronika K; Jäger, Manuel; Marrink, Siewert J; Slotboom, Dirk J; Hirsch, Anna K H
An Efficient Way to Screen Inhibitors of Energy-Coupling Factor (ECF) Transporters in a Bacterial Uptake Assay
2022 Bousis, Spyridon; Winkler, Steffen; Haupenthal, Jörg; Fulco, Francesco; Diamanti, Eleonora; Hirsch, Anna K H
Frontiers in Medicinal Chemistry 2022 Goes Virtual
2022 Diamanti, Eleonora; Méndez, María; Ross, Tatjana; Kuttruff, Christian A; Lefranc, Julien; Klingler, Franca-Maria; von Nussbaum, Franz; Jung, Manfred; Gehringer, Matthias
Structure-Guided Optimization of Small-Molecule Folate Uptake Inhibitors Targeting the Energy-Coupling Factor Transporters
2022 Kiefer, Alexander F; Bousis, Spyridon; Hamed, Mostafa M; Diamanti, Eleonora; Haupenthal, Jörg; Hirsch, Anna K H
Targeting the IspD Enzyme in the MEP Pathway: Identification of a Novel Fragment Class
2022 Diamanti, Eleonora; Hamed, Mostafa M; Lacour, Antoine; Bravo, Patricia; Illarionov, Boris; Fischer, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H
Assessment of the rules related to gaining activity against Gram-negative bacteria
2021 Ropponen, Henni-Karoliina; Diamanti, Eleonora; Siemens, Alexandra; Illarionov, Boris; Haupenthal, Jörg; Fischer, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H
Bacteriomimetic Liposomes Improve Antibiotic Activity of a Novel Energy-Coupling Factor Transporter Inhibitor
2021 Drost, M; Diamanti, E; Fuhrmann, K; Goes, A; Shams, A; Haupenthal, J; Koch, M; Hirsch, AKH; Fuhrmann, G
Search for the Active Ingredients from a 2-Aminothiazole DMSO Stock Solution with Antimalarial Activity
2021 Ropponen, Henni-Karoliina; Bader, Chantal D; Diamanti, Eleonora; Illarionov, Boris; Rottmann, Matthias; Fischer, Markus; Witschel, Matthias; Müller, Rolf; Hirsch, Anna K H
Energy-Coupling Factor Transporters as Novel Antimicrobial Targets
2019 Spyridon Bousis; Inda Setyawati; Eleonora Diamanti; Dirk J. Slotboom; Anna K. H. Hirsch
CD1b Tetramers Identify T Cells that Recognize Natural and Synthetic Diacylated Sulfoglycolipids from Mycobacterium tuberculosis
2018 James, Charlotte A; Yu, Krystle K Q; Gilleron, Martine; Prandi, Jacques; Yedulla, Vijayendar R; Moleda, Zuzanna Z; Diamanti, Eleonora; Khan, Momin; Aggarwal, Varinder K; Reijneveld, Josephine F; Reinink, Peter; Lenz, Stefanie; Emerson, Ryan O; Scriba, Thomas J; Souter, Michael N T; Godfrey, Dale I; Pellicci, Daniel G; Moody, D Branch; Minnaard, Adriaan J; Seshadri, Chetan; Van Rhijn, Ildiko
DXS as a target for structure-based drug design
2017 Gierse, Robin Matthias; Redeem, Eswar; Diamanti, Eleonora; Wrenger, Carsten; Groves, Matthew R; Hirsch, Anna Kh
Combined Interactions with I1-, I2-Imidazoline Binding Sites and α2-Adrenoceptors To Manage Opioid Addiction
2016 Giusepponi, Maria Elena; Cifani, Carlo; Micioni Di Bonaventura, Maria Vittoria; Mattioli, Laura; Hudson, Alan; Diamanti, Eleonora; Del Bello, Fabio; Giannella, Mario; Mammoli, Valerio; Paoletti, Corinne Dalila; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma
Pyrazole-Based Acid Ceramidase Inhibitors: Design, Synthesis, and Structure-Activity Relationships
2016 Diamanti, E; Bottegoni, G; Goldoni, L; Realini, N; Pagliuca, C; Bertozzi, F; Piomelli, D; Pizzirani, D
The Versatile 2-Substituted Imidazoline Nucleus as a Structural Motif of Ligands Directed to the Serotonin 5-HT1A Receptor
2016 Del Bello, Fabio; Cilia, Antonio; Carrieri, Antonio; Fasano, Domenico Claudio; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Micheli, Laura; Santini, Carlo; Diamanti, Eleonora; Giannella, Mario; Giorgioni, Gianfabio; Mammoli, Valerio; Paoletti, Corinne Dalila; Petrelli, Riccardo; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria
Antagonism/Agonism modulation to build novel antihypertensives selectively triggering i1-imidazoline receptor activation
2015 Del Bello, Fabio; Bargelli, Valentina; Cifani, Carlo; Gratteri, Paola; Bazzicalupi, Carla; Diamanti, Eleonora; Giannella, Mario; Mammoli, Valerio; Matucci, Rosanna; Micioni Di Bonaventura, Maria Vittoria; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria
| Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
|---|---|---|---|---|---|---|
| Harnessing the 12 Green Chemistry Principles for Sustainable Antiparasitic Drugs: Toward the One Health Approach | Martinengo, Bianca; Diamanti, Eleonora; Uliassi, Elisa; Bolognesi, Maria Laura | 2024-01-01 | ACS INFECTIOUS DISEASES | - | 1.01 Articolo in rivista | - |
| Hit optimization by dynamic combinatorial chemistry on Streptococcus pneumoniae energy-coupling factor transporter ECF-PanT | Exapicheidou, Ioulia Antonia; Shams, Atanaz; Ibrahim, Hamza; Tsarenko, Aleksei; Backenköhler, Mic...hael; Hamed, Mostafa M.; Diamanti, Eleonora; Volkamer, Andrea; Slotboom, Dirk J.; Hirsch, Anna K. H. | 2024-01-01 | CHEMICAL COMMUNICATIONS | - | 1.01 Articolo in rivista | - |
| Back in Person: Frontiers in Medicinal Chemistry 2023 | Gehringer, Matthias; Pape, Felix; Méndez, María; Barbie, Philipp; Unzue Lopez, Andrea; Lefranc, J...ulien; Klingler, Franca-Maria; Hessler, Gerhard; Langer, Thierry; Diamanti, Eleonora; Schiedel, Matthias | 2023-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2023 - Gehringer - Back in Person Frontiers in Medicinal Chemistry 2023.pdf |
| Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists? | Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria | 2023-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2023 - Pasieka - Click Chemistry and Targeted Degradation A Winning Combination for Medicinal Chemists.pdf |
| Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors | Ropponen, Henni-Karoliina; Diamanti, Eleonora; Johannsen, Sandra; Illarionov, Boris; Hamid, Rawia...; Jaki, Miriam; Sass, Peter; Fischer, Markus; Haupenthal, Jörg; Hirsch, Anna K H | 2023-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2023 - Ropponen - Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors.pdf; downloadSupplement.pdf |
| Identification of inhibitors targeting the energy-coupling factor (ECF) transporters | Diamanti, Eleonora; Souza, Paulo C T; Setyawati, Inda; Bousis, Spyridon; Gómez, Leticia M; Swier,... Lotteke J Y M; Shams, Atanaz; Tsarenko, Aleksei; Stanek, Weronika K; Jäger, Manuel; Marrink, Siewert J; Slotboom, Dirk J; Hirsch, Anna K H | 2023-01-01 | COMMUNICATIONS BIOLOGY | - | 1.01 Articolo in rivista | s42003-023-05555-x (5).pdf; 42003_2023_5555_MOESM1_ESM.pdf; 42003_2023_5555_MOESM3_ESM.xlsx |
| An Efficient Way to Screen Inhibitors of Energy-Coupling Factor (ECF) Transporters in a Bacterial Uptake Assay | Bousis, Spyridon; Winkler, Steffen; Haupenthal, Jörg; Fulco, Francesco; Diamanti, Eleonora; Hirsc...h, Anna K H | 2022-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | ijms-23-02637.pdf; ijms-23-02637-s001.zip |
| Frontiers in Medicinal Chemistry 2022 Goes Virtual | Diamanti, Eleonora; Méndez, María; Ross, Tatjana; Kuttruff, Christian A; Lefranc, Julien; Klingle...r, Franca-Maria; von Nussbaum, Franz; Jung, Manfred; Gehringer, Matthias | 2022-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
| Structure-Guided Optimization of Small-Molecule Folate Uptake Inhibitors Targeting the Energy-Coupling Factor Transporters | Kiefer, Alexander F; Bousis, Spyridon; Hamed, Mostafa M; Diamanti, Eleonora; Haupenthal, Jörg; Hi...rsch, Anna K H | 2022-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | kiefer-et-al-2022-structure-guided-optimization-of-small-molecule-folate-uptake-inhibitors-targeting-the-energy.pdf; From Bitter to Sweet_ a preliminary study towards a patient-friendly Praziquantel dosage form.pdf; jm1c02114_si_001.pdf |
| Targeting the IspD Enzyme in the MEP Pathway: Identification of a Novel Fragment Class | Diamanti, Eleonora; Hamed, Mostafa M; Lacour, Antoine; Bravo, Patricia; Illarionov, Boris; Fische...r, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H | 2022-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2021 - Diamanti - Targeting the IspD Enzyme in the MEP Pathway Identification of a Novel Fragment Class (1).pdf |
| Assessment of the rules related to gaining activity against Gram-negative bacteria | Ropponen, Henni-Karoliina; Diamanti, Eleonora; Siemens, Alexandra; Illarionov, Boris; Haupenthal,... Jörg; Fischer, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H | 2021-01-01 | RSC MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
| Bacteriomimetic Liposomes Improve Antibiotic Activity of a Novel Energy-Coupling Factor Transporter Inhibitor | Drost, M; Diamanti, E; Fuhrmann, K; Goes, A; Shams, A; Haupenthal, J; Koch, M; Hirsch, AKH; Fuhrm...ann, G | 2021-01-01 | PHARMACEUTICS | - | 1.01 Articolo in rivista | pharmaceutics-14-00004.pdf; pharmaceutics-14-00004-s001.zip |
| Search for the Active Ingredients from a 2-Aminothiazole DMSO Stock Solution with Antimalarial Activity | Ropponen, Henni-Karoliina; Bader, Chantal D; Diamanti, Eleonora; Illarionov, Boris; Rottmann, Mat...thias; Fischer, Markus; Witschel, Matthias; Müller, Rolf; Hirsch, Anna K H | 2021-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | CMDC-16-2089.pdf; downloadSupplement.pdf |
| Energy-Coupling Factor Transporters as Novel Antimicrobial Targets | Spyridon Bousis; Inda Setyawati; Eleonora Diamanti; Dirk J. Slotboom; Anna K. H. Hirsch | 2019-01-01 | ADVANCED THERAPEUTICS | - | 1.01 Articolo in rivista | - |
| CD1b Tetramers Identify T Cells that Recognize Natural and Synthetic Diacylated Sulfoglycolipids from Mycobacterium tuberculosis | James, Charlotte A; Yu, Krystle K Q; Gilleron, Martine; Prandi, Jacques; Yedulla, Vijayendar R; M...oleda, Zuzanna Z; Diamanti, Eleonora; Khan, Momin; Aggarwal, Varinder K; Reijneveld, Josephine F; Reinink, Peter; Lenz, Stefanie; Emerson, Ryan O; Scriba, Thomas J; Souter, Michael N T; Godfrey, Dale I; Pellicci, Daniel G; Moody, D Branch; Minnaard, Adriaan J; Seshadri, Chetan; Van Rhijn, Ildiko | 2018-01-01 | CELL CHEMICAL BIOLOGY | - | 1.01 Articolo in rivista | - |
| DXS as a target for structure-based drug design | Gierse, Robin Matthias; Redeem, Eswar; Diamanti, Eleonora; Wrenger, Carsten; Groves, Matthew R; H...irsch, Anna Kh | 2017-01-01 | FUTURE MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
| Combined Interactions with I1-, I2-Imidazoline Binding Sites and α2-Adrenoceptors To Manage Opioid Addiction | Giusepponi, Maria Elena; Cifani, Carlo; Micioni Di Bonaventura, Maria Vittoria; Mattioli, Laura; ...Hudson, Alan; Diamanti, Eleonora; Del Bello, Fabio; Giannella, Mario; Mammoli, Valerio; Paoletti, Corinne Dalila; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma | 2016-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
| Pyrazole-Based Acid Ceramidase Inhibitors: Design, Synthesis, and Structure-Activity Relationships | Diamanti, E; Bottegoni, G; Goldoni, L; Realini, N; Pagliuca, C; Bertozzi, F; Piomelli, D; Pizzira...ni, D | 2016-01-01 | SYNTHESIS | - | 1.01 Articolo in rivista | - |
| The Versatile 2-Substituted Imidazoline Nucleus as a Structural Motif of Ligands Directed to the Serotonin 5-HT1A Receptor | Del Bello, Fabio; Cilia, Antonio; Carrieri, Antonio; Fasano, Domenico Claudio; Ghelardini, Carla;... Di Cesare Mannelli, Lorenzo; Micheli, Laura; Santini, Carlo; Diamanti, Eleonora; Giannella, Mario; Giorgioni, Gianfabio; Mammoli, Valerio; Paoletti, Corinne Dalila; Petrelli, Riccardo; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria | 2016-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
| Antagonism/Agonism modulation to build novel antihypertensives selectively triggering i1-imidazoline receptor activation | Del Bello, Fabio; Bargelli, Valentina; Cifani, Carlo; Gratteri, Paola; Bazzicalupi, Carla; Diaman...ti, Eleonora; Giannella, Mario; Mammoli, Valerio; Matucci, Rosanna; Micioni Di Bonaventura, Maria Vittoria; Piergentili, Alessandro; Quaglia, Wilma; Pigini, Maria | 2015-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |