DIAMANTI, ELEONORA
DIAMANTI, ELEONORA
DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Ricercatori a tempo determinato
Benign-by-Design SAHA Analogues for Human and Animal Vector-Borne Parasitic Diseases
2024 Rossi, Michele; Martinengo, Bianca; Diamanti, Eleonora; Salerno, Alessandra; Rizzardi, Nicola; Fato, Romana; Bergamini, Christian; Souza de Oliveira, Andressa; de Araújo Marques Ferreira, Thais; Andrade Holanda, Cleonice; Romeiro, Luiz Antonio Soares; Soeiro, Maria de Nazaré Correia; Nunes, Krislayne; Ferreira de Almeida Fiuza, Ludmila; Meuser Batista, Marcos; Fraga, Carlos A. M.; E. A. Alkhalaf, Hamed; Elmahallawy, Ehab Kotb; Ebiloma, Godwin U.; De Koning, Harry P.; Vittorio, Serena; Vistoli, Giulio; Blanquart, Christophe; Bertrand, Philippe; Bolognesi, Maria Laura
Expression and characterization of pantothenate energy‐coupling factor transporters as an anti‐infective drug target
2024 Shams, Atanaz; Bousis, Spyridon; Diamanti, Eleonora; Elgaher, Walid A. M.; Zeimetz, Lucie; Haupenthal, Jörg; Slotboom, Dirk J.; Hirsch, Anna K. H.
Harnessing the 12 Green Chemistry Principles for Sustainable Antiparasitic Drugs: Toward the One Health Approach
2024 Martinengo, Bianca; Diamanti, Eleonora; Uliassi, Elisa; Bolognesi, Maria Laura
Hit optimization by dynamic combinatorial chemistry on Streptococcus pneumoniae energy-coupling factor transporter ECF-PanT
2024 Exapicheidou, Ioulia Antonia; Shams, Atanaz; Ibrahim, Hamza; Tsarenko, Aleksei; Backenköhler, Michael; Hamed, Mostafa M.; Diamanti, Eleonora; Volkamer, Andrea; Slotboom, Dirk J.; Hirsch, Anna K. H.
IspE kinase as an anti-infective target: Role of a hydrophobic pocket in inhibitor binding
2024 Hamid, Rawia; Walsh, Danica J.; Diamanti, Eleonora; Aguilar, Diana; Lacour, Antoine; Hamed, Mostafa M.; Hirsch, Anna K.H.
Target-Directed Dynamic Combinatorial Chemistry Affords Binders of Mycobacterium tuberculosis IspE
2024 Braun-Cornejo, Maria; Ornago, Camilla; Sonawane, Vidhisha; Haupenthal, Jörg; Kany, Andreas M.; Diamanti, Eleonora; Jézéquel, Gwenaëlle; Reiling, Norbert; Blankenfeldt, Wulf; Maas, Peter; Hirsch, Anna K. H.
Targeting Plasmodium falciparum IspD in the Methyl-d-erythritol Phosphate Pathway: Urea-Based Compounds with Nanomolar Potency on Target and Low-Micromolar Whole-Cell Activity
2024 Willocx, Daan; Bizzarri, Lorenzo; Alhayek, Alaa; Kannan, Deepika; Bravo, Patricia; Illarionov, Boris; Rox, Katharina; Lohse, Jonas; Fischer, Markus; Kany, Andreas M.; Hahne, Hannes; Rottmann, Matthias; Witschel, Matthias; Odom John, Audrey; Hamed, Mostafa M.; Diamanti, Eleonora; Hirsch, Anna K. H.
Targeting the Plasmodium falciparum IspE Enzyme
2024 Diamanti, Eleonora; Steinbach, Annina M.; de Carvalho, Lais P.; Ropponen, Henni-Karoliina; Lacour, Antoine; Hamid, Rawia; Eisa, Sidra; Bravo, Patricia; Bousis, Spyridon; Illarionov, Boris; Fischer, Markus; Hamed, Mostafa M.; Bach, Nina C.; Rottmann, Matthias; Held, Jana; Witschel, Matthias; Sieber, Stephan A.; Hirsch, Anna K. H.
Back in Person: Frontiers in Medicinal Chemistry 2023
2023 Gehringer, Matthias; Pape, Felix; Méndez, María; Barbie, Philipp; Unzue Lopez, Andrea; Lefranc, Julien; Klingler, Franca-Maria; Hessler, Gerhard; Langer, Thierry; Diamanti, Eleonora; Schiedel, Matthias
Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists?
2023 Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria
Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors
2023 Ropponen, Henni-Karoliina; Diamanti, Eleonora; Johannsen, Sandra; Illarionov, Boris; Hamid, Rawia; Jaki, Miriam; Sass, Peter; Fischer, Markus; Haupenthal, Jörg; Hirsch, Anna K H
Identification of inhibitors targeting the energy-coupling factor (ECF) transporters
2023 Diamanti, Eleonora; Souza, Paulo C T; Setyawati, Inda; Bousis, Spyridon; Gómez, Leticia M; Swier, Lotteke J Y M; Shams, Atanaz; Tsarenko, Aleksei; Stanek, Weronika K; Jäger, Manuel; Marrink, Siewert J; Slotboom, Dirk J; Hirsch, Anna K H
An Efficient Way to Screen Inhibitors of Energy-Coupling Factor (ECF) Transporters in a Bacterial Uptake Assay
2022 Bousis, Spyridon; Winkler, Steffen; Haupenthal, Jörg; Fulco, Francesco; Diamanti, Eleonora; Hirsch, Anna K H
Frontiers in Medicinal Chemistry 2022 Goes Virtual
2022 Diamanti, Eleonora; Méndez, María; Ross, Tatjana; Kuttruff, Christian A; Lefranc, Julien; Klingler, Franca-Maria; von Nussbaum, Franz; Jung, Manfred; Gehringer, Matthias
Structure-Guided Optimization of Small-Molecule Folate Uptake Inhibitors Targeting the Energy-Coupling Factor Transporters
2022 Kiefer, Alexander F; Bousis, Spyridon; Hamed, Mostafa M; Diamanti, Eleonora; Haupenthal, Jörg; Hirsch, Anna K H
Targeting the IspD Enzyme in the MEP Pathway: Identification of a Novel Fragment Class
2022 Diamanti, Eleonora; Hamed, Mostafa M; Lacour, Antoine; Bravo, Patricia; Illarionov, Boris; Fischer, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H
Assessment of the rules related to gaining activity against Gram-negative bacteria
2021 Ropponen, Henni-Karoliina; Diamanti, Eleonora; Siemens, Alexandra; Illarionov, Boris; Haupenthal, Jörg; Fischer, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H
Bacteriomimetic Liposomes Improve Antibiotic Activity of a Novel Energy-Coupling Factor Transporter Inhibitor
2021 Drost, M; Diamanti, E; Fuhrmann, K; Goes, A; Shams, A; Haupenthal, J; Koch, M; Hirsch, AKH; Fuhrmann, G
Search for the Active Ingredients from a 2-Aminothiazole DMSO Stock Solution with Antimalarial Activity
2021 Ropponen, Henni-Karoliina; Bader, Chantal D; Diamanti, Eleonora; Illarionov, Boris; Rottmann, Matthias; Fischer, Markus; Witschel, Matthias; Müller, Rolf; Hirsch, Anna K H
Energy-Coupling Factor Transporters as Novel Antimicrobial Targets
2019 Spyridon Bousis; Inda Setyawati; Eleonora Diamanti; Dirk J. Slotboom; Anna K. H. Hirsch
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Benign-by-Design SAHA Analogues for Human and Animal Vector-Borne Parasitic Diseases | Rossi, Michele; Martinengo, Bianca; Diamanti, Eleonora; Salerno, Alessandra; Rizzardi, Nicola; Fa...to, Romana; Bergamini, Christian; Souza de Oliveira, Andressa; de Araújo Marques Ferreira, Thais; Andrade Holanda, Cleonice; Romeiro, Luiz Antonio Soares; Soeiro, Maria de Nazaré Correia; Nunes, Krislayne; Ferreira de Almeida Fiuza, Ludmila; Meuser Batista, Marcos; Fraga, Carlos A. M.; E. A. Alkhalaf, Hamed; Elmahallawy, Ehab Kotb; Ebiloma, Godwin U.; De Koning, Harry P.; Vittorio, Serena; Vistoli, Giulio; Blanquart, Christophe; Bertrand, Philippe; Bolognesi, Maria Laura | 2024-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
Expression and characterization of pantothenate energy‐coupling factor transporters as an anti‐infective drug target | Shams, Atanaz; Bousis, Spyridon; Diamanti, Eleonora; Elgaher, Walid A. M.; Zeimetz, Lucie; Haupen...thal, Jörg; Slotboom, Dirk J.; Hirsch, Anna K. H. | 2024-01-01 | PROTEIN SCIENCE | - | 1.01 Articolo in rivista | 10.1002_pro.5195.pdf |
Harnessing the 12 Green Chemistry Principles for Sustainable Antiparasitic Drugs: Toward the One Health Approach | Martinengo, Bianca; Diamanti, Eleonora; Uliassi, Elisa; Bolognesi, Maria Laura | 2024-01-01 | ACS INFECTIOUS DISEASES | - | 1.01 Articolo in rivista | martinengo-et-al-2024-harnessing-the-12-green-chemistry-principles-for-sustainable-antiparasitic-drugs-toward-the-one.pdf; id4c00172_si_001.pdf |
Hit optimization by dynamic combinatorial chemistry on Streptococcus pneumoniae energy-coupling factor transporter ECF-PanT | Exapicheidou, Ioulia Antonia; Shams, Atanaz; Ibrahim, Hamza; Tsarenko, Aleksei; Backenköhler, Mic...hael; Hamed, Mostafa M.; Diamanti, Eleonora; Volkamer, Andrea; Slotboom, Dirk J.; Hirsch, Anna K. H. | 2024-01-01 | CHEMICAL COMMUNICATIONS | - | 1.01 Articolo in rivista | - |
IspE kinase as an anti-infective target: Role of a hydrophobic pocket in inhibitor binding | Hamid, Rawia; Walsh, Danica J.; Diamanti, Eleonora; Aguilar, Diana; Lacour, Antoine; Hamed, Mosta...fa M.; Hirsch, Anna K.H. | 2024-01-01 | STRUCTURE | - | 1.01 Articolo in rivista | - |
Target-Directed Dynamic Combinatorial Chemistry Affords Binders of Mycobacterium tuberculosis IspE | Braun-Cornejo, Maria; Ornago, Camilla; Sonawane, Vidhisha; Haupenthal, Jörg; Kany, Andreas M.; Di...amanti, Eleonora; Jézéquel, Gwenaëlle; Reiling, Norbert; Blankenfeldt, Wulf; Maas, Peter; Hirsch, Anna K. H. | 2024-01-01 | ACS OMEGA | - | 1.01 Articolo in rivista | - |
Targeting Plasmodium falciparum IspD in the Methyl-d-erythritol Phosphate Pathway: Urea-Based Compounds with Nanomolar Potency on Target and Low-Micromolar Whole-Cell Activity | Willocx, Daan; Bizzarri, Lorenzo; Alhayek, Alaa; Kannan, Deepika; Bravo, Patricia; Illarionov, Bo...ris; Rox, Katharina; Lohse, Jonas; Fischer, Markus; Kany, Andreas M.; Hahne, Hannes; Rottmann, Matthias; Witschel, Matthias; Odom John, Audrey; Hamed, Mostafa M.; Diamanti, Eleonora; Hirsch, Anna K. H. | 2024-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | JMedChem-2024.pdf; jm4c00212_si_001.pdf |
Targeting the Plasmodium falciparum IspE Enzyme | Diamanti, Eleonora; Steinbach, Annina M.; de Carvalho, Lais P.; Ropponen, Henni-Karoliina; Lacour..., Antoine; Hamid, Rawia; Eisa, Sidra; Bravo, Patricia; Bousis, Spyridon; Illarionov, Boris; Fischer, Markus; Hamed, Mostafa M.; Bach, Nina C.; Rottmann, Matthias; Held, Jana; Witschel, Matthias; Sieber, Stephan A.; Hirsch, Anna K. H. | 2024-01-01 | ACS OMEGA | - | 1.01 Articolo in rivista | - |
Back in Person: Frontiers in Medicinal Chemistry 2023 | Gehringer, Matthias; Pape, Felix; Méndez, María; Barbie, Philipp; Unzue Lopez, Andrea; Lefranc, J...ulien; Klingler, Franca-Maria; Hessler, Gerhard; Langer, Thierry; Diamanti, Eleonora; Schiedel, Matthias | 2023-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2023 - Gehringer - Back in Person Frontiers in Medicinal Chemistry 2023.pdf |
Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists? | Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria | 2023-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2023 - Pasieka - Click Chemistry and Targeted Degradation A Winning Combination for Medicinal Chemists.pdf |
Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors | Ropponen, Henni-Karoliina; Diamanti, Eleonora; Johannsen, Sandra; Illarionov, Boris; Hamid, Rawia...; Jaki, Miriam; Sass, Peter; Fischer, Markus; Haupenthal, Jörg; Hirsch, Anna K H | 2023-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2023 - Ropponen - Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors.pdf; downloadSupplement.pdf |
Identification of inhibitors targeting the energy-coupling factor (ECF) transporters | Diamanti, Eleonora; Souza, Paulo C T; Setyawati, Inda; Bousis, Spyridon; Gómez, Leticia M; Swier,... Lotteke J Y M; Shams, Atanaz; Tsarenko, Aleksei; Stanek, Weronika K; Jäger, Manuel; Marrink, Siewert J; Slotboom, Dirk J; Hirsch, Anna K H | 2023-01-01 | COMMUNICATIONS BIOLOGY | - | 1.01 Articolo in rivista | s42003-023-05555-x (5).pdf; 42003_2023_5555_MOESM1_ESM.pdf; 42003_2023_5555_MOESM3_ESM.xlsx |
An Efficient Way to Screen Inhibitors of Energy-Coupling Factor (ECF) Transporters in a Bacterial Uptake Assay | Bousis, Spyridon; Winkler, Steffen; Haupenthal, Jörg; Fulco, Francesco; Diamanti, Eleonora; Hirsc...h, Anna K H | 2022-01-01 | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - | 1.01 Articolo in rivista | ijms-23-02637.pdf; ijms-23-02637-s001.zip |
Frontiers in Medicinal Chemistry 2022 Goes Virtual | Diamanti, Eleonora; Méndez, María; Ross, Tatjana; Kuttruff, Christian A; Lefranc, Julien; Klingle...r, Franca-Maria; von Nussbaum, Franz; Jung, Manfred; Gehringer, Matthias | 2022-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
Structure-Guided Optimization of Small-Molecule Folate Uptake Inhibitors Targeting the Energy-Coupling Factor Transporters | Kiefer, Alexander F; Bousis, Spyridon; Hamed, Mostafa M; Diamanti, Eleonora; Haupenthal, Jörg; Hi...rsch, Anna K H | 2022-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | kiefer-et-al-2022-structure-guided-optimization-of-small-molecule-folate-uptake-inhibitors-targeting-the-energy.pdf; From Bitter to Sweet_ a preliminary study towards a patient-friendly Praziquantel dosage form.pdf; jm1c02114_si_001.pdf |
Targeting the IspD Enzyme in the MEP Pathway: Identification of a Novel Fragment Class | Diamanti, Eleonora; Hamed, Mostafa M; Lacour, Antoine; Bravo, Patricia; Illarionov, Boris; Fische...r, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H | 2022-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2021 - Diamanti - Targeting the IspD Enzyme in the MEP Pathway Identification of a Novel Fragment Class (1).pdf |
Assessment of the rules related to gaining activity against Gram-negative bacteria | Ropponen, Henni-Karoliina; Diamanti, Eleonora; Siemens, Alexandra; Illarionov, Boris; Haupenthal,... Jörg; Fischer, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H | 2021-01-01 | RSC MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Bacteriomimetic Liposomes Improve Antibiotic Activity of a Novel Energy-Coupling Factor Transporter Inhibitor | Drost, M; Diamanti, E; Fuhrmann, K; Goes, A; Shams, A; Haupenthal, J; Koch, M; Hirsch, AKH; Fuhrm...ann, G | 2021-01-01 | PHARMACEUTICS | - | 1.01 Articolo in rivista | pharmaceutics-14-00004.pdf; pharmaceutics-14-00004-s001.zip |
Search for the Active Ingredients from a 2-Aminothiazole DMSO Stock Solution with Antimalarial Activity | Ropponen, Henni-Karoliina; Bader, Chantal D; Diamanti, Eleonora; Illarionov, Boris; Rottmann, Mat...thias; Fischer, Markus; Witschel, Matthias; Müller, Rolf; Hirsch, Anna K H | 2021-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | CMDC-16-2089.pdf; downloadSupplement.pdf |
Energy-Coupling Factor Transporters as Novel Antimicrobial Targets | Spyridon Bousis; Inda Setyawati; Eleonora Diamanti; Dirk J. Slotboom; Anna K. H. Hirsch | 2019-01-01 | ADVANCED THERAPEUTICS | - | 1.01 Articolo in rivista | - |