CACIOLLA, JESSICA

CACIOLLA, JESSICA  

DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE  

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Risultati 1 - 7 di 7 (tempo di esecuzione: 0.097 secondi).
Titolo Autore(i) Anno Periodico Editore Tipo File
Balanced dual acting compounds targeting aromatase and estrogen receptor α as an emerging therapeutic opportunity to counteract estrogen responsive breast cancer Caciolla J.; Martini S.; Spinello A.; Pavlin M.; Turrini E.; Simonelli F.; Belluti F.; Rampa A.; ...Bisi A.; Fimognari C.; Zaffaroni N.; Gobbi S.; Magistrato A. 2021-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Fragment Merging, Growing, and Linking Identify New Trypanothione Reductase Inhibitors for Leishmaniasis Exertier, Cécile; Salerno, Alessandra; Antonelli, Lorenzo; Fiorillo, Annarita; Ocello, Riccardo; ...Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Masetti, Matteo; Fiorentino, Eleonora; Orsini, Stefania; Di Muccio, Trentina; Ilari, Andrea; Bolognesi, Maria Laura 2024-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista exertier-et-al-2024-fragment-merging-growing-and-linking-identify-new-trypanothione-reductase-inhibitors-for.pdfjm3c01439_si_001.pdf
Multifaceted activity of polyciclic MDR revertant agents in drug-resistant leukemic cells: Role of the spacer Caciolla J.; Picone G.; Farruggia G.; Valenti D.; Rampa A.; Malucelli E.; Belluti F.; Trezza A.; ...Spiga O.; Iotti S.; Gobbi S.; Cappadone C.; Bisi A. 2021-01-01 BIOORGANIC CHEMISTRY - 1.01 Articolo in rivista Bioorg Chem.pdf
Reconsidering Aromatase for Breast Cancer Treatment: New Roles for an Old Target Caciolla J.; Bisi A.; Belluti F.; Rampa A.; Gobbi S. 2020-01-01 MOLECULES - 1.01 Articolo in rivista Molecules review 2020.pdf
Single-digit nanomolar inhibitors lock the aromatase active site via a dualsteric targeting strategy Caciolla J.; Martini S.; Spinello A.; Belluti F.; Bisi A.; Zaffaroni N.; Magistrato A.; Gobbi S. 2022-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Switching from Aromatase Inhibitors to Dual Targeting Flavonoid-Based Compounds for Breast Cancer Treatment Gobbi S.; Martini S.; Rozza R.; Spinello A.; Caciolla J.; Rampa A.; Belluti F.; Zaffaroni N.; Mag...istrato A.; Bisi A. 2023-01-01 MOLECULES - 1.01 Articolo in rivista 2023 Molecules.pdfmolecules-28-03047-s001.zip
Targeting Orthosteric and Allosteric Pockets of Aromatase via Dual-Mode Novel Azole Inhibitors Caciolla J.; Spinello A.; Martini S.; Bisi A.; Zaffaroni N.; Gobbi S.; Magistrato A. 2020-01-01 ACS MEDICINAL CHEMISTRY LETTERS - 1.01 Articolo in rivista -