CACIOLLA, JESSICA
CACIOLLA, JESSICA
DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Balanced dual acting compounds targeting aromatase and estrogen receptor α as an emerging therapeutic opportunity to counteract estrogen responsive breast cancer
2021 Caciolla J.; Martini S.; Spinello A.; Pavlin M.; Turrini E.; Simonelli F.; Belluti F.; Rampa A.; Bisi A.; Fimognari C.; Zaffaroni N.; Gobbi S.; Magistrato A.
Fragment Merging, Growing, and Linking Identify New Trypanothione Reductase Inhibitors for Leishmaniasis
2024 Exertier, Cécile; Salerno, Alessandra; Antonelli, Lorenzo; Fiorillo, Annarita; Ocello, Riccardo; Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Masetti, Matteo; Fiorentino, Eleonora; Orsini, Stefania; Di Muccio, Trentina; Ilari, Andrea; Bolognesi, Maria Laura
Multifaceted activity of polyciclic MDR revertant agents in drug-resistant leukemic cells: Role of the spacer
2021 Caciolla J.; Picone G.; Farruggia G.; Valenti D.; Rampa A.; Malucelli E.; Belluti F.; Trezza A.; Spiga O.; Iotti S.; Gobbi S.; Cappadone C.; Bisi A.
Reconsidering Aromatase for Breast Cancer Treatment: New Roles for an Old Target
2020 Caciolla J.; Bisi A.; Belluti F.; Rampa A.; Gobbi S.
Single-digit nanomolar inhibitors lock the aromatase active site via a dualsteric targeting strategy
2022 Caciolla J.; Martini S.; Spinello A.; Belluti F.; Bisi A.; Zaffaroni N.; Magistrato A.; Gobbi S.
Switching from Aromatase Inhibitors to Dual Targeting Flavonoid-Based Compounds for Breast Cancer Treatment
2023 Gobbi S.; Martini S.; Rozza R.; Spinello A.; Caciolla J.; Rampa A.; Belluti F.; Zaffaroni N.; Magistrato A.; Bisi A.
Targeting Orthosteric and Allosteric Pockets of Aromatase via Dual-Mode Novel Azole Inhibitors
2020 Caciolla J.; Spinello A.; Martini S.; Bisi A.; Zaffaroni N.; Gobbi S.; Magistrato A.
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
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Balanced dual acting compounds targeting aromatase and estrogen receptor α as an emerging therapeutic opportunity to counteract estrogen responsive breast cancer | Caciolla J.; Martini S.; Spinello A.; Pavlin M.; Turrini E.; Simonelli F.; Belluti F.; Rampa A.; ...Bisi A.; Fimognari C.; Zaffaroni N.; Gobbi S.; Magistrato A. | 2021-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Fragment Merging, Growing, and Linking Identify New Trypanothione Reductase Inhibitors for Leishmaniasis | Exertier, Cécile; Salerno, Alessandra; Antonelli, Lorenzo; Fiorillo, Annarita; Ocello, Riccardo; ...Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Masetti, Matteo; Fiorentino, Eleonora; Orsini, Stefania; Di Muccio, Trentina; Ilari, Andrea; Bolognesi, Maria Laura | 2024-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | exertier-et-al-2024-fragment-merging-growing-and-linking-identify-new-trypanothione-reductase-inhibitors-for.pdf; jm3c01439_si_001.pdf |
Multifaceted activity of polyciclic MDR revertant agents in drug-resistant leukemic cells: Role of the spacer | Caciolla J.; Picone G.; Farruggia G.; Valenti D.; Rampa A.; Malucelli E.; Belluti F.; Trezza A.; ...Spiga O.; Iotti S.; Gobbi S.; Cappadone C.; Bisi A. | 2021-01-01 | BIOORGANIC CHEMISTRY | - | 1.01 Articolo in rivista | Bioorg Chem.pdf |
Reconsidering Aromatase for Breast Cancer Treatment: New Roles for an Old Target | Caciolla J.; Bisi A.; Belluti F.; Rampa A.; Gobbi S. | 2020-01-01 | MOLECULES | - | 1.01 Articolo in rivista | Molecules review 2020.pdf |
Single-digit nanomolar inhibitors lock the aromatase active site via a dualsteric targeting strategy | Caciolla J.; Martini S.; Spinello A.; Belluti F.; Bisi A.; Zaffaroni N.; Magistrato A.; Gobbi S. | 2022-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Switching from Aromatase Inhibitors to Dual Targeting Flavonoid-Based Compounds for Breast Cancer Treatment | Gobbi S.; Martini S.; Rozza R.; Spinello A.; Caciolla J.; Rampa A.; Belluti F.; Zaffaroni N.; Mag...istrato A.; Bisi A. | 2023-01-01 | MOLECULES | - | 1.01 Articolo in rivista | 2023 Molecules.pdf; molecules-28-03047-s001.zip |
Targeting Orthosteric and Allosteric Pockets of Aromatase via Dual-Mode Novel Azole Inhibitors | Caciolla J.; Spinello A.; Martini S.; Bisi A.; Zaffaroni N.; Gobbi S.; Magistrato A. | 2020-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |