DE MARCO, ROSSELLA
DE MARCO, ROSSELLA
DIPARTIMENTO DI CHIMICA "GIACOMO CIAMICIAN"
Assegnisti
5-aminomethyloxazolidine-2,4-dione hybrid α/β-dipeptide scaffolds as inductors of constrained conformations: Applications to the synthesis of integrin antagonists
2015 De Marco, Rossella; Mazzotti, Giacomo; Dattoli, Samantha D.; Baiula, Monica; Spampinato, Santi; Greco, Arianna; Gentilucci, Luca
A new generation of opioid peptidomimetics acting as central and/or peripheral analgesics
2012 R. De Marco; A. Tolomelli; A. Bedini; S. Spampinato; L. Gentilucci
A novel family of minimalist opioid peptides deprived of the classic pharmacophores
2011 L. Gentilucci; R. de Marco; A. Tolomelli; S. Feddersen; S. Spampinato; A. Bedini; R. Artali
A simple route towards peptide analogues containing substituted (S)- or (R)-tryptophans
2010 L. Gentilucci; L. Cerisoli; R. De Marco; A. Tolomelli
Ac-D-Trp-PheNH2 AND Ac-D-Trp-Phe-GlyNH2 - A NEW CLASS OF UNUSUAL OPIOID PEPTIDES
2010 L. Gentilucci; R. De Marco; A. Tolomelli; S. Spampinato; A. Bedini; R. Artali
Analytical pyrolysis of dipeptides containing proline and amino acids with polar side chains. Novel 2,5-diketopiperazine markers in the pyrolysates of proteins
2012 D. Fabbri; A.Adamiano; G. Falini; R. De Marco; I. Mancini
Antiangiogenic Effect of Dual/Selective α5β1/αvβ3 Integrin Antagonists Designed on Partially Modified Retro-Inverso Cyclotetrapeptide Mimetics
2010 L. Gentilucci; G. Cardillo; S. Spampinato; A. Tolomelli; F. Squassabia; R. De Marco; A. Bedini; M. Baiula; L. Belvisi; M. Civera
Chemical Modifications Designed to Improve Peptide Stability: Incorporation of Non-Natural Amino Acids, Pseudo-Peptide Bonds, and Cyclization
2010 L. Gentilucci; R. De Marco; L. Cerisoli
Constraining Endomorphin-1 by β,α-Hybrid Dipeptide/Heterocycle Scaffolds: Identification of a Novel κ-Opioid Receptor Selective Partial Agonist
2018 De Marco, Rossella; Bedini, Andrea; Spampinato, Santi*; Comellini, Lorenzo; Zhao, Junwei; Artali, Roberto; Gentilucci, Luca
Controlled solid phase peptide bond formation using N-carboxyanhydrides and PEG resins in water.
2013 De Marco R; Tolomelli A; Greco A; Gentilucci L
Controlling Cyclopeptide Backbone Conformation with β/α-Hybrid Peptide–Heterocycle Scaffolds
2016 Gentilucci, Luca; Gallo, Francesca; Meloni, Fernanda; Mastandrea, Marco; Del Secco, Benedetta; de Marco, Rossella
Convenient Synthesis of the Antibiotic Linezolid via an Oxazolidine-2,4-dione Intermediate Derived from the Chiral Building Block Isoserine
2014 Greco, A.; De Marco, R.; Tani, S.; Giacomini, D.; Galletti, P.; Tolomelli, A.; Juaristi, E.; Gentilucci, L.
Cyclic side-chain-linked opioid analogs utilizing cis- and trans-4-aminocyclohexyl-d-alanine
2014 Piekielna, J.; Gentilucci, L.; De Marco, R.; Perlikowska, R.; Adamska, A.; Olczak, J.; Mazur, M.; Artali, R.; Modranka, J.; Janecki, T.; Tomboly, C.; Janecka, A.
Cyclopeptide analogs for generating new molecular and 3D diversity
2009 L. Gentilucci; G. Cardillo; A. Tolomelli; F. Squassabia; R. De Marco; G. Chiriano
Dehydro-beta-amino acid containing peptidomimetics as integrin receptor ligands
2012 A. Tolomelli; A. Viola; L. Gentilucci; E. Mosconi; R. De Marco; M. Baiula; S. Spampinato; L. Belvisi; M. Civera
Design and characterization of opioid ligands based on cycle-in-macrocycle scaffold
2017 Adamska-Bartłomiejczyk, Anna; De Marco, Rossella; Gentilucci, Luca; Kluczyk, Alicja; Janecka, Anna
DESIGN AND SYNTHESIS OF OPIOID PEPTIDE ANALOGUES AND MIMETICS
2011 R.De Marco; L. Gentilucci; A. Tolomelli; S. Feddersen; S. Spampinato; A. Bedini; R. Artali.
DETERMINATION OF THE BIOLOGICALLY ACTIVE STRUCTURE OF THE ATYPICAL MOR-LIGAND c[D-Asp-1-amide-beta-Ala-D-Trp-Phe] AND ANALOGUES BY NMR AND MOLECULAR DOCKING
2010 L. Gentilucci; A.Tolomelli; S. Spampinato; A. Bedini; R. De Marco; R. Artali
Development and characterization of Endomorphin-1 analogues as novel potential analgesic drugs.
2009 Bedini A; Gentilucci L; Demarco R; Spampinato S
Diagnostic implementation of fast and selective integrin-mediated adhesion of cancer cells on functionalized zeolite L monolayers
2015 Greco, A.; Maggini, L.; De Cola, L.; De Marco, R.; Gentilucci, L.