Sfoglia per Autore
Discovery of Sustainable Drugs for Neglected Tropical Diseases: Cashew Nut Shell Liquid (CNSL)-Based Hybrids Target Mitochondrial Function and ATP Production in Trypanosoma brucei
2019 Cerone M.; Uliassi E.; Prati F.; Ebiloma G.U.; Lemgruber L.; Bergamini C.; Watson D.G.; de A. M. Ferreira T.; Roth Cardoso G.S.H.; Soares Romeiro L.A.; de Koning H.P.; Bolognesi M.L.
Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease
2019 Chalupova K.; Korabecny J.; Bartolini M.; Monti B.; Lamba D.; Caliandro R.; Pesaresi A.; Brazzolotto X.; Gastellier A.-J.; Nachon F.; Pejchal J.; Jarosova M.; Hepnarova V.; Jun D.; Hrabinova M.; Dolezal R.; Zdarova Karasova J.; Mzik M.; Kristofikova Z.; Misik J.; Muckova L.; Jost P.; Soukup O.; Benkova M.; Setnicka V.; Habartova L.; Chvojkova M.; Kleteckova L.; Vales K.; Mezeiova E.; Uliassi E.; Valis M.; Nepovimova E.; Bolognesi M.L.; Kuca K.
Cashew nut shell liquid (Cnsl) as a source of drugs for alzheimer’s disease
2021 Uliassi E.; de Oliveira A.S.; Nascente L.C.; Romeiro L.A.S.; Bolognesi M.L.
Sustainable production of pharmaceutical, nutraceutical and bioactive compounds from biomass and waste
2021 Espro C.; Paone E.; Mauriello F.; Gotti R.; Uliassi E.; Bolognesi M.L.; Rodriguez-Padron D.; Luque R.
Discovery of sustainable drugs for Alzheimer's disease: cardanol-derived cholinesterase inhibitors with antioxidant and anti-amyloid properties
2021 Ramos, GD; de Oliveira, AS; Bartolini, M; Naldi, M; Liparulo, I; Bergamini, C; Uliassi, E; Wu, L; Fraser, PE; Abreu, M; Kiametis, AS; Gargano, R; Silveira, ER; Brand, GD; Prchal, L; Soukup, O; Korabecny, J; Bolognesi, ML; Romeiro, LAS
Turning Donepezil into a Multi-Target-Directed Ligand through a Merging Strategy
2021 Perone R.; Albertini C.; Uliassi E.; Di Pietri F.; de Sena Murteira Pinheiro P.; Petralla S.; Rizzardi N.; Fato R.; Pulkrabkova L.; Soukup O.; Tramarin A.; Bartolini M.; Bolognesi M.L.
Phenothiazine-Tacrine Heterodimers: Pursuing Multitarget Directed Approach in Alzheimer's Disease
2021 Gorecki L.; Uliassi E.; Bartolini M.; Janockova J.; Hrabinova M.; Hepnarova V.; Prchal L.; Muckova L.; Pejchal J.; Karasova J.Z.; Mezeiova E.; Benkova M.; Kobrlova T.; Soukup O.; Petralla S.; Monti B.; Korabecny J.; Bolognesi M.L.
Riluzole-Rasagiline Hybrids: Toward the Development of Multi-Target-Directed Ligands for Amyotrophic Lateral Sclerosis
2022 Albertini, C; Salerno, A; Atzenti, S; Uliassi, E; Massenzio, F; Maruca, A; Rocca, R; Mecava, M; Silva, FSG; Mena, D; Valente, P; Duarte, AI; Chavarria, D; Bissaro, M; Moro, S; Federico, S; Spalluto, G; Soukup, O; Borges, F; Alcaro, S; Monti, B; Oliveira, PJ; Menendez, JC; Bolognesi, ML
The Use of Zidovudine Pharmacophore in Multi-Target-Directed Ligands for AIDS Therapy
2022 Bianco M.D.C.A.D.; Inacio Leite D.; Silva Castelo Branco F.; Boechat N.; Uliassi E.; Bolognesi M.L.; Bastos M.M.
Therapeutic strategies for identifying small molecules against prion diseases
2022 Uliassi, Elisa; Nikolic, Lea; Bolognesi, Maria Laura; Legname, Giuseppe
Identification of a Quinone Derivative as a YAP/TEAD Activity Modulator from a Repurposing Library
2022 Lauriola A.; Uliassi E.; Santucci M.; Bolognesi M.L.; Mor M.; Scalvini L.; Elisi G.M.; Gozzi G.; Tagliazucchi L.; Marverti G.; Ferrari S.; Losi L.; D'Arca D.; Costi M.P.
Enriching Proteolysis Targeting Chimeras with a Second Modality: When Two Are Better Than One
2022 Salerno, Alessandra; Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Testi, Eleonora; Guardigni, Melissa; Roberti, Marinella; Milelli, Andrea; Bolognesi, Maria Laura
PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease
2023 Guardigni M.; Pruccoli L.; Santini A.; Simone A.D.; Bersani M.; Spyrakis F.; Frabetti F.; Uliassi E.; Andrisano V.; Pagliarani B.; Fernández-Gómez P.; Palomo V.; Bolognesi M.L.; Tarozzi A.; Milelli A.
Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists?
2023 Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria
Targeted Protein Degradation for Infectious Diseases: from Basic Biology to Drug Discovery
2023 Rocío Marisol Espinoza Chávez; Salerno A.; Liuzzi A.; Ilari A.; Milelli A.; Uliassi E.; Bolognesi M.L.
Quinolinetrione-tacrine hybrids as multi-target-directed ligands against Alzheimer's disease
2023 Uliassi, E; Bergamini, C; Rizzardi, N; Naldi, M; Cores, A; Bartolini, M; Menéndez, JC; Bolognesi, ML
Fragment Merging, Growing, and Linking Identify New Trypanothione Reductase Inhibitors for Leishmaniasis
2024 Exertier, Cécile; Salerno, Alessandra; Antonelli, Lorenzo; Fiorillo, Annarita; Ocello, Riccardo; Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Masetti, Matteo; Fiorentino, Eleonora; Orsini, Stefania; Di Muccio, Trentina; Ilari, Andrea; Bolognesi, Maria Laura
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
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Discovery of Sustainable Drugs for Neglected Tropical Diseases: Cashew Nut Shell Liquid (CNSL)-Based Hybrids Target Mitochondrial Function and ATP Production in Trypanosoma brucei | Cerone M.; Uliassi E.; Prati F.; Ebiloma G.U.; Lemgruber L.; Bergamini C.; Watson D.G.; de A. M. ...Ferreira T.; Roth Cardoso G.S.H.; Soares Romeiro L.A.; de Koning H.P.; Bolognesi M.L. | 2019-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease | Chalupova K.; Korabecny J.; Bartolini M.; Monti B.; Lamba D.; Caliandro R.; Pesaresi A.; Brazzolo...tto X.; Gastellier A.-J.; Nachon F.; Pejchal J.; Jarosova M.; Hepnarova V.; Jun D.; Hrabinova M.; Dolezal R.; Zdarova Karasova J.; Mzik M.; Kristofikova Z.; Misik J.; Muckova L.; Jost P.; Soukup O.; Benkova M.; Setnicka V.; Habartova L.; Chvojkova M.; Kleteckova L.; Vales K.; Mezeiova E.; Uliassi E.; Valis M.; Nepovimova E.; Bolognesi M.L.; Kuca K. | 2019-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | Novel tacrine-tryptophan hybrids_ Multi-target directed ligands as potential treatment for Alzheimer_s disease.pdf |
Cashew nut shell liquid (Cnsl) as a source of drugs for alzheimer’s disease | Uliassi E.; de Oliveira A.S.; Nascente L.C.; Romeiro L.A.S.; Bolognesi M.L. | 2021-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-26-05441.pdf |
Sustainable production of pharmaceutical, nutraceutical and bioactive compounds from biomass and waste | Espro C.; Paone E.; Mauriello F.; Gotti R.; Uliassi E.; Bolognesi M.L.; Rodriguez-Padron D.; Luqu...e R. | 2021-01-01 | CHEMICAL SOCIETY REVIEWS | - | 1.01 Articolo in rivista | Chem Soc Rev_revised-FINAL (2).pdf |
Discovery of sustainable drugs for Alzheimer's disease: cardanol-derived cholinesterase inhibitors with antioxidant and anti-amyloid properties | Ramos, GD; de Oliveira, AS; Bartolini, M; Naldi, M; Liparulo, I; Bergamini, C; Uliassi, E; Wu, L;... Fraser, PE; Abreu, M; Kiametis, AS; Gargano, R; Silveira, ER; Brand, GD; Prchal, L; Soukup, O; Korabecny, J; Bolognesi, ML; Romeiro, LAS | 2021-01-01 | RSC MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | GAR_RSC_Med_Chem_merged(1).pdf |
Turning Donepezil into a Multi-Target-Directed Ligand through a Merging Strategy | Perone R.; Albertini C.; Uliassi E.; Di Pietri F.; de Sena Murteira Pinheiro P.; Petralla S.; Riz...zardi N.; Fato R.; Pulkrabkova L.; Soukup O.; Tramarin A.; Bartolini M.; Bolognesi M.L. | 2021-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | Turning Donepezil into a Multi-Target Post print.pdf |
Phenothiazine-Tacrine Heterodimers: Pursuing Multitarget Directed Approach in Alzheimer's Disease | Gorecki L.; Uliassi E.; Bartolini M.; Janockova J.; Hrabinova M.; Hepnarova V.; Prchal L.; Muckov...a L.; Pejchal J.; Karasova J.Z.; Mezeiova E.; Benkova M.; Kobrlova T.; Soukup O.; Petralla S.; Monti B.; Korabecny J.; Bolognesi M.L. | 2021-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | acschemneuro.1c00184.pdf |
Riluzole-Rasagiline Hybrids: Toward the Development of Multi-Target-Directed Ligands for Amyotrophic Lateral Sclerosis | Albertini, C; Salerno, A; Atzenti, S; Uliassi, E; Massenzio, F; Maruca, A; Rocca, R; Mecava, M; S...ilva, FSG; Mena, D; Valente, P; Duarte, AI; Chavarria, D; Bissaro, M; Moro, S; Federico, S; Spalluto, G; Soukup, O; Borges, F; Alcaro, S; Monti, B; Oliveira, PJ; Menendez, JC; Bolognesi, ML | 2022-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | acschemneuro.2c00261.pdf |
The Use of Zidovudine Pharmacophore in Multi-Target-Directed Ligands for AIDS Therapy | Bianco M.D.C.A.D.; Inacio Leite D.; Silva Castelo Branco F.; Boechat N.; Uliassi E.; Bolognesi M....L.; Bastos M.M. | 2022-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-27-08502-v3.pdf |
Therapeutic strategies for identifying small molecules against prion diseases | Uliassi, Elisa; Nikolic, Lea; Bolognesi, Maria Laura; Legname, Giuseppe | 2022-01-01 | CELL & TISSUE RESEARCH | - | 1.01 Articolo in rivista | - |
Identification of a Quinone Derivative as a YAP/TEAD Activity Modulator from a Repurposing Library | Lauriola A.; Uliassi E.; Santucci M.; Bolognesi M.L.; Mor M.; Scalvini L.; Elisi G.M.; Gozzi G.; ...Tagliazucchi L.; Marverti G.; Ferrari S.; Losi L.; D'Arca D.; Costi M.P. | 2022-01-01 | PHARMACEUTICS | - | 1.01 Articolo in rivista | pharmaceutics-14-00391-v2.pdf |
Enriching Proteolysis Targeting Chimeras with a Second Modality: When Two Are Better Than One | Salerno, Alessandra; Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Testi, Eleonora; Gua...rdigni, Melissa; Roberti, Marinella; Milelli, Andrea; Bolognesi, Maria Laura | 2022-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | acs.jmedchem.2c00302.pdf |
PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease | Guardigni M.; Pruccoli L.; Santini A.; Simone A.D.; Bersani M.; Spyrakis F.; Frabetti F.; Uliassi... E.; Andrisano V.; Pagliarani B.; Fernández-Gómez P.; Palomo V.; Bolognesi M.L.; Tarozzi A.; Milelli A. | 2023-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | acschemneuro.3c00096.pdf; cn3c00096_si_001.pdf |
Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists? | Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria | 2023-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | ChemMedChem - 2023 - Pasieka - Click Chemistry and Targeted Degradation A Winning Combination for Medicinal Chemists.pdf |
Targeted Protein Degradation for Infectious Diseases: from Basic Biology to Drug Discovery | Rocío Marisol Espinoza Chávez; Salerno A.; Liuzzi A.; Ilari A.; Milelli A.; Uliassi E.; Bolognesi... M.L. | 2023-01-01 | ACS BIO & MED CHEM AU | - | 1.01 Articolo in rivista | acsbiomedchemau.2c00063.pdf |
Quinolinetrione-tacrine hybrids as multi-target-directed ligands against Alzheimer's disease | Uliassi, E; Bergamini, C; Rizzardi, N; Naldi, M; Cores, A; Bartolini, M; Menéndez, JC; Bolognesi, ML | 2023-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | 1-s2.0-S0968089623002675-main.pdf; 1-s2.0-S0968089623002675-mmc1.docx |
Fragment Merging, Growing, and Linking Identify New Trypanothione Reductase Inhibitors for Leishmaniasis | Exertier, Cécile; Salerno, Alessandra; Antonelli, Lorenzo; Fiorillo, Annarita; Ocello, Riccardo; ...Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Masetti, Matteo; Fiorentino, Eleonora; Orsini, Stefania; Di Muccio, Trentina; Ilari, Andrea; Bolognesi, Maria Laura | 2024-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | exertier-et-al-2024-fragment-merging-growing-and-linking-identify-new-trypanothione-reductase-inhibitors-for.pdf; jm3c01439_si_001.pdf |
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