Sfoglia per Autore
Novel Class of Quinone-Bearing Polyamines as Multi-Target-Directed Ligands To Combat Alzheimer's Disease
2007 Bolognesi ML; Banzi R; Bartolini M; Cavalli A; Tarozzi A; Andrisano V; Minarini A; Rosini M; Tumiatti V; Bergamini C; Fato R; Lenaz G; Hrelia P; Cattaneo A; Recanatini M; Melchiorre C.
A new EGFR inhibitor induces apoptosis in colon cancer cells.
2007 Calonghi N; Pagnotta E; Parolin C; Mangano C; Bolognesi ML; Melchiorre C; Masotti L.
Progettazione e sintesi di derivati poliamminici per il trattamento della malattia di Alzheimer
2007 V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; V. Andrisano; M. Bartolini; F. Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre
Memoquine derivatives as potent inhibitors of AChE-induced amyloid-beta aggregation
2007 Bolognesi ML; Cavalli A; Andrisano V; Bartolini M; Minarini A; Melchiorre C
Multi-target-directed small molecules to combat neurodegenerative diseases
2007 Melchiorre C
Reversible HSA binding of lipocrine: a circular dichroism study.
2007 Pistolozzi M.; Rosini M.; Melchiorre C.; Bertucci C.
Beta-secretase monolithic micro-IMER (immobilized enzyme reactor) for on-line HPLC screening of quinone-bearing polyamine inhibitors.
2007 Mancini F.; Bolognesi ML.; Minarini A.; Melchiorre C.; Andrisano V.
New quinazoline compounds as non-peptidomimetic BACE-1 inhibitors in the treatment of Alzheimer's disease
2007 Matera R; Minarini A; Rosini M; Andrisano V; Mancini F; Melchiorre C.
Structure-activity relationships of methoctramine-related polyamines as muscarinic antagonist: Effect of replacing the inner polymethylene chain with cyclic moieties
2007 V. Tumiatti; A. Minarini; A. Milelli; M. Rosini; M. Buccioni; G. Marucci; C. Ghelardini; C. Bellucci; C. Melchiorre
Insight Into the Kinetic of Amyloid beta (1-42) Peptide Self-Aggregation: Elucidation of Inhibitors' Mechanism of Action
2007 M. Bartolini; C. Bertucci; M.L. Bolognesi; A. Cavalli; C. Melchiorre; V. Andrisano
Multi-Target-Directed Drug Design Strategy: From a Dual Binding Site Acetylcholinesterase Inhibitor to a Trifunctional Compound against Alzheimer's Disease
2007 Bolognesi ML; Cavalli A; Valgimigli L; Bartolini M; Rosini M; Andrisano V; Recanatini M; Melchiorre C
Monolithic stationary phase coupled with coulometric detection: development of an ion-pair HPLC method for the analysis of quinone-bearing compounds.
2007 F. Mancini; ML Bolognesi; C. Melchiorre; A. Cavalli; V. Andrisano
Synthesis of monomeric derivatives to probe Memoquin bivalent interactions
2008 ML. Bolognesi; A. Minarini; M. Bartolini; A. Cavalli; F. Mancini; V. Andrisano; M. Rosini; V. Tumiatti; C. Melchiorre
From the universal template strategy to multi-site-directed ligands for the treatment of Alzheimer’s disease
2008 C. Melchiorre
Novel class of quinone-bearing polyamines as multi-target-directed ligands to combat Alzheimer’s disease
2008 C. Melchiorre
Structure-Activity Relationships of New Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone
2008 V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; M. Micco; V. Andrisano; M. Bartolini; F. Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre
A rational approach to multi-site-directed ligands for the treatment of Alzheimer’s disease
2008 C. Melchiorre
Synthesis of doxazosin analogues as alpha-1 adrenoceptor antagonists with prostate antitumor activity
2008 Giardinà D.; Martarelli D.; Sagratini G.; Angeli P.; Ballinari D.; Gulini U.; Medori E.; Melchiorre C.; Pompei L.
CYTOTOXICITY EVALUATION OF A POLYAMINE-QUINONE LIBRARY CONJUGATES IN HUMAN COLON CARCINOMA CELLS
2008 C. Mangano; N. Calonghi; C. Parolin; C. Cappadone; F. Di Giorgio; J. Hysomema; M.L. Bolognesi; C. Melchiorre; L. Masotti
Inhibition of Acetylcholinesterase, Beta-Amyloid Aggregation, and NMDA Receptors in Alzheimer's Disease: A Promising Direction for the Multi-target-Directed Ligands Gold Rush
2008 M. Rosini; E. Simoni; M. Bartolini; A. Cavalli; L. Ceccarini; N. Pascu; D. W. McClymont; A. Tarozzi; M. L. Bolognesi; A. Minarini; V. Tumiatti; V. Andrisano; I. R. Mellor; C. Melchiorre
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Novel Class of Quinone-Bearing Polyamines as Multi-Target-Directed Ligands To Combat Alzheimer's Disease | Bolognesi ML; Banzi R; Bartolini M; Cavalli A; Tarozzi A; Andrisano V; Minarini A; Rosini M; Tumi...atti V; Bergamini C; Fato R; Lenaz G; Hrelia P; Cattaneo A; Recanatini M; Melchiorre C. | 2007-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A new EGFR inhibitor induces apoptosis in colon cancer cells. | Calonghi N; Pagnotta E; Parolin C; Mangano C; Bolognesi ML; Melchiorre C; Masotti L. | 2007-01-01 | BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS | - | 1.01 Articolo in rivista | - |
Progettazione e sintesi di derivati poliamminici per il trattamento della malattia di Alzheimer | V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; V. Andrisano; M. Bartolini; F. ...Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Memoquine derivatives as potent inhibitors of AChE-induced amyloid-beta aggregation | Bolognesi ML; Cavalli A; Andrisano V; Bartolini M; Minarini A; Melchiorre C | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Multi-target-directed small molecules to combat neurodegenerative diseases | Melchiorre C | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Reversible HSA binding of lipocrine: a circular dichroism study. | Pistolozzi M.; Rosini M.; Melchiorre C.; Bertucci C. | 2007-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Beta-secretase monolithic micro-IMER (immobilized enzyme reactor) for on-line HPLC screening of quinone-bearing polyamine inhibitors. | Mancini F.; Bolognesi ML.; Minarini A.; Melchiorre C.; Andrisano V. | 2007-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
New quinazoline compounds as non-peptidomimetic BACE-1 inhibitors in the treatment of Alzheimer's disease | Matera R; Minarini A; Rosini M; Andrisano V; Mancini F; Melchiorre C. | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Structure-activity relationships of methoctramine-related polyamines as muscarinic antagonist: Effect of replacing the inner polymethylene chain with cyclic moieties | V. Tumiatti; A. Minarini; A. Milelli; M. Rosini; M. Buccioni; G. Marucci; C. Ghelardini; C. Bellu...cci; C. Melchiorre | 2007-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Insight Into the Kinetic of Amyloid beta (1-42) Peptide Self-Aggregation: Elucidation of Inhibitors' Mechanism of Action | M. Bartolini; C. Bertucci; M.L. Bolognesi; A. Cavalli; C. Melchiorre; V. Andrisano | 2007-01-01 | CHEMBIOCHEM | - | 1.01 Articolo in rivista | - |
Multi-Target-Directed Drug Design Strategy: From a Dual Binding Site Acetylcholinesterase Inhibitor to a Trifunctional Compound against Alzheimer's Disease | Bolognesi ML; Cavalli A; Valgimigli L; Bartolini M; Rosini M; Andrisano V; Recanatini M; Melchior...re C | 2007-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Monolithic stationary phase coupled with coulometric detection: development of an ion-pair HPLC method for the analysis of quinone-bearing compounds. | F. Mancini; ML Bolognesi; C. Melchiorre; A. Cavalli; V. Andrisano | 2007-01-01 | JOURNAL OF SEPARATION SCIENCE | - | 1.01 Articolo in rivista | - |
Synthesis of monomeric derivatives to probe Memoquin bivalent interactions | ML. Bolognesi; A. Minarini; M. Bartolini; A. Cavalli; F. Mancini; V. Andrisano; M. Rosini; V. Tum...iatti; C. Melchiorre | 2008-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
From the universal template strategy to multi-site-directed ligands for the treatment of Alzheimer’s disease | C. Melchiorre | 2008-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Novel class of quinone-bearing polyamines as multi-target-directed ligands to combat Alzheimer’s disease | C. Melchiorre | 2008-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Structure-Activity Relationships of New Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone | V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; M. Micco; V. Andrisano; M. Bart...olini; F. Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre | 2008-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
A rational approach to multi-site-directed ligands for the treatment of Alzheimer’s disease | C. Melchiorre | 2008-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Synthesis of doxazosin analogues as alpha-1 adrenoceptor antagonists with prostate antitumor activity | Giardinà D.; Martarelli D.; Sagratini G.; Angeli P.; Ballinari D.; Gulini U.; Medori E.; Melchior...re C.; Pompei L. | 2008-01-01 | DRUGS OF THE FUTURE | - | 4.02 Riassunto (Abstract) | - |
CYTOTOXICITY EVALUATION OF A POLYAMINE-QUINONE LIBRARY CONJUGATES IN HUMAN COLON CARCINOMA CELLS | C. Mangano; N. Calonghi; C. Parolin; C. Cappadone; F. Di Giorgio; J. Hysomema; M.L. Bolognesi; C.... Melchiorre; L. Masotti | 2008-01-01 | - | Firenze, university press | 4.02 Riassunto (Abstract) | - |
Inhibition of Acetylcholinesterase, Beta-Amyloid Aggregation, and NMDA Receptors in Alzheimer's Disease: A Promising Direction for the Multi-target-Directed Ligands Gold Rush | M. Rosini; E. Simoni; M. Bartolini; A. Cavalli; L. Ceccarini; N. Pascu; D. W. McClymont; A. Taroz...zi; M. L. Bolognesi; A. Minarini; V. Tumiatti; V. Andrisano; I. R. Mellor; C. Melchiorre | 2008-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile