Sfoglia per Autore
Preparation of (hetero)aromatic (hetero)cyclic carboxamides for the treatment of Alzheimer's disease
2006 M. Rosini; V. Andrisano; M. Bartolini; C. Melchiorre
Recent advances in the design and synthesis of prazosin derivatives
2006 A. Minarini; M.L. Bolognesi; V. Tumiatti; C. Melchiorre.
Design, synthesis, and biological evaluation of substituted 2,3-dihydro-1H-cyclopenta[b]quinolin-9-ylamine related compounds as fructose-1,6-bisphosphatase inhibitors
2006 M. Rosini; F. Mancini; A. Tarozzi; F. Colizzi; V. Andrisano; M.L. Bolognesi; P. Hrelia; C. Melchiorre.
A NEW EPIDERMAL GROWTH FACTOR RECEPTOR INHIBITOR IN COLON CANCER CELLS
2006 Parolin C.; Calonghi N.; Pagnotta E.; Mangano C.; Bolognesi M.L.; Melchiorre C.; Masotti L.
Process for preparation of 1,4-benzoquinone-2,5-diamines by reaction of amines with 1,4-benzoquinones bearing leaving groups at the 2- and 5-positions
2006 M.L. Bolognesi; R. Banzi; A. Minarini; C. Melchiorre
Methoctramine analogues inhibit capsaicin induced currents in dorsal root ganglia and Xenopus oocytes expressing TRPV1
2006 Mellor IR; Rosini M; Minarini A; Tumiatti V; Melchiorre C
Progettazione e sintesi di poliammine a potenziale attività antitumorale
2006 Tumiatti V; Milelli A; Minarini A; Bolognesi M; Baiocchi D; Roncuzzi L; Gasperi-Campani A; Melchiorre C
One-molecule-multiple-target strategy: a novel multifunctional molecule designed to block EGF-r and to exert pro-apoptotic effects
2006 M.L. Bolognesi; A. Antonello; A. Tarozzi; M. Rosini; A. Minarini; V. Tumiatti; P. Hrelia; C. Melchiorre.
Multitarget-directed drug design strategy: a novel molecule designed to block epidermal growth factor receptor (EGFR) and to exert proapoptotic effects
2006 A. Antonello; A. Tarozzi; F. Morroni; A. Cavalli; M. Rosini; P. Hrelia; M.L. Bolognesi; C. Melchiorre.
Lipoic acid, a lead structure for multi-target-directed drugs for neurodegeneration
2006 M.L. Bolognesi; A. Minarini; V. Tumiatti; C. Melchiorre
Progress in acetylcholinesterase inhibitors for Alzheimer's disease
2006 M.L. Bolognesi; A. Minarini; V. Tumiatti; C. Melchiorre
Multitarget-directed drug design strategy: novel hybrid compounds between lipocrine and carvedilol
2007 Rosini M; Simoni E; Bolognesi ML; Andrisano V; Bartolini M; Tarozzi a; Hrelia P; Mellor I; Melchiorre C.
Multi-target-directed drug design strategy: quinone derivatives designed to block amyloid-beta aggregation and to exert antioxidant effects
2007 Bolognesi ML; Lizzi F; Andrisano V; Bartolini M; Hrelia P; Tarozzi A; Tumiatti V; Melchiorre C.
Characterization of Cholinesterase inhibitors by means of immobilized enzyme reactor
2007 M. Bartolini; M.L. Bolognesi; A. Cavalli; C. Melchiorre; A. Rampa; M. Recanatini; V. Andrisano
Strategie farmacologiche per il trattamento della malattia di Alzheimer
2007 M.L. Bolognesi; C. Melchiorre
Multi-target-directed drugs for neurodegeneration
2007 C. Melchiorre
Quinone-bearing polyamines are AChE inhibitors endowed with multifunctional properties
2007 M.L. Bolognesi; R. Banzi; A. Cavalli; A. Minarini; M. Bartolini; V. Andrisano; M. Recanatini; C. Melchiorre
Multi-Target-Directed Drug Design Strategy: From a Dual Binding Site Acetylcholinesterase Inhibitor to a Trifunctional Compound against Alzheimer's Disease
2007 Bolognesi ML; Cavalli A; Valgimigli L; Bartolini M; Rosini M; Andrisano V; Recanatini M; Melchiorre C
A new EGFR inhibitor induces apoptosis in colon cancer cells.
2007 Calonghi N; Pagnotta E; Parolin C; Mangano C; Bolognesi ML; Melchiorre C; Masotti L.
Progettazione e sintesi di derivati poliamminici per il trattamento della malattia di Alzheimer
2007 V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; V. Andrisano; M. Bartolini; F. Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Preparation of (hetero)aromatic (hetero)cyclic carboxamides for the treatment of Alzheimer's disease | M. Rosini; V. Andrisano; M. Bartolini; C. Melchiorre | 2006-01-01 | - | - | 6.01 Brevetto | - |
Recent advances in the design and synthesis of prazosin derivatives |
A. Minarini; M.L. Bolognesi; V. Tumiatti; C. Melchiorre. |
2006-01-01 | EXPERT OPINION ON DRUG DISCOVERY | - | 1.01 Articolo in rivista | - |
Design, synthesis, and biological evaluation of substituted 2,3-dihydro-1H-cyclopenta[b]quinolin-9-ylamine related compounds as fructose-1,6-bisphosphatase inhibitors |
M. Rosini; F. Mancini; A. Tarozzi; F. Colizzi; V. Andrisano; M.L. Bolognesi; P. Hrelia; C.... Melchiorre. |
2006-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A NEW EPIDERMAL GROWTH FACTOR RECEPTOR INHIBITOR IN COLON CANCER CELLS | Parolin C.; Calonghi N.; Pagnotta E.; Mangano C.; Bolognesi M.L.; Melchiorre C.; Masotti L. | 2006-01-01 | ITALIAN JOURNAL OF BIOCHEMISTRY | - | 4.02 Riassunto (Abstract) | - |
Process for preparation of 1,4-benzoquinone-2,5-diamines by reaction of amines with 1,4-benzoquinones bearing leaving groups at the 2- and 5-positions |
M.L. Bolognesi; R. Banzi; A. Minarini; C. Melchiorre |
2006-01-01 | - | - | 6.01 Brevetto | - |
Methoctramine analogues inhibit capsaicin induced currents in dorsal root ganglia and Xenopus oocytes expressing TRPV1 | Mellor IR; Rosini M; Minarini A; Tumiatti V; Melchiorre C | 2006-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Progettazione e sintesi di poliammine a potenziale attività antitumorale | Tumiatti V; Milelli A; Minarini A; Bolognesi M; Baiocchi D; Roncuzzi L; Gasperi-Campani A; Melchi...orre C | 2006-01-01 | - | Società di chimica Italiana | 4.02 Riassunto (Abstract) | - |
One-molecule-multiple-target strategy: a novel multifunctional molecule designed to block EGF-r and to exert pro-apoptotic effects |
M.L. Bolognesi; A. Antonello; A. Tarozzi; M. Rosini; A. Minarini; V. Tumiatti; P. Hrelia; C.... Melchiorre. |
2006-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Multitarget-directed drug design strategy: a novel molecule designed to block epidermal growth factor receptor (EGFR) and to exert proapoptotic effects |
A. Antonello; A. Tarozzi; F. Morroni; A. Cavalli; M. Rosini; P. Hrelia; M.L. Bolognesi; C.... Melchiorre. |
2006-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Lipoic acid, a lead structure for multi-target-directed drugs for neurodegeneration | M.L. Bolognesi; A. Minarini; V. Tumiatti; C. Melchiorre | 2006-01-01 | MINI-REVIEWS IN MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Progress in acetylcholinesterase inhibitors for Alzheimer's disease | M.L. Bolognesi; A. Minarini; V. Tumiatti; C. Melchiorre | 2006-01-01 | EXPERT OPINION ON THERAPEUTIC PATENTS | - | 1.01 Articolo in rivista | - |
Multitarget-directed drug design strategy: novel hybrid compounds between lipocrine and carvedilol | Rosini M; Simoni E; Bolognesi ML; Andrisano V; Bartolini M; Tarozzi a; Hrelia P; Mellor I; Melchi...orre C. | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Multi-target-directed drug design strategy: quinone derivatives designed to block amyloid-beta aggregation and to exert antioxidant effects | Bolognesi ML; Lizzi F; Andrisano V; Bartolini M; Hrelia P; Tarozzi A; Tumiatti V; Melchiorre C. | 2007-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Characterization of Cholinesterase inhibitors by means of immobilized enzyme reactor | M. Bartolini; M.L. Bolognesi; A. Cavalli; C. Melchiorre; A. Rampa; M. Recanatini; V. Andrisano | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Strategie farmacologiche per il trattamento della malattia di Alzheimer | M.L. Bolognesi; C. Melchiorre | 2007-01-01 | NEW ENTRIES IN PHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Multi-target-directed drugs for neurodegeneration | C. Melchiorre | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Quinone-bearing polyamines are AChE inhibitors endowed with multifunctional properties | M.L. Bolognesi; R. Banzi; A. Cavalli; A. Minarini; M. Bartolini; V. Andrisano; M. Recanatini; C. ...Melchiorre | 2007-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Multi-Target-Directed Drug Design Strategy: From a Dual Binding Site Acetylcholinesterase Inhibitor to a Trifunctional Compound against Alzheimer's Disease | Bolognesi ML; Cavalli A; Valgimigli L; Bartolini M; Rosini M; Andrisano V; Recanatini M; Melchior...re C | 2007-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A new EGFR inhibitor induces apoptosis in colon cancer cells. | Calonghi N; Pagnotta E; Parolin C; Mangano C; Bolognesi ML; Melchiorre C; Masotti L. | 2007-01-01 | BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS | - | 1.01 Articolo in rivista | - |
Progettazione e sintesi di derivati poliamminici per il trattamento della malattia di Alzheimer | V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; V. Andrisano; M. Bartolini; F. ...Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre | 2007-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
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