Sfoglia per Autore
Benextramine derivatives as probes to target human monoamine oxidases
2015 Maria Luisa Di Paolo; Andrea Milelli; Giorgio Cozza; Monica Rossetto; Michela Rosini; Anna Minarini
Natural polyamines and synthetic analogs modify the growth and the morphology of Pyrus communis pollen tubes affecting ROS levels and causing cell death
2015 Aloisi, I.; Cai, G.; Tumiatti, V.; Minarini, A.; Del Duca, S.
Macrocyclic naphthalene diimides as G-quadruplex binders
2015 Marchetti, C.; Minarini, A.; Tumiatti, V.; Moraca, F.; Parrotta, L.; Alcaro, S.; Rigo, R.; Sissi, C.; Gunaratnam, M.; Ohnmacht, S.A.; Neidle, S.; Milelli, A.
Nature-Inspired Multifunctional Ligands: Focusing on Amyloid-Based Molecular Mechanisms of Alzheimer’s Disease
2016 Simoni, Elena; Serafini, Melania M.; Bartolini, Manuela; Caporaso, Roberta; Pinto, Antonella; Necchi, Daniela; Fiori, Jessica; Vincenza, Andrisano; Minarini, Anna; Lanni, Cristina; Rosini, Michela
Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate.
2016 Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E; Lodola, A; Mor, M; Milelli, A; Minarini, A.
4-AMINO-2-PYRIDO-BICYCLIC PYRIMIDINES AND USE THEREOF AS MEDICAMENTS - 4 AMINO-2-PIRIDO-BICICLO PIRIMIDINE E LORO USO COME MEDICAMENTI
2016 Marco, DE VIVO; Antonio, ORTEGA MARTINEZ JOSE; Manuel, ARENCIBIA JIMENEZ JOSE; Minarini, Anna; Claudia, Sissi
In vivo characterization of ARN14140, a memantine/galantamine-based multi-target compound for Alzheimer's disease
2016 Reggiani, Angelo M.; Simoni, Elena; Caporaso, Roberta; Meunier, Johann; Keller, Emeline; Maurice, Tangui; Minarini, Anna; Rosini, Michela; Cavalli, Andrea
Polyamine Conjugation as a Promising Strategy To Target Amyloid Aggregation in the Framework of Alzheimer’s Disease
2016 Simoni, Elena; Caporaso, Roberta; Bergamini, Christian; Fiori, Jessica; Fato, Romana; Miszta, Przemyslaw; Filipek, Sławomir; Caraci, Filippo; Giuffrida, Maria Laura; Andrisano, Vincenza; Minarini, Anna; Bartolini, Manuela; Rosini, Michela
Multitarget strategies in Alzheimer's disease: benefits and challenges on the road to therapeutics
2016 Rosini, M; Simoni, E; Caporaso, R; Minarini, A
Farmaci che agiscono sul sistema renina-angiotensina
2017 Minarini, Anna
Naphthalene diimide-polyamine hybrids as antiproliferative agents: Focus on the architecture of the polyamine chains
2017 Milelli, Andrea; Marchetti, Chiara; Greco, Maria Laura; Moraca, Federica; Costa, Giosuè; Turrini, Eleonora; Catanzaro, Elena; Betari, Nibal; Calcabrini, Cinzia; Sissi, Claudia; Alcaro, Stefano; Fimognari, Carmela; Tumiatti, Vincenzo; Minarini, Anna
Targeting the Nrf2/Amyloid-Beta Liaison in Alzheimer's Disease: A Rational Approach
2017 Simoni, Elena; Serafini, Melania M; Caporaso, Roberta; Marchetti, Chiara; Racchi, Marco; Minarini, Anna; Bartolini, Manuela; Lanni, Cristina; Rosini, Michela
Quinazoline based α1-adrenoreceptor antagonists with potent antiproliferative activity in human prostate cancer cell lines
2017 Maestri, Valentina; Tarozzi, Andrea; Simoni, Elena; Cilia, Antonio; Poggesi, Elena; Naldi, Marina; Nicolini, Benedetta; Pruccoli, Letizia; Rosini, Michela; Minarini, Anna
Novel xanthone-polyamine conjugates as catalytic inhibitors of human topoisomerase IIα
2017 Minniti, Elirosa; Byl, Jo Ann W.; Riccardi, Laura; Sissi, Claudia; Rosini, Michela; De Vivo, Marco; Minarini, Anna; Osheroff, Neil
Multitarget drug design strategy in Alzheimer's disease: focus on cholinergic transmission and amyloid-beta aggregation
2017 Simoni, Elena; Bartolini, Manuela; Abu, Izuddin F; Blockley, Alix; Gotti, Cecilia; Bottegoni, Giovanni; Caporaso, Roberta; Bergamini, Christian; Andrisano, Vincenza; Cavalli, Andrea; Mellor, Ian R; Minarini, Anna; Rosini, Michela
Novel Polyamine–Naphthalene Diimide Conjugates Targeting Histone Deacetylases and DNA for Cancer Phenotype Reprogramming
2017 Alice, Pasini; Chiara, Marchetti; Claudia, Sissi; Marilisa, Cortesi; Emanuele, Giordano; Anna, Minarini; Andrea, Milelli
Novel targets for “old” polyamine analogues: monoamine oxidases and benextramine derivatives
2018 Maria Luisa Di Paolo, Giorgio Cozza, Andrea Milelli, Francesca Zonta, Stefania Sarno, Elirosa Minniti, Michela Rosini, Anna Minarini
Novel polyamine-based Histone deacetylases-Lysine demethylase 1 dual binding inhibitors
2018 Andrea Milelli, Chiara Marchetti, Eleonora Turrini, Elena Catanzaro, Roberta Mazzone, Daniela Tomaselli, Carmela FImognari, Vincenzo Tumiatti, Anna MInarini
Pharmacophore Hybridization To Discover Novel Topoisomerase II Poisons with Promising Antiproliferative Activity
2018 Ortega, Jose Antonio; Riccardi, Laura; Minniti, Elirosa; Borgogno, Marco; Arencibia, Jose M; Greco, Maria L; Minarini, Anna; Sissi, Claudia; De Vivo, Marco
Polyamine-containing etoposide derivatives as poisons of human type II topoisomerases: Differential effects on topoisomerase IIα and IIβ
2018 Oviatt A.A., Kuriappan J.A., Minniti E., Vann K.R. , Onuorah P. , Minarini A., M. De Vivo, Osheroff N.
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Benextramine derivatives as probes to target human monoamine oxidases | Maria Luisa Di Paolo; Andrea Milelli; Giorgio Cozza; Monica Rossetto; Michela Rosini; Anna Minarini | 2015-01-01 | AMINO ACIDS | - | 1.06 Abstract in rivista | - |
Natural polyamines and synthetic analogs modify the growth and the morphology of Pyrus communis pollen tubes affecting ROS levels and causing cell death | Aloisi, I.; Cai, G.; Tumiatti, V.; Minarini, A.; Del Duca, S. | 2015-01-01 | PLANT SCIENCE | - | 1.01 Articolo in rivista | 83.Plant Science 2015.pdf |
Macrocyclic naphthalene diimides as G-quadruplex binders | Marchetti, C.; Minarini, A.; Tumiatti, V.; Moraca, F.; Parrotta, L.; Alcaro, S.; Rigo, R.; Sissi,... C.; Gunaratnam, M.; Ohnmacht, S.A.; Neidle, S.; Milelli, A. | 2015-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | AM11585-516279.pdf |
Nature-Inspired Multifunctional Ligands: Focusing on Amyloid-Based Molecular Mechanisms of Alzheimer’s Disease | Simoni, Elena; Serafini, Melania M.; Bartolini, Manuela; Caporaso, Roberta; Pinto, Antonella; Nec...chi, Daniela; Fiori, Jessica; Vincenza, Andrisano; Minarini, Anna; Lanni, Cristina; Rosini, Michela | 2016-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | Simoni E. et al..pdf |
Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate. | Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E...; Lodola, A; Mor, M; Milelli, A; Minarini, A. | 2016-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
4-AMINO-2-PYRIDO-BICYCLIC PYRIMIDINES AND USE THEREOF AS MEDICAMENTS - 4 AMINO-2-PIRIDO-BICICLO PIRIMIDINE E LORO USO COME MEDICAMENTI | Marco, DE VIVO; Antonio, ORTEGA MARTINEZ JOSE; Manuel, ARENCIBIA JIMENEZ JOSE; Minarini, Anna; Cl...audia, Sissi | 2016-01-01 | - | - | 6.01 Brevetto | - |
In vivo characterization of ARN14140, a memantine/galantamine-based multi-target compound for Alzheimer's disease | Reggiani, Angelo M.; Simoni, Elena; Caporaso, Roberta; Meunier, Johann; Keller, Emeline; Maurice,... Tangui; Minarini, Anna; Rosini, Michela; Cavalli, Andrea | 2016-01-01 | SCIENTIFIC REPORTS | - | 1.01 Articolo in rivista | 88. Sc.Rep 2016.pdf |
Polyamine Conjugation as a Promising Strategy To Target Amyloid Aggregation in the Framework of Alzheimer’s Disease | Simoni, Elena; Caporaso, Roberta; Bergamini, Christian; Fiori, Jessica; Fato, Romana; Miszta, Prz...emyslaw; Filipek, Sławomir; Caraci, Filippo; Giuffrida, Maria Laura; Andrisano, Vincenza; Minarini, Anna; Bartolini, Manuela; Rosini, Michela | 2016-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
Multitarget strategies in Alzheimer's disease: benefits and challenges on the road to therapeutics | Rosini, M; Simoni, E; Caporaso, R; Minarini, A | 2016-01-01 | FUTURE MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Farmaci che agiscono sul sistema renina-angiotensina | Minarini, Anna | 2017-01-01 | - | Piccin Nuova Libraria | 5.02 Contributo in volume (Traduzione) | - |
Naphthalene diimide-polyamine hybrids as antiproliferative agents: Focus on the architecture of the polyamine chains | Milelli, Andrea; Marchetti, Chiara; Greco, Maria Laura; Moraca, Federica; Costa, Giosuè; Turrini,... Eleonora; Catanzaro, Elena; Betari, Nibal; Calcabrini, Cinzia; Sissi, Claudia; Alcaro, Stefano; Fimognari, Carmela; Tumiatti, Vincenzo; Minarini, Anna | 2017-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Targeting the Nrf2/Amyloid-Beta Liaison in Alzheimer's Disease: A Rational Approach | Simoni, Elena; Serafini, Melania M; Caporaso, Roberta; Marchetti, Chiara; Racchi, Marco; Minarini..., Anna; Bartolini, Manuela; Lanni, Cristina; Rosini, Michela | 2017-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | - |
Quinazoline based α1-adrenoreceptor antagonists with potent antiproliferative activity in human prostate cancer cell lines | Maestri, Valentina; Tarozzi, Andrea; Simoni, Elena; Cilia, Antonio; Poggesi, Elena; Naldi, Marina...; Nicolini, Benedetta; Pruccoli, Letizia; Rosini, Michela; Minarini, Anna | 2017-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Novel xanthone-polyamine conjugates as catalytic inhibitors of human topoisomerase IIα | Minniti, Elirosa; Byl, Jo Ann W.; Riccardi, Laura; Sissi, Claudia; Rosini, Michela; De Vivo, Marc...o; Minarini, Anna; Osheroff, Neil | 2017-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
Multitarget drug design strategy in Alzheimer's disease: focus on cholinergic transmission and amyloid-beta aggregation | Simoni, Elena; Bartolini, Manuela; Abu, Izuddin F; Blockley, Alix; Gotti, Cecilia; Bottegoni, Gio...vanni; Caporaso, Roberta; Bergamini, Christian; Andrisano, Vincenza; Cavalli, Andrea; Mellor, Ian R; Minarini, Anna; Rosini, Michela | 2017-01-01 | FUTURE MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Novel Polyamine–Naphthalene Diimide Conjugates Targeting Histone Deacetylases and DNA for Cancer Phenotype Reprogramming | Alice, Pasini; Chiara, Marchetti; Claudia, Sissi; Marilisa, Cortesi; Emanuele, Giordano; Anna, Mi...narini; Andrea, Milelli | 2017-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | Novel Polyamine–Naphthalene Diimide Conjugates Targeting Histone Deacetylases and DNA for Cancer Phenotype Reprogramming.pdf |
Novel targets for “old” polyamine analogues: monoamine oxidases and benextramine derivatives | Maria Luisa Di Paolo, Giorgio Cozza, Andrea Milelli, Francesca Zonta, Stefania Sarno, Elirosa Min...niti, Michela Rosini, Anna Minarini | 2018-01-01 | - | - | 4.03 Poster | - |
Novel polyamine-based Histone deacetylases-Lysine demethylase 1 dual binding inhibitors | Andrea Milelli, Chiara Marchetti, Eleonora Turrini, Elena Catanzaro, Roberta Mazzone, Daniela Tom...aselli, Carmela FImognari, Vincenzo Tumiatti, Anna MInarini | 2018-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
Pharmacophore Hybridization To Discover Novel Topoisomerase II Poisons with Promising Antiproliferative Activity | Ortega, Jose Antonio; Riccardi, Laura; Minniti, Elirosa; Borgogno, Marco; Arencibia, Jose M; Grec...o, Maria L; Minarini, Anna; Sissi, Claudia; De Vivo, Marco | 2018-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | 96.J.Med.Chem.2018.pdf |
Polyamine-containing etoposide derivatives as poisons of human type II topoisomerases: Differential effects on topoisomerase IIα and IIβ | Oviatt A.A., Kuriappan J.A., Minniti E., Vann K.R. , Onuorah P. , Minarini A., M. De Vivo, Osher...off N. | 2018-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
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