GIOIA, DARIO
GIOIA, DARIO
FABIT - DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Innovative Strategy toward Mutant CFTR Rescue in Cystic Fibrosis: Design and Synthesis of Thiadiazole Inhibitors of the E3 Ligase RNF5
2023 Brusa, Irene; Sondo, Elvira; Pesce, Emanuela; Tomati, Valeria; Gioia, Dario; Falchi, Federico; Balboni, Beatrice; Ortega Martínez, Jose Antonio; Veronesi, Marina; Romeo, Elisa; Margaroli, Natasha; Recanatini, Maurizio; Girotto, Stefania; Pedemonte, Nicoletta; Roberti, Marinella; Cavalli, Andrea
Watching the release of a photopharmacological drug from tubulin using time-resolved serial crystallography
2023 Wranik, Maximilian; Weinert, Tobias; Slavov, Chavdar; Masini, Tiziana; Furrer, Antonia; Gaillard, Natacha; Gioia, Dario; Ferrarotti, Marco; James, Daniel; Glover, Hannah; Carrillo, Melissa; Kekilli, Demet; Stipp, Robin; Skopintsev, Petr; Brünle, Steffen; Mühlethaler, Tobias; Beale, John; Gashi, Dardan; Nass, Karol; Ozerov, Dmitry; Johnson, Philip J. M.; Cirelli, Claudio; Bacellar, Camila; Braun, Markus; Wang, Meitian; Dworkowski, Florian; Milne, Chris; Cavalli, Andrea; Wachtveitl, Josef; Steinmetz, Michel O.; Standfuss, Jörg
Identification of RAD51-BRCA2 inhibitors using N-acylhydrazone-based dynamic combinatorial chemistry
2022 Bagnolini, Greta; Balboni, Beatrice; Schipani, Fabrizio; Gioia, Dario; Veronesi, Marina; De Franco, Francesca; Kaya, Cansu; Jumde, Ravindra P.; Antonio Ortega, Jose; Girotto, Stefania; Hirsch, Anna K. H.; Roberti, Marinella; Cavalli, Andrea
Rational Design of a Novel Tubulin Inhibitor with a Unique Mechanism of Action
2022 Muhlethaler, T.; Milanos, L.; Ortega, J. A.; Blum, T. B.; Gioia, D.; Roy, B.; Prota, A. E.; Cavalli, A.; Steinmetz, M. O.
Comprehensive Analysis of Binding Sites in Tubulin
2021 Muhlethaler T.; Gioia D.; Prota A.E.; Sharpe M.E.; Cavalli A.; Steinmetz M.O.
Dihydroquinoline pyrazoline-based compound as a new RAD51-BRCA2 protein-protein disruptor to trigger synthetic lethality in pancreatic cancer
2020 Bagnolini, Greta; Manerba, Marcella; Balboni, Andrea; Antonio Ortega, Jose; Gioia, Dario; De Franco, Francesca; Roberti, Marinella; Cavalli, Andrea
Synthetic Lethality in Pancreatic Cancer: Discovery of a New RAD51-BRCA2 Small Molecule Disruptor That Inhibits Homologous Recombination and Synergizes with Olaparib
2020 Bagnolini G.; Milano D.; Manerba M.; Schipani F.; Ortega J.A.; Gioia D.; Falchi F.; Balboni A.; Farabegoli F.; De Franco F.; Robertson J.; Pellicciari R.; Pallavicini I.; Peri S.; Minucci S.; Girotto S.; Di Stefano G.; Roberti M.; Cavalli A.
Dynamic Docking: A Paradigm Shift in Computational Drug Discovery
2017 Gioia, Dario; Bertazzo, Martina; Recanatini, Maurizio; Masetti, Matteo; Cavalli, Andrea
Protein Tunnels: The Case of Urease Accessory Proteins
2017 Musiani, Francesco; Gioia, Dario; Masetti, Matteo; Falchi, Federico; Cavalli, Andrea; Recanatini, Maurizio; Ciurli, Stefano