VIOLA, ANGELO
VIOLA, ANGELO
DIPARTIMENTO DI CHIMICA "GIACOMO CIAMICIAN"
A straightforward route to enantiopure 2-substituted-3,4-dehydro-beta-proline via ring closing metathesis
2011 A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; E. Paradisi
Alkylidene malonamides and acetacetamides as intermediates for the preparation of constrained dipeptide mimetics.
2012 A. Tolomelli; L. Gentilucci; A. Viola
An improved microwave assisted protocol for Yonemitsu-type trimolecular condensation
2014 Angelo Viola;Lucia Ferrazzano;Giulia Martelli;Sebastiano Ancona;Luca Gentilucci;Alessandra Tolomelli
An improved protocol for Yonemitsu-type trimolecular condensation
2012 A. Tolomelli; L. Gentilucci; A.Viola
Dehydro-beta-amino acid as building blocks for bioactive compounds
2012 G. Cardillo; L. Gentilucci; E. Mosconi; A. Tolomelli; A. Viola
Dehydro-beta-amino acid containing peptidomimetics as integrin receptor ligands
2012 A. Tolomelli; A. Viola; L. Gentilucci; E. Mosconi; R. De Marco; M. Baiula; S. Spampinato; L. Belvisi; M. Civera
Dehydro-beta-amino acids as scaffolds for the preparation of alpha-v-beta-3, alpha-5-beta-1 and alpha-4-beta-1 integrin ligands
2011 A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; M. Baiula; S. Spampinato; L. Belvisi; M. Civera
Dehydro-beta-proline Containing Alpha-4-beta-1 Integrin Antagonists: Stereochemical Recognition in Ligand-Receptor Interplay
2015 Tolomelli, Alessandra; Baiula, Monica; Viola, Angelo; Ferrazzano, Lucia; Gentilucci, Luca; Dattoli, Samantha Deianira; Spampinato, Santi; Juaristi, Eusebio; Escudero, Margarita
Design and synthesis of Alpha-v-beta-3 and Alpha-5-beta-1 integrin ligands as delivery systems for fluorescent molecules
2014 Tolomelli, Alessandra; Gentilucci, Luca; Viola, Angelo; Dattoli, Samantha Deianira; Baiula, Monica; Spampinato, Santi; Petkau-Milroy, Katja; Brunsveld, Luc
Design and synthesis of integrin ligands as «molecular shuttles» for drugs and fluorescent molecules delivery
2015 Ferrazzano, L.; Viola, A.; Tolomelli, A.
Design and synthesis of integrin ligands as «molecular shuttles» for drugs and fluorescent molecules delivery
2015 Ferrazzano, L.; Viola, A.; Tolomelli, A.
Design and Synthesis of Integrin Ligands αvβ3 and α5β1 as delivery systems for fluorescent molecules
2014 L. Ferrazzano; A. Tolomelli; A. Viola
Design, synthesis and in vitro evaluation of tumor homing agents by conjugation of integrin ligands to diagnostics and cytotoxic drugs
2014 A. Tolomelli; L. Gentilucci; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Belvisi; M.Civera
Development of isoxazoline-containing peptidomimetics as dual alpha-v-beta-3 and alpha-5-beta-1 integrin ligands.
2011 A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Belvisi; M. Civera
Exploring the reactivity of alkylidene malonamides: synthesis of polyfunctionalized isoxazolidinones, aziridines and oxazolines
2012 A. Tolomelli; G. Cardillo; L. Gentilucci; R. Juris; A. Viola; E. Juaristi
Modulation of αvβ3- and α5β1-integrin-mediated adhesion by dehydro-β-amino acids containing peptidomimetics
2013 TOLOMELLI A.; BAIULA M.; BELVISI L.; VIOLA A.; GENTILUCCI L.; TROISI S.; DATTOLI S. D.; SPAMPINATO S.; CIVERA M.; JUARISTI E.; ESCUDERO M.
New isoxazolidinone and 3,4-dehydro-β-proline derivatives as antibacterial agents and MAO-inhibitors: A complex balance between two activities
2016 Ferrazzano, Lucia; Viola, Angelo; Lonati, Elena; Bulbarelli, Alessandra; Musumeci, Rosario; Cocuzza, Clementina; Lombardo, Marco; Tolomelli, Alessandra
NEW PEPTIDOMIMETIC α4β1-INTEGRIN ANTAGONISTS FOR REDUCING INFLAMMATION AND ALLERGIC REACTIONS
2012 A. Greco; R. De Marco; A. Tolomelli; A. Viola; S. Spampinato; M. Baiula; S. Dattoli; L. Gentilucci
Novel tools against antibiotic resistance: design and synthesis of Linezolid analogues
2014 L. Ferrazzano; A. Tolomelli; A. Viola
One-Pot Two-Step Microwave-Assisted Synthesis of Alkylidene Acetoacetamido Esters, Useful Intermediates for β-Dehydropeptides
2016 Viola, Angelo; Ferrazzano, Lucia; Greco, Roberto; Cerisoli, Lucia; Caldi, Jonathan; Tolomelli, Alessandra
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
A straightforward route to enantiopure 2-substituted-3,4-dehydro-beta-proline via ring closing metathesis | A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; E. Paradisi | 2011-01-01 | AMINO ACIDS | - | 1.01 Articolo in rivista | - |
Alkylidene malonamides and acetacetamides as intermediates for the preparation of constrained dipeptide mimetics. | A. Tolomelli; L. Gentilucci; A. Viola | 2012-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
An improved microwave assisted protocol for Yonemitsu-type trimolecular condensation | Angelo Viola;Lucia Ferrazzano;Giulia Martelli;Sebastiano Ancona;Luca Gentilucci;Alessandra Tolomelli | 2014-01-01 | TETRAHEDRON | - | 1.01 Articolo in rivista | - |
An improved protocol for Yonemitsu-type trimolecular condensation | A. Tolomelli; L. Gentilucci; A.Viola | 2012-01-01 | - | Società Chimica Italiana | 4.02 Riassunto (Abstract) | - |
Dehydro-beta-amino acid as building blocks for bioactive compounds | G. Cardillo; L. Gentilucci; E. Mosconi; A. Tolomelli; A. Viola | 2012-01-01 | - | cietà Chimica Itlaiana -Divisione Chimica farmaceutica | 4.02 Riassunto (Abstract) | - |
Dehydro-beta-amino acid containing peptidomimetics as integrin receptor ligands | A. Tolomelli; A. Viola; L. Gentilucci; E. Mosconi; R. De Marco; M. Baiula; S. Spampinato; L. Belv...isi; M. Civera | 2012-01-01 | - | Europan Assciation for Chemical and Molecular Sciences | 4.02 Riassunto (Abstract) | - |
Dehydro-beta-amino acids as scaffolds for the preparation of alpha-v-beta-3, alpha-5-beta-1 and alpha-4-beta-1 integrin ligands | A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; M. Baiula; S. Spampinato; L. Belvisi; M. Civera | 2011-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Dehydro-beta-proline Containing Alpha-4-beta-1 Integrin Antagonists: Stereochemical Recognition in Ligand-Receptor Interplay | Tolomelli, Alessandra; Baiula, Monica; Viola, Angelo; Ferrazzano, Lucia; Gentilucci, Luca; Dattol...i, Samantha Deianira; Spampinato, Santi; Juaristi, Eusebio; Escudero, Margarita | 2015-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | accepmanus 519198.pdf |
Design and synthesis of Alpha-v-beta-3 and Alpha-5-beta-1 integrin ligands as delivery systems for fluorescent molecules | Tolomelli, Alessandra; Gentilucci, Luca; Viola, Angelo; Dattoli, Samantha Deianira; Baiula, Monic...a; Spampinato, Santi; Petkau-Milroy, Katja; Brunsveld, Luc | 2014-01-01 | LA CHIMICA E L'INDUSTRIA | - | 1.01 Articolo in rivista | - |
Design and synthesis of integrin ligands as «molecular shuttles» for drugs and fluorescent molecules delivery | Ferrazzano, L.; Viola, A.; Tolomelli, A. | 2015-01-01 | - | // | 4.02 Riassunto (Abstract) | - |
Design and synthesis of integrin ligands as «molecular shuttles» for drugs and fluorescent molecules delivery | Ferrazzano, L.; Viola, A.; Tolomelli, A. | 2015-01-01 | - | SCI | 4.02 Riassunto (Abstract) | - |
Design and Synthesis of Integrin Ligands αvβ3 and α5β1 as delivery systems for fluorescent molecules | L. Ferrazzano; A. Tolomelli; A. Viola | 2014-01-01 | - | European Association of Chemical and Molecular Sciences | 4.02 Riassunto (Abstract) | - |
Design, synthesis and in vitro evaluation of tumor homing agents by conjugation of integrin ligands to diagnostics and cytotoxic drugs | A. Tolomelli; L. Gentilucci; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Belvisi; M.Civera | 2014-01-01 | - | Elsevier | 4.02 Riassunto (Abstract) | - |
Development of isoxazoline-containing peptidomimetics as dual alpha-v-beta-3 and alpha-5-beta-1 integrin ligands. | A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Be...lvisi; M. Civera | 2011-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
Exploring the reactivity of alkylidene malonamides: synthesis of polyfunctionalized isoxazolidinones, aziridines and oxazolines | A. Tolomelli; G. Cardillo; L. Gentilucci; R. Juris; A. Viola; E. Juaristi | 2012-01-01 | ARKIVOC | - | 1.01 Articolo in rivista | - |
Modulation of αvβ3- and α5β1-integrin-mediated adhesion by dehydro-β-amino acids containing peptidomimetics | TOLOMELLI A.; BAIULA M.; BELVISI L.; VIOLA A.; GENTILUCCI L.; TROISI S.; DATTOLI S. D.; SPAMPINAT...O S.; CIVERA M.; JUARISTI E.; ESCUDERO M. | 2013-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
New isoxazolidinone and 3,4-dehydro-β-proline derivatives as antibacterial agents and MAO-inhibitors: A complex balance between two activities | Ferrazzano, Lucia; Viola, Angelo; Lonati, Elena; Bulbarelli, Alessandra; Musumeci, Rosario; Cocuz...za, Clementina; Lombardo, Marco; Tolomelli, Alessandra | 2016-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
NEW PEPTIDOMIMETIC α4β1-INTEGRIN ANTAGONISTS FOR REDUCING INFLAMMATION AND ALLERGIC REACTIONS | A. Greco; R. De Marco; A. Tolomelli; A. Viola; S. Spampinato; M. Baiula; S. Dattoli; L. Gentilucci | 2012-01-01 | - | SCI | 4.01 Contributo in Atti di convegno | - |
Novel tools against antibiotic resistance: design and synthesis of Linezolid analogues | L. Ferrazzano; A. Tolomelli; A. Viola | 2014-01-01 | - | European Association for Chemical and Molecular Sciences | 4.02 Riassunto (Abstract) | - |
One-Pot Two-Step Microwave-Assisted Synthesis of Alkylidene Acetoacetamido Esters, Useful Intermediates for β-Dehydropeptides | Viola, Angelo; Ferrazzano, Lucia; Greco, Roberto; Cerisoli, Lucia; Caldi, Jonathan; Tolomelli, Al...essandra | 2016-01-01 | EUROPEAN JOURNAL OF ORGANIC CHEMISTRY | - | 1.01 Articolo in rivista | - |