Sfoglia per Autore
Dehydro-beta-amino acids as scaffolds for the preparation of alpha-v-beta-3, alpha-5-beta-1 and alpha-4-beta-1 integrin ligands
2011 A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; M. Baiula; S. Spampinato; L. Belvisi; M. Civera
Eosinophil as a cellular target of the ocular anti-allergic action of mapracorat, a novel selective glucocorticoid receptor agonist
2011 Baiula M; Spartà A; Bedini A; Carbonari G; Bucolo C; Ward KW; Zhang JZ; Govoni P; Spampinato S
Development of isoxazoline-containing peptidomimetics as dual alpha-v-beta-3 and alpha-5-beta-1 integrin ligands.
2011 A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Belvisi; M. Civera
TNF-alpha-induced MOR up-regulation in human glioblastoma cells is coupled to a loss of MOR-activated signalling to intracellular effectors
2012 Bedini A; Vincelli G; Baiula M; Spampinato S
Dehydro-beta-amino acid containing peptidomimetics as integrin receptor ligands
2012 A. Tolomelli; A. Viola; L. Gentilucci; E. Mosconi; R. De Marco; M. Baiula; S. Spampinato; L. Belvisi; M. Civera
Pro-inflammatory stimuli increase mu-opioid receptor (MOR) number on cell surface of human glioblastoma cells but hamper opioid agonist-induced intracellular signaling. G-protein-coupled-receptors: from structural insights to functional mechanisms
2012 Bedini A; Vincelli G; Baiula M; Spampinato S
Peptidomimetic probes for modulating α4β1 integrin activity
2012 A. Greco; R. De Marco; A. Tolomelli; S. Spampinato; M. Baiula; S. Dattoli
NEW PEPTIDOMIMETIC α4β1-INTEGRIN ANTAGONISTS FOR REDUCING INFLAMMATION AND ALLERGIC REACTIONS
2012 A. Greco; R. De Marco; A. Tolomelli; A. Viola; S. Spampinato; M. Baiula; S. Dattoli; L. Gentilucci
Therapeutic Targeting of Eosinophil Adhesion and Accumulation in Allergic Conjunctivitis
2012 Baiula M; Bedini A; Carbonari G; Dattoli SD; Spampinato S
Molecular Mechanisms Mediating Nociceptin/Orphanin FQ Receptor Signaling, Desensitization and Internalization.
2012 Baiula M; Bedini A; Carbonari G.
REST is up-regulated by epidermal growth factor in HeLa cells and inhibits apoptosis by influencing histone H3 acetylation
2012 Baiula M; Carbonari G; Dattoli SD; Calienni M; Bedini A; Spampinato S.
Functional cross-talk between TLR4 and NOPr in human glial cells.
2013 Baiula M; Bedini A; Baldi J; Caprini M; Spampinato S
Ocular anti-allergic action of mapracorat, a novel selective glucocorticoid receptor agonist, involves eosinophil's apoptosis.
2013 Baiula M; Bedini A; Carbonari G; Dattoli SD; Govoni P; Cavet ME; Spampinato S
Prodynorphin-derived peptides
2013 S. Spampinato; A. Bedini; M. Baiula
Modulation of αvβ3- and α5β1-integrin-mediated adhesion by dehydro-β-amino acids containing peptidomimetics
2013 TOLOMELLI A.; BAIULA M.; BELVISI L.; VIOLA A.; GENTILUCCI L.; TROISI S.; DATTOLI S. D.; SPAMPINATO S.; CIVERA M.; JUARISTI E.; ESCUDERO M.
Inhibition of Toll-like Receptor 4 (TLR4)-induced NF-kB activation by NOP is lost in human glioblastoma cells chronically exposed to LPS.
2013 Bedini A; Baiula M; Vincelli G; Spampinato S
Design, synthesis and in vitro evaluation of tumor homing agents by conjugation of integrin ligands to diagnostics and cytotoxic drugs
2014 A. Tolomelli; L. Gentilucci; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Belvisi; M.Civera
Design and synthesis of Alpha-v-beta-3 and Alpha-5-beta-1 integrin ligands as delivery systems for fluorescent molecules
2014 Tolomelli, Alessandra; Gentilucci, Luca; Viola, Angelo; Dattoli, Samantha Deianira; Baiula, Monica; Spampinato, Santi; Petkau-Milroy, Katja; Brunsveld, Luc
Mapracorat, a selective glucocorticoid receptor agonist, causes apoptosis of eosinophils infiltrating the conjunctiva in late phase experimental ocular allergy
2014 Baiula M; Bedini A; Baldi J; Govoni P; Spampinato S
Synthesis and assay of retro-α4β1 integrin-targeting motifs
2014 S. D. Dattoli ; R. De Marco; M. Baiula; S. Spampinato; A. Greco; A. Tolomelli; L. Gentilucci
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Dehydro-beta-amino acids as scaffolds for the preparation of alpha-v-beta-3, alpha-5-beta-1 and alpha-4-beta-1 integrin ligands | A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; M. Baiula; S. Spampinato; L. Belvisi; M. Civera | 2011-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Eosinophil as a cellular target of the ocular anti-allergic action of mapracorat, a novel selective glucocorticoid receptor agonist | Baiula M; Spartà A; Bedini A; Carbonari G; Bucolo C; Ward KW; Zhang JZ; Govoni P; Spampinato S | 2011-01-01 | MOLECULAR VISION | - | 1.01 Articolo in rivista | - |
Development of isoxazoline-containing peptidomimetics as dual alpha-v-beta-3 and alpha-5-beta-1 integrin ligands. | A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Be...lvisi; M. Civera | 2011-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
TNF-alpha-induced MOR up-regulation in human glioblastoma cells is coupled to a loss of MOR-activated signalling to intracellular effectors | Bedini A; Vincelli G; Baiula M; Spampinato S | 2012-01-01 | - | - | 4.03 Poster | - |
Dehydro-beta-amino acid containing peptidomimetics as integrin receptor ligands | A. Tolomelli; A. Viola; L. Gentilucci; E. Mosconi; R. De Marco; M. Baiula; S. Spampinato; L. Belv...isi; M. Civera | 2012-01-01 | - | Europan Assciation for Chemical and Molecular Sciences | 4.02 Riassunto (Abstract) | - |
Pro-inflammatory stimuli increase mu-opioid receptor (MOR) number on cell surface of human glioblastoma cells but hamper opioid agonist-induced intracellular signaling. G-protein-coupled-receptors: from structural insights to functional mechanisms | Bedini A; Vincelli G; Baiula M; Spampinato S | 2012-01-01 | - | - | 4.03 Poster | - |
Peptidomimetic probes for modulating α4β1 integrin activity | A. Greco; R. De Marco; A. Tolomelli; S. Spampinato; M. Baiula; S. Dattoli | 2012-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
NEW PEPTIDOMIMETIC α4β1-INTEGRIN ANTAGONISTS FOR REDUCING INFLAMMATION AND ALLERGIC REACTIONS | A. Greco; R. De Marco; A. Tolomelli; A. Viola; S. Spampinato; M. Baiula; S. Dattoli; L. Gentilucci | 2012-01-01 | - | SCI | 4.01 Contributo in Atti di convegno | - |
Therapeutic Targeting of Eosinophil Adhesion and Accumulation in Allergic Conjunctivitis | Baiula M; Bedini A; Carbonari G; Dattoli SD; Spampinato S | 2012-01-01 | FRONTIERS IN PHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Molecular Mechanisms Mediating Nociceptin/Orphanin FQ Receptor Signaling, Desensitization and Internalization. | Baiula M; Bedini A; Carbonari G. | 2012-01-01 | CURRENT MOLECULAR PHARMACOLOGY | - | 1.01 Articolo in rivista | - |
REST is up-regulated by epidermal growth factor in HeLa cells and inhibits apoptosis by influencing histone H3 acetylation | Baiula M; Carbonari G; Dattoli SD; Calienni M; Bedini A; Spampinato S. | 2012-01-01 | BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR CELL RESEARCH | - | 1.01 Articolo in rivista | - |
Functional cross-talk between TLR4 and NOPr in human glial cells. | Baiula M; Bedini A; Baldi J; Caprini M; Spampinato S | 2013-01-01 | - | - | 4.03 Poster | - |
Ocular anti-allergic action of mapracorat, a novel selective glucocorticoid receptor agonist, involves eosinophil's apoptosis. | Baiula M; Bedini A; Carbonari G; Dattoli SD; Govoni P; Cavet ME; Spampinato S | 2013-01-01 | - | - | 4.03 Poster | - |
Prodynorphin-derived peptides | S. Spampinato; A. Bedini; M. Baiula | 2013-01-01 | - | Academic Press | 2.01 Capitolo / saggio in libro | - |
Modulation of αvβ3- and α5β1-integrin-mediated adhesion by dehydro-β-amino acids containing peptidomimetics | TOLOMELLI A.; BAIULA M.; BELVISI L.; VIOLA A.; GENTILUCCI L.; TROISI S.; DATTOLI S. D.; SPAMPINAT...O S.; CIVERA M.; JUARISTI E.; ESCUDERO M. | 2013-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Inhibition of Toll-like Receptor 4 (TLR4)-induced NF-kB activation by NOP is lost in human glioblastoma cells chronically exposed to LPS. | Bedini A; Baiula M; Vincelli G; Spampinato S | 2013-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
Design, synthesis and in vitro evaluation of tumor homing agents by conjugation of integrin ligands to diagnostics and cytotoxic drugs | A. Tolomelli; L. Gentilucci; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Belvisi; M.Civera | 2014-01-01 | - | Elsevier | 4.02 Riassunto (Abstract) | - |
Design and synthesis of Alpha-v-beta-3 and Alpha-5-beta-1 integrin ligands as delivery systems for fluorescent molecules | Tolomelli, Alessandra; Gentilucci, Luca; Viola, Angelo; Dattoli, Samantha Deianira; Baiula, Monic...a; Spampinato, Santi; Petkau-Milroy, Katja; Brunsveld, Luc | 2014-01-01 | LA CHIMICA E L'INDUSTRIA | - | 1.01 Articolo in rivista | - |
Mapracorat, a selective glucocorticoid receptor agonist, causes apoptosis of eosinophils infiltrating the conjunctiva in late phase experimental ocular allergy | Baiula M; Bedini A; Baldi J; Govoni P; Spampinato S | 2014-01-01 | DRUG DESIGN, DEVELOPMENT AND THERAPY | - | 1.01 Articolo in rivista | - |
Synthesis and assay of retro-α4β1 integrin-targeting motifs | S. D. Dattoli ; R. De Marco; M. Baiula; S. Spampinato; A. Greco; A. Tolomelli; L. Gentilucci | 2014-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
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