Sfoglia per Autore
Location of the Polyamine Binding Site in the Vestibule of the Nicotinic Acetylcholine Receptor Ion Channel
2001 Bixel M.G.; Weise C.; Bolognesi M.L.; Rosini M.; Brierly M.J.; Mellor I.R.; Usherwood P.N.R.; Melchiorre C.; Hucho F.
Binding of polyamine-containing toxins in the vestibule of the nicotinic acetylcholine receptor ion channel
2001 Bixel M.Gabriele; Krauss M.; Weise C.; Bolognesi M.L.; Rosini M.; Usherwood P.N.R.; Melchiorre C.; Hucho F.
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure
2002 Bolognesi M.L.; Bixel M.G.; Marucci G.; Bartolini M.; Krauss M.; Angeli P.; Antonello A.; Rosini M.; Tumiatti V.; Hucho F.; Melchiorre C.
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 2. Role of polymethylene chain lengths separating amine functions and of substituents on the terminal nitrogen atoms
2002 Rosini M.; Bixel M.G.; Marucci G.; Budriesi R.; Krauss M.; Bolognesi M.L.; Minarini A.; Tumiatti V.; Hucho F.; Melchiorre C.
Polymethylene tetraamine backbone as template for the development of biologically active polyamines
2003 Melchiorre C.; Antonello A.; Banzi R.; Bolognesi M.L.; Minarini A.; Rosini M.; Tumiatti V.
Memoquin: a new compound to attack Alzheimer's disease drug discovery
2004 Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Capsoni S.; Cattaneo A.
Memoquin: a new therapeutic poly-agent for Alzheimer's disease
2004 Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Margotti E.; Capsoni S.; Cattaneo A.
Progettazione e sintesi di analoghi rigidi di metoctramina nello studio dei recettori muscarinici
2004 Tumiatti V.; Bolognesi M.L.; Minarini A.; Rosini M.; Angeli A.; Buccioni M.; Marucci G.; Melchiorre C.
MEMOQUIN: A MULTIPOTENT ACETYLCHOLINESTERASE INHIBITOR WITH EXCELLENT IN VIVO ACTIVITY
2004 A.Cavalli; ML Bolognesi; M.Bartolini; V.Andrisano; C.Melchiorre; M.Recanatini; S.Capsoni; A.Cattaneo
Polyamines may modulate both G protein-coupled receptors and G proteins
2004 MARUCCI G.; NOVI F.; BANZI R.; BOLOGNESI M. L.; BUCCIONI M.; MINARINI A.; ROSINI M.; ANGELI P.; MAGGIO R.; MELCHIORRE C.
Design, synthesis, and biological evaluation of conformationally restricted rivastigmine analogues
2004 Bolognesi M. L.; Bartolini M.; Cavalli A.; Andrisano V.; Rosini M.; Minarini A.; Melchiorre C.
Methoctramine analogues inhibit responses to capsaicin in DRG neurons and cloned TRPV1
2005 Minarini A.; Mellor I.; Bolognesi M.L.; Ogilvie J.; Rosini M.; Tumiatti V.; Melchiorre C.
Methoctramine-related polyamines as antinociceptive agents
2005 Tumiatti V.; Minarini A.; Rosini M.; Bolognesi M.L.; Marucci G.; Buccioni M.; Ghelardini C.; Melchiorre C.
Memoquin: an up-date on preclinical studies
2005 Capsoni S.; Cavalli A.; Andrisano V.; Bolognesi M. L.; Recanatini M.; Melchiorre C.; Margotti E.; Cattaneo A.
Rational approach to discover multipotent anti-Alzheimer drugs
2005 Bolognesi M.L.; Cavalli A.; Andrisano V.; Banzi R.; Bartolini M.; Capsoni S.; Cattaneo A.; Minarini A.; Recanatini M.; Melchiorre C.
Bivalent tacrine-based acetylcholinesterase inhibitors: role of the spacer in the recognition process of the enzyme gorge
2005 Bolognesi M.L.; Bartolini M.; Cavalli A.; Rosini M.; Andrisano V.; Melchiorre C.
Lipocrine, a multipotent drug for the investigation of Alzheimer's disease
2005 Rosini M.; Andrisano V.; Bartolini M.; Bolognesi M.L.; Hrelia P.; Minarini A.; Tarozzi A.; Melchiorre C.
Heterocyclic inhibitors of AChE acylation and peripheral sites.
2005 Bolognesi M. L.; Andrisano V.; Bartolini M.; Cavalli A.; Minarini A.; Recanatini M.; Rosini M.; Tumiatti V.; Melchiorre C.
HPLC screening of a chemical library for Alzheimer's disease drug discovery
2005 Bartolini M.; Bolognesi M.L.; Cavrini V.; Melchiorre C.; Andrisano V.
Discovery of multipotent drugs for the teratment of Alzheimer's disease
2005 Rosini M.; Andrisano V.; Bartolini M.; Bolognesi M.L.; Cavalli A.; Minarini A.; Recanatini M.; Tumiatti V.; Melchiorre C.
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Location of the Polyamine Binding Site in the Vestibule of the Nicotinic Acetylcholine Receptor Ion Channel | Bixel M.G.; Weise C.; Bolognesi M.L.; Rosini M.; Brierly M.J.; Mellor I.R.; Usherwood P.N.R.; Mel...chiorre C.; Hucho F. | 2001-01-01 | THE JOURNAL OF BIOLOGICAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Binding of polyamine-containing toxins in the vestibule of the nicotinic acetylcholine receptor ion channel | Bixel M.Gabriele; Krauss M.; Weise C.; Bolognesi M.L.; Rosini M.; Usherwood P.N.R.; Melchiorre C....; Hucho F. | 2001-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure | Bolognesi M.L.; Bixel M.G.; Marucci G.; Bartolini M.; Krauss M.; Angeli P.; Antonello A.; Rosini ...M.; Tumiatti V.; Hucho F.; Melchiorre C. | 2002-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 2. Role of polymethylene chain lengths separating amine functions and of substituents on the terminal nitrogen atoms | Rosini M.; Bixel M.G.; Marucci G.; Budriesi R.; Krauss M.; Bolognesi M.L.; Minarini A.; Tumiatti ...V.; Hucho F.; Melchiorre C. | 2002-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Polymethylene tetraamine backbone as template for the development of biologically active polyamines | Melchiorre C.; Antonello A.; Banzi R.; Bolognesi M.L.; Minarini A.; Rosini M.; Tumiatti V. | 2003-01-01 | MEDICINAL RESEARCH REVIEWS | - | 1.01 Articolo in rivista | - |
Memoquin: a new compound to attack Alzheimer's disease drug discovery | Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Capsoni S.;... Cattaneo A. | 2004-01-01 | - | s.l. | 4.02 Riassunto (Abstract) | - |
Memoquin: a new therapeutic poly-agent for Alzheimer's disease | Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Margotti E....; Capsoni S.; Cattaneo A. | 2004-01-01 | NEUROBIOLOGY OF AGING | - | 4.02 Riassunto (Abstract) | - |
Progettazione e sintesi di analoghi rigidi di metoctramina nello studio dei recettori muscarinici | Tumiatti V.; Bolognesi M.L.; Minarini A.; Rosini M.; Angeli A.; Buccioni M.; Marucci G.; Melchior...re C. | 2004-01-01 | - | Grafiche Caroti | 4.02 Riassunto (Abstract) | - |
MEMOQUIN: A MULTIPOTENT ACETYLCHOLINESTERASE INHIBITOR WITH EXCELLENT IN VIVO ACTIVITY | A.Cavalli; ML Bolognesi; M.Bartolini; V.Andrisano; C.Melchiorre; M.Recanatini; S.Capsoni; A.Cattaneo | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Polyamines may modulate both G protein-coupled receptors and G proteins | MARUCCI G.; NOVI F.; BANZI R.; BOLOGNESI M. L.; BUCCIONI M.; MINARINI A.; ROSINI M.; ANGELI P.; M...AGGIO R.; MELCHIORRE C. | 2004-01-01 | MEDICINAL CHEMISTRY RESEARCH | - | 1.01 Articolo in rivista | - |
Design, synthesis, and biological evaluation of conformationally restricted rivastigmine analogues | Bolognesi M. L.; Bartolini M.; Cavalli A.; Andrisano V.; Rosini M.; Minarini A.; Melchiorre C. | 2004-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Methoctramine analogues inhibit responses to capsaicin in DRG neurons and cloned TRPV1 | Minarini A.; Mellor I.; Bolognesi M.L.; Ogilvie J.; Rosini M.; Tumiatti V.; Melchiorre C. | 2005-01-01 | - | s.l. | 4.02 Riassunto (Abstract) | - |
Methoctramine-related polyamines as antinociceptive agents | Tumiatti V.; Minarini A.; Rosini M.; Bolognesi M.L.; Marucci G.; Buccioni M.; Ghelardini C.; Melc...hiorre C. | 2005-01-01 | - | Università di Modena e Reggio Emilia | 4.02 Riassunto (Abstract) | - |
Memoquin: an up-date on preclinical studies | Capsoni S.; Cavalli A.; Andrisano V.; Bolognesi M. L.; Recanatini M.; Melchiorre C.; Margotti E.;... Cattaneo A. | 2005-01-01 | - | Medimond S.r.l. - Monduzzi Editore | 4.02 Riassunto (Abstract) | - |
Rational approach to discover multipotent anti-Alzheimer drugs | Bolognesi M.L.; Cavalli A.; Andrisano V.; Banzi R.; Bartolini M.; Capsoni S.; Cattaneo A.; Minari...ni A.; Recanatini M.; Melchiorre C. | 2005-01-01 | - | s.l. | 4.02 Riassunto (Abstract) | - |
Bivalent tacrine-based acetylcholinesterase inhibitors: role of the spacer in the recognition process of the enzyme gorge | Bolognesi M.L.; Bartolini M.; Cavalli A.; Rosini M.; Andrisano V.; Melchiorre C. | 2005-01-01 | - | s.l. | 4.02 Riassunto (Abstract) | - |
Lipocrine, a multipotent drug for the investigation of Alzheimer's disease | Rosini M.; Andrisano V.; Bartolini M.; Bolognesi M.L.; Hrelia P.; Minarini A.; Tarozzi A.; Melchi...orre C. | 2005-01-01 | - | s.l. | 4.02 Riassunto (Abstract) | - |
Heterocyclic inhibitors of AChE acylation and peripheral sites. | Bolognesi M. L.; Andrisano V.; Bartolini M.; Cavalli A.; Minarini A.; Recanatini M.; Rosini M.; T...umiatti V.; Melchiorre C. | 2005-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |
HPLC screening of a chemical library for Alzheimer's disease drug discovery | Bartolini M.; Bolognesi M.L.; Cavrini V.; Melchiorre C.; Andrisano V. | 2005-01-01 | - | s.l. | 4.02 Riassunto (Abstract) | - |
Discovery of multipotent drugs for the teratment of Alzheimer's disease | Rosini M.; Andrisano V.; Bartolini M.; Bolognesi M.L.; Cavalli A.; Minarini A.; Recanatini M.; Tu...miatti V.; Melchiorre C. | 2005-01-01 | SCIENTIA PHARMACEUTICA | - | 4.02 Riassunto (Abstract) | - |
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