Sfoglia per Autore
Prejunctional muscarinic inhibitory control of acetylcholine release in the human isolated detrusor: Involvement of the M4 receptor subtype
2000 D'Agostino G.; Bolognesi M.L.; Lucchelli A.; Vicini D.; Balestra B.; Spelta V.; Melchiorre C.; Tonini M.
Structure-activity relationship and site of binding of polyamine derivatives at the nicotinic acetylcholine receptor
2000 Bixel M.G.; Krauss M.; Liu Y.; Bolognesi M.L.; Rosini M.; Mellor I.S.; Usherwood P.N.R.; Melchiorre C.; Koji N.; Hucho F.
Analogues of prazosin that bear a benextramine-related polyamine backbone exhibit different antagonism toward α1-adrenoreceptor subtypes
2001 Bolognesi M.L.; Marucci G.; Angeli P.; Buccioni M.; Minarini A.; Rosini M.; Tumiatti V.; Melchiorre C.
Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines
2001 Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Spampinato S.; Tumiatti V.; Melchiorre C.
Binding of polyamine-containing toxins in the vestibule of the nicotinic acetylcholine receptor ion channel
2001 Bixel M.Gabriele; Krauss M.; Weise C.; Bolognesi M.L.; Rosini M.; Usherwood P.N.R.; Melchiorre C.; Hucho F.
Location of the Polyamine Binding Site in the Vestibule of the Nicotinic Acetylcholine Receptor Ion Channel
2001 Bixel M.G.; Weise C.; Bolognesi M.L.; Rosini M.; Brierly M.J.; Mellor I.R.; Usherwood P.N.R.; Melchiorre C.; Hucho F.
Analogues of polyamine alkaloids and their synthetic advantages
2001 Li Y.; Popaj K.; Lochner M.; Geneste H.; Budriesi R.; Chiarini A.; Melchiorre C.; Hesse M.
Design, synthesis, and biological activity of methoctramine-related polyamines as putative Gi protein activators
2001 Melchiorre C.; Bolognesi M.L.; Budriesi R.; Ghelardini C.; Chiarini A.; Minarini A.; Rosini M.; Tumiatti V.; Wade E.J.
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure
2002 Bolognesi M.L.; Bixel M.G.; Marucci G.; Bartolini M.; Krauss M.; Angeli P.; Antonello A.; Rosini M.; Tumiatti V.; Hucho F.; Melchiorre C.
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 2. Role of polymethylene chain lengths separating amine functions and of substituents on the terminal nitrogen atoms
2002 Rosini M.; Bixel M.G.; Marucci G.; Budriesi R.; Krauss M.; Bolognesi M.L.; Minarini A.; Tumiatti V.; Hucho F.; Melchiorre C.
Polymethylene tetraamine backbone as template for the development of biologically active polyamines
2003 Melchiorre C.; Antonello A.; Banzi R.; Bolognesi M.L.; Minarini A.; Rosini M.; Tumiatti V.
Memoquin: a new compound to attack Alzheimer's disease drug discovery
2004 Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Capsoni S.; Cattaneo A.
Studio della configurazione dell'antagonista alfa 1B-adrenergico (+)-cyclazosin
2004 Sagratini G.; Grelli M.; Gulini U.; Melchiorre C.; Antolini L.; Giardinà D.
Absolute configuration of alpha 1B-adrenoceptor antagonist (+)-cyclazosin
2004 Giardinà D.; Sagratini G.; Grelli M.; Gulini U.; Melchiorre C.; Antolini L.
Memoquin: a new therapeutic poly-agent for Alzheimer's disease
2004 Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Margotti E.; Capsoni S.; Cattaneo A.
Studio farmacologico del (+)-cyclazosin, un antagonista selettivo del recettore alfa 1B-adrenergico
2004 Marucci G.; Sagratini G.; Angeli P.; Buccioni M.; Gulini U.; Melchiorre C.; Testa R.; Giardinà D.
Progettazione e sintesi di analoghi rigidi di metoctramina nello studio dei recettori muscarinici
2004 Tumiatti V.; Bolognesi M.L.; Minarini A.; Rosini M.; Angeli A.; Buccioni M.; Marucci G.; Melchiorre C.
MEMOQUIN: A MULTIPOTENT ACETYLCHOLINESTERASE INHIBITOR WITH EXCELLENT IN VIVO ACTIVITY
2004 A.Cavalli; ML Bolognesi; M.Bartolini; V.Andrisano; C.Melchiorre; M.Recanatini; S.Capsoni; A.Cattaneo
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 3. Effect of replacing the inner polymethylene chain with cyclic moieties
2004 TUMIATTI V.; ANDRISANO V.; BANZI R.; BARTOLINI M.; MINARINI A.; ROSINI M.; MELCHIORRE C.
Polyamines may modulate both G protein-coupled receptors and G proteins
2004 MARUCCI G.; NOVI F.; BANZI R.; BOLOGNESI M. L.; BUCCIONI M.; MINARINI A.; ROSINI M.; ANGELI P.; MAGGIO R.; MELCHIORRE C.
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Prejunctional muscarinic inhibitory control of acetylcholine release in the human isolated detrusor: Involvement of the M4 receptor subtype | D'Agostino G.; Bolognesi M.L.; Lucchelli A.; Vicini D.; Balestra B.; Spelta V.; Melchiorre C.; To...nini M. | 2000-01-01 | BRITISH JOURNAL OF PHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Structure-activity relationship and site of binding of polyamine derivatives at the nicotinic acetylcholine receptor | Bixel M.G.; Krauss M.; Liu Y.; Bolognesi M.L.; Rosini M.; Mellor I.S.; Usherwood P.N.R.; Melchior...re C.; Koji N.; Hucho F. | 2000-01-01 | EUROPEAN JOURNAL OF BIOCHEMISTRY | - | 1.01 Articolo in rivista | - |
Analogues of prazosin that bear a benextramine-related polyamine backbone exhibit different antagonism toward α1-adrenoreceptor subtypes | Bolognesi M.L.; Marucci G.; Angeli P.; Buccioni M.; Minarini A.; Rosini M.; Tumiatti V.; Melchior...re C. | 2001-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines | Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Sp...ampinato S.; Tumiatti V.; Melchiorre C. | 2001-01-01 | BRITISH JOURNAL OF PHARMACOLOGY | - | 1.01 Articolo in rivista | British J Pharmacology - 2009 - Budriesi - Analysis of the muscarinic receptor subtype mediating inhibition of the.pdf |
Binding of polyamine-containing toxins in the vestibule of the nicotinic acetylcholine receptor ion channel | Bixel M.Gabriele; Krauss M.; Weise C.; Bolognesi M.L.; Rosini M.; Usherwood P.N.R.; Melchiorre C....; Hucho F. | 2001-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |
Location of the Polyamine Binding Site in the Vestibule of the Nicotinic Acetylcholine Receptor Ion Channel | Bixel M.G.; Weise C.; Bolognesi M.L.; Rosini M.; Brierly M.J.; Mellor I.R.; Usherwood P.N.R.; Mel...chiorre C.; Hucho F. | 2001-01-01 | THE JOURNAL OF BIOLOGICAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Analogues of polyamine alkaloids and their synthetic advantages | Li Y.; Popaj K.; Lochner M.; Geneste H.; Budriesi R.; Chiarini A.; Melchiorre C.; Hesse M. | 2001-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |
Design, synthesis, and biological activity of methoctramine-related polyamines as putative Gi protein activators | Melchiorre C.; Bolognesi M.L.; Budriesi R.; Ghelardini C.; Chiarini A.; Minarini A.; Rosini M.; T...umiatti V.; Wade E.J. | 2001-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | J. Med. Chem. 2001, 44, 24, 4035–4038.pdf |
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure | Bolognesi M.L.; Bixel M.G.; Marucci G.; Bartolini M.; Krauss M.; Angeli P.; Antonello A.; Rosini ...M.; Tumiatti V.; Hucho F.; Melchiorre C. | 2002-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 2. Role of polymethylene chain lengths separating amine functions and of substituents on the terminal nitrogen atoms | Rosini M.; Bixel M.G.; Marucci G.; Budriesi R.; Krauss M.; Bolognesi M.L.; Minarini A.; Tumiatti ...V.; Hucho F.; Melchiorre C. | 2002-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Polymethylene tetraamine backbone as template for the development of biologically active polyamines | Melchiorre C.; Antonello A.; Banzi R.; Bolognesi M.L.; Minarini A.; Rosini M.; Tumiatti V. | 2003-01-01 | MEDICINAL RESEARCH REVIEWS | - | 1.01 Articolo in rivista | - |
Memoquin: a new compound to attack Alzheimer's disease drug discovery | Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Capsoni S.;... Cattaneo A. | 2004-01-01 | - | s.l. | 4.02 Riassunto (Abstract) | - |
Studio della configurazione dell'antagonista alfa 1B-adrenergico (+)-cyclazosin | Sagratini G.; Grelli M.; Gulini U.; Melchiorre C.; Antolini L.; Giardinà D. | 2004-01-01 | - | Grafiche Caroti | 4.02 Riassunto (Abstract) | - |
Absolute configuration of alpha 1B-adrenoceptor antagonist (+)-cyclazosin | Giardinà D.; Sagratini G.; Grelli M.; Gulini U.; Melchiorre C.; Antolini L. | 2004-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |
Memoquin: a new therapeutic poly-agent for Alzheimer's disease | Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Margotti E....; Capsoni S.; Cattaneo A. | 2004-01-01 | NEUROBIOLOGY OF AGING | - | 4.02 Riassunto (Abstract) | - |
Studio farmacologico del (+)-cyclazosin, un antagonista selettivo del recettore alfa 1B-adrenergico | Marucci G.; Sagratini G.; Angeli P.; Buccioni M.; Gulini U.; Melchiorre C.; Testa R.; Giardinà D. | 2004-01-01 | - | Grafiche Caroti | 4.02 Riassunto (Abstract) | - |
Progettazione e sintesi di analoghi rigidi di metoctramina nello studio dei recettori muscarinici | Tumiatti V.; Bolognesi M.L.; Minarini A.; Rosini M.; Angeli A.; Buccioni M.; Marucci G.; Melchior...re C. | 2004-01-01 | - | Grafiche Caroti | 4.02 Riassunto (Abstract) | - |
MEMOQUIN: A MULTIPOTENT ACETYLCHOLINESTERASE INHIBITOR WITH EXCELLENT IN VIVO ACTIVITY | A.Cavalli; ML Bolognesi; M.Bartolini; V.Andrisano; C.Melchiorre; M.Recanatini; S.Capsoni; A.Cattaneo | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 3. Effect of replacing the inner polymethylene chain with cyclic moieties | TUMIATTI V.; ANDRISANO V.; BANZI R.; BARTOLINI M.; MINARINI A.; ROSINI M.; MELCHIORRE C. | 2004-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Polyamines may modulate both G protein-coupled receptors and G proteins | MARUCCI G.; NOVI F.; BANZI R.; BOLOGNESI M. L.; BUCCIONI M.; MINARINI A.; ROSINI M.; ANGELI P.; M...AGGIO R.; MELCHIORRE C. | 2004-01-01 | MEDICINAL CHEMISTRY RESEARCH | - | 1.01 Articolo in rivista | - |
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