ROBERTI, MARINELLA
ROBERTI, MARINELLA
DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di IIa fascia
A Focused Library of Psychotropic Analogues with Neuroprotective and Neuroregenerative Potential
2019 Uliassi, Elisa; Pena-Altamira, Luis Emiliano; Morales, Aixa V.; Massenzio, Francesca; Petralla, Sabrina; Rossi, Michele; Roberti, Marinella; Martinez Gonzalez, Loreto; Martinez, Ana; Monti, Barbara; Bolognesi, Maria Laura*
A ligand-based virtual screening approach to identify small molecules as hERG channel activators
2015 Giacomini, E.; Buonfiglio, R.; Masetti, M.; Wang, Y.; Tseng, G.-N.; Roberti, M.; Recanatini, M.
A natural-like synthetic small molecule impairs bcr-abl signaling cascades and induces megakaryocyte differentiation in erythroleukemia cells
2013 Turroni S.; Tolomeo M.; Mamone G.; Picariello G.; Giacomini E.; Brigidi P.; Roberti M.; Grimaudo S.; Pipitone R.M.; Di Cristina A.; Recanatini M.
A RAD51/BRCA2 small molecule inhibitor enhances the antineoplastic effect of the PARPi talazoparib in pancreatic cancer
2023 Laura Poppi, Samuel H Myers, Viola Previtali, Francesco Rinaldi, Fulvia Farabegoli, Giuseppina Di Stefano, Naomi Walsh, Marinella Roberti, Andrea Cavalli
A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation
2012 G. P. Chiriano; A. De Simone; F. Mancini; D. I. Perez; A. Cavalli; M. L. Bolognesi; G. Legname; A. Martinez; V. Andrisano; P. Carloni; M. Roberti
An 19F NMR fragment-based approach for the discovery and development of BRCA2-RAD51 inhibitors to pursuit synthetic lethality in combination with PARP inhibition in pancreatic cancer
2023 Myers S. H., Poppi L., Rinaldi F., Veronesi M., Ciamarone A., Previtali V., Bagnolini G., Schipani F., Ortega Martínez J. A., Girotto S., Di Stefano G., Farabegoli F., Walsh N., De Franco F., Roberti M., Cavalli A.
Antioxidant Activity of Hydroxystilbene Derivatives in Homogeneous Solution
2004 AMORATI R.; LUCARINI M.; MUGNAINI V.; PEDULLI G.F.; ROBERTI M.; PIZZIRANI D.
Antiparasitic effect of stilbene and terphenyl compounds against trypanosoma cruzi parasites
2021 Bruno F.; Castelli G.; Vitale F.; Catanzaro S.; Badaco V.V.; Roberti M.; Colomba C.; Cascio A.; Tolomeo M.
Antiproliferative agents that interfere with the cell cycle at the G(1)-->S transition: further development and characterization of a small library of stilbene-derived compounds
2008 Pizzirani D.; Roberti M.; Cavalli A.; Grimaudo S.; Di Cristina A.; Pipitone R.M.; Gebbia N.; Tolomeo M.; Recanatini M.
Application of an “inhalation by design” approach to the identification and in-vitro evaluation of novel purine based PI3Kδ inhibitors
2023 Mazzucato R.; Roberti M.; Capelli A.M.; Rancati F.; Biagetti M.; Fiorelli C.; Bruno P.; Ronchi P.; Bertolini S.; Corsi M.; Pala D.
Arylsulphones: A Promising Class on Non-Nucleoside Antiviral Agents
2005 L. Garuti; M. Roberti; D. Pizzirani; G. Poggi
Benzimidazole derivatives as kinase inhibitors
2014 Garuti L; Roberti M; Bottegoni G.
Berberine and its metabolites: Relationship between physicochemical properties and plasma levels after administration to human subjects
2014 Spinozzi, S.; Colliva, C.; Camborata, C.; Roberti, M.; Ianni, C.; Neri, F.; Calvarese, C.; Lisotti, A.; Mazzella, G.; Roda, A.
Capitolo 2. Proprietà chimico-fisiche e attività biologica
2015 Bolognesi, Maria Laura; Roberti, Marinella
Characterisation of bioactive compounds in wine by-products: toward the valorisation of sustainable resources
2019 Camilla Marasca, Irene Brusa, Chiara Cabrelle, Michele Protti, Matteo Micucci, Laura Mercolini, Marinella Roberti, Roberta Budriesi, Maurizio Recanatini
Combined analytical approaches to define biodistribution and biological activity of semi-synthetic berberrubine, the active metabolite of natural berberine
2018 Porru, Emanuele; Franco, Placido; Calabria, Donato; Spinozzi, Silvia; Roberti, Marinella; Caliceti, Cristiana; Roda, Aldo
Computational design and discovery of "minimally structured" hERG blockers.
2012 Cavalli A.; Buonfiglio R.; Ianni C.; Masetti M.; Ceccarini L.; Caves R.; Chang M.W.; Mitcheson J.S.; Roberti M.; Recanatini M.
DESIGN OF LIGANDS WITH A HIGH AFFINITY TO PrPC
2008 A. Kranjc; S. Bongarzone; G. Chiriano; G. Rossetti; X. Biarnés; A. Cavalli; M.L. Bolognesi; M. Roberti; G. Legname; P. Carloni
Diaryl Urea: A Privileged Structure in Anticancer Agents
2016 Garuti, Laura; Roberti, Marinella; Ferraro, Mariarosaria; Bottegoni, Giovanni
Differential antiproliferative activity of new benzimidazole- 4,7-diones.
2004 L. Garuti; M. Roberti; D. Pizzirani; A. Pession; E. Leoncini; V. Cenci; S. Hrelia.
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
A Focused Library of Psychotropic Analogues with Neuroprotective and Neuroregenerative Potential | Uliassi, Elisa; Pena-Altamira, Luis Emiliano; Morales, Aixa V.; Massenzio, Francesca; Petralla, S...abrina; Rossi, Michele; Roberti, Marinella; Martinez Gonzalez, Loreto; Martinez, Ana; Monti, Barbara; Bolognesi, Maria Laura* | 2019-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | - |
A ligand-based virtual screening approach to identify small molecules as hERG channel activators | Giacomini, E.; Buonfiglio, R.; Masetti, M.; Wang, Y.; Tseng, G.-N.; Roberti, M.; Recanatini, M. | 2015-01-01 | COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING | - | 1.01 Articolo in rivista | - |
A natural-like synthetic small molecule impairs bcr-abl signaling cascades and induces megakaryocyte differentiation in erythroleukemia cells | Turroni S.; Tolomeo M.; Mamone G.; Picariello G.; Giacomini E.; Brigidi P.; Roberti M.; Grimaudo ...S.; Pipitone R.M.; Di Cristina A.; Recanatini M. | 2013-01-01 | PLOS ONE | - | 1.01 Articolo in rivista | PLoS_One_2013.pdf |
A RAD51/BRCA2 small molecule inhibitor enhances the antineoplastic effect of the PARPi talazoparib in pancreatic cancer | Laura Poppi, Samuel H Myers, Viola Previtali, Francesco Rinaldi, Fulvia Farabegoli, Giuseppina Di... Stefano, Naomi Walsh, Marinella Roberti, Andrea Cavalli | 2023-01-01 | - | FEBS PRESS | 4.03 Poster | - |
A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation | G. P. Chiriano; A. De Simone; F. Mancini; D. I. Perez; A. Cavalli; M. L. Bolognesi; G. Legname; A.... Martinez; V. Andrisano; P. Carloni; M. Roberti | 2012-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
An 19F NMR fragment-based approach for the discovery and development of BRCA2-RAD51 inhibitors to pursuit synthetic lethality in combination with PARP inhibition in pancreatic cancer | Myers S. H., Poppi L., Rinaldi F., Veronesi M., Ciamarone A., Previtali V., Bagnolini G., Schipan...i F., Ortega Martínez J. A., Girotto S., Di Stefano G., Farabegoli F., Walsh N., De Franco F., Roberti M., Cavalli A. | 2023-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Antioxidant Activity of Hydroxystilbene Derivatives in Homogeneous Solution | AMORATI R.; LUCARINI M.; MUGNAINI V.; PEDULLI G.F.; ROBERTI M.; PIZZIRANI D. | 2004-01-01 | JOURNAL OF ORGANIC CHEMISTRY | - | 1.01 Articolo in rivista | - |
Antiparasitic effect of stilbene and terphenyl compounds against trypanosoma cruzi parasites | Bruno F.; Castelli G.; Vitale F.; Catanzaro S.; Badaco V.V.; Roberti M.; Colomba C.; Cascio A.; T...olomeo M. | 2021-01-01 | PHARMACEUTICALS | - | 1.01 Articolo in rivista | pharmaceuticals 2020.pdf |
Antiproliferative agents that interfere with the cell cycle at the G(1)-->S transition: further development and characterization of a small library of stilbene-derived compounds | Pizzirani D.; Roberti M.; Cavalli A.; Grimaudo S.; Di Cristina A.; Pipitone R.M.; Gebbia N.; Tolo...meo M.; Recanatini M. | 2008-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
Application of an “inhalation by design” approach to the identification and in-vitro evaluation of novel purine based PI3Kδ inhibitors | Mazzucato R.; Roberti M.; Capelli A.M.; Rancati F.; Biagetti M.; Fiorelli C.; Bruno P.; Ronchi P....; Bertolini S.; Corsi M.; Pala D. | 2023-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Arylsulphones: A Promising Class on Non-Nucleoside Antiviral Agents | L. Garuti; M. Roberti; D. Pizzirani; G. Poggi | 2005-01-01 | CURRENT MEDICINAL CHEMISTRY ANTI-INFECTIVE AGENTS | - | 1.01 Articolo in rivista | - |
Benzimidazole derivatives as kinase inhibitors | Garuti L; Roberti M; Bottegoni G. | 2014-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Berberine and its metabolites: Relationship between physicochemical properties and plasma levels after administration to human subjects | Spinozzi, S.; Colliva, C.; Camborata, C.; Roberti, M.; Ianni, C.; Neri, F.; Calvarese, C.; Lisott...i, A.; Mazzella, G.; Roda, A. | 2014-01-01 | JOURNAL OF NATURAL PRODUCTS | - | 1.01 Articolo in rivista | - |
Capitolo 2. Proprietà chimico-fisiche e attività biologica | Bolognesi, Maria Laura; Roberti, Marinella | 2015-01-01 | - | Casa Editrice Ambrosiana | 2.01 Capitolo / saggio in libro | - |
Characterisation of bioactive compounds in wine by-products: toward the valorisation of sustainable resources | Camilla Marasca, Irene Brusa, Chiara Cabrelle, Michele Protti, Matteo Micucci, Laura Mercolini, M...arinella Roberti, Roberta Budriesi, Maurizio Recanatini | 2019-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
Combined analytical approaches to define biodistribution and biological activity of semi-synthetic berberrubine, the active metabolite of natural berberine | Porru, Emanuele; Franco, Placido; Calabria, Donato; Spinozzi, Silvia; Roberti, Marinella; Calicet...i, Cristiana; Roda, Aldo | 2018-01-01 | ANALYTICAL AND BIOANALYTICAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Computational design and discovery of "minimally structured" hERG blockers. | Cavalli A.; Buonfiglio R.; Ianni C.; Masetti M.; Ceccarini L.; Caves R.; Chang M.W.; Mitcheson J....S.; Roberti M.; Recanatini M. | 2012-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
DESIGN OF LIGANDS WITH A HIGH AFFINITY TO PrPC | A. Kranjc; S. Bongarzone; G. Chiriano; G. Rossetti; X. Biarnés; A. Cavalli; M.L. Bolognesi; M. Ro...berti; G. Legname; P. Carloni | 2008-01-01 | - | s. n. | 4.02 Riassunto (Abstract) | - |
Diaryl Urea: A Privileged Structure in Anticancer Agents | Garuti, Laura; Roberti, Marinella; Ferraro, Mariarosaria; Bottegoni, Giovanni | 2016-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Differential antiproliferative activity of new benzimidazole- 4,7-diones. | L. Garuti; M. Roberti; D. Pizzirani; A. Pession; E. Leoncini; V. Cenci; S. Hrelia. | 2004-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |