BUDRIESI, ROBERTA
BUDRIESI, ROBERTA
DIPARTIMENTO DI FARMACIA E BIOTECNOLOGIE
Docenti di ruolo di IIa fascia
α1 - and α2-Adrenoreceptor Antagonist Profiles of 1- and 2-[ω -(4-Arylpiperazin-1-yl)alkyl]-1,2,3-benzotriazoles
2005 A. Boido; R. Budriesi; C. Canu Boido; P. Ioan; E. Terranova; A. Chiarini; F. Sparatore.
1,4-DHP scaffold: calcium channel ligand based approach from cardiovascular to neuroprotective activity.
2012 Budriesi R
1,4-Dihydropyridine bearing a pharmacophoric fragment of lidoflazine
1996 Chiarini A.; Rampa A.; Budriesi R.; Bisi A.; Fabbri G.; Valenti P.
1,4-dihydropyridine derivatives as calcium channel modulators: the role of 3-methoxy-flavone moiety
2005 R. Budriesi; A. Bisi; P. Ioan; A. Rampa; S. Gobbi; F. Belluti; L. Piazzi; P. Valenti; A. Chiarini
1,4-Dihydropyridine Scaffold in Medicinal Chemistry, The Story So Far And Perspectives (Part 2): Action in Other Targets and Antitargets
2012 E Carosati; P Ioan; M Micucci; F Broccatelli; G Cruciani; BS Zhorov; A Chiarini; R Budriesi
1,4-Dihydropyridine Scaffold in Medicinal Chemistry, The Story so Far And Perspectives. (Part 1): Action in Ion Channels and GPCRs.
2011 Ioan P; Carosati E; Micucci M;Cruciani G; Broccatelli F; ZhorovBS; Chiarini A ; Budriesi R
1,4-Dihydropyridines Active on the SIRT1/AMPK Pathway Ameliorate Skin Repair and Mitochondrial Function and Exhibit Inhibition of Proliferation in Cancer Cells
2016 Valente, Sergio; Mellini, Paolo; Spallotta, Francesco; Carafa, Vincenzo; Nebbioso, Angela; Polletta, Lucia; Carnevale, Ilaria; Saladini, Serena; Trisciuoglio, Daniela; Gabellini, Chiara; Tardugno, Maria; Zwergel, Clemens; Cencioni, Chiara; Atlante, Sandra; Moniot, Sébastien; Steegborn, Clemens; Budriesi, Roberta; Tafani, Marco; Del Bufalo, Donatella; Altucci, Lucia; Gaetano, Carlo; Mai, Antonello
1,4-Dihydropyridines containing R-NNO-azoxy moieties
1995 Gasco A.M.; Ermondi G.; Gasco A.; Budriesi R.; Chiarini A.
3-Aryl-4-nitrobenzothiochromans S,S-dioxide: From Calcium-Channel Modulators Properties to Multidrug-Resistance Reverting Activity
2020 Micucci, Matteo; Viale, Maurizio; Chiarini, Alberto; Spinelli, Domenico; Frosini, Maria; Tavani, Cinzia; Maccagno, Massimo; Bianchi, Lara; Gangemi, Rosaria; Budriesi, Roberta
4-Heterotricyclic substituted 1,4-dihydropyridines with a potent selective bradycardic effect
1991 Rampa A.; Chiarini A.; Bisi A.; Budriesi R.; Valenti P.
4-Imidazo[2,1-b]thiazole-1,4-DHPs and neuroprotection: preliminary study in hits searching
2019 Leoni, Alberto; Frosini, Maria; Locatelli, Alessandra; Micucci, Matteo; Carotenuto, Claudio; Durante, Miriam; Cosconati, Sandro; Budriesi, Roberta*
6-Methoxy7-benzofuranoxy and 6-methoxy-7-indolyloxy analogues of WB4101: discovery of a potent and selective a1D-adrenoceptor antagonist.
2013 Fumagalli L.; Pallavicini M.; Budriesi R.; Bolchi C.; Chiarini A.; Chiodini G.; Gobbi M.; Laurino P.; Micucci M.; Straniero V.; Valoti E.
A new class of selective myocardial calcium channel modulators 2. Role of the acetal chain in oxadiazol-3-one derivatives
2005 R. BUDRIESI; E. CAROSATI; A. CHIARINI; B. COSIMELLI; G. CRUCIANI; P. IOAN; SPINELLI D.; R. SPISANI
A New Class of Selective Myocardial Calcium Channel Modulators: Oxadiazol-1-one Derivatives
2004 R. Budriesi; E. Carosati; A. Chiarini; B. Cosimelli; G. Cruciani; P. Ioan; D. Spinelli; R. Spisani.
A potential host and virus targeting tool against COVID-19: Chemical characterization, antiviral, cytoprotective, antioxidant, respiratory smooth muscle relaxant effects of Paulownia tomentosa Steud
2023 Magurano F.; Micucci M.; Nuzzo D.; Baggieri M.; Picone P.; Gioacchini S.; Fioravanti R.; Bucci P.; Kojouri M.; Mari M.; Retini M.; Budriesi R.; Mattioli L.B.; Corazza I.; Di Liberto V.; Todaro L.; Giuseppetti R.; D'Ugo E.; Marchi A.; Mecca M.; D'Auria M.
Absolute configuration and biological profile of two thiazinooxadiazol-3-ones with L-type calcium channel activity: a study of the structural effects
2012 Pierfranco Ioan; Alessia Ciogli; Francesco Sirci; Roberta Budriesi; Barbara Cosimelli; Marco Pierini; Elda Severi; Alberto Chiarini; Gabriele Cruciani; Francesco Gasparrini; Domenico Spinelli; Emanuele Carosati
Acacia catechu wild extract: A nutraceutical approach to gastrointestinal pathologies
2016 Micucci, M.; Chiarini, A.; Budriesi, R.
Acacia catechu willd. Extract protects neuronal cells from oxidative stress-induced damage
2022 Chiaino E.; Stella R.; Peggion C.; Micucci M.; Budriesi R.; Mattioli L.B.; Marzetti C.; Pessina F.; Valoti M.; Frosini M.
Activity of Antioxidants from Crocus sativus L. Petals: Potential Preventive Effects towards Cardiovascular System
2020 Zeka K, Marrazzo P, Micucci M, Ruparelia KC, Arroo RRJ, Macchiarelli G, Nottola SA, Continenza MA, Chiarini A, Angeloni C, Hrelia S, Budriesi R.
Affinity and activity profiling of unichiral 8-substituted 1,4-benzodioxane analogues of WB4101 reveals a potent and selective α1B-adrenoceptor antagonist.
2012 Fumagalli L; Pallavicini M; Budriesi R; Gobbi M; Straniero V; Zagami M; Chiodini G; Bolchi C; Chiarini A; Micucci M; Valoti E
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
α1 - and α2-Adrenoreceptor Antagonist Profiles of 1- and 2-[ω -(4-Arylpiperazin-1-yl)alkyl]-1,2,3-benzotriazoles | A. Boido; R. Budriesi; C. Canu Boido; P. Ioan; E. Terranova; A. Chiarini; F. Sparatore. | 2005-01-01 | CHEMISTRY & BIODIVERSITY | - | 1.01 Articolo in rivista | - |
1,4-DHP scaffold: calcium channel ligand based approach from cardiovascular to neuroprotective activity. | Budriesi R | 2012-01-01 | - | s.n. | 4.02 Riassunto (Abstract) | - |
1,4-Dihydropyridine bearing a pharmacophoric fragment of lidoflazine | Chiarini A.; Rampa A.; Budriesi R.; Bisi A.; Fabbri G.; Valenti P. | 1996-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
1,4-dihydropyridine derivatives as calcium channel modulators: the role of 3-methoxy-flavone moiety | R. Budriesi; A. Bisi; P. Ioan; A. Rampa; S. Gobbi; F. Belluti; L. Piazzi; P. Valenti; A. Chiarini | 2005-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
1,4-Dihydropyridine Scaffold in Medicinal Chemistry, The Story So Far And Perspectives (Part 2): Action in Other Targets and Antitargets | E Carosati; P Ioan; M Micucci; F Broccatelli; G Cruciani; BS Zhorov; A Chiarini; R Budriesi | 2012-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
1,4-Dihydropyridine Scaffold in Medicinal Chemistry, The Story so Far And Perspectives. (Part 1): Action in Ion Channels and GPCRs. | Ioan P; Carosati E; Micucci M;Cruciani G; Broccatelli F; ZhorovBS; Chiarini A ; Budriesi R | 2011-01-01 | CURRENT MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
1,4-Dihydropyridines Active on the SIRT1/AMPK Pathway Ameliorate Skin Repair and Mitochondrial Function and Exhibit Inhibition of Proliferation in Cancer Cells | Valente, Sergio; Mellini, Paolo; Spallotta, Francesco; Carafa, Vincenzo; Nebbioso, Angela; Pollet...ta, Lucia; Carnevale, Ilaria; Saladini, Serena; Trisciuoglio, Daniela; Gabellini, Chiara; Tardugno, Maria; Zwergel, Clemens; Cencioni, Chiara; Atlante, Sandra; Moniot, Sébastien; Steegborn, Clemens; Budriesi, Roberta; Tafani, Marco; Del Bufalo, Donatella; Altucci, Lucia; Gaetano, Carlo; Mai, Antonello | 2016-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
1,4-Dihydropyridines containing R-NNO-azoxy moieties | Gasco A.M.; Ermondi G.; Gasco A.; Budriesi R.; Chiarini A. | 1995-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |
3-Aryl-4-nitrobenzothiochromans S,S-dioxide: From Calcium-Channel Modulators Properties to Multidrug-Resistance Reverting Activity | Micucci, Matteo; Viale, Maurizio; Chiarini, Alberto; Spinelli, Domenico; Frosini, Maria; Tavani, ...Cinzia; Maccagno, Massimo; Bianchi, Lara; Gangemi, Rosaria; Budriesi, Roberta | 2020-01-01 | MOLECULES | - | 1.01 Articolo in rivista | molecules-25-01056-v2.pdf |
4-Heterotricyclic substituted 1,4-dihydropyridines with a potent selective bradycardic effect | Rampa A.; Chiarini A.; Bisi A.; Budriesi R.; Valenti P. | 1991-01-01 | ARZNEIMITTEL-FORSCHUNG | - | 1.01 Articolo in rivista | - |
4-Imidazo[2,1-b]thiazole-1,4-DHPs and neuroprotection: preliminary study in hits searching | Leoni, Alberto; Frosini, Maria; Locatelli, Alessandra; Micucci, Matteo; Carotenuto, Claudio; Dura...nte, Miriam; Cosconati, Sandro; Budriesi, Roberta* | 2019-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | copertina e proof pubblicazione Leoni(1).pdf |
6-Methoxy7-benzofuranoxy and 6-methoxy-7-indolyloxy analogues of WB4101: discovery of a potent and selective a1D-adrenoceptor antagonist. | Fumagalli L.; Pallavicini M.; Budriesi R.; Bolchi C.; Chiarini A.; Chiodini G.; Gobbi M.; Laurino... P.; Micucci M.; Straniero V.; Valoti E. | 2013-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A new class of selective myocardial calcium channel modulators 2. Role of the acetal chain in oxadiazol-3-one derivatives | R. BUDRIESI; E. CAROSATI; A. CHIARINI; B. COSIMELLI; G. CRUCIANI; P. IOAN; SPINELLI D.; R. SPISANI | 2005-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A New Class of Selective Myocardial Calcium Channel Modulators: Oxadiazol-1-one Derivatives | R. Budriesi; E. Carosati; A. Chiarini; B. Cosimelli; G. Cruciani; P. Ioan; D. Spinelli; R. Spisani. | 2004-01-01 | DRUGS OF THE FUTURE | - | 4.02 Riassunto (Abstract) | - |
A potential host and virus targeting tool against COVID-19: Chemical characterization, antiviral, cytoprotective, antioxidant, respiratory smooth muscle relaxant effects of Paulownia tomentosa Steud | Magurano F.; Micucci M.; Nuzzo D.; Baggieri M.; Picone P.; Gioacchini S.; Fioravanti R.; Bucci P....; Kojouri M.; Mari M.; Retini M.; Budriesi R.; Mattioli L.B.; Corazza I.; Di Liberto V.; Todaro L.; Giuseppetti R.; D'Ugo E.; Marchi A.; Mecca M.; D'Auria M. | 2023-01-01 | BIOMÉDECINE & PHARMACOTHÉRAPIE | - | 1.01 Articolo in rivista | 1-s2.0-S075333222201472X-main(1).pdf |
Absolute configuration and biological profile of two thiazinooxadiazol-3-ones with L-type calcium channel activity: a study of the structural effects | Pierfranco Ioan; Alessia Ciogli; Francesco Sirci; Roberta Budriesi; Barbara Cosimelli; Marco Pier...ini; Elda Severi; Alberto Chiarini; Gabriele Cruciani; Francesco Gasparrini; Domenico Spinelli; Emanuele Carosati | 2012-01-01 | ORGANIC & BIOMOLECULAR CHEMISTRY | - | 1.01 Articolo in rivista | - |
Acacia catechu wild extract: A nutraceutical approach to gastrointestinal pathologies | Micucci, M.; Chiarini, A.; Budriesi, R. | 2016-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
Acacia catechu willd. Extract protects neuronal cells from oxidative stress-induced damage | Chiaino E.; Stella R.; Peggion C.; Micucci M.; Budriesi R.; Mattioli L.B.; Marzetti C.; Pessina F....; Valoti M.; Frosini M. | 2022-01-01 | ANTIOXIDANTS | - | 1.01 Articolo in rivista | antioxidants-11-00081-v2.pdf |
Activity of Antioxidants from Crocus sativus L. Petals: Potential Preventive Effects towards Cardiovascular System | Zeka K, Marrazzo P, Micucci M, Ruparelia KC, Arroo RRJ, Macchiarelli G, Nottola SA, Continenza M...A, Chiarini A, Angeloni C, Hrelia S, Budriesi R. | 2020-01-01 | ANTIOXIDANTS | - | 1.01 Articolo in rivista | antioxidants-2020.pdf |
Affinity and activity profiling of unichiral 8-substituted 1,4-benzodioxane analogues of WB4101 reveals a potent and selective α1B-adrenoceptor antagonist. | Fumagalli L; Pallavicini M; Budriesi R; Gobbi M; Straniero V; Zagami M; Chiodini G; Bolchi C; Chi...arini A; Micucci M; Valoti E | 2012-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |