ANDRISANO, VINCENZA
ANDRISANO, VINCENZA
DIPARTIMENTO DI SCIENZE PER LA QUALITA' DELLA VITA
Docenti di ruolo di Ia fascia
ANDRISANO V.; V. ANDRISANO.; Andrisano; E. ANDRISANO; ANDRISANO VINCENZA; Vincenza Andrisano
'Enzymes' immobilization on monolithic matrices: applications in drug discovery'
2010 Vincenza Andrisano; Manuela Bartolini
(±)- BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3β Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease
2021 Ismaili L.; Monnin J.; Etievant A.; Arribas R.L.; Viejo L.; Refouvelet B.; Soukup O.; Janockova J.; Hepnarova V.; Korabecny J.; Kucera T.; Jun D.; Andrys R.; Musilek K.; Baguet A.; Garcia-Frutos E.M.; De Simone A.; Andrisano V.; Bartolini M.; De Los Rios C.; Marco-Contelles J.; Haffen E.
- Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors.
2016 Angela, De Simone; Andrea, Milelli; Marina, Naldi; Vincenza, Andrisano
1,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: synthesis, pharmacological evaluation and mechanistic studies
2014 O Di Pietro; E Viayna; E Vicente-García; M Bartolini; Rosario Ramón; J Juárez-Jiménez; M. V Clos; B Pérez; V Andrisano; F. Javier Luque; R Lavilla; D Muñoz-Torrero
2-Arylbenzofuran-based molecules as multipotent Alzheimer's disease modifying agents
2012 S. Rizzo; A. Tarozzi; M. Bartolini; G. Da Costa; A. Bisi; S. Gobbi; F. Belluti; A. Ligresti; M. Allarà; J-P. Monti; V. Andrisano; V. Di Marzo; P. Hrelia; A. Rampa
20079SLZMC - PRIN 2007-Metodologie analitiche avanzate nelle ricerca e sviluppo di farmaci.
2009 Andrisano V.
3,4-Dihydro-1,3,5-triazin-2(1H)-ones as the First Dual BACE-1/GSK-3β Fragment Hits against Alzheimer's Disease
2015 Prati, Federica; De Simone, Angela; Armirotti, Andrea; Summa, Maria; Pizzirani, Daniela; Scarpelli, Rita; Bertozzi, Sine Mandrup; Perez, Daniel I.; Andrisano, Vincenza; Perez-Castillo, Ana; Monti, Barbara; Massenzio, Francesca; Polito, Letizia; Racchi, Marco; Sabatino, Piera; Bottegoni, Giovanni; Martinez, Ana; Cavalli, Andrea; Bolognesi, Maria L.
3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy
2003 Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valenti P.; Recanatini M.
A Fluorescent Styrylquinoline with Combined Therapeutic and Diagnostic Activities against Alzheimer's and Prion Diseases
2013 Staderini, M; Aulic, S; Bartolini, M; Hoang, NAT; Gonzalez-Ruiz, V; Perez, DI; Cabezas, N; Martinez, A; Martin, MA; Andrisano; Legname, G; Menendez, JC; Bolognesi, ML
A multi-approach study for BACE-1 inhibitors characterization.
2010 Angela De Simone; F. Mancini; C. Bertucci; V. Andrisano
A MULTI-METHODOLOGICAL APPROACH FOR BETA-AMYLOID AGGREGATION AND INHIBITION STUDIES
2010 Bartolini M.; Naldi M.; Fiori J.; Valle F.; Biscarini F.; Nicolau D.V.; Andrisano V.
A multi-methodological approach for the investigation of β-Amyloid-CORMs interaction: an LC-ESI/MS and Circular Dichroism study.
2018 de simone a, naldi m, tedesco d, bartolini m, andrisano v
A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors
2019 Perez-Areales F.J.; Turcu A.L.; Barniol-Xicota M.; Pont C.; Pivetta D.; Espargaro A.; Bartolini M.; De Simone A.; Andrisano V.; Perez B.; Sabate R.; Sureda F.X.; Vazquez S.; Munoz-Torrero D.
A patent review of butyrylcholinesterase inhibitors and reactivators 2010–2017
2018 Andrisano, Vincenza*; Naldi, Marina; De Simone, Angela; Bartolini, Manuela
A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation
2012 G. P. Chiriano; A. De Simone; F. Mancini; D. I. Perez; A. Cavalli; M. L. Bolognesi; G. Legname; A. Martinez; V. Andrisano; P. Carloni; M. Roberti
A small molecule targeting the multifactorial nature of Alzheimer's disease
2007 Cavalli A.; Bolognesi M. L.; Capsoni S.; Andrisano V.; Bartolini M.; Margotti E.; Cattaneo A.; Recanatini M.; Melchiorre C.
Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: Molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives
2000 Rampa A.; Bisi A.; Belluti F.; Gobbi S.; Valenti P.; Andrisano V.; Cavrini V.; Cavalli A.; Recanatini M.
Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives
2001 Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Cavalli A.; Recanatini M.; Valenti P.
Acetylcholinesterase oriented immobilization on nanopatterned bilayered surfaces for biosensing devices
2010 M. Bartolini; M. Naldi; D. V. Nicolau; F.C.M.J.M. van Delft; J. van Zijl; J. Snijder; F.C. van den Heuvel; V. Andrisano
ACETYLCHOLINESTERASE-BASED ANALYTICAL TOOLS FOR DRUG SCREENING
2012 M. Bartolini; M. Naldi; D.V. Nicolau; F.C.M.J.M. van Delft; J. van Zijl; J. Snijder; F.C. van den Heuvel; V. Andrisano
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
'Enzymes' immobilization on monolithic matrices: applications in drug discovery' | Vincenza Andrisano; Manuela Bartolini | 2010-01-01 | - | ILM Publications | 2.01 Capitolo / saggio in libro | - |
(±)- BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3β Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease | Ismaili L.; Monnin J.; Etievant A.; Arribas R.L.; Viejo L.; Refouvelet B.; Soukup O.; Janockova J....; Hepnarova V.; Korabecny J.; Kucera T.; Jun D.; Andrys R.; Musilek K.; Baguet A.; Garcia-Frutos E.M.; De Simone A.; Andrisano V.; Bartolini M.; De Los Rios C.; Marco-Contelles J.; Haffen E. | 2021-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | - |
- Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors. | Angela, De Simone; Andrea, Milelli; Marina, Naldi; Vincenza, Andrisano | 2016-01-01 | - | - | 4.03 Poster | - |
1,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: synthesis, pharmacological evaluation and mechanistic studies | O Di Pietro; E Viayna; E Vicente-García; M Bartolini; Rosario Ramón; J Juárez-Jiménez; M. V Clos;... B Pérez; V Andrisano; F. Javier Luque; R Lavilla; D Muñoz-Torrero | 2014-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
2-Arylbenzofuran-based molecules as multipotent Alzheimer's disease modifying agents | S. Rizzo; A. Tarozzi; M. Bartolini; G. Da Costa; A. Bisi; S. Gobbi; F. Belluti; A. Ligresti; M. A...llarà; J-P. Monti; V. Andrisano; V. Di Marzo; P. Hrelia; A. Rampa | 2012-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
20079SLZMC - PRIN 2007-Metodologie analitiche avanzate nelle ricerca e sviluppo di farmaci. | Andrisano V. | 2009-01-01 | - | - | 8.04 Coordinamento di progetti di ricerca | - |
3,4-Dihydro-1,3,5-triazin-2(1H)-ones as the First Dual BACE-1/GSK-3β Fragment Hits against Alzheimer's Disease | Prati, Federica; De Simone, Angela; Armirotti, Andrea; Summa, Maria; Pizzirani, Daniela; Scarpell...i, Rita; Bertozzi, Sine Mandrup; Perez, Daniel I.; Andrisano, Vincenza; Perez-Castillo, Ana; Monti, Barbara; Massenzio, Francesca; Polito, Letizia; Racchi, Marco; Sabatino, Piera; Bottegoni, Giovanni; Martinez, Ana; Cavalli, Andrea; Bolognesi, Maria L. | 2015-01-01 | ACS CHEMICAL NEUROSCIENCE | - | 1.01 Articolo in rivista | accepted11585-546374.pdf |
3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy | Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valen...ti P.; Recanatini M. | 2003-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A Fluorescent Styrylquinoline with Combined Therapeutic and Diagnostic Activities against Alzheimer's and Prion Diseases | Staderini, M; Aulic, S; Bartolini, M; Hoang, NAT; Gonzalez-Ruiz, V; Perez, DI; Cabezas, N; Martin...ez, A; Martin, MA; Andrisano; Legname, G; Menendez, JC; Bolognesi, ML | 2013-01-01 | ACS MEDICINAL CHEMISTRY LETTERS | - | 1.01 Articolo in rivista | - |
A multi-approach study for BACE-1 inhibitors characterization. | Angela De Simone; F. Mancini; C. Bertucci; V. Andrisano | 2010-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
A MULTI-METHODOLOGICAL APPROACH FOR BETA-AMYLOID AGGREGATION AND INHIBITION STUDIES | Bartolini M.; Naldi M.; Fiori J.; Valle F.; Biscarini F.; Nicolau D.V.; Andrisano V. | 2010-01-01 | - | CLEUP sc | 4.02 Riassunto (Abstract) | - |
A multi-methodological approach for the investigation of β-Amyloid-CORMs interaction: an LC-ESI/MS and Circular Dichroism study. | de simone a, naldi m, tedesco d, bartolini m, andrisano v | 2018-01-01 | - | - | 4.01 Contributo in Atti di convegno | - |
A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors | Perez-Areales F.J.; Turcu A.L.; Barniol-Xicota M.; Pont C.; Pivetta D.; Espargaro A.; Bartolini M....; De Simone A.; Andrisano V.; Perez B.; Sabate R.; Sureda F.X.; Vazquez S.; Munoz-Torrero D. | 2019-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A patent review of butyrylcholinesterase inhibitors and reactivators 2010–2017 | Andrisano, Vincenza*; Naldi, Marina; De Simone, Angela; Bartolini, Manuela | 2018-01-01 | EXPERT OPINION ON THERAPEUTIC PATENTS | - | 1.01 Articolo in rivista | - |
A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation | G. P. Chiriano; A. De Simone; F. Mancini; D. I. Perez; A. Cavalli; M. L. Bolognesi; G. Legname; A.... Martinez; V. Andrisano; P. Carloni; M. Roberti | 2012-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A small molecule targeting the multifactorial nature of Alzheimer's disease | Cavalli A.; Bolognesi M. L.; Capsoni S.; Andrisano V.; Bartolini M.; Margotti E.; Cattaneo A.; Re...canatini M.; Melchiorre C. | 2007-01-01 | ANGEWANDTE CHEMIE. INTERNATIONAL EDITION | - | 1.01 Articolo in rivista | - |
Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: Molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives | Rampa A.; Bisi A.; Belluti F.; Gobbi S.; Valenti P.; Andrisano V.; Cavrini V.; Cavalli A.; Recana...tini M. | 2000-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives | Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Caval...li A.; Recanatini M.; Valenti P. | 2001-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Acetylcholinesterase oriented immobilization on nanopatterned bilayered surfaces for biosensing devices | M. Bartolini; M. Naldi; D. V. Nicolau; F.C.M.J.M. van Delft; J. van Zijl; J. Snijder; F.C. van de...n Heuvel; V. Andrisano | 2010-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
ACETYLCHOLINESTERASE-BASED ANALYTICAL TOOLS FOR DRUG SCREENING | M. Bartolini; M. Naldi; D.V. Nicolau; F.C.M.J.M. van Delft; J. van Zijl; J. Snijder; F.C. van den... Heuvel; V. Andrisano | 2012-01-01 | - | bestprint | 4.02 Riassunto (Abstract) | - |