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Mostrati risultati da 1 a 20 di 223
Titolo Autore(i) Anno Periodico Editore Tipo File
Negative inotropic and calcium antagonistic activity of alkyl and arylalkyl phosphonates Bellucci C.; Gualtieri F.; Scapecchi S.; Teodori E.; Budriesi R.; Chiarini A. 1989-01-01 IL FARMACO - 1.01 Articolo in rivista -
Xanthone 1,4-dihydropyridine derivatives with a potent selective bradycardic effect Valenti P.; Chiarini A.; Gasperi F.; Budriesi R. 1990-01-01 ARZNEIMITTEL-FORSCHUNG - 1.01 Articolo in rivista -
Molecular properties of the histamine H2-receptor. Covalent inhibition by tetraamine disulfides Chiarini A.; Minarini A.; Budriesi R.; Melchiorre C. 1990-01-01 IL FARMACO - 1.01 Articolo in rivista -
Further investigation on methoctramine-related tetraamines: Effects of terminal N-substitution and of chain length separating the four nitrogens on M2 muscarinic receptor blocking activity Minarini A.; Budriesi R.; Chiarini A.; Melchiorre C.; Tumiatti V. 1991-01-01 IL FARMACO - 1.01 Articolo in rivista -
4-Heterotricyclic substituted 1,4-dihydropyridines with a potent selective bradycardic effect Rampa A.; Chiarini A.; Bisi A.; Budriesi R.; Valenti P. 1991-01-01 ARZNEIMITTEL-FORSCHUNG - 1.01 Articolo in rivista -
Synthesis and cardiovascular properties of fluorenyl derivatives related to verapamil Novella Romanelli M.; Teodori E.; Scapecchi S.; Dei S.; Budriesi R.; Chiarini A. 1991-01-01 IL FARMACO - 1.01 Articolo in rivista -
Fluorenone and benzophenone 1,4-dihydropyridine derivatives with cardiodepressant activity Rampa A.; Budriesi R.; Bisi A.; Chiarini A.; Valenti P. 1992-01-01 ARZNEIMITTEL-FORSCHUNG - 1.01 Articolo in rivista -
Synthesis and biological evaluation of some new phosphonates Garuti L.; Ferranti A.; Ronerti M.; Katz E.; Budriesi R.; Chiarini A. 1992-01-01 PHARMAZIE - 1.01 Articolo in rivista -
Affinity and selectivity at M2 and M3 muscarinic receptor subtypes of cyclic and open oxygenated analogues of 4-DAMP Tumiatti V.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R.; Bolognesi M.L. 1992-01-01 IL FARMACO - 1.01 Articolo in rivista -
Negative inotropic and chronotropic activity of calcium channel ligands possessing a xanthone 1,4-dihydropyridine backbone Chiarini A.; Rampa A.; Bisi A.; Budriesi R.; Valenti P. 1992-01-01 ARZNEIMITTEL-FORSCHUNG - 1.01 Articolo in rivista -
Synthesis and cardiovascular properties of furazanyl-1,4-dihydropyridines and of furoxanyl analogues Gasco A.M.; Fruttero R.; Sorba G.; Gasco A.; Budriesi R.; Chiarini A. 1992-01-01 ARZNEIMITTEL-FORSCHUNG - 1.01 Articolo in rivista -
Xanthone analogues of milrinone Montanari P.; Chiarini A.; Budriesi R.; Valenti P. 1992-01-01 JOURNAL OF HETEROCYCLIC CHEMISTRY - 1.01 Articolo in rivista -
SAR studies in the field of Ca-antagonists: 2-substituted 1,4-dihydropyridines with a xanthone backbone Bisi A.; Budriesi R.; Chiarini A.; Rampa A.; Valenti P. 1993-01-01 IL FARMACO - 1.01 Articolo in rivista -
Semi-rigid analogues of the calcium antagonist verapamil: A molecular modelling study Romanelli M.N.; Dei S.; Scapecchi S.; Teodori E.; Gualtieri F.; Budriesi R.; Mannhold R. 1994-01-01 JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN - 1.01 Articolo in rivista -
Synthesis and pharmacological evaluation of verapamil analogs with restricted molecular flexibility Teodori E.; Dei S.; Romanelli M.; Scapecchi S.; Gualtieri F.; Budriesi R.; Chiarini A.; Lemoine H....; Mannhold R. 1994-01-01 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Synthesis and "in vitro" cardiovascular activity of 4-aryl-2,3,3a,4-tetrahydro-1h-pyrrolo[2,1-c][1,4]benzothiazin-1-ones and 7-acetoxy-6-phenyl-7a,8,9,10-tetrahydropyrrolo [2,1,-d][1,5]benzothiazepin-10-one Campiani G.; Garofalo A.; Fiorini I.; Nacci V.; Botta M.; Tafi A.; Chiarini A.; Budriesi R.; Brun...i G.; Romeo M.R. 1994-01-01 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS - 1.01 Articolo in rivista -
Design, Synthesis, and Biological Activity of Methoctramine-Related Tetraamines Bearing an 11-Acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one Moiety: Structural Requirements for Optimum Occupancy of Muscarinic Receptor Subtypes As Revealed by Symmetrical and Unsymmetrical Polyamines Minarini A.; Bolognesi M.L.; Budriesi R.; Canossa M.; Chiarini A.; Spampinato S.; Melchiorre C. 1994-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Design, synthesis and biological activity of some 4-DAMP- related compounds Tumiatti V.; Santi S.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R. 1995-01-01 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS - 1.01 Articolo in rivista -
Structure-activity relationship studies in the field of calcium antagonists. Xanthone 1,4-dihydropyridines bearing a 2,3-lactone ring Rampa A.; Budriesi R.; Bisi A.; Fabbri G.; Barili P.L.; Chiarini A.; Valenti P. 1995-01-01 ARZNEIMITTEL-FORSCHUNG - 1.01 Articolo in rivista -
The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists Melchiorre C.; Minarini A.; Budriesi R.; Chiarini A.; Spampinato S.; Tumiatti V. 1995-01-01 LIFE SCIENCES - 1.01 Articolo in rivista -
Mostrati risultati da 1 a 20 di 223
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