Sfoglia per Autore
Characterisation of the conjugate of the (6-maleimidocaproyl)hydrazone derivative of doxorubicin with lactosaminated human albumin by 13C NMR spectroscopy.
2009-01-01 Boga C.; Fiume L.; Baglioni M.; Bertucci C.; Farina C.; Kratz F.; Manerba M.; Naldi M.; Di Stefano G.
The enhancement of interstitial transport of a doxorubicin-lactosaminated albumin conjugate by imatinib: in rat hepatocellular carcinoma it is not preferentially higher than that in liver and bone marrow.
2009-01-01 Fiume L.; Baglioni M.; Busi C.; Manerba M.; Di Stefano G.
Effect of copper on extracellular levels of key pro-inflammatory molecules in hypothalamic GN11 and primary neurons.
2009-01-01 Spisni E; Valerii MC; Manerba M; Strillacci A; Polazzi E; Mattia T; Griffoni C; Tomasi V.
Altered glycosylation profile of purified plasma ACT from Alzheimer's disease.
2010-01-01 Ianni M; Manerba M; Di Stefano G; Porcellini E; Chiappelli M; Carbone I; Licastro F.
Impairment of aerobic glycolysis by inhibitors of lactic dehydrogenase hinders the growth of human hepatocellular carcinoma cell lines.
2010-01-01 Fiume L; Manerba M; Vettraino M; Di Stefano G
Inhibition of lactic dehydrogenase as a way to increase the anti-proliferative effect of multi-targeted kinase inhibitors.
2011-01-01 Fiume L.; Vettraino M.; Manerba M.; Di Stefano G.
Effect of sorafenib on the energy metabolism of hepatocellular carcinoma cells.
2011-01-01 Fiume L.; Manerba M.; Vettraino M.; Di Stefano G.
Galloflavin (CAS 568-80-9), a novel inhibitor of lactate dehydrogenase.
2012-01-01 Manerba M.; Vettraino M.; Fiume L.; Di Stefano G.; Sartini A.; Giacomini E.; Buonfiglio R.; Roberti M.; Recanatini M.
Galloflavin, a new lactate dehydrogenase inhibitor, induces the death of human breast cancer cells with different glycolytic attitude by affecting distinct signaling pathways.
2012-01-01 Farabegoli F.; Vettraino M.; Manerba M.; Fiume L.; Roberti M.; Di Stefano G.
Galloflavin suppresses lactate dehydrogenase activity and causes MYC downregulationin Burkitt lymphoma cells via NAD/NADH-dependent inhibition of sirtuin-1
2013-01-01 Vettraino M; Manerba M; Govoni M; Di Stefano G.
NAD metabolism and functions: a common therapeutic target for neoplastic, metabolic and neurodegenerative diseases
2013-01-01 Di Stefano G; Manerba M; Vettraino M
Inhibition of lactate dehydrogenase activity as an approach to cancer therapy
2014-01-01 Luigi FIUME; Marcella MANERBA; Marina VETTRAINO; Giuseppina DI STEFANO
Albumin-drug conjugates in the treatment of hepatic disorders.
2014-01-01 Fiume L;Manerba M;Di Stefano G
Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors
2015-01-01 Sebastiano Rupiani; Rosa Buonfiglio; Marcella Manerba; Lorenza Di Ianni; Marina Vettraino; Elisa Giacomini; Matteo Masetti; Federico Falchi; Giuseppina Di Stefano; Marinella Roberti; Maurizio Recanatini
Lactate dehydrogenase inhibitors sensitize lymphoma cells to cisplatin without enhancing the drug effects on immortalized normal lymphocytes.
2015-01-01 M. Manerba; L. Di Ianni; L. Fiume; M. Roberti; M. Recanatini; G. Di Stefano
Lactate dehydrogenase inhibition: Exploring possible applications beyond cancer treatment
2016-01-01 Di Stefano, Giuseppina; Manerba, Marcella; Di Ianni, Lorenza; Fiume, Luigi
Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A
2016-01-01 Rupiani, Sebastiano; Guidotti, Laura; Manerba, Marcella; Di Ianni, Lorenza; Giacomini, Elisa; Falchi, Federico; Di Stefano, Giuseppina; Roberti, Marinella; Recanatini, Maurizio
Synthetic Lethality Triggered by Combining Olaparib with BRCA2-Rad51 Disruptors
2017-01-01 Falchi, Federico; Giacomini, Elisa; Masini, Tiziana; Boutard, Nicolas; Di Ianni, Lorenza; Manerba, Marcella; Farabegoli, Fulvia; Rossini, Lara; Robertson, Janet; Minucci, Saverio; Pallavicini, Isabella; Di Stefano, Giuseppina; Roberti, Marinella; Pellicciari, Roberto; Cavalli, Andrea
LDH inhibition impacts on heat shock response and induces senescence of hepatocellular carcinoma cells
2017-01-01 Manerba, Marcella; Di Ianni, Lorenza; Govoni, Marzia; Roberti, Marinella; Recanatini, Maurizio; Di Stefano, Giuseppina
Lactate dehydrogenase inhibitors can reverse inflammation induced changes in colon cancer cells
2017-01-01 Manerba, Marcella; Di Ianni, Lorenza; Govoni, Marzia; Roberti, Marinella; Recanatini, Maurizio; Di Stefano, Giuseppina
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Characterisation of the conjugate of the (6-maleimidocaproyl)hydrazone derivative of doxorubicin with lactosaminated human albumin by 13C NMR spectroscopy. | Boga C.; Fiume L.; Baglioni M.; Bertucci C.; Farina C.; Kratz F.; Manerba M.; Naldi M.; Di Stefano G. | 2009-01-01 | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | - | 1.01 Articolo in rivista | - |
The enhancement of interstitial transport of a doxorubicin-lactosaminated albumin conjugate by imatinib: in rat hepatocellular carcinoma it is not preferentially higher than that in liver and bone marrow. | Fiume L.; Baglioni M.; Busi C.; Manerba M.; Di Stefano G. | 2009-01-01 | EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS | - | 1.01 Articolo in rivista | - |
Effect of copper on extracellular levels of key pro-inflammatory molecules in hypothalamic GN11 and primary neurons. | Spisni E; Valerii MC; Manerba M; Strillacci A; Polazzi E; Mattia T; Griffoni C; Tomasi V. | 2009-01-01 | NEUROTOXICOLOGY | - | 1.01 Articolo in rivista | - |
Altered glycosylation profile of purified plasma ACT from Alzheimer's disease. | Ianni M; Manerba M; Di Stefano G; Porcellini E; Chiappelli M; Carbone I; Licastro F. | 2010-01-01 | IMMUNITY & AGEING | - | 1.01 Articolo in rivista | 1742-4933-7-S1-S6.pdf |
Impairment of aerobic glycolysis by inhibitors of lactic dehydrogenase hinders the growth of human hepatocellular carcinoma cell lines. | Fiume L; Manerba M; Vettraino M; Di Stefano G | 2010-01-01 | PHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Inhibition of lactic dehydrogenase as a way to increase the anti-proliferative effect of multi-targeted kinase inhibitors. | Fiume L.; Vettraino M.; Manerba M.; Di Stefano G. | 2011-01-01 | PHARMACOLOGICAL RESEARCH | - | 1.01 Articolo in rivista | - |
Effect of sorafenib on the energy metabolism of hepatocellular carcinoma cells. | Fiume L.; Manerba M.; Vettraino M.; Di Stefano G. | 2011-01-01 | EUROPEAN JOURNAL OF PHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Galloflavin (CAS 568-80-9), a novel inhibitor of lactate dehydrogenase. | Manerba M.; Vettraino M.; Fiume L.; Di Stefano G.; Sartini A.; Giacomini E.; Buonfiglio R.; Roberti M.; Recanatini M. | 2012-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
Galloflavin, a new lactate dehydrogenase inhibitor, induces the death of human breast cancer cells with different glycolytic attitude by affecting distinct signaling pathways. | Farabegoli F.; Vettraino M.; Manerba M.; Fiume L.; Roberti M.; Di Stefano G. | 2012-01-01 | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | - | 1.01 Articolo in rivista | - |
Galloflavin suppresses lactate dehydrogenase activity and causes MYC downregulationin Burkitt lymphoma cells via NAD/NADH-dependent inhibition of sirtuin-1 | Vettraino M; Manerba M; Govoni M; Di Stefano G. | 2013-01-01 | ANTI-CANCER DRUGS | - | 1.01 Articolo in rivista | - |
NAD metabolism and functions: a common therapeutic target for neoplastic, metabolic and neurodegenerative diseases | Di Stefano G; Manerba M; Vettraino M | 2013-01-01 | CURRENT TOPICS IN MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Inhibition of lactate dehydrogenase activity as an approach to cancer therapy | Luigi FIUME; Marcella MANERBA; Marina VETTRAINO; Giuseppina DI STEFANO | 2014-01-01 | FUTURE MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Albumin-drug conjugates in the treatment of hepatic disorders. | Fiume L;Manerba M;Di Stefano G | 2014-01-01 | EXPERT OPINION ON DRUG DELIVERY | - | 1.01 Articolo in rivista | - |
Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors | Sebastiano Rupiani; Rosa Buonfiglio; Marcella Manerba; Lorenza Di Ianni; Marina Vettraino; Elisa Giacomini; Matteo Masetti; Federico Falchi; Giuseppina Di Stefano; Marinella Roberti; Maurizio Recanatini | 2015-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Lactate dehydrogenase inhibitors sensitize lymphoma cells to cisplatin without enhancing the drug effects on immortalized normal lymphocytes. | M. Manerba; L. Di Ianni; L. Fiume; M. Roberti; M. Recanatini; G. Di Stefano | 2015-01-01 | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | - | 1.01 Articolo in rivista | REVISED TEXT-1.pdf |
Lactate dehydrogenase inhibition: Exploring possible applications beyond cancer treatment | Di Stefano, Giuseppina; Manerba, Marcella; Di Ianni, Lorenza; Fiume, Luigi | 2016-01-01 | FUTURE MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A | Rupiani, Sebastiano; Guidotti, Laura; Manerba, Marcella; Di Ianni, Lorenza; Giacomini, Elisa; Falchi, Federico; Di Stefano, Giuseppina; Roberti, Marinella; Recanatini, Maurizio | 2016-01-01 | ORGANIC & BIOMOLECULAR CHEMISTRY | - | 1.01 Articolo in rivista | - |
Synthetic Lethality Triggered by Combining Olaparib with BRCA2-Rad51 Disruptors | Falchi, Federico; Giacomini, Elisa; Masini, Tiziana; Boutard, Nicolas; Di Ianni, Lorenza; Manerba, Marcella; Farabegoli, Fulvia; Rossini, Lara; Robertson, Janet; Minucci, Saverio; Pallavicini, Isabella; Di Stefano, Giuseppina; Roberti, Marinella; Pellicciari, Roberto; Cavalli, Andrea | 2017-01-01 | ACS CHEMICAL BIOLOGY | - | 1.01 Articolo in rivista | - |
LDH inhibition impacts on heat shock response and induces senescence of hepatocellular carcinoma cells | Manerba, Marcella; Di Ianni, Lorenza; Govoni, Marzia; Roberti, Marinella; Recanatini, Maurizio; Di Stefano, Giuseppina | 2017-01-01 | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | - | 1.01 Articolo in rivista | Bozza finale_PHASCI_4029_final.pdf |
Lactate dehydrogenase inhibitors can reverse inflammation induced changes in colon cancer cells | Manerba, Marcella; Di Ianni, Lorenza; Govoni, Marzia; Roberti, Marinella; Recanatini, Maurizio; Di Stefano, Giuseppina | 2017-01-01 | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | - | 1.01 Articolo in rivista | manerba_2107.pdf |
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