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Mostrati risultati da 1 a 20 di 60
Titolo Autore(i) Anno Periodico Editore Tipo File
Peptidomimetic Scaffolds for the Discovery of New Bioactive Compounds. Cyclotetrapeptide Analogues Based on a 13-Membered, Partially Modified Retro-Inverso Structure. Applications to the synthesis of Cancer Cell Adhesion Inhibitors L. Gentilucci; G. Cardillo; S. Spampinato; A. Tolomelli; F. Squassabia; R. De Marco; M. Baiula 2008-01-01 - s.n 4.02 Riassunto (Abstract) -
Investigation of the Interaction Between the Atypical Agonist c[YpwFG] and MOR L. Gentilucci; F. Squassabia; R. De Marco; R. Artali; G. Cardillo; A. Tolomelli; S. Spampinato; A.... Bedini. 2008-01-01 THE FEBS JOURNAL - 1.01 Articolo in rivista -
Investigation on MOR receptor activation by atypical mechanisms G. Bombieri; R. Artali; L. Gentilucci; R. De Marco; S. Spampinato; A. Bedini; 2008-01-01 - s.n 4.02 Riassunto (Abstract) -
Development and characterization of Endomorphin-1 analogues as novel potential analgesic drugs. Bedini A; Gentilucci L; Demarco R; Spampinato S 2009-01-01 - - 4.03 Poster -
Cyclopeptide analogs for generating new molecular and 3D diversity L. Gentilucci; G. Cardillo; A. Tolomelli; F. Squassabia; R. De Marco; G. Chiriano 2009-01-01 COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING - 1.01 Articolo in rivista -
Synthesis and Conformational Analysis of Cyclotetrapeptide Mimetic beta-Turn Templates and Validation as 3D Scaffolds L. Gentilucci; G. Cardillo; A. Tolomelli; R. De Marco; A. Garelli; S. Spampinato; A. Spartà; E. J...uaristi 2009-01-01 CHEMMEDCHEM - 1.01 Articolo in rivista -
DETERMINATION OF THE BIOLOGICALLY ACTIVE STRUCTURE OF THE ATYPICAL MOR-LIGAND c[D-Asp-1-amide-beta-Ala-D-Trp-Phe] AND ANALOGUES BY NMR AND MOLECULAR DOCKING L. Gentilucci; A.Tolomelli; S. Spampinato; A. Bedini; R. De Marco; R. Artali 2010-01-01 BOLETÍN DE LA SOCIEDAD QUÍMICA DE MÉXICO - 4.02 Riassunto (Abstract) -
Ac-D-Trp-PheNH2 AND Ac-D-Trp-Phe-GlyNH2 - A NEW CLASS OF UNUSUAL OPIOID PEPTIDES L. Gentilucci; R. De Marco; A. Tolomelli; S. Spampinato; A. Bedini; R. Artali 2010-01-01 - INRC 4.02 Riassunto (Abstract) -
A simple route towards peptide analogues containing substituted (S)- or (R)-tryptophans L. Gentilucci; L. Cerisoli; R. De Marco; A. Tolomelli 2010-01-01 TETRAHEDRON LETTERS - 1.01 Articolo in rivista -
Antiangiogenic Effect of Dual/Selective α5β1/αvβ3 Integrin Antagonists Designed on Partially Modified Retro-Inverso Cyclotetrapeptide Mimetics L. Gentilucci; G. Cardillo; S. Spampinato; A. Tolomelli; F. Squassabia; R. De Marco; A. Bedini; M.... Baiula; L. Belvisi; M. Civera 2010-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Peripheral antinociceptive effects of the cyclic endomorphin-1 analog c[YpwFG] in a mouse visceral pain model Bedini A; Baiula M; Gentilucci L; Tolomelli A; De Marco R; Spampinato S. 2010-01-01 PEPTIDES - 1.01 Articolo in rivista -
Interactions between atypical opioid agonists and MOR Gentilucci L.; De Marco R.; Tolomelli A.; Bedini A.; Spampinato S.; Artali R.; 2010-01-01 - s.n 4.02 Riassunto (Abstract) -
Chemical Modifications Designed to Improve Peptide Stability: Incorporation of Non-Natural Amino Acids, Pseudo-Peptide Bonds, and Cyclization L. Gentilucci; R. De Marco; L. Cerisoli 2010-01-01 CURRENT PHARMACEUTICAL DESIGN - 1.01 Articolo in rivista -
The Inverse Type II β-Turn on D-Trp-Phe, a Pharmacophoric Motif for MOR Agonists. Gentilucci L; Tolomelli A; De Marco R; Spampinato S; Bedini A; Artali R. 2011-01-01 CHEMMEDCHEM - 1.01 Articolo in rivista -
DESIGN AND SYNTHESIS OF OPIOID PEPTIDE ANALOGUES AND MIMETICS R.De Marco; L. Gentilucci; A. Tolomelli; S. Feddersen; S. Spampinato; A. Bedini; R. Artali. 2011-01-01 PHARMACOLOGICAL REPORTS - 1.06 Abstract in rivista -
Endomorphin-1 analogues as novel and highly selective MOPr agonists: design and characterization of innovative analgesic drugs Bedini A; Gentilucci L; De Marco R; Spampinato S 2011-01-01 - - 4.03 Poster -
Synthesis of Constrained Peptidomimetics Containing 2-Oxo-1,3-oxazolidine-4-carboxylic Acids L. Gentilucci; A. Tolomelli; R. De Marco; C. Tomasini; S. Feddersen 2011-01-01 EUROPEAN JOURNAL OF ORGANIC CHEMISTRY - 1.01 Articolo in rivista -
A novel family of minimalist opioid peptides deprived of the classic pharmacophores L. Gentilucci; R. de Marco; A. Tolomelli; S. Feddersen; S. Spampinato; A. Bedini; R. Artali 2011-01-01 PHARMACOLOGICAL REPORTS - 1.06 Abstract in rivista -
Opioid Activity Profiles of Oversimplified Peptides Lacking in the Protonable N-Terminus R. De Marco; A. Tolomelli; S. Spampinato; A. Bedini; L. Gentilucci 2012-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
One-step synthesis of constrained peptidomimetics including oxazolidinones and/or dehydro-amino acids, and application to the design of bioactive compounds R. De Marco; A. Tolomelli; M. Campitiello; P. Rubini; S. Rupiani; A. Greco; L. Gentilucci 2012-01-01 - SCI 4.01 Contributo in Atti di convegno -
Mostrati risultati da 1 a 20 di 60
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