Sfoglia per Autore
“Linear and Cyclic Dehydro-beta-Amino Acids as Conformationally Constrained Scaffolds for the Preparation of Bioactive Compounds”
2010 G. Cardillo; L. Gentilucci; E.Mosconi; A. Viola; A. Tolomelli
Stereoselective Synthesis of Linear and Cyclic Dehydro-beta-amino Acids for the Preparation of alpha-v-beta-3 and alpha-5-beta-1 Integrin Inhibitors
2010 G. Cardillo; L. Gentilucci; E.Mosconi; A. Viola; A. Tolomelli
Dehydro-beta-amino acids as scaffolds for the preparation of alpha-v-beta-3, alpha-5-beta-1 and alpha-4-beta-1 integrin ligands
2011 A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; M. Baiula; S. Spampinato; L. Belvisi; M. Civera
A straightforward route to enantiopure 2-substituted-3,4-dehydro-beta-proline via ring closing metathesis
2011 A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; E. Paradisi
Development of isoxazoline-containing peptidomimetics as dual alpha-v-beta-3 and alpha-5-beta-1 integrin ligands.
2011 A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Belvisi; M. Civera
Dehydro-beta-amino acid containing peptidomimetics as integrin receptor ligands
2012 A. Tolomelli; A. Viola; L. Gentilucci; E. Mosconi; R. De Marco; M. Baiula; S. Spampinato; L. Belvisi; M. Civera
Dehydro-beta-amino acid as building blocks for bioactive compounds
2012 G. Cardillo; L. Gentilucci; E. Mosconi; A. Tolomelli; A. Viola
NEW PEPTIDOMIMETIC α4β1-INTEGRIN ANTAGONISTS FOR REDUCING INFLAMMATION AND ALLERGIC REACTIONS
2012 A. Greco; R. De Marco; A. Tolomelli; A. Viola; S. Spampinato; M. Baiula; S. Dattoli; L. Gentilucci
Exploring the reactivity of alkylidene malonamides: synthesis of polyfunctionalized isoxazolidinones, aziridines and oxazolines
2012 A. Tolomelli; G. Cardillo; L. Gentilucci; R. Juris; A. Viola; E. Juaristi
An improved protocol for Yonemitsu-type trimolecular condensation
2012 A. Tolomelli; L. Gentilucci; A.Viola
Alkylidene malonamides and acetacetamides as intermediates for the preparation of constrained dipeptide mimetics.
2012 A. Tolomelli; L. Gentilucci; A. Viola
Modulation of αvβ3- and α5β1-integrin-mediated adhesion by dehydro-β-amino acids containing peptidomimetics
2013 TOLOMELLI A.; BAIULA M.; BELVISI L.; VIOLA A.; GENTILUCCI L.; TROISI S.; DATTOLI S. D.; SPAMPINATO S.; CIVERA M.; JUARISTI E.; ESCUDERO M.
Design, synthesis and in vitro evaluation of tumor homing agents by conjugation of integrin ligands to diagnostics and cytotoxic drugs
2014 A. Tolomelli; L. Gentilucci; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Belvisi; M.Civera
Design and Synthesis of Integrin Ligands αvβ3 and α5β1 as delivery systems for fluorescent molecules
2014 L. Ferrazzano; A. Tolomelli; A. Viola
Design and synthesis of Alpha-v-beta-3 and Alpha-5-beta-1 integrin ligands as delivery systems for fluorescent molecules
2014 Tolomelli, Alessandra; Gentilucci, Luca; Viola, Angelo; Dattoli, Samantha Deianira; Baiula, Monica; Spampinato, Santi; Petkau-Milroy, Katja; Brunsveld, Luc
Novel tools against antibiotic resistance: design and synthesis of Linezolid analogues
2014 L. Ferrazzano; A. Tolomelli; A. Viola
An improved microwave assisted protocol for Yonemitsu-type trimolecular condensation
2014 Angelo Viola;Lucia Ferrazzano;Giulia Martelli;Sebastiano Ancona;Luca Gentilucci;Alessandra Tolomelli
Toward the Development of Dual-Targeted Glyceraldehyde-3-phosphate Dehydrogenase/Trypanothione Reductase Inhibitors againstTrypanosoma bruceiandTrypanosoma cruzi
2014 Federica Belluti;Elisa Uliassi;Giacomo Veronesi;Christian Bergamini;Marcel Kaiser;Reto Brun;Angelo Viola;Romana Fato;Paul A. M. Michels;R. Luise Krauth-Siegel;Andrea Cavalli;Maria Laura Bolognesi
Design and synthesis of integrin ligands as «molecular shuttles» for drugs and fluorescent molecules delivery
2015 Ferrazzano, L.; Viola, A.; Tolomelli, A.
Design and synthesis of integrin ligands as «molecular shuttles» for drugs and fluorescent molecules delivery
2015 Ferrazzano, L.; Viola, A.; Tolomelli, A.
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
“Linear and Cyclic Dehydro-beta-Amino Acids as Conformationally Constrained Scaffolds for the Preparation of Bioactive Compounds” | G. Cardillo; L. Gentilucci; E.Mosconi; A. Viola; A. Tolomelli | 2010-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Stereoselective Synthesis of Linear and Cyclic Dehydro-beta-amino Acids for the Preparation of alpha-v-beta-3 and alpha-5-beta-1 Integrin Inhibitors | G. Cardillo; L. Gentilucci; E.Mosconi; A. Viola; A. Tolomelli | 2010-01-01 | BOLETÍN DE LA SOCIEDAD QUÍMICA DE MÉXICO | - | 4.02 Riassunto (Abstract) | - |
Dehydro-beta-amino acids as scaffolds for the preparation of alpha-v-beta-3, alpha-5-beta-1 and alpha-4-beta-1 integrin ligands | A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; M. Baiula; S. Spampinato; L. Belvisi; M. Civera | 2011-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
A straightforward route to enantiopure 2-substituted-3,4-dehydro-beta-proline via ring closing metathesis | A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; E. Paradisi | 2011-01-01 | AMINO ACIDS | - | 1.01 Articolo in rivista | - |
Development of isoxazoline-containing peptidomimetics as dual alpha-v-beta-3 and alpha-5-beta-1 integrin ligands. | A. Tolomelli; L. Gentilucci; E. Mosconi; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Be...lvisi; M. Civera | 2011-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
Dehydro-beta-amino acid containing peptidomimetics as integrin receptor ligands | A. Tolomelli; A. Viola; L. Gentilucci; E. Mosconi; R. De Marco; M. Baiula; S. Spampinato; L. Belv...isi; M. Civera | 2012-01-01 | - | Europan Assciation for Chemical and Molecular Sciences | 4.02 Riassunto (Abstract) | - |
Dehydro-beta-amino acid as building blocks for bioactive compounds | G. Cardillo; L. Gentilucci; E. Mosconi; A. Tolomelli; A. Viola | 2012-01-01 | - | cietà Chimica Itlaiana -Divisione Chimica farmaceutica | 4.02 Riassunto (Abstract) | - |
NEW PEPTIDOMIMETIC α4β1-INTEGRIN ANTAGONISTS FOR REDUCING INFLAMMATION AND ALLERGIC REACTIONS | A. Greco; R. De Marco; A. Tolomelli; A. Viola; S. Spampinato; M. Baiula; S. Dattoli; L. Gentilucci | 2012-01-01 | - | SCI | 4.01 Contributo in Atti di convegno | - |
Exploring the reactivity of alkylidene malonamides: synthesis of polyfunctionalized isoxazolidinones, aziridines and oxazolines | A. Tolomelli; G. Cardillo; L. Gentilucci; R. Juris; A. Viola; E. Juaristi | 2012-01-01 | ARKIVOC | - | 1.01 Articolo in rivista | - |
An improved protocol for Yonemitsu-type trimolecular condensation | A. Tolomelli; L. Gentilucci; A.Viola | 2012-01-01 | - | Società Chimica Italiana | 4.02 Riassunto (Abstract) | - |
Alkylidene malonamides and acetacetamides as intermediates for the preparation of constrained dipeptide mimetics. | A. Tolomelli; L. Gentilucci; A. Viola | 2012-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Modulation of αvβ3- and α5β1-integrin-mediated adhesion by dehydro-β-amino acids containing peptidomimetics | TOLOMELLI A.; BAIULA M.; BELVISI L.; VIOLA A.; GENTILUCCI L.; TROISI S.; DATTOLI S. D.; SPAMPINAT...O S.; CIVERA M.; JUARISTI E.; ESCUDERO M. | 2013-01-01 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Design, synthesis and in vitro evaluation of tumor homing agents by conjugation of integrin ligands to diagnostics and cytotoxic drugs | A. Tolomelli; L. Gentilucci; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Belvisi; M.Civera | 2014-01-01 | - | Elsevier | 4.02 Riassunto (Abstract) | - |
Design and Synthesis of Integrin Ligands αvβ3 and α5β1 as delivery systems for fluorescent molecules | L. Ferrazzano; A. Tolomelli; A. Viola | 2014-01-01 | - | European Association of Chemical and Molecular Sciences | 4.02 Riassunto (Abstract) | - |
Design and synthesis of Alpha-v-beta-3 and Alpha-5-beta-1 integrin ligands as delivery systems for fluorescent molecules | Tolomelli, Alessandra; Gentilucci, Luca; Viola, Angelo; Dattoli, Samantha Deianira; Baiula, Monic...a; Spampinato, Santi; Petkau-Milroy, Katja; Brunsveld, Luc | 2014-01-01 | LA CHIMICA E L'INDUSTRIA | - | 1.01 Articolo in rivista | - |
Novel tools against antibiotic resistance: design and synthesis of Linezolid analogues | L. Ferrazzano; A. Tolomelli; A. Viola | 2014-01-01 | - | European Association for Chemical and Molecular Sciences | 4.02 Riassunto (Abstract) | - |
An improved microwave assisted protocol for Yonemitsu-type trimolecular condensation | Angelo Viola;Lucia Ferrazzano;Giulia Martelli;Sebastiano Ancona;Luca Gentilucci;Alessandra Tolomelli | 2014-01-01 | TETRAHEDRON | - | 1.01 Articolo in rivista | - |
Toward the Development of Dual-Targeted Glyceraldehyde-3-phosphate Dehydrogenase/Trypanothione Reductase Inhibitors againstTrypanosoma bruceiandTrypanosoma cruzi | Federica Belluti;Elisa Uliassi;Giacomo Veronesi;Christian Bergamini;Marcel Kaiser;Reto Brun;Angel...o Viola;Romana Fato;Paul A. M. Michels;R. Luise Krauth-Siegel;Andrea Cavalli;Maria Laura Bolognesi | 2014-01-01 | CHEMMEDCHEM | - | 1.01 Articolo in rivista | - |
Design and synthesis of integrin ligands as «molecular shuttles» for drugs and fluorescent molecules delivery | Ferrazzano, L.; Viola, A.; Tolomelli, A. | 2015-01-01 | - | SCI | 4.02 Riassunto (Abstract) | - |
Design and synthesis of integrin ligands as «molecular shuttles» for drugs and fluorescent molecules delivery | Ferrazzano, L.; Viola, A.; Tolomelli, A. | 2015-01-01 | - | // | 4.02 Riassunto (Abstract) | - |
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