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Mostrati risultati da 1 a 20 di 109
Titolo Autore(i) Anno Periodico Editore Tipo File
Synthesis of flavone-2'-carboxylic acid analogues as potential antitumor agents Valenti P.; Bisi A.; Rampa A.; Gobbi S.; Belluti F.; Re P.D.; Cima L.; Carrara M. 1998-01-01 ANTI-CANCER DRUG DESIGN - 1.01 Articolo in rivista -
Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: Molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives Rampa A.; Bisi A.; Belluti F.; Gobbi S.; Valenti P.; Andrisano V.; Cavrini V.; Cavalli A.; Recana...tini M. 2000-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
SAR of 9-amino-1,2,3-4-tetrahydroacridine-based acetylcholinesterase inhibitors: Synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues Recanatini M.; Cavalli A.; Belluti F.; Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Valenti P.; Andris...ano V.; Bartolini M.; Cavrini V. 2000-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Synthesis and biological activity of some rigid analogues of flavone-8- acetic acid Valenti P.; Bisi A.; Rampa A.; Belluti F.; Gobbi S.; Zampiron A.; Carrara M. 2000-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Caval...li A.; Recanatini M.; Valenti P. 2001-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
A new class of nonsteroidal aromatase inhibitors: Design and synthesis of chromone and xanthone derivatives and inhibition of the P450 enzymes aromatase and 17α-hydroxylase/C17,20-lyase Recanatini M.; Hartmann R.W.; Bisi A.; Cavalli A.; Belluti F.; Gobbi S.; Rampa A.; Valenti P.; Pa...lzer M.; Palusczak A. 2001-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Synthesis and antitumor activity of new derivatives of xanthen-9-one-4-acetic acid Gobbi S.; Rampa A.; Bisi A.; Belluti F.; Valenti P.; Caputo A.; Zampiron A.; Carrara M. 2002-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valen...ti P.; Recanatini M. 2003-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Cardiovascular hybrid drugs: New benzazepinone derivatives as bradycardic agents endowed with selective β1-Non-competitive antagonism Bisi A.; Rampa A.; Budriesi R.; Gobbi S.; Belluti F.; Ioan P.; Valoti E.; Chiarini A.; Valenti P. 2003-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Synthesis and biological evaluation of 3-alkoxy analogues of flavone-8-acetic acid Gobbi S.; Rampa A.; Bisi A.; Belluti F.; Piazzi L.; Valenti P.; Caputo A.; Zampiron A.; Carrara M. 2003-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
In vitro biological activity of new analogues of flavon-8-acetic acid M. Carrara; A. Zampiron; M. Barbera; A. Caputo; S. Gobbi; F. Belluti; A. Bisi; L. Piazzi; A. Ramp...a; P. Valenti 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
Derivati a struttura benzofenonica come inibitori dell'acetilcolinesterasi F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; V. Andrisano; M. Bartolini; A. Cavalli; M. Re...canatini; P. Valenti 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
Analogues of the dual acetylcholinesterase inhibitor AP2238: synthesis and SAR L. Piazzi; M. Bartolini; F. Belluti; A. Bisi; A. Cavalli; S. Gobbi; A. Rampa; P. Valenti 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
Cholinesterase inhibitors: xanthostigmine derivatives blocking the acetylcholinesterase-induced beta-amyloid aggregation. Belluti F.; Rampa A.; Piazzi L.; Bisi A.; Gobbi S.; Bartolini M.; Andrisano V.; Cavalli A.; Recan...atini M.; Valenti P. 2005-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
1,4-dihydropyridine derivatives as calcium channel modulators: the role of 3-methoxy-flavone moiety R. Budriesi; A. Bisi; P. Ioan; A. Rampa; S. Gobbi; F. Belluti; L. Piazzi; P. Valenti; A. Chiarini 2005-01-01 BIOORGANIC & MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Nonsteroidal Aromatase inhibitors: synthesis and evaluation of new flavone derivatives S. Gobbi; A. Bisi; F. Belluti; L. Piazzi; A. Rampa; P. Valenti; A. Cavalli; A. Paluszcak; R.W. Ha...rtmann 2005-01-01 - s.n 4.02 Riassunto (Abstract) -
Studies on cytostatic and cytotoxic activity of new flavopiridol analogues M. Carrara; A. Zampiron; A. Caputo; F. Belluti; A. Bisi; S. Gobbi; L. Piazzi; A. Rampa; P. Valent...i; P. Da Re 2005-01-01 - s.n 4.02 Riassunto (Abstract) -
In vitro studies of flavon-8-acetic acid analogues M. Carrara; A. Zampiron; M. Barbera; A. Caputo; S. Gobbi; F. Belluti; A. Bisi; L. Piazzi; A. Ramp...a; P. Valenti 2005-01-01 - s.n 4.02 Riassunto (Abstract) -
Homopterocarpanes as bridged triarylethylene analogues: synthesis and antagonistic effects in human MCF-7 breast cancer cells A. Rampa; A. Bisi; F. Belluti; S. Gobbi; L. Piazzi; P. Valenti; A. Zampiron; A. Caputo; K. Varani...; P. A. Borea; M. Carrara 2005-01-01 IL FARMACO - 1.01 Articolo in rivista -
Benzophenone derivatives as Inhibitors of Acetylcholinesterase F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; M. Bartolini; A. Cavalli; P. Valenti 2005-01-01 - s.n 4.02 Riassunto (Abstract) -
Mostrati risultati da 1 a 20 di 109
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