Sfoglia per Autore
Synthesis of flavone-2'-carboxylic acid analogues as potential antitumor agents
1998 Valenti P.; Bisi A.; Rampa A.; Gobbi S.; Belluti F.; Re P.D.; Cima L.; Carrara M.
Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: Molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives
2000 Rampa A.; Bisi A.; Belluti F.; Gobbi S.; Valenti P.; Andrisano V.; Cavrini V.; Cavalli A.; Recanatini M.
SAR of 9-amino-1,2,3-4-tetrahydroacridine-based acetylcholinesterase inhibitors: Synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues
2000 Recanatini M.; Cavalli A.; Belluti F.; Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Valenti P.; Andrisano V.; Bartolini M.; Cavrini V.
Synthesis and biological activity of some rigid analogues of flavone-8- acetic acid
2000 Valenti P.; Bisi A.; Rampa A.; Belluti F.; Gobbi S.; Zampiron A.; Carrara M.
Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives
2001 Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Cavalli A.; Recanatini M.; Valenti P.
A new class of nonsteroidal aromatase inhibitors: Design and synthesis of chromone and xanthone derivatives and inhibition of the P450 enzymes aromatase and 17α-hydroxylase/C17,20-lyase
2001 Recanatini M.; Hartmann R.W.; Bisi A.; Cavalli A.; Belluti F.; Gobbi S.; Rampa A.; Valenti P.; Palzer M.; Palusczak A.
Synthesis and antitumor activity of new derivatives of xanthen-9-one-4-acetic acid
2002 Gobbi S.; Rampa A.; Bisi A.; Belluti F.; Valenti P.; Caputo A.; Zampiron A.; Carrara M.
3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy
2003 Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valenti P.; Recanatini M.
Cardiovascular hybrid drugs: New benzazepinone derivatives as bradycardic agents endowed with selective β1-Non-competitive antagonism
2003 Bisi A.; Rampa A.; Budriesi R.; Gobbi S.; Belluti F.; Ioan P.; Valoti E.; Chiarini A.; Valenti P.
Synthesis and biological evaluation of 3-alkoxy analogues of flavone-8-acetic acid
2003 Gobbi S.; Rampa A.; Bisi A.; Belluti F.; Piazzi L.; Valenti P.; Caputo A.; Zampiron A.; Carrara M.
In vitro biological activity of new analogues of flavon-8-acetic acid
2004 M. Carrara; A. Zampiron; M. Barbera; A. Caputo; S. Gobbi; F. Belluti; A. Bisi; L. Piazzi; A. Rampa; P. Valenti
Derivati a struttura benzofenonica come inibitori dell'acetilcolinesterasi
2004 F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; V. Andrisano; M. Bartolini; A. Cavalli; M. Recanatini; P. Valenti
Analogues of the dual acetylcholinesterase inhibitor AP2238: synthesis and SAR
2004 L. Piazzi; M. Bartolini; F. Belluti; A. Bisi; A. Cavalli; S. Gobbi; A. Rampa; P. Valenti
Cholinesterase inhibitors: xanthostigmine derivatives blocking the acetylcholinesterase-induced beta-amyloid aggregation.
2005 Belluti F.; Rampa A.; Piazzi L.; Bisi A.; Gobbi S.; Bartolini M.; Andrisano V.; Cavalli A.; Recanatini M.; Valenti P.
1,4-dihydropyridine derivatives as calcium channel modulators: the role of 3-methoxy-flavone moiety
2005 R. Budriesi; A. Bisi; P. Ioan; A. Rampa; S. Gobbi; F. Belluti; L. Piazzi; P. Valenti; A. Chiarini
Nonsteroidal Aromatase inhibitors: synthesis and evaluation of new flavone derivatives
2005 S. Gobbi; A. Bisi; F. Belluti; L. Piazzi; A. Rampa; P. Valenti; A. Cavalli; A. Paluszcak; R.W. Hartmann
Studies on cytostatic and cytotoxic activity of new flavopiridol analogues
2005 M. Carrara; A. Zampiron; A. Caputo; F. Belluti; A. Bisi; S. Gobbi; L. Piazzi; A. Rampa; P. Valenti; P. Da Re
In vitro studies of flavon-8-acetic acid analogues
2005 M. Carrara; A. Zampiron; M. Barbera; A. Caputo; S. Gobbi; F. Belluti; A. Bisi; L. Piazzi; A. Rampa; P. Valenti
Homopterocarpanes as bridged triarylethylene analogues: synthesis and antagonistic effects in human MCF-7 breast cancer cells
2005 A. Rampa; A. Bisi; F. Belluti; S. Gobbi; L. Piazzi; P. Valenti; A. Zampiron; A. Caputo; K. Varani; P. A. Borea; M. Carrara
Benzophenone derivatives as Inhibitors of Acetylcholinesterase
2005 F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; M. Bartolini; A. Cavalli; P. Valenti
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
Synthesis of flavone-2'-carboxylic acid analogues as potential antitumor agents | Valenti P.; Bisi A.; Rampa A.; Gobbi S.; Belluti F.; Re P.D.; Cima L.; Carrara M. | 1998-01-01 | ANTI-CANCER DRUG DESIGN | - | 1.01 Articolo in rivista | - |
Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: Molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives | Rampa A.; Bisi A.; Belluti F.; Gobbi S.; Valenti P.; Andrisano V.; Cavrini V.; Cavalli A.; Recana...tini M. | 2000-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
SAR of 9-amino-1,2,3-4-tetrahydroacridine-based acetylcholinesterase inhibitors: Synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues | Recanatini M.; Cavalli A.; Belluti F.; Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Valenti P.; Andris...ano V.; Bartolini M.; Cavrini V. | 2000-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Synthesis and biological activity of some rigid analogues of flavone-8- acetic acid | Valenti P.; Bisi A.; Rampa A.; Belluti F.; Gobbi S.; Zampiron A.; Carrara M. | 2000-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives | Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Caval...li A.; Recanatini M.; Valenti P. | 2001-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
A new class of nonsteroidal aromatase inhibitors: Design and synthesis of chromone and xanthone derivatives and inhibition of the P450 enzymes aromatase and 17α-hydroxylase/C17,20-lyase | Recanatini M.; Hartmann R.W.; Bisi A.; Cavalli A.; Belluti F.; Gobbi S.; Rampa A.; Valenti P.; Pa...lzer M.; Palusczak A. | 2001-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Synthesis and antitumor activity of new derivatives of xanthen-9-one-4-acetic acid | Gobbi S.; Rampa A.; Bisi A.; Belluti F.; Valenti P.; Caputo A.; Zampiron A.; Carrara M. | 2002-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy | Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valen...ti P.; Recanatini M. | 2003-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Cardiovascular hybrid drugs: New benzazepinone derivatives as bradycardic agents endowed with selective β1-Non-competitive antagonism | Bisi A.; Rampa A.; Budriesi R.; Gobbi S.; Belluti F.; Ioan P.; Valoti E.; Chiarini A.; Valenti P. | 2003-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Synthesis and biological evaluation of 3-alkoxy analogues of flavone-8-acetic acid | Gobbi S.; Rampa A.; Bisi A.; Belluti F.; Piazzi L.; Valenti P.; Caputo A.; Zampiron A.; Carrara M. | 2003-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
In vitro biological activity of new analogues of flavon-8-acetic acid | M. Carrara; A. Zampiron; M. Barbera; A. Caputo; S. Gobbi; F. Belluti; A. Bisi; L. Piazzi; A. Ramp...a; P. Valenti | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Derivati a struttura benzofenonica come inibitori dell'acetilcolinesterasi | F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; V. Andrisano; M. Bartolini; A. Cavalli; M. Re...canatini; P. Valenti | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Analogues of the dual acetylcholinesterase inhibitor AP2238: synthesis and SAR | L. Piazzi; M. Bartolini; F. Belluti; A. Bisi; A. Cavalli; S. Gobbi; A. Rampa; P. Valenti | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Cholinesterase inhibitors: xanthostigmine derivatives blocking the acetylcholinesterase-induced beta-amyloid aggregation. | Belluti F.; Rampa A.; Piazzi L.; Bisi A.; Gobbi S.; Bartolini M.; Andrisano V.; Cavalli A.; Recan...atini M.; Valenti P. | 2005-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
1,4-dihydropyridine derivatives as calcium channel modulators: the role of 3-methoxy-flavone moiety | R. Budriesi; A. Bisi; P. Ioan; A. Rampa; S. Gobbi; F. Belluti; L. Piazzi; P. Valenti; A. Chiarini | 2005-01-01 | BIOORGANIC & MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Nonsteroidal Aromatase inhibitors: synthesis and evaluation of new flavone derivatives | S. Gobbi; A. Bisi; F. Belluti; L. Piazzi; A. Rampa; P. Valenti; A. Cavalli; A. Paluszcak; R.W. Ha...rtmann | 2005-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Studies on cytostatic and cytotoxic activity of new flavopiridol analogues | M. Carrara; A. Zampiron; A. Caputo; F. Belluti; A. Bisi; S. Gobbi; L. Piazzi; A. Rampa; P. Valent...i; P. Da Re | 2005-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
In vitro studies of flavon-8-acetic acid analogues | M. Carrara; A. Zampiron; M. Barbera; A. Caputo; S. Gobbi; F. Belluti; A. Bisi; L. Piazzi; A. Ramp...a; P. Valenti | 2005-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Homopterocarpanes as bridged triarylethylene analogues: synthesis and antagonistic effects in human MCF-7 breast cancer cells | A. Rampa; A. Bisi; F. Belluti; S. Gobbi; L. Piazzi; P. Valenti; A. Zampiron; A. Caputo; K. Varani...; P. A. Borea; M. Carrara | 2005-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |
Benzophenone derivatives as Inhibitors of Acetylcholinesterase | F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; M. Bartolini; A. Cavalli; P. Valenti | 2005-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
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