Sfoglia per Autore
Molecular properties of the histamine H2-receptor. Covalent inhibition by tetraamine disulfides
1990 Chiarini A.; Minarini A.; Budriesi R.; Melchiorre C.
Further investigation on methoctramine-related tetraamines: Effects of terminal N-substitution and of chain length separating the four nitrogens on M2 muscarinic receptor blocking activity
1991 Minarini A.; Budriesi R.; Chiarini A.; Melchiorre C.; Tumiatti V.
Affinity and selectivity at M2 and M3 muscarinic receptor subtypes of cyclic and open oxygenated analogues of 4-DAMP
1992 Tumiatti V.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R.; Bolognesi M.L.
Synthesis and Biological Activity of Some Methoctramine-Related Tetraamines Bearing a 11-Acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4]-benzodiazepin-6-one Moiety as Antimuscarinics: A Second Generation of Highly Selective M2 Muscarinic Receptor Antagonists
1993 Melchiorre C.; Bolognesi M.L.; Chiarini A.; Minarini A.; Spampinato S.
Binding profile of the selective muscarinic receptor antagonist tripitramine
1994 Maggio R.; Barbier P.; Bolognesi M.L.; Minarini A.; Tedeschi D.; Melchiorre C.
Design, Synthesis, and Biological Activity of Methoctramine-Related Tetraamines Bearing an 11-Acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one Moiety: Structural Requirements for Optimum Occupancy of Muscarinic Receptor Subtypes As Revealed by Symmetrical and Unsymmetrical Polyamines
1994 Minarini A.; Bolognesi M.L.; Budriesi R.; Canossa M.; Chiarini A.; Spampinato S.; Melchiorre C.
Design, synthesis and biological activity of some tetraamines related to methoctramine and 4-DAMP
1995 Melchiorre C.; Minarini A.; Spampinato S.; Tumiatti V.
Design, synthesis and biological activity of some 4-DAMP- related compounds
1995 Tumiatti V.; Santi S.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R.
Synthesis, muscarinic blocking activity and molecular modeling studies of 4-DAMP-related compounds
1995 Recanatini M.; Tumiatti V.; Budriesi R.; Chiarini A.; Sabatino P.; Bolognesi M.L.; Melchiorre C.
The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists
1995 Melchiorre C.; Minarini A.; Budriesi R.; Chiarini A.; Spampinato S.; Tumiatti V.
In vitro characterization of tripitramine, a polymethylene tetraamine displaying high selectivity and affinity for muscarinic M2 receptors
1995 Chiarini A.; Budriesi R.; Bolognesi M.L.; Minarini A.; Melchiorre C.
Tetraamines as lead compounds for the design of neurotransmitter receptor ligands:Focus on α-adrenergic and muscarinic receptors recognition
1996 Melchiorre C.; Angeli P.; Bolognesi M.L.; Budriesi R.; Cacciaguerra S.; Chiarini A.; Crucianelli M.; Giardina D.; Gulini U.; Marucci G.; Minarini A.; Spampinato S.; Tumiatti V.
Universal template approach to drug design: Polyamines as selective muscarinic receptor antagonists
1998 Bolognesi M.L.; Minarini A.; Budriesi R.; Cacciaguerra S.; Chiarini A.; Spampinato S.; Tumiatti V.; Melchiorre C.
Antagonist binding profile of the split chimeric muscarinic m2-trunc/m3-tail receptor
1998 Barbier P.; Colelli A.; Bolognesi M.L.; Minarini A.; Tumiatti V.; Corsini G.U.; Melchiorre C.; Maggio R.
Search for selective antagonists at α1-adrenoreceptors: Neutral or negative antagonism?
1998 Melchiorre C.; Bolognesi M.L.; Budriesi R.; Chiarini A.; Giardina D.; Minarini A.; Quaglia W.; Leonardi A.
Search for α1-adrenoceptor subtypes selective antagonists: Design, synthesis and biological activity of cystazosin, an α(1D)-adrenoceptor antagonist
1998 Minarini A.; Budriesi R.; Chiarini A.; Leonardi A.; Melchiorre C.
Design, synthesis, and biological activity of prazosin-related antagonists. Role of the piperazine and furan units of prazosin on the selectivity for α1-adrenoreceptor subtypes
1998 Bolognesi M.L.; Budriesi R.; Chiarini A.; Poggesi E.; Leonardi A.; Melchiorre C.
WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for α1-adrenoreceptor subtypes and 5-HT(1A) receptors
1999 Bolognesi M.L.; Budriesi R.; Cavalli A.; Chiarini A.; Gotti R.; Leonardi A.; Minarini A.; Poggesi E.; Recanatini M.; Rosini M.; Tumiatti V.; Melchiorre C.
Design, synthesis, and biological evaluation of symmetrically and unsymmetrically substituted methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists
1999 Rosini M.; Budriesi R.; Bixel M.G.; Bolognesi M.L.; Chiarini A.; Hucho F.; Krogsgaard-Larsen P.; Mellor I.R.; Minarini A.; Tumiatti V.; Usherwood P.N.R.; Melchiorre C.
α1-Adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety
2000 Melchiorre C.; Angeli P.; Bolognesi M.L.; Chiarini A.; Giardina D.; Gulini U.; Leonardi A.; Marucci G.; Minarini A.; Pigini M.; Quaglia W.; Rosini M.; Tumiatti V.
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