Sfoglia per Autore
WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for α1-adrenoreceptor subtypes and 5-HT(1A) receptors
1999 Bolognesi M.L.; Budriesi R.; Cavalli A.; Chiarini A.; Gotti R.; Leonardi A.; Minarini A.; Poggesi E.; Recanatini M.; Rosini M.; Tumiatti V.; Melchiorre C.
Design, synthesis, and biological evaluation of symmetrically and unsymmetrically substituted methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists
1999 Rosini M.; Budriesi R.; Bixel M.G.; Bolognesi M.L.; Chiarini A.; Hucho F.; Krogsgaard-Larsen P.; Mellor I.R.; Minarini A.; Tumiatti V.; Usherwood P.N.R.; Melchiorre C.
Structure-activity relationship and site of binding of polyamine derivatives at the nicotinic acetylcholine receptor
2000 Bixel M.G.; Krauss M.; Liu Y.; Bolognesi M.L.; Rosini M.; Mellor I.S.; Usherwood P.N.R.; Melchiorre C.; Koji N.; Hucho F.
α1-Adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety
2000 Melchiorre C.; Angeli P.; Bolognesi M.L.; Chiarini A.; Giardina D.; Gulini U.; Leonardi A.; Marucci G.; Minarini A.; Pigini M.; Quaglia W.; Rosini M.; Tumiatti V.
Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines
2001 Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Spampinato S.; Tumiatti V.; Melchiorre C.
Binding of polyamine-containing toxins in the vestibule of the nicotinic acetylcholine receptor ion channel
2001 Bixel M.Gabriele; Krauss M.; Weise C.; Bolognesi M.L.; Rosini M.; Usherwood P.N.R.; Melchiorre C.; Hucho F.
Design, synthesis, and biological activity of methoctramine-related polyamines as putative Gi protein activators
2001 Melchiorre C.; Bolognesi M.L.; Budriesi R.; Ghelardini C.; Chiarini A.; Minarini A.; Rosini M.; Tumiatti V.; Wade E.J.
Location of the Polyamine Binding Site in the Vestibule of the Nicotinic Acetylcholine Receptor Ion Channel
2001 Bixel M.G.; Weise C.; Bolognesi M.L.; Rosini M.; Brierly M.J.; Mellor I.R.; Usherwood P.N.R.; Melchiorre C.; Hucho F.
Analogues of prazosin that bear a benextramine-related polyamine backbone exhibit different antagonism toward α1-adrenoreceptor subtypes
2001 Bolognesi M.L.; Marucci G.; Angeli P.; Buccioni M.; Minarini A.; Rosini M.; Tumiatti V.; Melchiorre C.
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure
2002 Bolognesi M.L.; Bixel M.G.; Marucci G.; Bartolini M.; Krauss M.; Angeli P.; Antonello A.; Rosini M.; Tumiatti V.; Hucho F.; Melchiorre C.
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 2. Role of polymethylene chain lengths separating amine functions and of substituents on the terminal nitrogen atoms
2002 Rosini M.; Bixel M.G.; Marucci G.; Budriesi R.; Krauss M.; Bolognesi M.L.; Minarini A.; Tumiatti V.; Hucho F.; Melchiorre C.
Polymethylene tetraamine backbone as template for the development of biologically active polyamines
2003 Melchiorre C.; Antonello A.; Banzi R.; Bolognesi M.L.; Minarini A.; Rosini M.; Tumiatti V.
Methoctramine analogues inhibit responses to capsaicin and protons in rat dorsal root ganglion neurons
2004 MELLOR I. R.; OGILVIE J.; PLUTEANU F.; CLOTHIER R. H.; PARKER T. L.; ROSINI M.; MINARINI A.; TUMIATTI V.; MELCHIORRE C.
Progettazione e sintesi di analoghi rigidi di metoctramina nello studio dei recettori muscarinici
2004 Tumiatti V.; Bolognesi M.L.; Minarini A.; Rosini M.; Angeli A.; Buccioni M.; Marucci G.; Melchiorre C.
Polyamines may modulate both G protein-coupled receptors and G proteins
2004 MARUCCI G.; NOVI F.; BANZI R.; BOLOGNESI M. L.; BUCCIONI M.; MINARINI A.; ROSINI M.; ANGELI P.; MAGGIO R.; MELCHIORRE C.
Design, synthesis, and biological evaluation of conformationally restricted rivastigmine analogues
2004 Bolognesi M. L.; Bartolini M.; Cavalli A.; Andrisano V.; Rosini M.; Minarini A.; Melchiorre C.
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 3. Effect of replacing the inner polymethylene chain with cyclic moieties
2004 TUMIATTI V.; ANDRISANO V.; BANZI R.; BARTOLINI M.; MINARINI A.; ROSINI M.; MELCHIORRE C.
Methoctramine analogues inhibit responses to capsaicin in DRG neurons and cloned TRPV1
2005 Minarini A.; Mellor I.; Bolognesi M.L.; Ogilvie J.; Rosini M.; Tumiatti V.; Melchiorre C.
Methoctramine-related polyamines as antinociceptive agents
2005 Tumiatti V.; Minarini A.; Rosini M.; Bolognesi M.L.; Marucci G.; Buccioni M.; Ghelardini C.; Melchiorre C.
Bivalent tacrine-based acetylcholinesterase inhibitors: role of the spacer in the recognition process of the enzyme gorge
2005 Bolognesi M.L.; Bartolini M.; Cavalli A.; Rosini M.; Andrisano V.; Melchiorre C.
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for α1-adrenoreceptor subtypes and 5-HT(1A) receptors | Bolognesi M.L.; Budriesi R.; Cavalli A.; Chiarini A.; Gotti R.; Leonardi A.; Minarini A.; Poggesi... E.; Recanatini M.; Rosini M.; Tumiatti V.; Melchiorre C. | 1999-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Design, synthesis, and biological evaluation of symmetrically and unsymmetrically substituted methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists | Rosini M.; Budriesi R.; Bixel M.G.; Bolognesi M.L.; Chiarini A.; Hucho F.; Krogsgaard-Larsen P.; ...Mellor I.R.; Minarini A.; Tumiatti V.; Usherwood P.N.R.; Melchiorre C. | 1999-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Structure-activity relationship and site of binding of polyamine derivatives at the nicotinic acetylcholine receptor | Bixel M.G.; Krauss M.; Liu Y.; Bolognesi M.L.; Rosini M.; Mellor I.S.; Usherwood P.N.R.; Melchior...re C.; Koji N.; Hucho F. | 2000-01-01 | EUROPEAN JOURNAL OF BIOCHEMISTRY | - | 1.01 Articolo in rivista | - |
α1-Adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety | Melchiorre C.; Angeli P.; Bolognesi M.L.; Chiarini A.; Giardina D.; Gulini U.; Leonardi A.; Maruc...ci G.; Minarini A.; Pigini M.; Quaglia W.; Rosini M.; Tumiatti V. | 2000-01-01 | PHARMACEUTICA ACTA HELVETIAE | - | 1.01 Articolo in rivista | - |
Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines | Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Sp...ampinato S.; Tumiatti V.; Melchiorre C. | 2001-01-01 | BRITISH JOURNAL OF PHARMACOLOGY | - | 1.01 Articolo in rivista | British J Pharmacology - 2009 - Budriesi - Analysis of the muscarinic receptor subtype mediating inhibition of the.pdf |
Binding of polyamine-containing toxins in the vestibule of the nicotinic acetylcholine receptor ion channel | Bixel M.Gabriele; Krauss M.; Weise C.; Bolognesi M.L.; Rosini M.; Usherwood P.N.R.; Melchiorre C....; Hucho F. | 2001-01-01 | IL FARMACO | - | 1.01 Articolo in rivista | - |
Design, synthesis, and biological activity of methoctramine-related polyamines as putative Gi protein activators | Melchiorre C.; Bolognesi M.L.; Budriesi R.; Ghelardini C.; Chiarini A.; Minarini A.; Rosini M.; T...umiatti V.; Wade E.J. | 2001-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | J. Med. Chem. 2001, 44, 24, 4035–4038.pdf |
Location of the Polyamine Binding Site in the Vestibule of the Nicotinic Acetylcholine Receptor Ion Channel | Bixel M.G.; Weise C.; Bolognesi M.L.; Rosini M.; Brierly M.J.; Mellor I.R.; Usherwood P.N.R.; Mel...chiorre C.; Hucho F. | 2001-01-01 | THE JOURNAL OF BIOLOGICAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Analogues of prazosin that bear a benextramine-related polyamine backbone exhibit different antagonism toward α1-adrenoreceptor subtypes | Bolognesi M.L.; Marucci G.; Angeli P.; Buccioni M.; Minarini A.; Rosini M.; Tumiatti V.; Melchior...re C. | 2001-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure | Bolognesi M.L.; Bixel M.G.; Marucci G.; Bartolini M.; Krauss M.; Angeli P.; Antonello A.; Rosini ...M.; Tumiatti V.; Hucho F.; Melchiorre C. | 2002-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 2. Role of polymethylene chain lengths separating amine functions and of substituents on the terminal nitrogen atoms | Rosini M.; Bixel M.G.; Marucci G.; Budriesi R.; Krauss M.; Bolognesi M.L.; Minarini A.; Tumiatti ...V.; Hucho F.; Melchiorre C. | 2002-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Polymethylene tetraamine backbone as template for the development of biologically active polyamines | Melchiorre C.; Antonello A.; Banzi R.; Bolognesi M.L.; Minarini A.; Rosini M.; Tumiatti V. | 2003-01-01 | MEDICINAL RESEARCH REVIEWS | - | 1.01 Articolo in rivista | - |
Methoctramine analogues inhibit responses to capsaicin and protons in rat dorsal root ganglion neurons | MELLOR I. R.; OGILVIE J.; PLUTEANU F.; CLOTHIER R. H.; PARKER T. L.; ROSINI M.; MINARINI A.; TUMI...ATTI V.; MELCHIORRE C. | 2004-01-01 | EUROPEAN JOURNAL OF PHARMACOLOGY | - | 1.01 Articolo in rivista | - |
Progettazione e sintesi di analoghi rigidi di metoctramina nello studio dei recettori muscarinici | Tumiatti V.; Bolognesi M.L.; Minarini A.; Rosini M.; Angeli A.; Buccioni M.; Marucci G.; Melchior...re C. | 2004-01-01 | - | Grafiche Caroti | 4.02 Riassunto (Abstract) | - |
Polyamines may modulate both G protein-coupled receptors and G proteins | MARUCCI G.; NOVI F.; BANZI R.; BOLOGNESI M. L.; BUCCIONI M.; MINARINI A.; ROSINI M.; ANGELI P.; M...AGGIO R.; MELCHIORRE C. | 2004-01-01 | MEDICINAL CHEMISTRY RESEARCH | - | 1.01 Articolo in rivista | - |
Design, synthesis, and biological evaluation of conformationally restricted rivastigmine analogues | Bolognesi M. L.; Bartolini M.; Cavalli A.; Andrisano V.; Rosini M.; Minarini A.; Melchiorre C. | 2004-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 3. Effect of replacing the inner polymethylene chain with cyclic moieties | TUMIATTI V.; ANDRISANO V.; BANZI R.; BARTOLINI M.; MINARINI A.; ROSINI M.; MELCHIORRE C. | 2004-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Methoctramine analogues inhibit responses to capsaicin in DRG neurons and cloned TRPV1 | Minarini A.; Mellor I.; Bolognesi M.L.; Ogilvie J.; Rosini M.; Tumiatti V.; Melchiorre C. | 2005-01-01 | - | s.l. | 4.02 Riassunto (Abstract) | - |
Methoctramine-related polyamines as antinociceptive agents | Tumiatti V.; Minarini A.; Rosini M.; Bolognesi M.L.; Marucci G.; Buccioni M.; Ghelardini C.; Melc...hiorre C. | 2005-01-01 | - | Università di Modena e Reggio Emilia | 4.02 Riassunto (Abstract) | - |
Bivalent tacrine-based acetylcholinesterase inhibitors: role of the spacer in the recognition process of the enzyme gorge | Bolognesi M.L.; Bartolini M.; Cavalli A.; Rosini M.; Andrisano V.; Melchiorre C. | 2005-01-01 | - | s.l. | 4.02 Riassunto (Abstract) | - |
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