Sfoglia per Autore
SAR of 9-amino-1,2,3-4-tetrahydroacridine-based acetylcholinesterase inhibitors: Synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues
2000 Recanatini M.; Cavalli A.; Belluti F.; Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Valenti P.; Andrisano V.; Bartolini M.; Cavrini V.
Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives
2001 Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Cavalli A.; Recanatini M.; Valenti P.
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure
2002 Bolognesi M.L.; Bixel M.G.; Marucci G.; Bartolini M.; Krauss M.; Angeli P.; Antonello A.; Rosini M.; Tumiatti V.; Hucho F.; Melchiorre C.
3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy
2003 Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valenti P.; Recanatini M.
Analytical methods for the determination of folic acid in a polymeric micellar carrier
2003 Andrisano V.; Bartolini M.; Bertucci C.; Cavrini V.; Luppi B.; Cerchiara T.
Analytical methods for the determination of folic acid in a polymeric micellar carrier
2003 Andrisano V.; Bartolini M.; Bertucci C.; Cavrini V.; Luppi B.; Cerchiara T.
Design, synthesis, and biological evaluation of conformationally restricted rivastigmine analogues
2004 Bolognesi M. L.; Bartolini M.; Cavalli A.; Andrisano V.; Rosini M.; Minarini A.; Melchiorre C.
Evaluation of the inhibitory potency of a new series of AChE-inhibitors by using a monolithic AChE-micro-IMER
2004 M. Bartolini; V. Tumiatti; V. Andrisano
METODI ANALITICI INTEGRATI PER LA VALUTAZIONE DEL PROFILO D’AZIONE DI NUOVI FARMACI ANTI-ALZHEIMER.
2004 M. Bartolini; C. Bertucci; V. Cavrini; V. Andrisano
Memoquin: a new compound to attack Alzheimer's disease drug discovery
2004 Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Capsoni S.; Cattaneo A.
INTEGRATED ANALYTICAL APPROACHES FOR ALZHEIMER’S DISEASE NEW DRUG DISCOVERY
2004 M. Bartolini; C. Bertucci; V. Cavrini; V. Andrisano.
CHOOSING THE RIGHT CHROMATOGRAPHIC SUPPORT FOR ENZYME-BASED MICRO-IMERS.
2004 M.Bartolini; V.Cavrini; V.Andrisano
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 3. Effect of replacing the inner polymethylene chain with cyclic moieties
2004 TUMIATTI V.; ANDRISANO V.; BANZI R.; BARTOLINI M.; MINARINI A.; ROSINI M.; MELCHIORRE C.
RAPID ON-LINE SCREENING AND CHARACTERIZATION OF NEW INHIBITORS BY USING AN ACHE-MICRO-REACTOR
2004 M.Bartolini; V.Cavrini; V.Andrisano
DEVELOPMENT AND CHARACTERIZATION OF A PACKED AChE-micro-IMER FOR DRUG DISCOVERY IN ALZHEIMER’S DISEASE
2004 M.Bartolini; V.Cavrini; V.Andrisano
MEMOQUIN: A MULTIPOTENT ACETYLCHOLINESTERASE INHIBITOR WITH EXCELLENT IN VIVO ACTIVITY
2004 A.Cavalli; ML Bolognesi; M.Bartolini; V.Andrisano; C.Melchiorre; M.Recanatini; S.Capsoni; A.Cattaneo
Memoquin: a new therapeutic poly-agent for Alzheimer's disease
2004 Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Margotti E.; Capsoni S.; Cattaneo A.
Derivati a struttura benzofenonica come inibitori dell'acetilcolinesterasi
2004 F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; V. Andrisano; M. Bartolini; A. Cavalli; M. Recanatini; P. Valenti
Analogues of the dual acetylcholinesterase inhibitor AP2238: synthesis and SAR
2004 L. Piazzi; M. Bartolini; F. Belluti; A. Bisi; A. Cavalli; S. Gobbi; A. Rampa; P. Valenti
Monolytic micro-immobilized-enzyme reactor with human recombinant acetylcholinesterase for on-line inhibition studies
2004 BARTOLINI M; CAVRINI V.; ANDRISANO V
Titolo | Autore(i) | Anno | Periodico | Editore | Tipo | File |
---|---|---|---|---|---|---|
SAR of 9-amino-1,2,3-4-tetrahydroacridine-based acetylcholinesterase inhibitors: Synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues | Recanatini M.; Cavalli A.; Belluti F.; Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Valenti P.; Andris...ano V.; Bartolini M.; Cavrini V. | 2000-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives | Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Caval...li A.; Recanatini M.; Valenti P. | 2001-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure | Bolognesi M.L.; Bixel M.G.; Marucci G.; Bartolini M.; Krauss M.; Angeli P.; Antonello A.; Rosini ...M.; Tumiatti V.; Hucho F.; Melchiorre C. | 2002-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy | Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valen...ti P.; Recanatini M. | 2003-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Analytical methods for the determination of folic acid in a polymeric micellar carrier | Andrisano V.; Bartolini M.; Bertucci C.; Cavrini V.; Luppi B.; Cerchiara T. | 2003-01-01 | JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS | - | 1.01 Articolo in rivista | 2003 Analytical methods for the determination of folic acid in a polymeric micellar carrier.pdf |
Analytical methods for the determination of folic acid in a polymeric micellar carrier | Andrisano V.; Bartolini M.; Bertucci C.; Cavrini V.; Luppi B.; Cerchiara T. | 2003-01-01 | JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS | - | 1.01 Articolo in rivista | - |
Design, synthesis, and biological evaluation of conformationally restricted rivastigmine analogues | Bolognesi M. L.; Bartolini M.; Cavalli A.; Andrisano V.; Rosini M.; Minarini A.; Melchiorre C. | 2004-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
Evaluation of the inhibitory potency of a new series of AChE-inhibitors by using a monolithic AChE-micro-IMER | M. Bartolini; V. Tumiatti; V. Andrisano | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
METODI ANALITICI INTEGRATI PER LA VALUTAZIONE DEL PROFILO D’AZIONE DI NUOVI FARMACI ANTI-ALZHEIMER. | M. Bartolini; C. Bertucci; V. Cavrini; V. Andrisano | 2004-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
Memoquin: a new compound to attack Alzheimer's disease drug discovery | Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Capsoni S.;... Cattaneo A. | 2004-01-01 | - | s.l. | 4.02 Riassunto (Abstract) | - |
INTEGRATED ANALYTICAL APPROACHES FOR ALZHEIMER’S DISEASE NEW DRUG DISCOVERY | M. Bartolini; C. Bertucci; V. Cavrini; V. Andrisano. | 2004-01-01 | - | s.n | 4.01 Contributo in Atti di convegno | - |
CHOOSING THE RIGHT CHROMATOGRAPHIC SUPPORT FOR ENZYME-BASED MICRO-IMERS. | M.Bartolini; V.Cavrini; V.Andrisano | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 3. Effect of replacing the inner polymethylene chain with cyclic moieties | TUMIATTI V.; ANDRISANO V.; BANZI R.; BARTOLINI M.; MINARINI A.; ROSINI M.; MELCHIORRE C. | 2004-01-01 | JOURNAL OF MEDICINAL CHEMISTRY | - | 1.01 Articolo in rivista | - |
RAPID ON-LINE SCREENING AND CHARACTERIZATION OF NEW INHIBITORS BY USING AN ACHE-MICRO-REACTOR | M.Bartolini; V.Cavrini; V.Andrisano | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
DEVELOPMENT AND CHARACTERIZATION OF A PACKED AChE-micro-IMER FOR DRUG DISCOVERY IN ALZHEIMER’S DISEASE | M.Bartolini; V.Cavrini; V.Andrisano | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
MEMOQUIN: A MULTIPOTENT ACETYLCHOLINESTERASE INHIBITOR WITH EXCELLENT IN VIVO ACTIVITY | A.Cavalli; ML Bolognesi; M.Bartolini; V.Andrisano; C.Melchiorre; M.Recanatini; S.Capsoni; A.Cattaneo | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Memoquin: a new therapeutic poly-agent for Alzheimer's disease | Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Margotti E....; Capsoni S.; Cattaneo A. | 2004-01-01 | NEUROBIOLOGY OF AGING | - | 4.02 Riassunto (Abstract) | - |
Derivati a struttura benzofenonica come inibitori dell'acetilcolinesterasi | F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; V. Andrisano; M. Bartolini; A. Cavalli; M. Re...canatini; P. Valenti | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Analogues of the dual acetylcholinesterase inhibitor AP2238: synthesis and SAR | L. Piazzi; M. Bartolini; F. Belluti; A. Bisi; A. Cavalli; S. Gobbi; A. Rampa; P. Valenti | 2004-01-01 | - | s.n | 4.02 Riassunto (Abstract) | - |
Monolytic micro-immobilized-enzyme reactor with human recombinant acetylcholinesterase for on-line inhibition studies | BARTOLINI M; CAVRINI V.; ANDRISANO V | 2004-01-01 | JOURNAL OF CHROMATOGRAPHY A | - | 1.01 Articolo in rivista | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile