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Mostrati risultati da 1 a 20 di 248
Titolo Autore(i) Anno Periodico Editore Tipo File
SAR of 9-amino-1,2,3-4-tetrahydroacridine-based acetylcholinesterase inhibitors: Synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues Recanatini M.; Cavalli A.; Belluti F.; Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Valenti P.; Andris...ano V.; Bartolini M.; Cavrini V. 2000-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Caval...li A.; Recanatini M.; Valenti P. 2001-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure Bolognesi M.L.; Bixel M.G.; Marucci G.; Bartolini M.; Krauss M.; Angeli P.; Antonello A.; Rosini ...M.; Tumiatti V.; Hucho F.; Melchiorre C. 2002-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valen...ti P.; Recanatini M. 2003-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Analytical methods for the determination of folic acid in a polymeric micellar carrier Andrisano V.; Bartolini M.; Bertucci C.; Cavrini V.; Luppi B.; Cerchiara T. 2003-01-01 JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS - 1.01 Articolo in rivista 2003 Analytical methods for the determination of folic acid in a polymeric micellar carrier.pdf
Analytical methods for the determination of folic acid in a polymeric micellar carrier Andrisano V.; Bartolini M.; Bertucci C.; Cavrini V.; Luppi B.; Cerchiara T. 2003-01-01 JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS - 1.01 Articolo in rivista -
Design, synthesis, and biological evaluation of conformationally restricted rivastigmine analogues Bolognesi M. L.; Bartolini M.; Cavalli A.; Andrisano V.; Rosini M.; Minarini A.; Melchiorre C. 2004-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
Evaluation of the inhibitory potency of a new series of AChE-inhibitors by using a monolithic AChE-micro-IMER M. Bartolini; V. Tumiatti; V. Andrisano 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
METODI ANALITICI INTEGRATI PER LA VALUTAZIONE DEL PROFILO D’AZIONE DI NUOVI FARMACI ANTI-ALZHEIMER. M. Bartolini; C. Bertucci; V. Cavrini; V. Andrisano 2004-01-01 - s.n 4.01 Contributo in Atti di convegno -
Memoquin: a new compound to attack Alzheimer's disease drug discovery Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Capsoni S.;... Cattaneo A. 2004-01-01 - s.l. 4.02 Riassunto (Abstract) -
INTEGRATED ANALYTICAL APPROACHES FOR ALZHEIMER’S DISEASE NEW DRUG DISCOVERY M. Bartolini; C. Bertucci; V. Cavrini; V. Andrisano. 2004-01-01 - s.n 4.01 Contributo in Atti di convegno -
CHOOSING THE RIGHT CHROMATOGRAPHIC SUPPORT FOR ENZYME-BASED MICRO-IMERS. M.Bartolini; V.Cavrini; V.Andrisano 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 3. Effect of replacing the inner polymethylene chain with cyclic moieties TUMIATTI V.; ANDRISANO V.; BANZI R.; BARTOLINI M.; MINARINI A.; ROSINI M.; MELCHIORRE C. 2004-01-01 JOURNAL OF MEDICINAL CHEMISTRY - 1.01 Articolo in rivista -
RAPID ON-LINE SCREENING AND CHARACTERIZATION OF NEW INHIBITORS BY USING AN ACHE-MICRO-REACTOR M.Bartolini; V.Cavrini; V.Andrisano 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
DEVELOPMENT AND CHARACTERIZATION OF A PACKED AChE-micro-IMER FOR DRUG DISCOVERY IN ALZHEIMER’S DISEASE M.Bartolini; V.Cavrini; V.Andrisano 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
MEMOQUIN: A MULTIPOTENT ACETYLCHOLINESTERASE INHIBITOR WITH EXCELLENT IN VIVO ACTIVITY A.Cavalli; ML Bolognesi; M.Bartolini; V.Andrisano; C.Melchiorre; M.Recanatini; S.Capsoni; A.Cattaneo 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
Memoquin: a new therapeutic poly-agent for Alzheimer's disease Cavalli A.; Bolognesi M.L.; Bartolini M.; Andrisano V.; Melchiorre C.; Recanatini M.; Margotti E....; Capsoni S.; Cattaneo A. 2004-01-01 NEUROBIOLOGY OF AGING - 4.02 Riassunto (Abstract) -
Derivati a struttura benzofenonica come inibitori dell'acetilcolinesterasi F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; V. Andrisano; M. Bartolini; A. Cavalli; M. Re...canatini; P. Valenti 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
Analogues of the dual acetylcholinesterase inhibitor AP2238: synthesis and SAR L. Piazzi; M. Bartolini; F. Belluti; A. Bisi; A. Cavalli; S. Gobbi; A. Rampa; P. Valenti 2004-01-01 - s.n 4.02 Riassunto (Abstract) -
Monolytic micro-immobilized-enzyme reactor with human recombinant acetylcholinesterase for on-line inhibition studies BARTOLINI M; CAVRINI V.; ANDRISANO V 2004-01-01 JOURNAL OF CHROMATOGRAPHY A - 1.01 Articolo in rivista -
Mostrati risultati da 1 a 20 di 248
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